ZA854364B - Avermectin and milbemycin 12-keto,12-imino and 13-amino derivatives - Google Patents
Avermectin and milbemycin 12-keto,12-imino and 13-amino derivativesInfo
- Publication number
- ZA854364B ZA854364B ZA854364A ZA854364A ZA854364B ZA 854364 B ZA854364 B ZA 854364B ZA 854364 A ZA854364 A ZA 854364A ZA 854364 A ZA854364 A ZA 854364A ZA 854364 B ZA854364 B ZA 854364B
- Authority
- ZA
- South Africa
- Prior art keywords
- milbemycin
- avermectin
- keto
- imino
- amino derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
- A01N47/34—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the groups, e.g. biuret; Thio analogues thereof; Urea-aldehyde condensation products
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Veterinary Medicine (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biochemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/619,238 US4579864A (en) | 1984-06-11 | 1984-06-11 | Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA854364B true ZA854364B (en) | 1986-02-26 |
Family
ID=24481058
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA854364A ZA854364B (en) | 1984-06-11 | 1985-06-10 | Avermectin and milbemycin 12-keto,12-imino and 13-amino derivatives |
Country Status (7)
Country | Link |
---|---|
US (1) | US4579864A (ja) |
EP (1) | EP0165029B1 (ja) |
JP (1) | JPH0753734B2 (ja) |
AU (1) | AU569624B2 (ja) |
DE (1) | DE3574019D1 (ja) |
NZ (1) | NZ212289A (ja) |
ZA (1) | ZA854364B (ja) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4587247A (en) * | 1985-02-25 | 1986-05-06 | Merck & Co., Inc. | Substituted and unsubstituted 13-(alkoxy)methoxy derivatives of the avermectin aglycones, compositions and use |
NZ219576A (en) * | 1986-03-12 | 1989-01-06 | Glaxo Group Ltd | Milbemycin derivatives and pharmaceutical, veterinary, and pesticidal compositions |
ES2054664T3 (es) * | 1986-03-12 | 1994-08-16 | American Cyanamid Co | Compuestos macrolidos. |
GB8606108D0 (en) * | 1986-03-12 | 1986-04-16 | Glaxo Group Ltd | Chemical compounds |
US5336789A (en) * | 1986-03-12 | 1994-08-09 | American Cyanamid Company | Macrolide compounds |
US5185456A (en) * | 1986-03-12 | 1993-02-09 | American Cyanamid Company | Macrolide compounds |
EP0342710B1 (en) * | 1986-03-25 | 1993-05-19 | Sankyo Company Limited | Macrolide compounds, their preparation and their use |
CA1296329C (en) * | 1986-06-06 | 1992-02-25 | Derek R. Sutherland | Macrolide compounds |
EP0253378A3 (de) * | 1986-07-18 | 1988-03-23 | Ciba-Geigy Ag | 13Beta-Alkyl-derivate von S541-Antibiotika zur Bekämpfung von Parasiten an Nutztieren und Pflanzen |
US4916154A (en) * | 1986-09-12 | 1990-04-10 | American Cyanamid Company | 23-Imino derivatives of LL-F28249 compounds |
US4831016A (en) * | 1986-10-31 | 1989-05-16 | Merck & Co., Inc. | Reduced avermectin derivatives |
IL85119A (en) * | 1987-01-23 | 1993-01-14 | Pfizer | Streptomyces avermitilis strains, their preparation and use in production of avermectins |
US4886829A (en) * | 1987-03-06 | 1989-12-12 | American Cyanamid Company | 23-Oxo (keto) and 23-imino derivatives of mono- and diepoxy LL-F28249 compounds |
US5192777A (en) * | 1987-09-11 | 1993-03-09 | American Cyanamid Company | Macrolide compounds |
GB8721375D0 (en) * | 1987-09-11 | 1987-10-21 | Glaxo Group Ltd | Chemical process |
GB8721378D0 (en) * | 1987-09-11 | 1987-10-21 | Glaxo Group Ltd | Chemical process |
DE3888936T2 (de) * | 1987-11-03 | 1994-07-21 | Beecham Group Plc | Zwischenprodukte für die Herstellung makrolider Antibiotika mit anthelmintischer Wirkung. |
GB8811037D0 (en) * | 1988-05-10 | 1988-06-15 | Glaxo Group Ltd | Chemical compounds |
US4873224A (en) * | 1988-05-23 | 1989-10-10 | Merck & Co., Inc. | Avermectin derivatives |
US5428034A (en) * | 1988-09-02 | 1995-06-27 | Sankyo Co., Ltd. | Milbemycin derivatives, their preparation and their use |
US5023241A (en) * | 1989-07-31 | 1991-06-11 | Merck & Co., Inc. | Avermectin derivatives |
JP2622197B2 (ja) * | 1990-03-01 | 1997-06-18 | 三共株式会社 | 13−エーテル置換ミルベマイシン誘導体 |
US5194301A (en) * | 1990-08-09 | 1993-03-16 | Investigacion Y Desarrollo, C.A. | Process for reducing scale formation in vinyl polymerization reactors |
EG19869A (en) * | 1991-12-18 | 1996-03-31 | Sankyo Co | Substituted thio acetoxymilbemycon derivatives their preparation and their agrochemical uses |
DK0765879T3 (da) * | 1995-09-29 | 2001-03-19 | Sankyo Co | 13-substituerede milbemycin 5-oximderivater, deres fremstilling og deres anvendelse over for insekter og andre skadedyr |
AT501406A1 (de) * | 1997-12-23 | 2006-08-15 | Syngenta Participations Ag | Verfahren zur bekämpfung von mollusken |
AU2001252613B2 (en) | 2000-04-27 | 2004-05-13 | Novartis Animal Health K.K. | 13-substituted milbemycin derivatives, their preparation and their use against insects and other pests |
CN103896961A (zh) * | 2014-03-25 | 2014-07-02 | 武汉大学 | 一种米尔贝肟类化合物及其制备方法 |
CN105037467A (zh) * | 2015-05-29 | 2015-11-11 | 河北威远生化农药有限公司 | 4”-脱氧-4”烷基化或酰基化胺基阿维菌素B2a/2b衍生物及其制备方法和用途 |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3950360A (en) * | 1972-06-08 | 1976-04-13 | Sankyo Company Limited | Antibiotic substances |
SE434277B (sv) * | 1976-04-19 | 1984-07-16 | Merck & Co Inc | Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis |
US4093629A (en) * | 1977-04-11 | 1978-06-06 | Merck & Co., Inc. | Derivatives of antibiotic substance milbemycin and processes therefor |
US4134973A (en) * | 1977-04-11 | 1979-01-16 | Merck & Co., Inc. | Carbohydrate derivatives of milbemycin and processes therefor |
US4199569A (en) * | 1977-10-03 | 1980-04-22 | Merck & Co., Inc. | Selective hydrogenation products of C-076 compounds and derivatives thereof |
US4201861A (en) * | 1977-10-03 | 1980-05-06 | Merck & Co., Inc. | Acyl derivatives of C-076 compounds |
US4206205A (en) * | 1977-10-03 | 1980-06-03 | Merck & Co., Inc. | Monosaccharide and aglycone derivatives of C-076 |
US4173571A (en) * | 1977-12-19 | 1979-11-06 | Merck & Co., Inc. | 13-Halo and 13-deoxy derivatives of C-076 compounds |
US4171314A (en) * | 1977-12-19 | 1979-10-16 | Merck & Co., Inc. | 13-Halo and 13-deoxy C-076 compounds |
US4289760A (en) * | 1980-05-02 | 1981-09-15 | Merck & Co., Inc. | 23-Keto derivatives of C-076 compounds |
NZ201681A (en) * | 1981-09-03 | 1985-11-08 | Merck & Co Inc | Avermectin derivatives and parasiticidal compositions |
US4427663A (en) * | 1982-03-16 | 1984-01-24 | Merck & Co., Inc. | 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof |
JPS5920285A (ja) * | 1982-07-23 | 1984-02-01 | Sankyo Co Ltd | ミルベマイシンdの5−二塩基酸エステル誘導体及びその塩 |
JPS59108785A (ja) * | 1982-11-25 | 1984-06-23 | Sankyo Co Ltd | ミルベマイシン類の5−オキシム誘導体 |
-
1984
- 1984-06-11 US US06/619,238 patent/US4579864A/en not_active Expired - Lifetime
-
1985
- 1985-06-04 NZ NZ212289A patent/NZ212289A/en unknown
- 1985-06-07 AU AU43409/85A patent/AU569624B2/en not_active Ceased
- 1985-06-07 EP EP85304063A patent/EP0165029B1/en not_active Expired
- 1985-06-07 DE DE8585304063T patent/DE3574019D1/de not_active Expired
- 1985-06-10 ZA ZA854364A patent/ZA854364B/xx unknown
- 1985-06-11 JP JP60125281A patent/JPH0753734B2/ja not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
JPS6122087A (ja) | 1986-01-30 |
US4579864A (en) | 1986-04-01 |
NZ212289A (en) | 1988-05-30 |
EP0165029B1 (en) | 1989-11-02 |
AU569624B2 (en) | 1988-02-11 |
AU4340985A (en) | 1985-12-19 |
DE3574019D1 (en) | 1989-12-07 |
EP0165029A1 (en) | 1985-12-18 |
JPH0753734B2 (ja) | 1995-06-07 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ZA854364B (en) | Avermectin and milbemycin 12-keto,12-imino and 13-amino derivatives | |
NZ216980A (en) | 25-substituted avermectin derivatives | |
NZ225542A (en) | Avermectin derivatives and parasiticidal compositions | |
AU2740188A (en) | N6-hydroxycycloalkyl and N6-hydroxycycloakenyl adenosine derivatives | |
NZ223272A (en) | Avermectin derivatives and parasiticidal compositions | |
AU1313288A (en) | Avermectin derivatives | |
AU574566B2 (en) | 13-akoxymethoxy avermectin aglycone derivatives | |
AU587200B2 (en) | Treatment of cancer with phlorizin and its derivatives | |
ZA89538B (en) | Avermectin derivatives | |
NZ225837A (en) | Avermectin derivatives and pesticidal compositions | |
NZ212673A (en) | Avermectin and milbemycin derivatives and parasiticidal compositions | |
NZ220587A (en) | Milbemycin derivatives and compositions | |
AU1907788A (en) | N-aminobutyl-n-phenylarylamide derivatives, their preparation and their application in therapy | |
ZA899818B (en) | Avermectin derivatives | |
NZ219577A (en) | Milbemycin derivatives and compositions | |
DE3560679D1 (en) | 4-hydroxy-2h-1-benzothiopyran-2-one derivatives, their preparation and uses | |
EP0172581A3 (en) | Disaccharide derivatives | |
AU7827687A (en) | Macrolide derivatives | |
IL75428A0 (en) | Milbemycin derivatives,their preparation and their use as pesticides | |
AU5668286A (en) | Carbohydrate derivatives and compositions thereof for therapeutic or diagnostic use, and methods for their use | |
NZ221350A (en) | Uridine derivatives and pharmaceutical preparation | |
NZ215917A (en) | 22-oh milbemycin derivatives and parasiticidal compositions | |
AU7888487A (en) | Morpholine and hydrogenated pyridine derivatives | |
AU578739B2 (en) | Vinyltetrazolylphenyl derivatives, their preparation and their use | |
NZ216908A (en) | Avermectin derivatives |