AR081769A1 - Derivados indazolicos e intermediarios para su produccion, utiles como agentes profilacticos o terapeuticos para enfermedades degenerativas coriorretinales - Google Patents

Derivados indazolicos e intermediarios para su produccion, utiles como agentes profilacticos o terapeuticos para enfermedades degenerativas coriorretinales

Info

Publication number
AR081769A1
AR081769A1 ARP110101839A ARP110101839A AR081769A1 AR 081769 A1 AR081769 A1 AR 081769A1 AR P110101839 A ARP110101839 A AR P110101839A AR P110101839 A ARP110101839 A AR P110101839A AR 081769 A1 AR081769 A1 AR 081769A1
Authority
AR
Argentina
Prior art keywords
production
useful
chorioretinal
formula
compound represented
Prior art date
Application number
ARP110101839A
Other languages
English (en)
Inventor
Akira Takama
Masahiko Hagihara
Koji Ohashi
Takeshi Matsugi
Yasunori Tsuzaki
Shinichiro Hirai
Hiroshi Nishida
Tomokazu Fujimoto
Kazutaka Kido
Ken-Ichi Komori
Original Assignee
Santen Pharmaceutical Co Ltd
Ube Industries
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Santen Pharmaceutical Co Ltd, Ube Industries filed Critical Santen Pharmaceutical Co Ltd
Publication of AR081769A1 publication Critical patent/AR081769A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cardiology (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Compuesto representado por la fórmula (1) o una sal farmacéuticamente aceptable del mismo que tiene un efecto supresor sobre la muerte de las células fotorreceptoras en un modelo en ratón de trastorno por la luz. Por lo tanto, es útil como agente profiláctico o terapéutico para una enfermedad degenerativa coriorretinal sustancialmente no acompañada de neovascularización, por ejemplo, degeneración macular de tipo seco relacionada con la edad, retinitis pigmentosa, atrofia girata de coroides y retina, y para un trastorno coriorretinal que acompaña a una enfermedad con dichas características. También se provee un compuesto representado por la fórmula (1) o una sal del mismo y un intermediario para su producción para utilizar en la profilaxis o terapia de la enfermedad degenerativa coriorretinal, y el uso de un compuesto representado por la fórmula (1) o una sal del mismo farmacéuticamente aceptable para la producción de un agente profiláctico o terapéutico para la enfermedad degenerativa coriorretinal.
ARP110101839A 2010-05-27 2011-05-27 Derivados indazolicos e intermediarios para su produccion, utiles como agentes profilacticos o terapeuticos para enfermedades degenerativas coriorretinales AR081769A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2010121821 2010-05-27

Publications (1)

Publication Number Publication Date
AR081769A1 true AR081769A1 (es) 2012-10-17

Family

ID=45003996

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP110101839A AR081769A1 (es) 2010-05-27 2011-05-27 Derivados indazolicos e intermediarios para su produccion, utiles como agentes profilacticos o terapeuticos para enfermedades degenerativas coriorretinales

Country Status (4)

Country Link
JP (1) JP2012006919A (es)
AR (1) AR081769A1 (es)
TW (1) TW201202214A (es)
WO (1) WO2011149010A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2656292T3 (es) * 2012-05-01 2018-02-26 Translatum Medicus Inc. Métodos de tratamiento y diagnóstico de enfermedades oculares que causan ceguera
AU2014285301A1 (en) * 2013-07-04 2016-01-21 Nippon Soda Co., Ltd. Phenylimidazole derivative, and therapeutic medicine or preventive medicine for inflammatory disease, etc.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002083175A1 (fr) * 2001-04-11 2002-10-24 Senju Pharmaceutical Co., Ltd. Agents ameliorant la fonction visuelle
KR101163800B1 (ko) * 2003-10-15 2012-07-09 산텐 세이야꾸 가부시키가이샤 신규 인다졸 유도체
WO2006112313A1 (ja) * 2005-04-13 2006-10-26 Ube Industries, Ltd. インダゾール誘導体を有効成分として含む網膜神経細胞保護剤

Also Published As

Publication number Publication date
TW201202214A (en) 2012-01-16
JP2012006919A (ja) 2012-01-12
WO2011149010A1 (ja) 2011-12-01

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