ZA904207B - Avermectin derivatives - Google Patents

Avermectin derivatives

Info

Publication number
ZA904207B
ZA904207B ZA904207A ZA904207A ZA904207B ZA 904207 B ZA904207 B ZA 904207B ZA 904207 A ZA904207 A ZA 904207A ZA 904207 A ZA904207 A ZA 904207A ZA 904207 B ZA904207 B ZA 904207B
Authority
ZA
South Africa
Prior art keywords
avermectin derivatives
avermectin
derivatives
Prior art date
Application number
ZA904207A
Other languages
English (en)
Inventor
Helmut Mrozik
Mrozik Helmut
Peter J Sinclair
J Sinclair Peter
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of ZA904207B publication Critical patent/ZA904207B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
ZA904207A 1989-06-02 1990-06-01 Avermectin derivatives ZA904207B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/360,620 US5030622A (en) 1989-06-02 1989-06-02 Avermectin derivatives

Publications (1)

Publication Number Publication Date
ZA904207B true ZA904207B (en) 1991-03-27

Family

ID=23418773

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA904207A ZA904207B (en) 1989-06-02 1990-06-01 Avermectin derivatives

Country Status (7)

Country Link
US (1) US5030622A (xx)
EP (1) EP0401029A1 (xx)
JP (1) JPH0374397A (xx)
AU (1) AU636613B2 (xx)
CA (1) CA2018097A1 (xx)
NZ (1) NZ233801A (xx)
ZA (1) ZA904207B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2387384T3 (es) * 1999-02-09 2012-09-21 The Kitasato Institute Derivados de avermectina
GB9926887D0 (en) * 1999-11-12 2000-01-12 Novartis Ag Organic compounds
US20040087519A1 (en) * 2000-08-09 2004-05-06 Satoshi Omura Avermectin derivatives
CA2418968C (en) * 2000-08-09 2009-11-24 The Kitasato Institute Avermectin derivatives
US8426460B2 (en) 2008-12-04 2013-04-23 Merial Limited Dimeric avermectin and milbemycin derivatives
US8980896B2 (en) 2009-12-17 2015-03-17 Merial, Inc. Compositions comprising macrocyclic lactone compounds and spirodioxepinoindoles
DK3351546T5 (da) 2011-12-02 2024-08-12 Boehringer Ingelheim Vetmedica Gmbh Langtidsvirkende injicerbare moxidectinformuleringer
CN103421065B (zh) * 2013-07-03 2016-05-18 大庆志飞生物化工有限公司 一类新型阿维菌素衍生物及其制备方法
BR112019011502A2 (pt) * 2016-12-09 2019-11-05 Bayer Animal Health Gmbh preparação farmacêutica e método para sua fabricação

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
ES8800986A1 (es) * 1985-07-27 1987-12-01 Pfizer Un procedimiento para la produccion de un nuevo derivado de avermectina
US4831016A (en) * 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
IN167980B (xx) * 1987-01-23 1991-01-19 Pfizer
ES2058244T3 (es) * 1987-01-23 1994-11-01 Pfizer Procedimiento para produccion de avermectinas y cultivos para el mismo.
US4806527A (en) * 1987-03-16 1989-02-21 Merck & Co., Inc. Avermectin derivatives
US4874749A (en) * 1987-07-31 1989-10-17 Merck & Co., Inc. 4"-Deoxy-4-N-methylamino avermectin Bla/Blb
US4873224A (en) * 1988-05-23 1989-10-10 Merck & Co., Inc. Avermectin derivatives
US4906619A (en) * 1988-07-22 1990-03-06 Merck & Co., Inc. Alkyl avermectin derivatives

Also Published As

Publication number Publication date
JPH0374397A (ja) 1991-03-28
AU5622190A (en) 1990-12-06
US5030622A (en) 1991-07-09
CA2018097A1 (en) 1990-12-02
AU636613B2 (en) 1993-05-06
NZ233801A (en) 1992-06-25
EP0401029A1 (en) 1990-12-05

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