ZA886120B - New avermectin derivatives,a process for their preparation and their use - Google Patents
New avermectin derivatives,a process for their preparation and their useInfo
- Publication number
- ZA886120B ZA886120B ZA886120A ZA886120A ZA886120B ZA 886120 B ZA886120 B ZA 886120B ZA 886120 A ZA886120 A ZA 886120A ZA 886120 A ZA886120 A ZA 886120A ZA 886120 B ZA886120 B ZA 886120B
- Authority
- ZA
- South Africa
- Prior art keywords
- preparation
- avermectin derivatives
- new avermectin
- new
- derivatives
- Prior art date
Links
- RRZXIRBKKLTSOM-XPNPUAGNSA-N avermectin B1a Chemical class C1=C[C@H](C)[C@@H]([C@@H](C)CC)O[C@]11O[C@H](C\C=C(C)\[C@@H](O[C@@H]2O[C@@H](C)[C@H](O[C@@H]3O[C@@H](C)[C@H](O)[C@@H](OC)C3)[C@@H](OC)C2)[C@@H](C)\C=C\C=C/2[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\2)O)C[C@H]4C1 RRZXIRBKKLTSOM-XPNPUAGNSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19873727648 DE3727648A1 (de) | 1987-08-19 | 1987-08-19 | Neue avermectin derivate, verfahren zu ihrer herstellung und ihre verwendung |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA886120B true ZA886120B (en) | 1989-05-30 |
Family
ID=6334058
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA886120A ZA886120B (en) | 1987-08-19 | 1988-08-18 | New avermectin derivatives,a process for their preparation and their use |
Country Status (8)
Country | Link |
---|---|
US (1) | US4916120A (pt) |
EP (1) | EP0303933A3 (pt) |
JP (1) | JPS6468378A (pt) |
AU (1) | AU2114088A (pt) |
BR (1) | BR8804191A (pt) |
DE (1) | DE3727648A1 (pt) |
NZ (1) | NZ225837A (pt) |
ZA (1) | ZA886120B (pt) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8801908D0 (en) * | 1988-01-28 | 1988-02-24 | Glaxo Group Ltd | Chemical compounds |
NZ228866A (en) * | 1988-05-02 | 1991-10-25 | Merck & Co Inc | Fluoro-substituted milbemycins and avermectins for combatting parasites and insects |
US6001822A (en) * | 1989-04-11 | 1999-12-14 | Pfizer Inc. | Antiparasitic formulations |
US5057499A (en) * | 1989-06-02 | 1991-10-15 | Merck & Co. Inc. | Avermectin derivatives |
US5830875A (en) * | 1989-10-30 | 1998-11-03 | Merck & Co., Inc. | 24-and 25-substituted avermectin and milbemycin derivatives |
US5208222A (en) * | 1991-03-28 | 1993-05-04 | Merck & Co., Inc. | 4"-and 4'-alkylthio avermectin derivatives |
US5290804A (en) * | 1991-05-01 | 1994-03-01 | Merck & Co., Inc. | Anthelmintic milbemycin analogs of novel microorganisms |
US5189026A (en) * | 1991-06-07 | 1993-02-23 | Fractal Laboratories, Inc. | Treatment of human diseases involving dysregulation or dysfunction of the nervous system |
US5262400A (en) * | 1991-06-20 | 1993-11-16 | Merck & Co., Inc. | 4α-substituted avermectin derivatives |
US5240915A (en) * | 1991-10-15 | 1993-08-31 | Merck & Co., Inc. | Avermectin derivatives |
PL174488B1 (pl) * | 1993-05-10 | 1998-08-31 | Merck & Co Inc | Preparat do zwalczania pasożytów zwierząt oraz sposób wytwarzania preparatu do zwalczania pasożytów zwierząt |
US5602107A (en) * | 1993-05-10 | 1997-02-11 | Merck & Co., Inc. | Pour-on formulations consisting of gylcols, glycerides and avermectin compounds |
GB9312154D0 (en) * | 1993-06-12 | 1993-07-28 | Pfizer Ltd | Antiparasitic agents |
US5606517A (en) * | 1994-06-08 | 1997-02-25 | Exa Corporation | Viscosity reduction in physical process simulation |
DE69636706T2 (de) * | 1995-09-25 | 2007-10-11 | Ashmont Holdings Ltd., Takapuna | Makrocyclische lacton anthelmintika |
US5773422A (en) * | 1996-01-29 | 1998-06-30 | Komer; Gene | Avermectin formulation |
DE19613972A1 (de) * | 1996-04-09 | 1997-10-16 | Bayer Ag | Injektionsformulierungen von Avermectinen und Milbemycinen auf Basis von Rizinusöl |
KR100483912B1 (ko) * | 1996-04-09 | 2005-08-31 | 바이엘 악티엔게젤샤프트 | 피마자유를기초로한아버멕틴과밀베마이신의주사제제 |
US5788978A (en) * | 1996-12-17 | 1998-08-04 | Passeron; Eduardo Julio | Injectable pulsatile ivermectin composition |
US6054140A (en) * | 1997-03-21 | 2000-04-25 | Biogenesis S.A. | Long acting injectable parasiticidal composition and the process for its preparation |
GB9825402D0 (en) † | 1998-11-19 | 1999-01-13 | Pfizer Ltd | Antiparasitic formulations |
BRPI0509673A (pt) * | 2004-04-07 | 2007-10-09 | Intervet Int Bv | composição para o tratamento de parasitas, forma de dosagem farmacêutica, método para tratar um organismo, e, processos para introduzir pelo menos um aditivo em um organismo, para fabricar uma composição, para liberar um aditivo em um organismo, e, para conformar um produto macio mastigável |
DE102004053964A1 (de) * | 2004-11-09 | 2006-05-11 | Bayer Healthcare Ag | Mittel gegen Demodikose |
RU2688919C1 (ru) | 2013-12-20 | 2019-05-23 | Интервет Интернэшнл Б.В. | Изоксазолиновые композиции и их применение в провилактике или лечении паразитарных инвазий животных |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5663993A (en) * | 1979-10-30 | 1981-05-30 | Microbial Chem Res Found | Novel preparation of tobramycin |
US4333925A (en) * | 1981-05-11 | 1982-06-08 | Merck & Co., Inc. | Derivatives of C-076 compounds |
US4423209A (en) * | 1982-02-26 | 1983-12-27 | Merck & Co., Inc. | Processes for the interconversion of avermectin compounds |
-
1987
- 1987-08-19 DE DE19873727648 patent/DE3727648A1/de not_active Withdrawn
-
1988
- 1988-08-01 US US07/230,221 patent/US4916120A/en not_active Expired - Fee Related
- 1988-08-08 EP EP88112884A patent/EP0303933A3/de not_active Withdrawn
- 1988-08-16 NZ NZ225837A patent/NZ225837A/xx unknown
- 1988-08-18 AU AU21140/88A patent/AU2114088A/en not_active Abandoned
- 1988-08-18 BR BR8804191A patent/BR8804191A/pt unknown
- 1988-08-18 ZA ZA886120A patent/ZA886120B/xx unknown
- 1988-08-19 JP JP63204836A patent/JPS6468378A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
DE3727648A1 (de) | 1989-03-02 |
NZ225837A (en) | 1990-04-26 |
EP0303933A2 (de) | 1989-02-22 |
AU2114088A (en) | 1989-02-23 |
EP0303933A3 (de) | 1989-10-25 |
BR8804191A (pt) | 1989-03-14 |
US4916120A (en) | 1990-04-10 |
JPS6468378A (en) | 1989-03-14 |
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