AR091679A1 - Modulares alostericos positivos del receptor de acetilcolina nicotinico - Google Patents
Modulares alostericos positivos del receptor de acetilcolina nicotinicoInfo
- Publication number
- AR091679A1 AR091679A1 ARP130102397A AR091679A1 AR 091679 A1 AR091679 A1 AR 091679A1 AR P130102397 A ARP130102397 A AR P130102397A AR 091679 A1 AR091679 A1 AR 091679A1
- Authority
- AR
- Argentina
- Prior art keywords
- acetilcoline
- nicotinic
- receiver
- positive allosteric
- modular
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/EP2012/063219 WO2013007621A1 (fr) | 2011-07-08 | 2012-07-06 | Modulateurs allostériques positifs des récepteurs nicotiniques d'acétylcholine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR091679A1 true AR091679A1 (es) | 2015-02-18 |
Family
ID=48745970
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP130102397 AR091679A1 (es) | 2012-07-06 | 2013-07-05 | Modulares alostericos positivos del receptor de acetilcolina nicotinico |
| ARP130102396 AR091678A1 (es) | 2012-07-06 | 2013-07-05 | Modulares alostericos positivos del receptor de acetilcolina nicotinico |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP130102396 AR091678A1 (es) | 2012-07-06 | 2013-07-05 | Modulares alostericos positivos del receptor de acetilcolina nicotinico |
Country Status (2)
| Country | Link |
|---|---|
| AR (2) | AR091679A1 (fr) |
| WO (2) | WO2014006120A1 (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GEP20207149B (en) | 2016-03-22 | 2020-09-10 | Merck Sharp & Dohme | Allosteric modulators of nicotinic acetylcholine receptors |
| TWI839355B (zh) | 2018-05-01 | 2024-04-21 | 美商默沙東有限責任公司 | 菸鹼乙醯膽鹼受體之螺哌啶異位調節劑 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2010003155A (es) | 2007-10-04 | 2010-04-01 | Hoffmann La Roche | Derivados de ciclopropil aril amida y uso de los mismos. |
| CN105130957A (zh) | 2009-05-29 | 2015-12-09 | 拉夸里亚创药株式会社 | 作为钙或钠通道阻滞剂的芳基取代羧酰胺衍生物 |
| US8497271B2 (en) * | 2009-10-07 | 2013-07-30 | Bristol-Myers Squibb Company | Modulators of G protein-coupled receptor 88 |
| UA111746C2 (uk) | 2011-07-08 | 2016-06-10 | Х. Луннбек А/С | Позитивні алостеричні модулятори нікотинового рецептора ацетилхоліну |
-
2013
- 2013-07-04 WO PCT/EP2013/064093 patent/WO2014006120A1/fr active Application Filing
- 2013-07-04 WO PCT/EP2013/064088 patent/WO2014006117A1/fr active Application Filing
- 2013-07-05 AR ARP130102397 patent/AR091679A1/es unknown
- 2013-07-05 AR ARP130102396 patent/AR091678A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2014006117A1 (fr) | 2014-01-09 |
| WO2014006120A1 (fr) | 2014-01-09 |
| AR091678A1 (es) | 2015-02-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |