AP2008004602A0 - Melanocortin type 4 receptor agonist piperidinoylpyrrolidines - Google Patents

Melanocortin type 4 receptor agonist piperidinoylpyrrolidines

Info

Publication number
AP2008004602A0
AP2008004602A0 AP2008004602A AP2008004602A AP2008004602A0 AP 2008004602 A0 AP2008004602 A0 AP 2008004602A0 AP 2008004602 A AP2008004602 A AP 2008004602A AP 2008004602 A AP2008004602 A AP 2008004602A AP 2008004602 A0 AP2008004602 A0 AP 2008004602A0
Authority
AP
ARIPO
Prior art keywords
piperidinoylpyrrolidines
receptor agonist
melanocortin type
melanocortin
type
Prior art date
Application number
AP2008004602A
Other languages
English (en)
Inventor
Mark David Andrews
Alan Daniel Brown
Mark I Lansdell
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of AP2008004602A0 publication Critical patent/AP2008004602A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AP2008004602A 2006-02-23 2007-02-19 Melanocortin type 4 receptor agonist piperidinoylpyrrolidines AP2008004602A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US77629506P 2006-02-23 2006-02-23
US88784007P 2007-02-02 2007-02-02
PCT/IB2007/000456 WO2007096763A2 (fr) 2006-02-23 2007-02-19 Pipéridinoylpyrrolidines en tant qu'agonistes du récepteur de la mélanocortine de type 4

Publications (1)

Publication Number Publication Date
AP2008004602A0 true AP2008004602A0 (en) 2008-10-31

Family

ID=38169450

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2008004602A AP2008004602A0 (en) 2006-02-23 2007-02-19 Melanocortin type 4 receptor agonist piperidinoylpyrrolidines

Country Status (22)

Country Link
US (1) US8138188B2 (fr)
EP (1) EP1989196B1 (fr)
KR (1) KR101036981B1 (fr)
AP (1) AP2008004602A0 (fr)
AU (1) AU2007219236B2 (fr)
BR (1) BRPI0708264A2 (fr)
CA (1) CA2642922C (fr)
CR (1) CR10219A (fr)
DK (1) DK1989196T3 (fr)
EA (1) EA200801738A1 (fr)
EC (1) ECSP088688A (fr)
ES (1) ES2402581T3 (fr)
HK (1) HK1126489A1 (fr)
IL (1) IL193279A (fr)
MA (1) MA30228B1 (fr)
ME (1) MEP6808A (fr)
MX (1) MX2008010899A (fr)
NO (1) NO20083480L (fr)
RS (1) RS20080371A (fr)
SG (1) SG185849A1 (fr)
TN (1) TNSN08337A1 (fr)
WO (1) WO2007096763A2 (fr)

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EP2025674A1 (fr) 2007-08-15 2009-02-18 sanofi-aventis Tetrahydronaphthaline substituée, son procédé de fabrication et son utilisation en tant que médicament
US8737295B2 (en) 2007-11-16 2014-05-27 Qualcomm Incorporated Sector identification using sector parameters signatures
US8848656B2 (en) 2007-11-16 2014-09-30 Qualcomm Incorporated Utilizing broadcast signals to convey restricted association information
US9603062B2 (en) 2007-11-16 2017-03-21 Qualcomm Incorporated Classifying access points using pilot identifiers
US8902867B2 (en) 2007-11-16 2014-12-02 Qualcomm Incorporated Favoring access points in wireless communications
EP2103614A1 (fr) * 2008-03-18 2009-09-23 Santhera Pharmaceuticals (Schweiz) AG Dérivés d'imidazopyrimidine, d'imidazopyrazine et d' imidazopyridazine substitués en tant que modulateur de récepteur de la mélanocortine-4
US8588773B2 (en) 2008-08-04 2013-11-19 Qualcomm Incorporated System and method for cell search and selection in a wireless communication system
UA99555C2 (en) 2008-11-12 2012-08-27 Элджи Лайф Саенсез Лтд. Melanocortin receptor agonists
JP5890780B2 (ja) * 2009-11-18 2016-03-22 ヘルシン ヘルスケア ソシエテ アノニム 中枢を介する悪心および嘔吐を治療するための組成物および方法
EP2722045B1 (fr) 2009-11-18 2016-07-06 Helsinn Healthcare SA Compositions pour traiter les nausées et vomissements à médiation centrale
WO2012120054A1 (fr) 2011-03-08 2012-09-13 Sanofi Dérivés oxathiazine di- et tri-substitués, procédé pour leur préparation, utilisation en tant que médicament, agent pharmaceutique contenant ces dérivés et utilisation
US8901114B2 (en) 2011-03-08 2014-12-02 Sanofi Oxathiazine derivatives substituted with carbocycles or heterocycles, method for producing same, drugs containing said compounds, and use thereof
WO2012120053A1 (fr) 2011-03-08 2012-09-13 Sanofi Dérivés oxathiazine ramifiés, procédé pour leur préparation, utilisation en tant que médicament, agents pharmaceutiques contenant ces dérivés et leur utilisation
WO2012120056A1 (fr) 2011-03-08 2012-09-13 Sanofi Dérivés oxathiazine tétra-substitués, procédé pour leur préparation, utilisation en tant que médicament, agent pharmaceutique contenant ces dérivés et utilisation
WO2012120055A1 (fr) 2011-03-08 2012-09-13 Sanofi Dérivés oxathiazine di- et tri-substitués, procédé pour leur préparation, utilisation en tant que médicament, agent pharmaceutique contenant ces dérivés et utilisation
RU2731913C2 (ru) 2015-08-04 2020-09-09 Астеллас Фарма Инк. Пиперазиновое производное
MX2022015706A (es) 2020-06-09 2023-01-24 Pfizer Antagonistas del receptor de melanocortina 4 y usos de estos.
CA3241470A1 (fr) 2021-12-06 2023-06-15 Pfizer Inc. Antagonistes du recepteur 4 de la melanocortine et leurs utilisations

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CA2098167C (fr) * 1992-06-24 2006-12-19 Dorothea Isler Aliments pour humains et animaux contenant un inhibiteur de la lipase
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ES2421920T3 (es) 2008-08-06 2013-09-06 Pfizer Ltd Compuestos de diazepina y diazocano como agonistas de MC4

Also Published As

Publication number Publication date
EP1989196B1 (fr) 2013-02-13
TNSN08337A1 (fr) 2009-12-29
KR101036981B1 (ko) 2011-05-25
WO2007096763A2 (fr) 2007-08-30
RS20080371A (en) 2009-07-15
ES2402581T3 (es) 2013-05-06
MA30228B1 (fr) 2009-02-02
AU2007219236B2 (en) 2012-06-21
NO20083480L (no) 2008-09-10
ECSP088688A (es) 2008-10-31
AU2007219236A1 (en) 2007-08-30
CA2642922A1 (fr) 2007-08-30
IL193279A0 (en) 2009-02-11
EA200801738A1 (ru) 2008-12-30
US8138188B2 (en) 2012-03-20
DK1989196T3 (da) 2013-04-15
KR20080095918A (ko) 2008-10-29
HK1126489A1 (en) 2009-09-04
BRPI0708264A2 (pt) 2011-05-24
CA2642922C (fr) 2011-08-02
MEP6808A (xx) 2010-02-10
EP1989196A2 (fr) 2008-11-12
CR10219A (es) 2008-09-23
WO2007096763A3 (fr) 2007-10-18
IL193279A (en) 2012-12-31
MX2008010899A (es) 2008-11-27
US20090036459A1 (en) 2009-02-05
SG185849A1 (en) 2012-12-28

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