AR065352A1 - Derivados de piridil-triazolopirimidina, pesticidas que los contienen y proceso para prepararlos. - Google Patents
Derivados de piridil-triazolopirimidina, pesticidas que los contienen y proceso para prepararlos.Info
- Publication number
- AR065352A1 AR065352A1 ARP080100635A ARP080100635A AR065352A1 AR 065352 A1 AR065352 A1 AR 065352A1 AR P080100635 A ARP080100635 A AR P080100635A AR P080100635 A ARP080100635 A AR P080100635A AR 065352 A1 AR065352 A1 AR 065352A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- substituted
- aryl
- hydrogen
- nr4r5
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Veterinary Medicine (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Reivindicacion 1: Un derivado de piridil-triazolopirimidina representado por la formula (1) o su sal, en la cual R1 es hidrogeno, alquilo que puede estar sustituido con A, cicloalquilo que puede estar sustituido con A, alquenilo que puede estarsustituido con A, alquinilo que puede estar sustituido con A, halogeno, ciano, arilo, un grupo heterocíclico que puede estar sustituido con alquilo, OR2, S(O)nR3 o NR4R5; R2 es hidrogeno, alquilo, alquenilo, alquinilo, haloalquilo, alcoxialquilo,acetilo o arilo; R3 es alquilo o acetilo; R4 es hidrogeno o alquilo; R5 es hidrogeno, alquilo, acetilo, CH2CH2OR2 o CH2CN; A es halogeno, OR2, S(O)nR3, NR4R5, ciano, alquilo, cicloalquilo, arilo, un grupo heterocíclico, SCH2COOR2 o -CH(CN)2; X esalquilo, alquenilo, alquinilo, arilo, halogeno, haloalquilo, ciano, nitro, NR4R5, S(O)nR3, COR2 o COOR2; m es un entero de 1 a 4 y n es un entero de 0 a 2; siempre que se excluya la 7-(3-cloro-5-(trifluormetil)piridin-2-il)-[1,2,4)triazolo[1,5-a]pirimidina.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2007034371 | 2007-02-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR065352A1 true AR065352A1 (es) | 2009-06-03 |
Family
ID=39319691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080100635A AR065352A1 (es) | 2007-02-15 | 2008-02-14 | Derivados de piridil-triazolopirimidina, pesticidas que los contienen y proceso para prepararlos. |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US8124760B2 (es) |
| EP (1) | EP2118113B1 (es) |
| JP (1) | JP5231829B2 (es) |
| KR (1) | KR20090119854A (es) |
| CN (1) | CN101611037B (es) |
| AR (1) | AR065352A1 (es) |
| AU (1) | AU2008215426A1 (es) |
| BR (1) | BRPI0808126B1 (es) |
| CA (1) | CA2676736A1 (es) |
| CL (1) | CL2008000494A1 (es) |
| DK (1) | DK2118113T3 (es) |
| EG (1) | EG25529A (es) |
| ES (1) | ES2400574T3 (es) |
| HR (1) | HRP20130324T1 (es) |
| IL (1) | IL200416A0 (es) |
| MA (1) | MA31163B1 (es) |
| MX (1) | MX2009008772A (es) |
| NZ (1) | NZ578803A (es) |
| PL (1) | PL2118113T3 (es) |
| PT (1) | PT2118113E (es) |
| RS (1) | RS52789B (es) |
| SI (1) | SI2118113T1 (es) |
| TW (1) | TW200902535A (es) |
| WO (1) | WO2008099902A1 (es) |
| ZA (1) | ZA200905370B (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009067621A1 (en) | 2007-11-21 | 2009-05-28 | Decode Genetics Ehf | Biaryl pde4 inhibitors for treating pulmonary and cardiovascular disorders |
| JP2010065026A (ja) * | 2008-08-13 | 2010-03-25 | Ishihara Sangyo Kaisha Ltd | ピリジル−トリアゾロピリミジン誘導体又はその塩、並びにそれらを含有する有害生物防除剤 |
| WO2010059836A1 (en) * | 2008-11-20 | 2010-05-27 | Decode Genetics Ehf | Substituted aza-bridged bicyclics for cardiovascular and cns disease |
| TW201029575A (en) | 2009-01-29 | 2010-08-16 | Ishihara Sangyo Kaisha | Triazolopyrimidine derivative or its salt, process for producing the same and pesticide containing the same |
| JP2011168582A (ja) * | 2010-01-21 | 2011-09-01 | Ishihara Sangyo Kaisha Ltd | トリアゾロピリジン誘導体又はその塩、それらの製造方法及びそれらを含有する有害生物防除剤 |
| JP6086864B2 (ja) | 2010-08-18 | 2017-03-01 | サミュメッド リミテッド ライアビリティ カンパニー | カテニンシグナル伝達経路活性化剤としてのジケトンおよびヒドロキシケトン |
| EP2668177B1 (en) | 2011-01-28 | 2014-10-22 | Boehringer Ingelheim International GmbH | Substituted pyridinyl-pyrimidines and their use as medicaments |
| KR101339572B1 (ko) * | 2011-09-05 | 2013-12-10 | 이정은 | 초미립자 약제 살포기용 첨가제 |
| AU2014218720B2 (en) | 2013-02-22 | 2018-09-27 | Samumed, Llc | Gamma-diketones as Wnt/beta -catenin signaling pathway activators |
| HUE046741T2 (hu) | 2014-08-20 | 2020-03-30 | Samumed Llc | Gamma-diketonok bõröregedés és ráncok megelõzésére és kezelésére |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4209621A (en) | 1979-04-27 | 1980-06-24 | American Cyanamid Company | (Substituted-phenyl)-1,2,4-triazolo[4,3-a]-pyrimidines and (substituted-phenyl)-1,2,4-triazolo[1,5-a]pyrimidines |
| US4444774A (en) * | 1982-07-29 | 1984-04-24 | American Cyanamid Company | 7-Heteroaryl[1,2,4]triazolo[1,5-a]pyrimidines |
| US4562192A (en) | 1984-02-03 | 1985-12-31 | G. D. Searle & Co. | 6-Substituted-5-phenyltetrazolo[1,5-a][1,2,4]triazole[1,5-c]pyrimidines, and pharmaceutical compositions containing them |
| AU7306201A (en) * | 2000-06-30 | 2002-01-14 | American Home Prod | Substituted-triazolopyrimidines as anticancer agents |
| WO2004082383A1 (en) * | 2003-03-17 | 2004-09-30 | Basf Aktiengesellschaft | Use of triazolopyrimidines for combating nematode diseases of plants |
-
2008
- 2008-02-05 JP JP2008025572A patent/JP5231829B2/ja not_active Expired - Fee Related
- 2008-02-07 AU AU2008215426A patent/AU2008215426A1/en not_active Abandoned
- 2008-02-07 PT PT87113098T patent/PT2118113E/pt unknown
- 2008-02-07 ES ES08711309T patent/ES2400574T3/es active Active
- 2008-02-07 CA CA002676736A patent/CA2676736A1/en not_active Abandoned
- 2008-02-07 DK DK08711309.8T patent/DK2118113T3/da active
- 2008-02-07 PL PL08711309T patent/PL2118113T3/pl unknown
- 2008-02-07 RS RS20130033A patent/RS52789B/en unknown
- 2008-02-07 BR BRPI0808126A patent/BRPI0808126B1/pt not_active IP Right Cessation
- 2008-02-07 US US12/526,520 patent/US8124760B2/en not_active Expired - Fee Related
- 2008-02-07 KR KR1020097016972A patent/KR20090119854A/ko not_active Application Discontinuation
- 2008-02-07 SI SI200830935T patent/SI2118113T1/sl unknown
- 2008-02-07 ZA ZA200905370A patent/ZA200905370B/xx unknown
- 2008-02-07 EP EP08711309A patent/EP2118113B1/en active Active
- 2008-02-07 MX MX2009008772A patent/MX2009008772A/es active IP Right Grant
- 2008-02-07 WO PCT/JP2008/052475 patent/WO2008099902A1/en active Application Filing
- 2008-02-07 CN CN2008800050569A patent/CN101611037B/zh not_active Expired - Fee Related
- 2008-02-07 NZ NZ578803A patent/NZ578803A/en not_active IP Right Cessation
- 2008-02-14 AR ARP080100635A patent/AR065352A1/es not_active Application Discontinuation
- 2008-02-14 TW TW097105200A patent/TW200902535A/zh unknown
- 2008-02-15 CL CL200800494A patent/CL2008000494A1/es unknown
-
2009
- 2009-08-04 MA MA32139A patent/MA31163B1/fr unknown
- 2009-08-12 EG EG2009081217A patent/EG25529A/xx active
- 2009-08-13 IL IL200416A patent/IL200416A0/en unknown
-
2013
- 2013-04-10 HR HRP20130324AT patent/HRP20130324T1/hr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP2118113B1 (en) | 2013-01-30 |
| AU2008215426A1 (en) | 2008-08-21 |
| RS52789B (en) | 2013-10-31 |
| WO2008099902A1 (en) | 2008-08-21 |
| DK2118113T3 (da) | 2013-02-18 |
| CN101611037B (zh) | 2012-11-28 |
| CN101611037A (zh) | 2009-12-23 |
| CL2008000494A1 (es) | 2008-06-27 |
| KR20090119854A (ko) | 2009-11-20 |
| MA31163B1 (fr) | 2010-02-01 |
| PT2118113E (pt) | 2013-03-14 |
| CA2676736A1 (en) | 2008-08-21 |
| HRP20130324T1 (hr) | 2013-05-31 |
| JP5231829B2 (ja) | 2013-07-10 |
| EG25529A (en) | 2012-02-06 |
| SI2118113T1 (sl) | 2013-06-28 |
| JP2008222707A (ja) | 2008-09-25 |
| IL200416A0 (en) | 2010-04-29 |
| ZA200905370B (en) | 2010-10-27 |
| BRPI0808126A2 (pt) | 2014-09-16 |
| ES2400574T3 (es) | 2013-04-10 |
| BRPI0808126B1 (pt) | 2016-12-27 |
| PL2118113T3 (pl) | 2013-06-28 |
| US20100087452A1 (en) | 2010-04-08 |
| NZ578803A (en) | 2011-11-25 |
| EP2118113A1 (en) | 2009-11-18 |
| TW200902535A (en) | 2009-01-16 |
| MX2009008772A (es) | 2009-08-25 |
| US8124760B2 (en) | 2012-02-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |