AR026708A1 - Derivados de 5-hidroxi-indazol para el tratamiento de glaucoma - Google Patents
Derivados de 5-hidroxi-indazol para el tratamiento de glaucomaInfo
- Publication number
- AR026708A1 AR026708A1 ARP000106395A ARP000106395A AR026708A1 AR 026708 A1 AR026708 A1 AR 026708A1 AR P000106395 A ARP000106395 A AR P000106395A AR P000106395 A ARP000106395 A AR P000106395A AR 026708 A1 AR026708 A1 AR 026708A1
- Authority
- AR
- Argentina
- Prior art keywords
- indazol
- glaucoma
- treatment
- hydroxy
- derivatives
- Prior art date
Links
- 208000010412 Glaucoma Diseases 0.000 title abstract 2
- ZHDXWEPRYNHNDC-UHFFFAOYSA-N 1h-indazol-5-ol Chemical class OC1=CC=C2NN=CC2=C1 ZHDXWEPRYNHNDC-UHFFFAOYSA-N 0.000 title 1
- 125000000022 2-aminoethyl group Chemical group [H]C([*])([H])C([H])([H])N([H])[H] 0.000 abstract 1
- 230000004406 elevated intraocular pressure Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Ophthalmology & Optometry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US19028300P | 2000-03-17 | 2000-03-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR026708A1 true AR026708A1 (es) | 2003-02-26 |
Family
ID=22700701
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP000106395A AR026708A1 (es) | 2000-03-17 | 2000-12-01 | Derivados de 5-hidroxi-indazol para el tratamiento de glaucoma |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP1268439A1 (enExample) |
| JP (1) | JP2003535821A (enExample) |
| KR (1) | KR20030095183A (enExample) |
| CN (1) | CN1450995A (enExample) |
| AR (1) | AR026708A1 (enExample) |
| AU (2) | AU2001219180B2 (enExample) |
| BR (1) | BR0017163A (enExample) |
| CA (1) | CA2401959A1 (enExample) |
| MX (1) | MXPA02008825A (enExample) |
| PL (1) | PL365422A1 (enExample) |
| WO (1) | WO2001070701A1 (enExample) |
| ZA (1) | ZA200206853B (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6960579B1 (en) | 1998-05-19 | 2005-11-01 | Alcon Manufacturing, Ltd. | Serotonergic 5HT7 receptor compounds for treating ocular and CNS disorders |
| WO2002098350A2 (en) | 2001-06-01 | 2002-12-12 | Alcon, Inc. | Pyranoindazoles and their use for the treatment of glaucoma |
| TW593302B (en) | 2001-12-20 | 2004-06-21 | Alcon Inc | Novel benzodifuranimidazoline and benzofuranimidazoline derivatives and their use for the treatment of glaucoma |
| US7196082B2 (en) | 2002-11-08 | 2007-03-27 | Merck & Co. Inc. | Ophthalmic compositions for treating ocular hypertension |
| CN100384827C (zh) * | 2002-11-08 | 2008-04-30 | 默克公司 | 用于治疗高眼压症的眼用组合物 |
| CA2505127A1 (en) * | 2002-11-08 | 2004-05-27 | James B. Doherty | Ophthalmic compositions for treating ocular hypertension |
| EP1581209A4 (en) | 2002-12-13 | 2009-03-11 | Alcon Inc | NEW BENZOPYRAN ANALOGUE AND ITS USE FOR THE TREATMENT OF GLAUKOM |
| JP2004262812A (ja) * | 2003-02-28 | 2004-09-24 | Rohto Pharmaceut Co Ltd | 眼圧低下剤 |
| AU2004271978B2 (en) * | 2003-09-04 | 2009-02-05 | Merck & Co., Inc. | Ophthalmic compositions for treating ocular hypertension |
| AR046890A1 (es) | 2003-12-15 | 2005-12-28 | Alcon Inc | [1,4] oxazino [2,3-g] indazoles sustituidos para el tratamiento del glaucoma. |
| US7129257B1 (en) | 2003-12-15 | 2006-10-31 | Alcon, Inc. | Pyrazolo[3,4- e]benzoxazoles for the treatment of glaucoma |
| US7338972B1 (en) | 2003-12-15 | 2008-03-04 | Alcon, Inc. | Substituted 1-alkylamino-1H-indazoles for the treatment of glaucoma |
| AU2005308523B2 (en) | 2004-11-29 | 2010-01-07 | Warner-Lambert Company Llc | Therapeutic pyrazolo[3,4-b] pyridines and indazoles |
| US7425572B2 (en) | 2004-12-08 | 2008-09-16 | Alcon, Inc. | Use of dioxindoindazoles and dioxoloindazoles for treating glaucoma |
| KR100972921B1 (ko) * | 2009-12-02 | 2010-07-28 | 제이케이이앤씨 주식회사 | 회전 격판식 선회류 세정 및 탈취장치 |
| WO2025000053A1 (en) * | 2023-06-28 | 2025-01-02 | Psylo Pty Ltd | Compounds |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2680366B1 (fr) * | 1991-08-13 | 1995-01-20 | Adir | Nouveaux derives d'arylethylamines, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent. |
| WO1999059499A2 (en) * | 1998-05-19 | 1999-11-25 | Alcon Laboratories, Inc. | Serotonergic 5ht7 receptor compounds for treating ocular and cns disorders |
| GB9819020D0 (en) * | 1998-09-01 | 1998-10-28 | Cerebrus Ltd | Chemical compounds III |
| AU755119B2 (en) * | 1998-09-18 | 2002-12-05 | Alcon Laboratories, Inc. | Serotonergic 5HT2 agonists for treating glaucoma |
-
2000
- 2000-11-14 WO PCT/US2000/031143 patent/WO2001070701A1/en not_active Ceased
- 2000-11-14 JP JP2001568911A patent/JP2003535821A/ja active Pending
- 2000-11-14 KR KR1020027011862A patent/KR20030095183A/ko not_active Ceased
- 2000-11-14 AU AU2001219180A patent/AU2001219180B2/en not_active Ceased
- 2000-11-14 PL PL00365422A patent/PL365422A1/xx not_active Application Discontinuation
- 2000-11-14 CA CA002401959A patent/CA2401959A1/en not_active Abandoned
- 2000-11-14 CN CN00819348A patent/CN1450995A/zh active Pending
- 2000-11-14 MX MXPA02008825A patent/MXPA02008825A/es unknown
- 2000-11-14 BR BR0017163-8A patent/BR0017163A/pt not_active IP Right Cessation
- 2000-11-14 EP EP00982109A patent/EP1268439A1/en not_active Withdrawn
- 2000-11-14 AU AU1918001A patent/AU1918001A/xx active Pending
- 2000-12-01 AR ARP000106395A patent/AR026708A1/es unknown
-
2002
- 2002-08-27 ZA ZA200206853A patent/ZA200206853B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA02008825A (es) | 2004-10-15 |
| PL365422A1 (en) | 2005-01-10 |
| EP1268439A1 (en) | 2003-01-02 |
| WO2001070701A1 (en) | 2001-09-27 |
| AU2001219180B2 (en) | 2005-04-07 |
| JP2003535821A (ja) | 2003-12-02 |
| AU1918001A (en) | 2001-10-03 |
| KR20030095183A (ko) | 2003-12-18 |
| BR0017163A (pt) | 2003-01-14 |
| ZA200206853B (en) | 2004-11-02 |
| CA2401959A1 (en) | 2001-09-27 |
| CN1450995A (zh) | 2003-10-22 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR026708A1 (es) | Derivados de 5-hidroxi-indazol para el tratamiento de glaucoma | |
| BRPI0418245A (pt) | nitróxi-derivados de prostaglandina | |
| ATE340171T1 (de) | Piperazinderivate zur behandlung bakterieller infektionen | |
| CY1114048T1 (el) | Συνδυασμος βριμονιδινης και τιμολολης για τοπικη οφθαλμικη χρηση | |
| ATE202706T1 (de) | Verwendung von 9-deoxyprostaglandinderivaten zur behandlung von glaukom | |
| ECSP045081A (es) | Derivados de 1,8-naftiridina y su uso para el tratamiento de la diabetes y trastornos relacionados | |
| ES2191286T3 (es) | Moleculas pequeñas, utiles en el tratamiento de enfermedades inflamatorias. | |
| CY1112946T1 (el) | 4-υδροξυβενζομορφανια | |
| AR020442A1 (es) | Agonistas de 5ht2serotonergicos para el tratamiento de glaucoma | |
| PL374523A1 (en) | Calicheamicin derivative-carrier conjugates | |
| DE60023043T2 (de) | (S,S)-Reboxetin zur Behandlung von Inkontinenz | |
| DE60121988D1 (de) | Kombinationstherapie mit antidiabetischen und antikonvulsiven mitteln | |
| CY1108610T1 (el) | Πεπτιδια της il-2 και παραγωγα αυτων και χρηση αυτων ως θεραπευτικοι παραγοντες | |
| BR0017157A (pt) | Derivados de 6-hidroxi-indazol para o tratamento de glaucoma | |
| ES2191208T3 (es) | Oxiimino-pregnano-carbolactonas. | |
| DE60331638D1 (de) | Keratin-netzwerke enthaltende wundverbände für gewebedefekte | |
| ECSP044862A (es) | Pirenzepine ophthalmic gel | |
| EA200200742A1 (ru) | 1,2-диарилбензимидазолы для лечения заболеваний, связанных с активацией микроглии | |
| WO1998039293A3 (en) | 13-thia prostaglandins for use in glaucoma therapy | |
| DE60115466D1 (de) | Wirkstoffvorläufer von imidazopyridin-derivaten | |
| TR200101149T2 (tr) | Dış retina bozukluklarının tedavisi. | |
| ES2178765T3 (es) | Nuevos derivados de 1,7,7-trimetil-biciclo (2.2.1) heptano. | |
| AR026707A1 (es) | Agonistas de 5ht2 para el control de pio y para el tratamiento de glaucoma | |
| EA200300727A1 (ru) | Производные 2h-1-бензопирана, способы их получения и их фармацевтические композиции | |
| AR022321A1 (es) | Derivados de anticonvulsivo utiles para el tratamiento de la migrana transformada |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |