ZA838829B - Esters of 3-(3-substituted-amino-2-hydroxypropoxy)-4-substituted-1,2,5-thiadiazole derivatives - Google Patents

Esters of 3-(3-substituted-amino-2-hydroxypropoxy)-4-substituted-1,2,5-thiadiazole derivatives

Info

Publication number
ZA838829B
ZA838829B ZA838829A ZA838829A ZA838829B ZA 838829 B ZA838829 B ZA 838829B ZA 838829 A ZA838829 A ZA 838829A ZA 838829 A ZA838829 A ZA 838829A ZA 838829 B ZA838829 B ZA 838829B
Authority
ZA
South Africa
Prior art keywords
substituted
hydroxypropoxy
esters
amino
thiadiazole derivatives
Prior art date
Application number
ZA838829A
Other languages
English (en)
Inventor
William L Matier
Paul W Erhardt
Ghanshyam Patil
Original Assignee
American Hospital Supply Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Hospital Supply Corp filed Critical American Hospital Supply Corp
Publication of ZA838829B publication Critical patent/ZA838829B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ZA838829A 1982-12-22 1983-11-25 Esters of 3-(3-substituted-amino-2-hydroxypropoxy)-4-substituted-1,2,5-thiadiazole derivatives ZA838829B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/452,280 US4508725A (en) 1982-12-22 1982-12-22 Esters of 3-(3-substituted-amino-2-hydroxypropoxy)-4-substituted-1,2,5-thiadiazole derivatives

Publications (1)

Publication Number Publication Date
ZA838829B true ZA838829B (en) 1985-03-27

Family

ID=23795857

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA838829A ZA838829B (en) 1982-12-22 1983-11-25 Esters of 3-(3-substituted-amino-2-hydroxypropoxy)-4-substituted-1,2,5-thiadiazole derivatives

Country Status (14)

Country Link
US (1) US4508725A (fr)
EP (1) EP0131006B1 (fr)
JP (1) JPS60500288A (fr)
AU (1) AU567908B2 (fr)
CA (1) CA1230879A (fr)
DE (1) DE3382578T2 (fr)
ES (1) ES8504159A1 (fr)
IE (1) IE59617B1 (fr)
IT (1) IT1172381B (fr)
MX (1) MX156097A (fr)
NO (1) NO164095C (fr)
NZ (1) NZ206385A (fr)
WO (1) WO1984002525A1 (fr)
ZA (1) ZA838829B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623652A (en) 1981-11-12 1986-11-18 American Hospital Supply Corporation Esters of thiadiazole oxypropanolaine derivatives and pharmaceutical uses
CA2120603A1 (fr) * 1991-10-11 1993-04-15 Louis Desantis Jr. Compositions opthalmiques topiques comportant des 4-[(groupe amino substitueen 3)-2-hydroxypropoxy]-1,2,5-thiadiazoles et methodes pour leur utilisation
US5320839A (en) * 1991-10-11 1994-06-14 Alcon Laboratories, Inc. Topical ophthalmic compositions comprising 4-(3-substituted amino-2-hydroxypropoxy)-1,2,5-thiadiazoles and methods for their use
US5672709A (en) * 1994-10-24 1997-09-30 Eli Lilly And Company Heterocyclic compounds and their preparation and use
US6750238B1 (en) 2000-05-12 2004-06-15 The University Of Toledo Aralkyl ester soft drugs
US7049326B2 (en) 2000-05-12 2006-05-23 The University Of Toledo Method and compositions for temporarily incapacitating subjects
US6756047B2 (en) 2000-05-12 2004-06-29 The University Of Toledo Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
US20110092507A1 (en) * 2009-10-20 2011-04-21 Chin-Tsai Fan Process for preparing R-(+)-3-morpholino-4-(3- tert-butylamino-2-hydroxypropoxy)-1,2,5-thiadiazole

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4051144A (en) * 1968-05-22 1977-09-27 Charles E. Frosst & Co. Sinister-3,5-disubstituted oxozolidines their preparation and use
US3655663A (en) * 1969-04-21 1972-04-11 Burton K Wasson 4-(3-secondary amino-2-hydroxy-proxy) 1 2 5-thiadiazoles
FR2132570B1 (fr) * 1971-04-09 1974-08-02 Lipha
US3729477A (en) * 1971-09-09 1973-04-24 Frosst & Co Charles E Certain 4-(3-amino-2-hydroxypropoxy)-1,2,5-thiadiazole-3-carboxamides
US4083992A (en) * 1972-12-15 1978-04-11 Imperial Chemical Industries Limited Alkanolamine derivatives
US4011217A (en) * 1973-04-19 1977-03-08 Merck Sharp & Dohme (I.A.) Corporation 4-(3-amino-2-acyloxypropoxy)-1,2,5-thiadiazole compounds
US3891639A (en) * 1973-04-19 1975-06-24 Merck Sharp & Dohme 4-{8 3-Amino-2-acyloxypropoxy{9 -1,2,5-thiadiazole compounds
DE2609486A1 (de) * 1975-08-07 1977-05-12 Hoffmann La Roche Imidazo eckige klammer auf 1,5-a eckige klammer zu eckige klammer auf 1,4 eckige klammer zu diazepin-verbindungen und verfahren zu ihrer herstellung
US4127674A (en) * 1977-03-21 1978-11-28 Allergan Pharmaceuticals, Inc. Method of treatment for glaucoma
US4387103A (en) * 1980-11-28 1983-06-07 American Hospital Supply Corporation Method for treatment or prophylaxis of cardiac disorders
ZA827646B (en) * 1981-11-12 1983-08-31 American Hospital Supply Corp Esters of aryloxypropanolamine derivatives

Also Published As

Publication number Publication date
IT1172381B (it) 1987-06-18
AU567908B2 (en) 1987-12-10
WO1984002525A1 (fr) 1984-07-05
EP0131006A4 (fr) 1985-06-06
NO164095C (no) 1990-09-05
IE832730L (en) 1984-06-22
AU2334184A (en) 1984-07-17
EP0131006B1 (fr) 1992-06-10
NZ206385A (en) 1986-08-08
JPS60500288A (ja) 1985-03-07
ES528225A0 (es) 1985-04-16
DE3382578T2 (de) 1993-03-25
IT8349538A0 (it) 1983-12-19
ES8504159A1 (es) 1985-04-16
CA1230879A (fr) 1987-12-29
EP0131006A1 (fr) 1985-01-16
NO843352L (no) 1984-08-22
IE59617B1 (en) 1994-03-09
NO164095B (no) 1990-05-21
US4508725A (en) 1985-04-02
DE3382578D1 (de) 1992-07-16
MX156097A (es) 1988-07-07

Similar Documents

Publication Publication Date Title
AU522975B2 (en) Carbazolyl-(4)-oxypropanolamine derivatives
GR81098B (en) Derivatives of 2,2 - iminodisethanol
NZ191462A (en) Derivatives of 2 ,16 -bis-piperidino-3 -hydroxy-5 -androstane-3 -esters
IL59829A (en) Derivatives of 9,10-anthracene-bis-carboxaldehyde-bis-hydrazone
PH21897A (en) Process for the manufacture of 1 sulfo-2-oxoazetidine derivatives
AU517598B2 (en) Derivatives of 1-aza-(2,2,2)-bicyclo-octane
GB2045757B (en) 1,2,3-thiadiazole-5-carboxylic acid derivatives
ZA838829B (en) Esters of 3-(3-substituted-amino-2-hydroxypropoxy)-4-substituted-1,2,5-thiadiazole derivatives
GB2018775B (en) Process for the preparation of asymmetical n-phenyl n'-substituted- -phenylene diamenes
AU1666583A (en) 1,2,5-thiadiazole derivatives
IL59333A0 (en) 2,6-dibromo- or -dichloro-isonicontinoyl derivatives of aminoacids
GB8418085D0 (en) 1 3 4-thiadiazole derivatives
NZ197563A (en) 3-(1,2,4-triazinylthiomethyl)-3-cephem-1-sulphoxide derivatives
GB2036737B (en) Derivatives of 1,5-dimethylbicyclo(3,2,1)octaine
AU1521083A (en) Ethyl 3-(n-n-butyl-n-acetyl)-aminopropionate
AU557580B2 (en) 15-cycloaliphatic derivatives of 13,14-didehydro- carboprostacyclins
JPS5626875A (en) 44*naphthaleniloxy*piperidine derivatives
GB2056439B (en) Hexahydroazepine derivatives
AU522421B2 (en) "hydroisoquinolinium derivatives"
AU2028283A (en) Alkanolaminoxy derivatives of 3,4-dihydro-2h-1,4- benzothiazine-3-one
GB8311220D0 (en) 1 2 4-triazol-1-yl-propionitrile derivatives
JPS55127347A (en) 1*1**biphenyll22yllalkylamine derivative
AU1974283A (en) 2,3-dihydro-2,2-dimethyl-benzofuran derivatives
GB2122602B (en) Novel 2 3-dihydro-indene derivatives
GB8319575D0 (en) 6 beta-halopenicillanic acid derivatives