AR035948A1 - Compuestos analogos de la espinosina , composiciones insecticidas, acaricidas formuladas con dichos compuestos ,metodos acaricidas, insecticidas y /o de proteccion de lugares , de infestaciones mediadas por insectos y acaros, respectivamente de control de poblaciones de acaros o insectos utilizando - Google Patents
Compuestos analogos de la espinosina , composiciones insecticidas, acaricidas formuladas con dichos compuestos ,metodos acaricidas, insecticidas y /o de proteccion de lugares , de infestaciones mediadas por insectos y acaros, respectivamente de control de poblaciones de acaros o insectos utilizandoInfo
- Publication number
- AR035948A1 AR035948A1 ARP020101030A ARP020101030A AR035948A1 AR 035948 A1 AR035948 A1 AR 035948A1 AR P020101030 A ARP020101030 A AR P020101030A AR P020101030 A ARP020101030 A AR P020101030A AR 035948 A1 AR035948 A1 AR 035948A1
- Authority
- AR
- Argentina
- Prior art keywords
- compounds
- group
- insecticides
- insects
- insecticiated
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 241000238631 Hexapoda Species 0.000 title abstract 2
- 239000000642 acaricide Substances 0.000 title abstract 2
- 239000002917 insecticide Substances 0.000 title abstract 2
- 206010061217 Infestation Diseases 0.000 title 1
- 230000001404 mediated effect Effects 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- -1 1,3-butadienyl Chemical group 0.000 abstract 2
- 125000004973 1-butenyl group Chemical group C(=CCC)* 0.000 abstract 2
- 125000006017 1-propenyl group Chemical group 0.000 abstract 2
- 241000238876 Acari Species 0.000 abstract 1
- 241000254173 Coleoptera Species 0.000 abstract 1
- 241000255925 Diptera Species 0.000 abstract 1
- 241000258937 Hemiptera Species 0.000 abstract 1
- 241000255777 Lepidoptera Species 0.000 abstract 1
- 241000341865 Saccharopolyspora pogona Species 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000003120 macrolide antibiotic agent Substances 0.000 abstract 1
- 229940041033 macrolides Drugs 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 125000004108 n-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 abstract 1
- VGGSULWDCMWZPO-ODEMIOGVSA-N spinosin Chemical class O([C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]1C1=C(O)C=2C(=O)C=C(OC=2C=C1OC)C=1C=CC(O)=CC=1)[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O VGGSULWDCMWZPO-ODEMIOGVSA-N 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N45/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring
- A01N45/02—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring having three carbocyclic rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N63/00—Biocides, pest repellants or attractants, or plant growth regulators containing microorganisms, viruses, microbial fungi, animals or substances produced by, or obtained from, microorganisms, viruses, microbial fungi or animals, e.g. enzymes or fermentates
- A01N63/20—Bacteria; Substances produced thereby or obtained therefrom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P19/00—Preparation of compounds containing saccharide radicals
- C12P19/44—Preparation of O-glycosides, e.g. glucosides
- C12P19/60—Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin
- C12P19/62—Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin the hetero ring having eight or more ring members and only oxygen as ring hetero atoms, e.g. erythromycin, spiramycin, nystatin
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical & Material Sciences (AREA)
- Zoology (AREA)
- Organic Chemistry (AREA)
- Wood Science & Technology (AREA)
- Biotechnology (AREA)
- Pest Control & Pesticides (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Plant Pathology (AREA)
- Dentistry (AREA)
- Genetics & Genomics (AREA)
- Microbiology (AREA)
- Biochemistry (AREA)
- Virology (AREA)
- Molecular Biology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- General Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
- Saccharide Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Cosmetics (AREA)
Abstract
Se describen y reivindican compuestos de espinosina de fórmula (1), en donde R3 es un grupo seleccionado entre las fórmulas (2) a (7); R4 es un átomo de hidrógeno o un grupo hidroxilo; R5 es un átomo de hidrógeno o un grupo metilo; R8 es 1-butenilo, 1,3-butadienilo, n-butilo, 3-hidroxi-1-butenilo, o 1-propenilo; y R9 es un átomo de hidrógeno o un grupo seleccionado de fórmulas (8) a (16), siempre que: a) si R3 es un grupo de la fórmula (3) ó (4), R4 y R5 son H, y R8 es 1-butenilo, entonces R9 no es H ni un grupo de la fórmula (8); y b) si R3 es un grupo de la fórmula (2), entonces R4 y R5 son H, R8 es 1 propenilo, y R9 es H. Dichos compuestos son macrólidos obtenidos del cultivo de Saccharopolyspora pogona 30141.2, 30141.3, 30141.4, 30141.5, 30141.8, y 30141.13. Dichos compuestos, conforme a las experiencias realizadas, han demostrado ser útiles, en función de su eficacia para el control de ácaros e insectos, particularmente de especies de Lepidoptera, Coleoptera, Homoptera y Diptera y también como intermediarios para preparar otros insecticidas y miticidas. Se describen y reivindican los objetos restantes mencionados en el título.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27760101P | 2001-03-21 | 2001-03-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR035948A1 true AR035948A1 (es) | 2004-07-28 |
Family
ID=23061579
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP020101030A AR035948A1 (es) | 2001-03-21 | 2002-03-21 | Compuestos analogos de la espinosina , composiciones insecticidas, acaricidas formuladas con dichos compuestos ,metodos acaricidas, insecticidas y /o de proteccion de lugares , de infestaciones mediadas por insectos y acaros, respectivamente de control de poblaciones de acaros o insectos utilizando |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP1373290B1 (es) |
| JP (1) | JP4554158B2 (es) |
| KR (1) | KR100904941B1 (es) |
| CN (1) | CN1310935C (es) |
| AR (1) | AR035948A1 (es) |
| DK (1) | DK1373290T3 (es) |
| ES (1) | ES2496940T3 (es) |
| IL (2) | IL157974A0 (es) |
| MX (1) | MXPA03008460A (es) |
| WO (1) | WO2002077005A1 (es) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI275592B (en) * | 2001-03-21 | 2007-03-11 | Dow Agrosciences Llc | Synthetic derivatives of 21-butenyl and related spinosyns |
| DE10320505A1 (de) | 2003-05-08 | 2004-11-25 | Bayer Healthcare Ag | Mittel zum Bekämpfen von Parasiten an Tieren |
| TW201031327A (en) * | 2008-11-14 | 2010-09-01 | Bayer Cropscience Ag | Active compound combinations having insecticidal and acaricidal properties |
| CN101629203B (zh) * | 2008-12-09 | 2010-08-11 | 湖南师范大学 | 一种多杀菌素制备工艺 |
| CN101720766B (zh) * | 2009-12-29 | 2012-08-22 | 华南农业大学 | 茶皂素与多杀菌素的杀虫组合物 |
| EP2528587B1 (en) | 2010-01-25 | 2015-03-18 | Eli Lilly and Company | Spinosyns for use in internally controlling or treating equine bot larvae |
| AR081720A1 (es) * | 2010-02-19 | 2012-10-17 | Sumitomo Chemical Co | Composicion para el control de plagas |
| CN102190694B (zh) * | 2010-03-12 | 2015-09-09 | 中南大学 | 多杀菌素衍生物、制备方法及其作为杀虫剂的用途 |
| CN102286579B (zh) * | 2011-08-05 | 2013-05-22 | 牡丹江佰佳信生物科技有限公司 | 制备多杀霉素的方法及其所使用的培养基 |
| TW201416077A (zh) * | 2012-07-26 | 2014-05-01 | Lilly Co Eli | 單一劑量口服調配物及使用殺外寄生蟲劑賜諾殺（ｓｐｉｎｏｓａｄ）以治療貓之方法 |
| WO2014194503A1 (en) * | 2013-06-06 | 2014-12-11 | Eli Lilly And Company | Parasiticidal compounds, methods, and formulations |
| CN105283465A (zh) * | 2013-06-06 | 2016-01-27 | 伊莱利利公司 | 杀寄生虫的化合物、方法和制剂 |
| KR101716795B1 (ko) * | 2014-07-31 | 2017-03-16 | 우석대학교 산학협력단 | 스피노사드 생산 효율이 우수한 신규 사카로폴리스포라 스피노사(Saccharopolyspora spinosa) wsp8209 및 이를 이용한 스피노사드 생산방법 |
| CN110776536B (zh) * | 2019-09-20 | 2021-06-25 | 国家粮食和物资储备局科学研究院 | 一种从须糖多孢菌发酵液中提取丁烯基多杀菌素的工艺 |
| EP4079744B1 (en) | 2021-04-23 | 2025-08-06 | Acies Bio d.o.o. | Novel spinosyn compounds and their use as a pesticide |
| AR125402A1 (es) | 2021-04-23 | 2023-07-12 | Acies Bio D O O | Profármacos nuevos de espinosinas |
| EP4101858A1 (en) | 2021-06-08 | 2022-12-14 | Acies Bio d.o.o. | Novel spinosyn compounds |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MA21697A1 (fr) * | 1988-12-19 | 1990-07-01 | Dow Agrosciences Llc | Composes de macrolides. |
| US5362634A (en) | 1989-10-30 | 1994-11-08 | Dowelanco | Process for producing A83543 compounds |
| CN1073483A (zh) | 1991-11-08 | 1993-06-23 | 道伊兰科公司 | 一种发酵杀虫剂化合物及其制备方法 |
| BR9406587A (pt) | 1993-03-12 | 1996-01-02 | Dowelanco | Novos compostos a83543 e processo para a produção dos mesmos |
| JP4717163B2 (ja) * | 1995-06-14 | 2011-07-06 | ダウ・アグロサイエンス・エル・エル・シー | スピノシン化合物の合成的修飾 |
| JP2662941B2 (ja) * | 1995-08-11 | 1997-10-15 | アルプス電気株式会社 | 光学装置 |
| US6001981A (en) | 1996-06-13 | 1999-12-14 | Dow Agrosciences Llc | Synthetic modification of Spinosyn compounds |
| AU775637B2 (en) * | 1999-04-16 | 2004-08-12 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
| AU783734B2 (en) * | 1999-09-13 | 2005-12-01 | Dow Agrosciences Llc | Pesticidal macrolides |
| TWI275592B (en) * | 2001-03-21 | 2007-03-11 | Dow Agrosciences Llc | Synthetic derivatives of 21-butenyl and related spinosyns |
-
2002
- 2002-03-21 WO PCT/US2002/008957 patent/WO2002077005A1/en not_active Ceased
- 2002-03-21 MX MXPA03008460A patent/MXPA03008460A/es active IP Right Grant
- 2002-03-21 IL IL15797402A patent/IL157974A0/xx unknown
- 2002-03-21 DK DK02719327.5T patent/DK1373290T3/da active
- 2002-03-21 ES ES02719327.5T patent/ES2496940T3/es not_active Expired - Lifetime
- 2002-03-21 JP JP2002576263A patent/JP4554158B2/ja not_active Expired - Fee Related
- 2002-03-21 KR KR1020037012245A patent/KR100904941B1/ko not_active Expired - Fee Related
- 2002-03-21 EP EP02719327.5A patent/EP1373290B1/en not_active Expired - Lifetime
- 2002-03-21 CN CNB028084373A patent/CN1310935C/zh not_active Expired - Fee Related
- 2002-03-21 AR ARP020101030A patent/AR035948A1/es unknown
-
2003
- 2003-09-17 IL IL157974A patent/IL157974A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| EP1373290A1 (en) | 2004-01-02 |
| JP2004532836A (ja) | 2004-10-28 |
| CN1620463A (zh) | 2005-05-25 |
| ES2496940T3 (es) | 2014-09-22 |
| MXPA03008460A (es) | 2004-06-30 |
| DK1373290T3 (da) | 2014-12-01 |
| WO2002077005A1 (en) | 2002-10-03 |
| KR20030085023A (ko) | 2003-11-01 |
| KR100904941B1 (ko) | 2009-06-29 |
| IL157974A (en) | 2010-06-16 |
| JP4554158B2 (ja) | 2010-09-29 |
| EP1373290B1 (en) | 2014-08-20 |
| IL157974A0 (en) | 2004-03-28 |
| CN1310935C (zh) | 2007-04-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |