AR060412A1 - Una composicion farmaceutica utilizable para inhibir o evitar la formacion no deseada de tejido fibroso y uso de la n- sulfoetilnicotinamida para inhibir o evitar la formacion no deseada de tejido fibroso - Google Patents

Una composicion farmaceutica utilizable para inhibir o evitar la formacion no deseada de tejido fibroso y uso de la n- sulfoetilnicotinamida para inhibir o evitar la formacion no deseada de tejido fibroso

Info

Publication number
AR060412A1
AR060412A1 ARP070101508A ARP070101508A AR060412A1 AR 060412 A1 AR060412 A1 AR 060412A1 AR P070101508 A ARP070101508 A AR P070101508A AR P070101508 A ARP070101508 A AR P070101508A AR 060412 A1 AR060412 A1 AR 060412A1
Authority
AR
Argentina
Prior art keywords
inhibit
avoid
formation
fiber
sulfoetilnicotinamida
Prior art date
Application number
ARP070101508A
Other languages
English (en)
Inventor
Moises Gabriel Zeitune
Ruben Martin Laguens
Original Assignee
Creactivar S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Creactivar S A filed Critical Creactivar S A
Priority to ARP070101508A priority Critical patent/AR060412A1/es
Priority to PCT/MX2008/000049 priority patent/WO2008123759A1/es
Publication of AR060412A1 publication Critical patent/AR060412A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides
    • C07D213/82Amides; Imides in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4406Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 3, e.g. zimeldine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un compuesto que inhibe, evita, o previene la formacion no deseada de tejido fibroso que responde a la formula estructural (1), sulfoetilnicotinamida (NESA, ácido 2- (N-nicotinamido] etanosulfonico) y a los derivados farmacéuticamente aceptables del mismo. La composicion farmacéutica que comprende al compuesto N-sulfoetilnicotinamida (NESA) o un derivado farmacéuticamente aceptable del mismo.
ARP070101508A 2007-04-10 2007-04-10 Una composicion farmaceutica utilizable para inhibir o evitar la formacion no deseada de tejido fibroso y uso de la n- sulfoetilnicotinamida para inhibir o evitar la formacion no deseada de tejido fibroso AR060412A1 (es)

Priority Applications (2)

Application Number Priority Date Filing Date Title
ARP070101508A AR060412A1 (es) 2007-04-10 2007-04-10 Una composicion farmaceutica utilizable para inhibir o evitar la formacion no deseada de tejido fibroso y uso de la n- sulfoetilnicotinamida para inhibir o evitar la formacion no deseada de tejido fibroso
PCT/MX2008/000049 WO2008123759A1 (es) 2007-04-10 2008-04-10 N-sulfoetilnicotinamida, composiciones farmacéuticas que la contienen y uso de las mismas para inhibir o evitar la formación no deseada de tejido fibroso

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ARP070101508A AR060412A1 (es) 2007-04-10 2007-04-10 Una composicion farmaceutica utilizable para inhibir o evitar la formacion no deseada de tejido fibroso y uso de la n- sulfoetilnicotinamida para inhibir o evitar la formacion no deseada de tejido fibroso

Publications (1)

Publication Number Publication Date
AR060412A1 true AR060412A1 (es) 2008-06-18

Family

ID=39590600

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070101508A AR060412A1 (es) 2007-04-10 2007-04-10 Una composicion farmaceutica utilizable para inhibir o evitar la formacion no deseada de tejido fibroso y uso de la n- sulfoetilnicotinamida para inhibir o evitar la formacion no deseada de tejido fibroso

Country Status (2)

Country Link
AR (1) AR060412A1 (es)
WO (1) WO2008123759A1 (es)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1408481A (en) * 1973-02-15 1975-10-01 Seperic Beta-pyridyl-carbon-amido-alkane-sulphonic acid salts their preparation and their applications
US5840294A (en) * 1993-03-29 1998-11-24 Queen's University At Kingston Method for treating amyloidosis

Also Published As

Publication number Publication date
WO2008123759A1 (es) 2008-10-16

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