ZA869591B - Substituted 5,6-dialkoxyquinazoline derivatives - Google Patents

Substituted 5,6-dialkoxyquinazoline derivatives

Info

Publication number
ZA869591B
ZA869591B ZA869591A ZA869591A ZA869591B ZA 869591 B ZA869591 B ZA 869591B ZA 869591 A ZA869591 A ZA 869591A ZA 869591 A ZA869591 A ZA 869591A ZA 869591 B ZA869591 B ZA 869591B
Authority
ZA
South Africa
Prior art keywords
dialkoxyquinazoline
derivatives
substituted
dialkoxyquinazoline derivatives
Prior art date
Application number
ZA869591A
Other languages
English (en)
Inventor
Victor T Bandurco
Stanley C Bell
John H Dodd
Robert Faltico
Charles F Schwender
Alfonso J Tobia
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of ZA869591B publication Critical patent/ZA869591B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA869591A 1985-12-20 1986-12-19 Substituted 5,6-dialkoxyquinazoline derivatives ZA869591B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/811,233 US4672116A (en) 1985-12-20 1985-12-20 Substituted 5,6-dialkoxyquinazoline derivatives

Publications (1)

Publication Number Publication Date
ZA869591B true ZA869591B (en) 1988-07-27

Family

ID=25205964

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA869591A ZA869591B (en) 1985-12-20 1986-12-19 Substituted 5,6-dialkoxyquinazoline derivatives

Country Status (6)

Country Link
US (1) US4672116A (de)
EP (1) EP0227450A3 (de)
JP (1) JPS62187462A (de)
AU (1) AU6675186A (de)
DK (1) DK615186A (de)
ZA (1) ZA869591B (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU610328B2 (en) * 1987-12-03 1991-05-16 Smithkline Beckman Intercredit B.V. 2,4- diaminoquinazoline derivatives
US4877790A (en) * 1987-12-15 1989-10-31 Kanebo Limited Quinazoline derivative, processes for its production, and cerebral dysfunction remedying agent comprising it as active ingredient
DE68917485T2 (de) * 1988-01-23 1995-02-09 Kyowa Hakko Kogyo Kk Pyridazinon-Derivate und diese enthaltende pharmazeutische Zubereitungen.
US5411963A (en) * 1988-01-29 1995-05-02 Dowelanco Quinazoline derivatives
US5214144A (en) * 1991-10-07 1993-05-25 Dowelanco Process for the preparation of 4-haloquinazolines
CA2077252C (en) * 1992-08-31 2001-04-10 Khashayar Karimian Methods of making ureas and guanidines, and intermediates therefor
IL108630A0 (en) * 1993-02-18 1994-05-30 Fmc Corp Insecticidal substituted 2,4-diaminoquinazolines
TW334434B (en) * 1995-05-16 1998-06-21 Kanebo Ltd Novel quinazoline compound and anti-tumor agent
JP2006523640A (ja) * 2003-04-16 2006-10-19 エフ.ホフマン−ラ ロシュ アーゲー 置換7−アザ−キナゾリン化合物
CN1774425A (zh) * 2003-04-16 2006-05-17 霍夫曼-拉罗奇有限公司 喹唑啉化合物
WO2008084493A2 (en) * 2007-01-09 2008-07-17 Unichem Laboratories Limited A novel process for the preparation of 2-halo-4-aminoquinazolines
US9603848B2 (en) 2007-06-08 2017-03-28 Senomyx, Inc. Modulation of chemosensory receptors and ligands associated therewith
US7928111B2 (en) 2007-06-08 2011-04-19 Senomyx, Inc. Compounds including substituted thienopyrimidinone derivatives as ligands for modulating chemosensory receptors
CA2731800C (en) 2008-07-31 2018-03-20 Senomyx, Inc. Processes and intermediates for making sweet taste enhancers
MX354835B (es) 2012-08-06 2018-03-21 Senomyx Inc Modificador del sabor dulce.
JO3155B1 (ar) 2013-02-19 2017-09-20 Senomyx Inc معدِّل نكهة حلوة
MX2021001193A (es) 2018-08-07 2021-04-28 Firmenich Incorporated 2,2-dioxidos de 4-amino-1h-benzo[c][1,2,6]tiadiazina 5-sustituidos y formulaciones y usos de los mismos.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4287341A (en) * 1979-11-01 1981-09-01 Pfizer Inc. Alkoxy-substituted-6-chloro-quinazoline-2,4-diones
US4351832A (en) * 1980-04-18 1982-09-28 American Home Products Corporation 2-(Piperazinyl)-4-pyrimidinamines
US4634769A (en) * 1984-09-25 1987-01-06 Ortho Pharmaceutical Corporation Process for the preparation of 8-halo-5,6-dialkoxyquinazoline-2,4-diones and their salts

Also Published As

Publication number Publication date
US4672116A (en) 1987-06-09
JPS62187462A (ja) 1987-08-15
DK615186D0 (da) 1986-12-18
AU6675186A (en) 1987-06-25
EP0227450A2 (de) 1987-07-01
DK615186A (da) 1987-06-21
EP0227450A3 (de) 1988-01-07

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