ZA881226B - Labile ketone derivatives of 3-substituted-1-alkylamino 2-propanols and their use as beta-adrenergic blockers - Google Patents
Labile ketone derivatives of 3-substituted-1-alkylamino 2-propanols and their use as beta-adrenergic blockersInfo
- Publication number
- ZA881226B ZA881226B ZA881226A ZA881226A ZA881226B ZA 881226 B ZA881226 B ZA 881226B ZA 881226 A ZA881226 A ZA 881226A ZA 881226 A ZA881226 A ZA 881226A ZA 881226 B ZA881226 B ZA 881226B
- Authority
- ZA
- South Africa
- Prior art keywords
- beta
- alkylamino
- propanols
- substituted
- present
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
- C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/32—Oximes
- C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
- C07C251/36—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atoms of the oxyimino groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C251/38—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atoms of the oxyimino groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of a saturated carbon skeleton
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Ophthalmology & Optometry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Furan Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2600287A | 1987-03-16 | 1987-03-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA881226B true ZA881226B (en) | 1988-08-17 |
Family
ID=21829283
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA881226A ZA881226B (en) | 1987-03-16 | 1988-02-22 | Labile ketone derivatives of 3-substituted-1-alkylamino 2-propanols and their use as beta-adrenergic blockers |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP0283147B1 (xx) |
| JP (2) | JPH01501797A (xx) |
| KR (1) | KR960008766B1 (xx) |
| AT (1) | ATE105547T1 (xx) |
| AU (1) | AU609788B2 (xx) |
| CA (1) | CA1335286C (xx) |
| DE (2) | DE3889486T4 (xx) |
| DK (1) | DK626588A (xx) |
| ES (1) | ES2051831T3 (xx) |
| FI (1) | FI94337C (xx) |
| IE (1) | IE62828B1 (xx) |
| NO (1) | NO171312C (xx) |
| WO (1) | WO1988007036A1 (xx) |
| ZA (1) | ZA881226B (xx) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1988007036A1 (en) * | 1987-03-16 | 1988-09-22 | University Of Florida | LABILE KETONE DERIVATIVES OF 3-SUBSTITUTED-1-ALKYLAMINO-2-PROPANOLS AND THEIR USE AS beta-ADRENERGIC BLOCKERS |
| US5177064A (en) * | 1990-07-13 | 1993-01-05 | University Of Florida | Targeted drug delivery via phosphonate derivatives |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3619370A (en) * | 1969-04-21 | 1971-11-09 | Frosst & Co Charles E | Microbial reduction of thiadiazoles |
| DE2645710C2 (de) * | 1976-10-09 | 1985-06-27 | Merck Patent Gmbh, 6100 Darmstadt | Phenoxy-amino-propanole, Verfahren zu ihrer Herstellung und pharmazeutische Zubereitung |
| JPS563862A (en) * | 1979-06-26 | 1981-01-16 | Nippon Denso Co | Refrigeration device |
| IL65541A0 (en) * | 1981-05-06 | 1982-07-30 | Haessle Ab | Alkylamino-2-propanols,process for their preparation and pharmaceutical preparations containing same |
| US4521414A (en) * | 1981-06-18 | 1985-06-04 | The Texas A&M University System | Ophthalmic compositions and their use for treating elevated intraocular pressure and glaucoma |
| DE3270905D1 (en) * | 1981-12-17 | 1986-06-05 | Haessle Ab | Para-substituted 3-phenoxy-1-carbonylaminoalkylamino-propan-2-ols having beta receptor blocking properties |
| US4616022A (en) * | 1984-08-17 | 1986-10-07 | Warner-Lambert Company | Procaterol stabilization |
| WO1988007036A1 (en) * | 1987-03-16 | 1988-09-22 | University Of Florida | LABILE KETONE DERIVATIVES OF 3-SUBSTITUTED-1-ALKYLAMINO-2-PROPANOLS AND THEIR USE AS beta-ADRENERGIC BLOCKERS |
-
1988
- 1988-02-16 WO PCT/US1988/000386 patent/WO1988007036A1/en active IP Right Grant
- 1988-02-16 JP JP63501931A patent/JPH01501797A/ja active Granted
- 1988-02-16 AU AU13459/88A patent/AU609788B2/en not_active Expired
- 1988-02-22 IE IE47588A patent/IE62828B1/en not_active IP Right Cessation
- 1988-02-22 ZA ZA881226A patent/ZA881226B/xx unknown
- 1988-02-25 ES ES88301615T patent/ES2051831T3/es not_active Expired - Lifetime
- 1988-02-25 DE DE3889486T patent/DE3889486T4/de not_active Expired - Lifetime
- 1988-02-25 AT AT8888301615T patent/ATE105547T1/de not_active IP Right Cessation
- 1988-02-25 EP EP88301615A patent/EP0283147B1/en not_active Expired - Lifetime
- 1988-02-25 DE DE3889486A patent/DE3889486D1/de not_active Expired - Lifetime
- 1988-02-26 CA CA000560031A patent/CA1335286C/en not_active Expired - Fee Related
- 1988-11-10 DK DK626588A patent/DK626588A/da not_active Application Discontinuation
- 1988-11-15 FI FI885271A patent/FI94337C/fi active IP Right Grant
- 1988-11-15 NO NO885081A patent/NO171312C/no not_active IP Right Cessation
- 1988-12-16 KR KR1019880701483A patent/KR960008766B1/ko not_active IP Right Cessation
-
1992
- 1992-10-19 JP JP4306006A patent/JPH06122624A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| IE880475L (en) | 1988-09-16 |
| DE3889486T2 (de) | 1994-09-01 |
| KR960008766B1 (ko) | 1996-07-03 |
| NO171312B (no) | 1992-11-16 |
| JPH06122624A (ja) | 1994-05-06 |
| FI885271A0 (fi) | 1988-11-15 |
| NO171312C (no) | 1993-02-24 |
| JPH0518820B2 (xx) | 1993-03-15 |
| EP0283147A1 (en) | 1988-09-21 |
| FI94337B (fi) | 1995-05-15 |
| NO885081D0 (no) | 1988-11-15 |
| JPH01501797A (ja) | 1989-06-22 |
| ES2051831T3 (es) | 1994-07-01 |
| AU1345988A (en) | 1988-10-10 |
| IE62828B1 (en) | 1995-03-08 |
| DK626588A (da) | 1988-12-08 |
| EP0283147B1 (en) | 1994-05-11 |
| DE3889486D1 (de) | 1994-06-16 |
| DK626588D0 (da) | 1988-11-10 |
| CA1335286C (en) | 1995-04-18 |
| ATE105547T1 (de) | 1994-05-15 |
| FI885271A (fi) | 1988-11-15 |
| WO1988007036A1 (en) | 1988-09-22 |
| DE3889486T4 (de) | 1994-12-01 |
| KR890700573A (ko) | 1989-04-25 |
| FI94337C (fi) | 1995-08-25 |
| AU609788B2 (en) | 1991-05-09 |
| NO885081L (no) | 1989-01-13 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES8202546A1 (es) | Metodo de producir derivados de tiazolidina | |
| EP0251315A3 (en) | Naphthalene derivatives, process for their preparation and pharmaceutical compositions containing the same | |
| AU586691B2 (en) | Diamino-androstane derivatives, process for their preparation and pharmaceutical compositions containing them | |
| GR3024896T3 (en) | Steroid derivatives for the treatment of prostatic hypertrophy, their preparation and uses | |
| IL89929A0 (en) | Beta-lactam derivatives,their preparation and pharmaceutical compositions containing them | |
| KR910016915A (ko) | 과콜레스테롤혈증 치료제 | |
| HUT57694A (en) | Process for producing new beta-diketones and pharmaceutical compositions comprising same | |
| ZA881226B (en) | Labile ketone derivatives of 3-substituted-1-alkylamino 2-propanols and their use as beta-adrenergic blockers | |
| ES8705410A1 (es) | Un procedimiento para preparar un derivado de 1,5 beurotiarepina. | |
| GB2179653B (en) | Heterocyclic compounds | |
| HU910108D0 (en) | Process for the production of macrolide compounds | |
| HUT47923A (en) | Process for production of new derivatives of naphtotiazephin and medical compositions containing these substances | |
| AU623794B2 (en) | Method of treating diabetes mellitus with bisphenol derivatives | |
| DE3363575D1 (en) | Furyloxazolylacetic acid derivatives, process for preparing same and pharmaceutical compositions containing same | |
| NO974747L (no) | Fremgangsmåte for fremstilling av streptograminer | |
| JPS5649380A (en) | Cephalosporin analogue | |
| SE8205767D0 (sv) | A titre de medicaments, certains derives mono substitues de lacide 4-phenyl 4-oxo buten-2-oigue, ainsi que les compositions les renfermant | |
| ES8506679A2 (es) | Mejoras en el objeto de la patente de invencion n 514.340 que se refiere a: procedimiento de obtencion de nuevos derivados de piperazina | |
| EP0307221A3 (en) | Process for the preparation of macrolide compounds |