AR028983A1 - Composiciones farmaceuticas que contienen nicotina o un ligando de los receptores nicotinicos y un inhibidor de la monoamina oxidasa y su aplicacion en la abstinencia de tabaco - Google Patents
Composiciones farmaceuticas que contienen nicotina o un ligando de los receptores nicotinicos y un inhibidor de la monoamina oxidasa y su aplicacion en la abstinencia de tabacoInfo
- Publication number
- AR028983A1 AR028983A1 ARP000100404A ARP000100404A AR028983A1 AR 028983 A1 AR028983 A1 AR 028983A1 AR P000100404 A ARP000100404 A AR P000100404A AR P000100404 A ARP000100404 A AR P000100404A AR 028983 A1 AR028983 A1 AR 028983A1
- Authority
- AR
- Argentina
- Prior art keywords
- pharmaceutical compositions
- inhibitor
- monoamine
- oxidase
- bind
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/465—Nicotine; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Addiction (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9901144A FR2788982B1 (fr) | 1999-02-02 | 1999-02-02 | Compositions pharmaceutiques contenant de la nicotine et leur application dans le sevrage tabagique |
Publications (1)
Publication Number | Publication Date |
---|---|
AR028983A1 true AR028983A1 (es) | 2003-06-04 |
Family
ID=9541474
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP000100404A AR028983A1 (es) | 1999-02-02 | 2000-01-31 | Composiciones farmaceuticas que contienen nicotina o un ligando de los receptores nicotinicos y un inhibidor de la monoamina oxidasa y su aplicacion en la abstinencia de tabaco |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1150715A1 (fr) |
JP (1) | JP2002536342A (fr) |
AR (1) | AR028983A1 (fr) |
AU (1) | AU2298800A (fr) |
CA (1) | CA2361437A1 (fr) |
FR (1) | FR2788982B1 (fr) |
HU (1) | HUP0201279A2 (fr) |
WO (1) | WO2000045846A1 (fr) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6605610B1 (en) * | 1997-12-31 | 2003-08-12 | Pfizer Inc | Aryl fused azapolycyclic compounds |
ME00459B (me) | 1997-12-31 | 2011-10-10 | Pfizer Prod Inc | Aril fuzirana azapoliciklična jedinjenja |
NZ510287A (en) | 1998-11-27 | 2003-05-30 | Neurosearch As | 8-azabicyclo[3.2.1]oct-2-ene and -octane derivatives useful as cholinergic ligands at the nicotinic acetyl choline receptor |
IL137937A0 (en) * | 1999-08-27 | 2001-10-31 | Pfizer Prod Inc | A pharmaceutical composition for the prevention and treatment of nicotine addiction in a mammal |
DK1358177T3 (da) | 2000-10-13 | 2006-12-04 | Neurosearch As | Behandling af affektbetonede lidelser ved den kombinerede virkning af en nikotinreceptoragonist og et monoaminergt stof |
AU2002234836B2 (en) * | 2001-04-20 | 2007-08-23 | Pfizer Products Inc. | Process for the preparation of 1,3-substituted indenes and aryl-fused azapolycyclic compounds |
SE521512C2 (sv) | 2001-06-25 | 2003-11-11 | Niconovum Ab | Anordning för administrering av en substans till främre delen av en individs munhåla |
ATE427745T1 (de) | 2001-11-05 | 2009-04-15 | Krele Pharmaceuticals Llc | Zusammensetzungen und verfahren zur erhíhung der compliance mit therapien unter verwendung von aldehyddehydrogenase-hemmern und zur behandlung von alkoholsmus |
MXPA04010190A (es) * | 2002-04-18 | 2005-02-03 | Astrazeneca Ab | Compuestos heterociclicos. |
BR0309343A (pt) * | 2002-04-18 | 2005-02-15 | Astrazeneca Ab | Composto, composição farmacêutica, uso de um composto, e, método de tratamento ou profilaxia de doenças ou condições humanas |
BR0309342A (pt) * | 2002-04-18 | 2005-02-15 | Astrazeneca Ab | Composto, composição farmacêutica, uso de um composto, e, método de tratamento ou profilaxia de doenças ou condições humanas |
CA2495248A1 (fr) | 2002-08-30 | 2004-03-11 | Memory Pharmaceuticals Corporation | Derives d'anabaseine utiles pour le traitement de maladies neurodegeneratives |
CA2499128C (fr) | 2002-09-25 | 2012-07-31 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles et benzoisothiazoles, leur preparation et leurs utilisations |
JP4708795B2 (ja) | 2002-12-20 | 2011-06-22 | ニコノヴァム エービー | 物理的および化学的に安定なニコチン−含有粒状物質 |
IL155666A (en) * | 2003-04-29 | 2013-12-31 | Neurim Pharma 1991 | Insomnia treatment |
DE10338174A1 (de) * | 2003-08-20 | 2005-03-24 | Lts Lohmann Therapie-Systeme Ag | Transdermale Arzneimittelzubereitungen mit Wirkstoffkombinationen zur Behandlung der Parkinson-Krankheit |
US7396833B2 (en) | 2003-12-22 | 2008-07-08 | Memory Pharmaceuticals Corporation | Indoles, 1H-indazoles, 1,2-benzisoxazoles, and 1,2-benzisothiazoles, and preparation and uses thereof |
RU2417225C2 (ru) | 2004-03-25 | 2011-04-27 | Мемори Фармасьютиклз Корпорейшн | Индазолы, бензотиазолы, бензоизотиазолы, бензизоксазолы и их получение и применение |
ATE487716T1 (de) | 2004-04-22 | 2010-11-15 | Memory Pharm Corp | Indole, 1h-indazole, 1,2-benzisoxazole, 1,2- benzoisothiazole, deren herstellung und verwendungen |
AU2005243147A1 (en) | 2004-05-07 | 2005-11-24 | Memory Pharmaceuticals Corporation | 1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles, 1,2-benzoisothiazoles, and chromones and preparation and uses thereof |
US7459469B2 (en) | 2004-11-10 | 2008-12-02 | Targacept, Inc. | Hydroxybenzoate salts of metanicotine compounds |
JP2008525464A (ja) | 2004-12-22 | 2008-07-17 | メモリー・ファーマシューティカルズ・コーポレイション | α−7ニコチン性受容体リガンド並びにその製造及び使用 |
US8106066B2 (en) | 2005-09-23 | 2012-01-31 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof |
EP1976519A2 (fr) * | 2006-01-27 | 2008-10-08 | Yale University | Analogues de cystisine et d'acétylcholine et procédés de traitement des troubles de l'humeur |
AU2007224584A1 (en) | 2006-03-16 | 2007-09-20 | Niconovum Ab | Improved snuff composition |
US8017785B2 (en) | 2006-05-09 | 2011-09-13 | Astrazeneca Ab | Salt forms of (2S)-(4E)-N-methyl-5-[3-(5-isopropoxypyridin)y1]-4-penten 2-amine |
TWI389889B (zh) | 2006-05-09 | 2013-03-21 | Targacept Inc | (2s)-(4e)-n-甲基-5-〔3-(5-異丙氧基吡啶)基〕-4-戊烯-2-胺之新穎多晶型 |
US20100028447A1 (en) * | 2007-01-22 | 2010-02-04 | Targacept, Inc. | Intranasal, Buccal, And Sublingual Administration Of Metanicotine Analogs |
US8697722B2 (en) * | 2007-11-02 | 2014-04-15 | Sri International | Nicotinic acetylcholine receptor modulators |
WO2009058120A1 (fr) * | 2007-11-02 | 2009-05-07 | Sri International | Modulateurs des récepteurs nicotiniques de l'acétylcholine |
EP2523562B1 (fr) | 2010-01-11 | 2019-01-02 | Astraea Therapeutics, LLC | Modulateurs du récepteur nicotinique de l'acétylcholine |
MX2012013193A (es) | 2010-05-20 | 2012-12-17 | Astrazeneca Ab | Nuevo proceso para preparar aminas olefinicas sustituidas con arilo. |
US20130165511A1 (en) | 2010-09-01 | 2013-06-27 | TONIX Pharmaceuticals Holding Corp | Treatment for cocaine addiction |
US10653639B2 (en) * | 2016-05-16 | 2020-05-19 | Cv Sciences, Inc. | Pharmaceutical formulations containing cannabidiol and nicotine for treating smokeless tobacco addiction |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2446895A (en) * | 1994-04-22 | 1995-11-16 | Assistance Publique - Hopitaux De Paris | Use of mao-a inhibitors for the manufacture of a medicament in the treatment of tobacco withdrawal symptoms in smokers |
US5803081A (en) * | 1996-06-28 | 1998-09-08 | Regent Court Technologies | Tobacco and related products |
-
1999
- 1999-02-02 FR FR9901144A patent/FR2788982B1/fr not_active Expired - Fee Related
-
2000
- 2000-01-28 EP EP00901660A patent/EP1150715A1/fr not_active Withdrawn
- 2000-01-28 WO PCT/FR2000/000193 patent/WO2000045846A1/fr not_active Application Discontinuation
- 2000-01-28 JP JP2000596965A patent/JP2002536342A/ja not_active Withdrawn
- 2000-01-28 HU HU0201279A patent/HUP0201279A2/hu unknown
- 2000-01-28 CA CA002361437A patent/CA2361437A1/fr not_active Abandoned
- 2000-01-28 AU AU22988/00A patent/AU2298800A/en not_active Abandoned
- 2000-01-31 AR ARP000100404A patent/AR028983A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2000045846A1 (fr) | 2000-08-10 |
FR2788982B1 (fr) | 2002-08-02 |
AU2298800A (en) | 2000-08-25 |
JP2002536342A (ja) | 2002-10-29 |
EP1150715A1 (fr) | 2001-11-07 |
HUP0201279A2 (en) | 2002-09-28 |
CA2361437A1 (fr) | 2000-08-10 |
FR2788982A1 (fr) | 2000-08-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |