AR035491A1 - Tetrahidrocarbazoles, un procedimiento para su preparacion, usos de los mismos, preparacion para el cuidado personal, composicion oral, y medicamento - Google Patents
Tetrahidrocarbazoles, un procedimiento para su preparacion, usos de los mismos, preparacion para el cuidado personal, composicion oral, y medicamentoInfo
- Publication number
- AR035491A1 AR035491A1 ARP010104354A ARP010104354A AR035491A1 AR 035491 A1 AR035491 A1 AR 035491A1 AR P010104354 A ARP010104354 A AR P010104354A AR P010104354 A ARP010104354 A AR P010104354A AR 035491 A1 AR035491 A1 AR 035491A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- cycloalkyl
- alkoxy
- phenyl
- substituted
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q17/00—Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
- A61Q17/005—Antimicrobial preparations
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
- A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
- A61K8/492—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid having condensed rings, e.g. indol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
- A61K8/4933—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having sulfur as an exocyclic substituent, e.g. pyridinethione
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/69—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing fluorine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61L—METHODS OR APPARATUS FOR STERILISING MATERIALS OR OBJECTS IN GENERAL; DISINFECTION, STERILISATION OR DEODORISATION OF AIR; CHEMICAL ASPECTS OF BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES; MATERIALS FOR BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES
- A61L2/00—Methods or apparatus for disinfecting or sterilising materials or objects other than foodstuffs or contact lenses; Accessories therefor
- A61L2/16—Methods or apparatus for disinfecting or sterilising materials or objects other than foodstuffs or contact lenses; Accessories therefor using chemical substances
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q11/00—Preparations for care of the teeth, of the oral cavity or of dentures; Dentifrices, e.g. toothpastes; Mouth rinses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q15/00—Anti-perspirants or body deodorants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C11—ANIMAL OR VEGETABLE OILS, FATS, FATTY SUBSTANCES OR WAXES; FATTY ACIDS THEREFROM; DETERGENTS; CANDLES
- C11D—DETERGENT COMPOSITIONS; USE OF SINGLE SUBSTANCES AS DETERGENTS; SOAP OR SOAP-MAKING; RESIN SOAPS; RECOVERY OF GLYCEROL
- C11D3/00—Other compounding ingredients of detergent compositions covered in group C11D1/00
- C11D3/16—Organic compounds
- C11D3/26—Organic compounds containing nitrogen
- C11D3/28—Heterocyclic compounds containing nitrogen in the ring
-
- C—CHEMISTRY; METALLURGY
- C11—ANIMAL OR VEGETABLE OILS, FATS, FATTY SUBSTANCES OR WAXES; FATTY ACIDS THEREFROM; DETERGENTS; CANDLES
- C11D—DETERGENT COMPOSITIONS; USE OF SINGLE SUBSTANCES AS DETERGENTS; SOAP OR SOAP-MAKING; RESIN SOAPS; RECOVERY OF GLYCEROL
- C11D3/00—Other compounding ingredients of detergent compositions covered in group C11D1/00
- C11D3/48—Medical, disinfecting agents, disinfecting, antibacterial, germicidal or antimicrobial compositions
-
- D—TEXTILES; PAPER
- D21—PAPER-MAKING; PRODUCTION OF CELLULOSE
- D21H—PULP COMPOSITIONS; PREPARATION THEREOF NOT COVERED BY SUBCLASSES D21C OR D21D; IMPREGNATING OR COATING OF PAPER; TREATMENT OF FINISHED PAPER NOT COVERED BY CLASS B31 OR SUBCLASS D21G; PAPER NOT OTHERWISE PROVIDED FOR
- D21H21/00—Non-fibrous material added to the pulp, characterised by its function, form or properties; Paper-impregnating or coating material, characterised by its function, form or properties
- D21H21/14—Non-fibrous material added to the pulp, characterised by its function, form or properties; Paper-impregnating or coating material, characterised by its function, form or properties characterised by function or properties in or on the paper
- D21H21/36—Biocidal agents, e.g. fungicidal, bactericidal, insecticidal agents
-
- D—TEXTILES; PAPER
- D21—PAPER-MAKING; PRODUCTION OF CELLULOSE
- D21H—PULP COMPOSITIONS; PREPARATION THEREOF NOT COVERED BY SUBCLASSES D21C OR D21D; IMPREGNATING OR COATING OF PAPER; TREATMENT OF FINISHED PAPER NOT COVERED BY CLASS B31 OR SUBCLASS D21G; PAPER NOT OTHERWISE PROVIDED FOR
- D21H25/00—After-treatment of paper not provided for in groups D21H17/00 - D21H23/00
- D21H25/18—After-treatment of paper not provided for in groups D21H17/00 - D21H23/00 of old paper as in books, documents, e.g. restoring
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Birds (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Wood Science & Technology (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Dermatology (AREA)
- Oral & Maxillofacial Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Cosmetics (AREA)
Abstract
Tetrahidrocarbazoles que tienen la fórmula (1) (2) en las cuales R1 es hidrógeno, alquilo C1-20, cicloalquilo C3-12, alquenilo C2-20, cicloalquenilo C4-12, alquinilo C3-20, cicloalquinilo C4-12, fenilo o fenil-alquilo C1-5 cada uno de ellos no sustituido o sustituido con alquilo C1-5, cicloalquilo C3-12, alcoxi C1-5, cicloalcoxi C3-12, halógeno, carboxi, alquilcarbonilo C1-7, alcoxicarbonilo C1-7, cicloalquilcarbonilo C3-12, cicloalcoxicarbonilo C3-12, ciano, trifluormetilo, pentafluoretilo, amino, N,N-mono- o di-alquilamino C1-20 o nitro, R2 es hidrógeno, hidroxi, alquilo C1-20, cicloalquilo C3-12, hidroxialquilo C1-20, hidroxialcoxi C1-20, aminoalquilo C1-20, N-monoalquilamino C1-20-alquilo C1-20, N-monoalquilaminohidroxi C1-20-alcoxi C1-20, N,N-dialquilamino C1-20-alquilo C1-20, N,N-dialquilaminohidroxi C1-20-alcoxi C1-20, carboxi, carboxi-alquilo C1-20 éster, haloalquilo C1-20, haloalcoxi C1-20, alquenilo C2-20, cicloalquenilo C4-12, alquinilo C3-20, cicloalquinilo C4-12, alcoxi C1-20, alqueniloxi C2-20, alquiniloxi C2-20, halógeno, ciano, alquilcarbonilo C1-7, nitro, trifluormetilo o pentafluoretilo; R3 y R4 son cada uno independientemente hidrógeno o alquilo C1-20, o R3 y R4 conjuntamente denotan un radical alquileno C2-20, un radical alquenileno C2-20, un radical alquinileno C4-20 o un radical alquileno C3-20 interrumpido por -N(R6)-, donde es posible que dichos radicales divalentes estén adicionalmente sustituidos con uno o más de alquilo C1-20, cicloalquilo C3-12, alquenilo C2-20, cicloalquenilo C4-12, alquinilo C3-20, cicloalquinilo C4-12, alcoxicarbonilo C1-7, o fenilo o fenil-alquilo C1-5 cada uno no sustituido o sustituido con alquilo C1-5, cicloalquilo C3-12, alcoxi C1-5, cicloalcoxi C3-12, halógeno, carboxi, alcoxicarbonilo C1-7, cicloalcoxicarbonilo C3-12, ciano, trifluormetilo, pentafluoretilo, amino, N,N-mono- o di-alquilamino C1-20 o nitro, o R3 y R4 conjuntamente denotan un biciclo [x.y.z] alquileno C4-20 o biciclo [x.y.z] alquileno C4-20 interrumpido con -N(R6)-, donde x, y y z son cada uno independientemente uno del otro de 0 a 10, R5 es hidrógeno, hidroxi, alquilo C1-20, alcoxi C1-20, cicloalquilo C3-12, alquenilo C2-20, cicloalquenilo C4-12, alquinilo C3-20, cicloalquinilo C4-12, fenilo o fenilo-alquilo C1-5, cada uno no sustituido o sustituido con alquilo C1-5, cicloalquilo C3-12, alcoxi C1-5, cicloalcoxi C3-12, halógeno, carboxi, alcoxicarbonilo C1-7, cicloalcoxicarbonilo C3-12, ciano, trifluormetilo, pentafluoretilo, amino, N,N-mono- o di-alquilamino C1-20 o nitro; R6 es hidrógeno, alquilo C1-20, cicloalquilo C3-12, alquenilo C2-20, cicloalquenilo C4-12, alquinilo C3-20, cicloalquinilo C4-12, alcoxicarbonilo C1-7, fenilo o fenilo-alquilo C1-5, cada uno no sustituido o sustituido con alquilo C1-5, cicloalquilo C3-12, alcoxi c1-5, cicloalcoxi C3-12, halógeno, carboxi, alcoxicarbonilo C1-7, cicloalcoxicarbonilo C3-12, ciano, trifluormetilo, pentafluoretilo, N,N-mono- o di-alquilamino C1-20 o nitro; Q es -SO2-, -O- o -(CO)-; X es -CH- o -N-; m es 1 a 3; y t es 0 a 1; que son apropiados como ingredientes activos antimicrobianos, procedimiento para su preparación, usos de los mismos, preparación para el cuidado personal, composición oral, y medicamento.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00810844 | 2000-09-18 | ||
| CH8432001 | 2001-05-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR035491A1 true AR035491A1 (es) | 2004-06-02 |
Family
ID=25738650
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP010104354A AR035491A1 (es) | 2000-09-18 | 2001-09-14 | Tetrahidrocarbazoles, un procedimiento para su preparacion, usos de los mismos, preparacion para el cuidado personal, composicion oral, y medicamento |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US6967215B2 (es) |
| EP (1) | EP1319006B1 (es) |
| AR (1) | AR035491A1 (es) |
| AT (1) | ATE282620T1 (es) |
| AU (1) | AU2002214977A1 (es) |
| DE (1) | DE60107275T2 (es) |
| ES (1) | ES2231564T3 (es) |
| WO (1) | WO2002024699A1 (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105307731B (zh) | 2013-06-27 | 2019-09-24 | 宝洁公司 | 防腐性个人护理组合物 |
| WO2019100106A1 (en) * | 2017-11-24 | 2019-05-31 | The University Of Sydney | Antibacterial compounds and methods of use thereof |
| CN112851680B (zh) * | 2021-01-21 | 2021-12-24 | 河南科技大学第一附属医院 | 一种医用护理杀菌消毒的吲哚类药物分子及其制备方法和应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH653675A5 (en) | 1983-05-26 | 1986-01-15 | Ciba Geigy Ag | Microbicides |
| US5645988A (en) | 1991-05-08 | 1997-07-08 | The United States Of America As Represented By The Department Of Health And Human Services | Methods of identifying drugs with selective effects against cancer cells |
-
2001
- 2001-09-11 WO PCT/EP2001/010479 patent/WO2002024699A1/en active IP Right Grant
- 2001-09-11 US US10/380,573 patent/US6967215B2/en not_active Expired - Fee Related
- 2001-09-11 AU AU2002214977A patent/AU2002214977A1/en not_active Abandoned
- 2001-09-11 EP EP01983479A patent/EP1319006B1/en not_active Expired - Lifetime
- 2001-09-11 AT AT01983479T patent/ATE282620T1/de not_active IP Right Cessation
- 2001-09-11 ES ES01983479T patent/ES2231564T3/es not_active Expired - Lifetime
- 2001-09-11 DE DE60107275T patent/DE60107275T2/de not_active Expired - Fee Related
- 2001-09-14 AR ARP010104354A patent/AR035491A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ATE282620T1 (de) | 2004-12-15 |
| WO2002024699A1 (en) | 2002-03-28 |
| DE60107275T2 (de) | 2005-12-01 |
| DE60107275D1 (de) | 2004-12-23 |
| ES2231564T3 (es) | 2005-05-16 |
| AU2002214977A1 (en) | 2002-04-02 |
| US20040097535A1 (en) | 2004-05-20 |
| EP1319006B1 (en) | 2004-11-17 |
| EP1319006A1 (en) | 2003-06-18 |
| US6967215B2 (en) | 2005-11-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure | ||
| FC | Refusal |