MX2009012374A - Compuestos novedosos como ligandos del receptor de canabinoides. - Google Patents

Compuestos novedosos como ligandos del receptor de canabinoides.

Info

Publication number
MX2009012374A
MX2009012374A MX2009012374A MX2009012374A MX2009012374A MX 2009012374 A MX2009012374 A MX 2009012374A MX 2009012374 A MX2009012374 A MX 2009012374A MX 2009012374 A MX2009012374 A MX 2009012374A MX 2009012374 A MX2009012374 A MX 2009012374A
Authority
MX
Mexico
Prior art keywords
novel compounds
receptor ligands
cannabinoid receptor
compounds
compositions
Prior art date
Application number
MX2009012374A
Other languages
English (en)
Inventor
Michael J Dart
William A Carroll
Jennifer M Frost
Sridhar Peddi
Arturo Perez-Medrano
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of MX2009012374A publication Critical patent/MX2009012374A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Circuit Arrangement For Electric Light Sources In General (AREA)
  • Led Devices (AREA)

Abstract

La presente solicitud se refiere a compuestos que contienen tiazolilideno de la fórmula (I) en donde R1, R2, R3 y R4 son como se definieron en la descripción. La presente solicitud también se refiere a la composición que comprende dichos compuestos, y los métodos de tratamiento de los padecimientos y enfermedades utilizando dichos compuestos y composiciones.
MX2009012374A 2007-05-18 2008-05-15 Compuestos novedosos como ligandos del receptor de canabinoides. MX2009012374A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US93883807P 2007-05-18 2007-05-18
PCT/US2008/063648 WO2008144360A1 (en) 2007-05-18 2008-05-15 Novel compounds as cannabinoid receptor ligands

Publications (1)

Publication Number Publication Date
MX2009012374A true MX2009012374A (es) 2009-12-01

Family

ID=39552291

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009012374A MX2009012374A (es) 2007-05-18 2008-05-15 Compuestos novedosos como ligandos del receptor de canabinoides.

Country Status (7)

Country Link
US (1) US8735434B2 (es)
EP (1) EP2160393A1 (es)
JP (1) JP2010527929A (es)
CN (1) CN101711253A (es)
CA (1) CA2683086A1 (es)
MX (1) MX2009012374A (es)
WO (1) WO2008144360A1 (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20090018685A (ko) 2006-05-31 2009-02-20 아보트 러보러터리즈 칸나비노이드 수용체 리간드로서의 티아졸 화합물 및 이의 용도
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JP2011513495A (ja) 2008-03-11 2011-04-28 アボット・ラボラトリーズ カンナビノイド受容体リガンドとしての新規な化合物
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EP2428507B1 (en) 2008-09-16 2015-10-21 AbbVie Bahamas Ltd. Cannabinoid receptor ligands
PA8854001A1 (es) * 2008-12-16 2010-07-27 Abbott Lab Compuestos novedosos como ligandos de receptores de canabinoides
TW201130855A (en) 2009-12-16 2011-09-16 Abbott Lab Prodrug compounds useful as cannabinoid ligands

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Also Published As

Publication number Publication date
CN101711253A (zh) 2010-05-19
WO2008144360A1 (en) 2008-11-27
US8735434B2 (en) 2014-05-27
US20080287510A1 (en) 2008-11-20
JP2010527929A (ja) 2010-08-19
EP2160393A1 (en) 2010-03-10
CA2683086A1 (en) 2008-11-18

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