AR068439A1 - Derivado de 6-pirimidinil-pirimid-2-ona - Google Patents
Derivado de 6-pirimidinil-pirimid-2-onaInfo
- Publication number
- AR068439A1 AR068439A1 ARP080103982A ARP080103982A AR068439A1 AR 068439 A1 AR068439 A1 AR 068439A1 AR P080103982 A ARP080103982 A AR P080103982A AR P080103982 A ARP080103982 A AR P080103982A AR 068439 A1 AR068439 A1 AR 068439A1
- Authority
- AR
- Argentina
- Prior art keywords
- pirimid
- pirimidinil
- ona
- derived
- disease
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Diabetes (AREA)
- Ophthalmology & Optometry (AREA)
- Physical Education & Sports Medicine (AREA)
- Hematology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Obesity (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Endocrinology (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Dermatology (AREA)
- Cardiology (AREA)
- Emergency Medicine (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Un compuesto representado por la formula (1) o una sal farmacéuticamente aceptable de él: que se usa para el tratamiento preventivo y/o terapéutico de una enfermedad provocada por la actividad anormal de la tau proteína cinasa 1 tal como enfermedades neurodegenerativas (por ejemplo, la enfermedad de Alzheimer).
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2007269485 | 2007-09-14 | ||
JP2007275713 | 2007-09-25 | ||
EP08290028A EP2078717A1 (en) | 2008-01-11 | 2008-01-11 | 6-Pyrimidinyl-pyrimid-2-one derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
AR068439A1 true AR068439A1 (es) | 2009-11-18 |
Family
ID=39874051
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP080103982A AR068439A1 (es) | 2007-09-14 | 2008-09-12 | Derivado de 6-pirimidinil-pirimid-2-ona |
Country Status (15)
Country | Link |
---|---|
US (2) | US8198437B2 (es) |
EP (1) | EP2193129B1 (es) |
JP (1) | JP5249320B2 (es) |
KR (1) | KR20100074182A (es) |
CN (1) | CN101883770A (es) |
AR (1) | AR068439A1 (es) |
AU (1) | AU2008297817A1 (es) |
BR (1) | BRPI0816705A2 (es) |
CA (1) | CA2698819A1 (es) |
EA (1) | EA201070367A1 (es) |
MX (1) | MX2010002765A (es) |
NZ (1) | NZ584277A (es) |
TW (1) | TW200927134A (es) |
WO (1) | WO2009035162A1 (es) |
ZA (1) | ZA201002213B (es) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200813015A (en) * | 2006-03-15 | 2008-03-16 | Mitsubishi Pharma Corp | 2-(cyclic amino)-pyrimidone derivatives |
MX2010002765A (es) | 2007-09-14 | 2010-05-19 | Mitsubishi Tanabe Pharma Corp | Derivado de 6-pirimidinil-pirimid-4-ona. |
TW201043618A (en) | 2009-03-10 | 2010-12-16 | Sanofi Aventis | Intermediate compound for synthesizing pharmaceutical agent and production method thereof |
EP2464632A1 (en) | 2009-08-13 | 2012-06-20 | Mitsubishi Tanabe Pharma Corporation | Pyrimidone derivatives used as tau protein kinase 1 inhibitors |
WO2011019089A1 (en) * | 2009-08-13 | 2011-02-17 | Mitsubishi Tanabe Pharma Corporation | Pyrimidone derivatives used as tau protein kinase 1 inhibitors |
EP2567959B1 (en) | 2011-09-12 | 2014-04-16 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
EP3453706A1 (en) | 2017-09-08 | 2019-03-13 | Basf Se | Pesticidal imidazole compounds |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2116460A1 (en) | 1993-03-02 | 1994-09-03 | Mitsubishi Chemical Corporation | Preventive or therapeutic agents for alzheimer's disease, a screening method of alzheimer's disease and tau-protein kinase i originated from human being |
MXPA04002662A (es) * | 2001-09-21 | 2004-11-22 | Sanofi Aventis | Derivados de 3-substituida-4-pirimidona. |
AR036604A1 (es) * | 2001-09-21 | 2004-09-22 | Mitsubishi Pharma Corp | Derivados de 4-pirimidona 3-sustituida |
TWI357408B (en) * | 2003-03-26 | 2012-02-01 | Mitsubishi Tanabe Pharma Corp | 3-substituted-4-pyrimidone derivatives |
TW200621760A (en) * | 2004-09-09 | 2006-07-01 | Mitsubishi Pharma Corp | 2-morpholino-4-pyrimidone compound |
ZA200703383B (en) | 2004-09-29 | 2009-05-27 | Mitsubishi Pharma Corp | 6-(pyridinyl)-4-pyrimidone derivates as tau protein kinase 1 inhibitors |
TW200740779A (en) | 2005-07-22 | 2007-11-01 | Mitsubishi Pharma Corp | Intermediate compound for synthesizing pharmaceutical agent and production method thereof |
TW200813015A (en) | 2006-03-15 | 2008-03-16 | Mitsubishi Pharma Corp | 2-(cyclic amino)-pyrimidone derivatives |
AR064660A1 (es) * | 2006-12-26 | 2009-04-15 | Mitsubishi Tanabe Pharma Corp | Derivados de pirimidinona 6-heterociclica 2-sustituida, medicamentos que los contienen y usos para prevenir y/o tratar enfermedades neurodegenerativas entre otras |
MX2010002765A (es) | 2007-09-14 | 2010-05-19 | Mitsubishi Tanabe Pharma Corp | Derivado de 6-pirimidinil-pirimid-4-ona. |
AR076014A1 (es) | 2009-04-02 | 2011-05-11 | Sanofi Aventis | Derivados de 3- (1,4) oxazepan -4-pirimidona |
-
2008
- 2008-09-12 MX MX2010002765A patent/MX2010002765A/es not_active Application Discontinuation
- 2008-09-12 TW TW097135175A patent/TW200927134A/zh unknown
- 2008-09-12 CA CA2698819A patent/CA2698819A1/en not_active Abandoned
- 2008-09-12 BR BRPI0816705 patent/BRPI0816705A2/pt not_active IP Right Cessation
- 2008-09-12 JP JP2010510582A patent/JP5249320B2/ja not_active Expired - Fee Related
- 2008-09-12 NZ NZ584277A patent/NZ584277A/en not_active IP Right Cessation
- 2008-09-12 US US12/677,213 patent/US8198437B2/en not_active Expired - Fee Related
- 2008-09-12 AU AU2008297817A patent/AU2008297817A1/en not_active Abandoned
- 2008-09-12 WO PCT/JP2008/066936 patent/WO2009035162A1/en active Application Filing
- 2008-09-12 EP EP08831179A patent/EP2193129B1/en active Active
- 2008-09-12 KR KR1020107008065A patent/KR20100074182A/ko not_active Application Discontinuation
- 2008-09-12 EA EA201070367A patent/EA201070367A1/ru unknown
- 2008-09-12 CN CN2008801137447A patent/CN101883770A/zh active Pending
- 2008-09-12 AR ARP080103982A patent/AR068439A1/es not_active Application Discontinuation
-
2010
- 2010-03-29 ZA ZA2010/02213A patent/ZA201002213B/en unknown
-
2012
- 2012-05-09 US US13/467,302 patent/US8518939B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP2193129A1 (en) | 2010-06-09 |
WO2009035162A1 (en) | 2009-03-19 |
TW200927134A (en) | 2009-07-01 |
KR20100074182A (ko) | 2010-07-01 |
US20110021773A1 (en) | 2011-01-27 |
AU2008297817A1 (en) | 2009-03-19 |
CA2698819A1 (en) | 2009-03-19 |
EP2193129B1 (en) | 2012-10-24 |
NZ584277A (en) | 2011-11-25 |
JP2010538969A (ja) | 2010-12-16 |
US8198437B2 (en) | 2012-06-12 |
US8518939B2 (en) | 2013-08-27 |
EA201070367A1 (ru) | 2010-08-30 |
MX2010002765A (es) | 2010-05-19 |
BRPI0816705A2 (pt) | 2015-03-17 |
JP5249320B2 (ja) | 2013-07-31 |
CN101883770A (zh) | 2010-11-10 |
ZA201002213B (en) | 2011-06-29 |
US20120252812A1 (en) | 2012-10-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |