AR065352A1 - Derivados de piridil-triazolopirimidina, pesticidas que los contienen y proceso para prepararlos. - Google Patents
Derivados de piridil-triazolopirimidina, pesticidas que los contienen y proceso para prepararlos.Info
- Publication number
- AR065352A1 AR065352A1 ARP080100635A ARP080100635A AR065352A1 AR 065352 A1 AR065352 A1 AR 065352A1 AR P080100635 A ARP080100635 A AR P080100635A AR P080100635 A ARP080100635 A AR P080100635A AR 065352 A1 AR065352 A1 AR 065352A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- substituted
- aryl
- hydrogen
- nr4r5
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Veterinary Medicine (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Reivindicacion 1: Un derivado de piridil-triazolopirimidina representado por la formula (1) o su sal, en la cual R1 es hidrogeno, alquilo que puede estar sustituido con A, cicloalquilo que puede estar sustituido con A, alquenilo que puede estarsustituido con A, alquinilo que puede estar sustituido con A, halogeno, ciano, arilo, un grupo heterocíclico que puede estar sustituido con alquilo, OR2, S(O)nR3 o NR4R5; R2 es hidrogeno, alquilo, alquenilo, alquinilo, haloalquilo, alcoxialquilo,acetilo o arilo; R3 es alquilo o acetilo; R4 es hidrogeno o alquilo; R5 es hidrogeno, alquilo, acetilo, CH2CH2OR2 o CH2CN; A es halogeno, OR2, S(O)nR3, NR4R5, ciano, alquilo, cicloalquilo, arilo, un grupo heterocíclico, SCH2COOR2 o -CH(CN)2; X esalquilo, alquenilo, alquinilo, arilo, halogeno, haloalquilo, ciano, nitro, NR4R5, S(O)nR3, COR2 o COOR2; m es un entero de 1 a 4 y n es un entero de 0 a 2; siempre que se excluya la 7-(3-cloro-5-(trifluormetil)piridin-2-il)-[1,2,4)triazolo[1,5-a]pirimidina.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2007034371 | 2007-02-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR065352A1 true AR065352A1 (es) | 2009-06-03 |
Family
ID=39319691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080100635A AR065352A1 (es) | 2007-02-15 | 2008-02-14 | Derivados de piridil-triazolopirimidina, pesticidas que los contienen y proceso para prepararlos. |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US8124760B2 (es) |
| EP (1) | EP2118113B1 (es) |
| JP (1) | JP5231829B2 (es) |
| KR (1) | KR20090119854A (es) |
| CN (1) | CN101611037B (es) |
| AR (1) | AR065352A1 (es) |
| AU (1) | AU2008215426A1 (es) |
| BR (1) | BRPI0808126B1 (es) |
| CA (1) | CA2676736A1 (es) |
| CL (1) | CL2008000494A1 (es) |
| DK (1) | DK2118113T3 (es) |
| EG (1) | EG25529A (es) |
| ES (1) | ES2400574T3 (es) |
| HR (1) | HRP20130324T1 (es) |
| IL (1) | IL200416A0 (es) |
| MA (1) | MA31163B1 (es) |
| MX (1) | MX2009008772A (es) |
| NZ (1) | NZ578803A (es) |
| PL (1) | PL2118113T3 (es) |
| PT (1) | PT2118113E (es) |
| RS (1) | RS52789B (es) |
| SI (1) | SI2118113T1 (es) |
| TW (1) | TW200902535A (es) |
| WO (1) | WO2008099902A1 (es) |
| ZA (1) | ZA200905370B (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2222639A1 (en) | 2007-11-21 | 2010-09-01 | Decode Genetics EHF | Biaryl pde4 inhibitors for treating pulmonary and cardiovascular disorders |
| JP2010065026A (ja) * | 2008-08-13 | 2010-03-25 | Ishihara Sangyo Kaisha Ltd | ピリジル−トリアゾロピリミジン誘導体又はその塩、並びにそれらを含有する有害生物防除剤 |
| WO2010059836A1 (en) * | 2008-11-20 | 2010-05-27 | Decode Genetics Ehf | Substituted aza-bridged bicyclics for cardiovascular and cns disease |
| TW201029575A (en) | 2009-01-29 | 2010-08-16 | Ishihara Sangyo Kaisha | Triazolopyrimidine derivative or its salt, process for producing the same and pesticide containing the same |
| JP2011168582A (ja) * | 2010-01-21 | 2011-09-01 | Ishihara Sangyo Kaisha Ltd | トリアゾロピリジン誘導体又はその塩、それらの製造方法及びそれらを含有する有害生物防除剤 |
| US8609717B2 (en) * | 2010-08-18 | 2013-12-17 | Samumed, Llc | β- and γ-diketones and γ-hydroxyketones as WNT/β-catenin signaling pathway activators |
| JP5959537B2 (ja) | 2011-01-28 | 2016-08-02 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 置換ピリジニル−ピリミジン及び医薬としてのその使用 |
| KR101339572B1 (ko) * | 2011-09-05 | 2013-12-10 | 이정은 | 초미립자 약제 살포기용 첨가제 |
| ES2709824T3 (es) | 2013-02-22 | 2019-04-17 | Samumed Llc | Gamma-dicetonas como activadores de la ruta de señalización Wnt/beta-catenina |
| RU2727039C2 (ru) | 2014-08-20 | 2020-07-17 | СЭМЬЮМЕД, ЭлЭлСи | Гамма-дикетоны для лечения и профилактики старения кожи и морщин |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4209621A (en) | 1979-04-27 | 1980-06-24 | American Cyanamid Company | (Substituted-phenyl)-1,2,4-triazolo[4,3-a]-pyrimidines and (substituted-phenyl)-1,2,4-triazolo[1,5-a]pyrimidines |
| US4444774A (en) * | 1982-07-29 | 1984-04-24 | American Cyanamid Company | 7-Heteroaryl[1,2,4]triazolo[1,5-a]pyrimidines |
| US4562192A (en) | 1984-02-03 | 1985-12-31 | G. D. Searle & Co. | 6-Substituted-5-phenyltetrazolo[1,5-a][1,2,4]triazole[1,5-c]pyrimidines, and pharmaceutical compositions containing them |
| HUP0300798A3 (en) * | 2000-06-30 | 2006-02-28 | Wyeth Corp | Substituted-triazolopyrimidines and their use as anticancer agents and pharmaceutical compositions containing them |
| WO2004082383A1 (en) * | 2003-03-17 | 2004-09-30 | Basf Aktiengesellschaft | Use of triazolopyrimidines for combating nematode diseases of plants |
-
2008
- 2008-02-05 JP JP2008025572A patent/JP5231829B2/ja not_active Expired - Fee Related
- 2008-02-07 CA CA002676736A patent/CA2676736A1/en not_active Abandoned
- 2008-02-07 CN CN2008800050569A patent/CN101611037B/zh not_active Expired - Fee Related
- 2008-02-07 AU AU2008215426A patent/AU2008215426A1/en not_active Abandoned
- 2008-02-07 PT PT87113098T patent/PT2118113E/pt unknown
- 2008-02-07 WO PCT/JP2008/052475 patent/WO2008099902A1/en active Application Filing
- 2008-02-07 US US12/526,520 patent/US8124760B2/en not_active Expired - Fee Related
- 2008-02-07 SI SI200830935T patent/SI2118113T1/sl unknown
- 2008-02-07 KR KR1020097016972A patent/KR20090119854A/ko not_active Application Discontinuation
- 2008-02-07 EP EP08711309A patent/EP2118113B1/en active Active
- 2008-02-07 BR BRPI0808126A patent/BRPI0808126B1/pt not_active IP Right Cessation
- 2008-02-07 MX MX2009008772A patent/MX2009008772A/es active IP Right Grant
- 2008-02-07 RS RS20130033A patent/RS52789B/en unknown
- 2008-02-07 NZ NZ578803A patent/NZ578803A/en not_active IP Right Cessation
- 2008-02-07 DK DK08711309.8T patent/DK2118113T3/da active
- 2008-02-07 ES ES08711309T patent/ES2400574T3/es active Active
- 2008-02-07 PL PL08711309T patent/PL2118113T3/pl unknown
- 2008-02-07 ZA ZA200905370A patent/ZA200905370B/xx unknown
- 2008-02-14 TW TW097105200A patent/TW200902535A/zh unknown
- 2008-02-14 AR ARP080100635A patent/AR065352A1/es not_active Application Discontinuation
- 2008-02-15 CL CL200800494A patent/CL2008000494A1/es unknown
-
2009
- 2009-08-04 MA MA32139A patent/MA31163B1/fr unknown
- 2009-08-12 EG EG2009081217A patent/EG25529A/xx active
- 2009-08-13 IL IL200416A patent/IL200416A0/en unknown
-
2013
- 2013-04-10 HR HRP20130324AT patent/HRP20130324T1/hr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX2009008772A (es) | 2009-08-25 |
| HRP20130324T1 (hr) | 2013-05-31 |
| IL200416A0 (en) | 2010-04-29 |
| BRPI0808126B1 (pt) | 2016-12-27 |
| MA31163B1 (fr) | 2010-02-01 |
| CN101611037B (zh) | 2012-11-28 |
| US20100087452A1 (en) | 2010-04-08 |
| JP5231829B2 (ja) | 2013-07-10 |
| EG25529A (en) | 2012-02-06 |
| KR20090119854A (ko) | 2009-11-20 |
| DK2118113T3 (da) | 2013-02-18 |
| NZ578803A (en) | 2011-11-25 |
| SI2118113T1 (sl) | 2013-06-28 |
| EP2118113B1 (en) | 2013-01-30 |
| CA2676736A1 (en) | 2008-08-21 |
| CN101611037A (zh) | 2009-12-23 |
| BRPI0808126A2 (pt) | 2014-09-16 |
| ES2400574T3 (es) | 2013-04-10 |
| PT2118113E (pt) | 2013-03-14 |
| TW200902535A (en) | 2009-01-16 |
| PL2118113T3 (pl) | 2013-06-28 |
| RS52789B (en) | 2013-10-31 |
| JP2008222707A (ja) | 2008-09-25 |
| EP2118113A1 (en) | 2009-11-18 |
| WO2008099902A1 (en) | 2008-08-21 |
| US8124760B2 (en) | 2012-02-28 |
| ZA200905370B (en) | 2010-10-27 |
| AU2008215426A1 (en) | 2008-08-21 |
| CL2008000494A1 (es) | 2008-06-27 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR065352A1 (es) | Derivados de piridil-triazolopirimidina, pesticidas que los contienen y proceso para prepararlos. | |
| ES2452299T3 (es) | Compuestos heterocíclicos fungicidas | |
| AR047533A1 (es) | Proceso para preparar carboxamidas 2-aminotiazol-5-aromaticas como inhibidores de la quinasa | |
| PE20181094A1 (es) | Derivados heterociclicos condensados sustituidos por 2-(het)arilo como pesticidas | |
| AR075635A1 (es) | N-alcoxiamidas de 6-(fenil sustituido)-4-aminopicolinatos y 2-(fenil sustituido)-6-amino-4-pirimidina carboxilatos, su uso como herbicidas selectivos para las cosechas y proceso de preparacion de dichos compuestos | |
| PE20171514A1 (es) | Heterociclos biciclicos como inhibidores de fgfr | |
| CU23926B1 (es) | Derivado de oxopirazina y herbicida | |
| UY33458A (es) | Derivados de metoxifenilo heterocíclicamente sustituidos con un grupo oxo, procedimientos para su preparación y uso de los mismos como medicamentos | |
| PE20190339A1 (es) | 1h-pirazolo[4,3-b] piridinas como inhibidores de pde1 | |
| AR056888A1 (es) | Derivados de heterociclil imidazol | |
| AR058562A1 (es) | Derivados de pirimido [4,5 b] (1,4) oxazinas , procedimientos de obtencion y su uso como inhibidores de acetil coa y dgat 1 | |
| AR047456A1 (es) | Derivados de amidas, procesos para su preparacion y uso como insecticidas | |
| AR054369A1 (es) | Compuestos de imidazol condensado y su uso como inhibidores de aldosterona sintasa | |
| AR080785A1 (es) | Derivados de imidazo[1,2-a]pirimidina ,proceso para prepararlos e intermediarios de dicha sintesis, composiciones farmaceuticas que los contienen y uso de los mismos en el tratamiento de patologias del sistema nervioso central,tales como esquizofrenia y parkinson, entre otros. | |
| AR060591A1 (es) | Compuestos imidazo | |
| AR086474A1 (es) | Compuestos de pirazol pesticidas | |
| ES2530943T3 (es) | Derivados de la cromenona con actividad antitumoral | |
| CR10346A (es) | Derivados de azabiciclo[3.1.0]hexil como modulares de los receptores de dopamina d3 | |
| ECSP099394A (es) | Derivados de quinuclidinol como antogonistas de receptores muscarínicos | |
| DOP2012000318A (es) | Compuestos heterociclicos fusionados | |
| AR080596A1 (es) | Compuestos alquilamido y composiciones farmaceuticas | |
| AR069531A1 (es) | Derivados de indolinona y procedimiento para su fabricacion | |
| NI201500134A (es) | Derivados de 2-((4-amino-3-(3-flúor-5-hidroxifenil)-1h-pirazolo[3,4-d]pirimidin-1-il) metil)-3-(2-(trifluorometil)bencil)quinazolina-4(3h)-ona y su uso como inhibidores de fosfoinositida 3-quinasas | |
| WO2009010789A3 (en) | Pyrimidine derivatives 934 | |
| CO6230982A2 (es) | Compuestos triciclicos que contienen actividad antagonista de factor de liberacion de corticotropina y composiciones farmaceuticas que los contienen |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |