ZA722627B - 4h-5-triazolo(4,3-a)(1,4)benzodiazepines - Google Patents

4h-5-triazolo(4,3-a)(1,4)benzodiazepines

Info

Publication number
ZA722627B
ZA722627B ZA722627A ZA722627A ZA722627B ZA 722627 B ZA722627 B ZA 722627B ZA 722627 A ZA722627 A ZA 722627A ZA 722627 A ZA722627 A ZA 722627A ZA 722627 B ZA722627 B ZA 722627B
Authority
ZA
South Africa
Prior art keywords
benzodiazepines
triazolo
Prior art date
Application number
ZA722627A
Other languages
English (en)
Inventor
J Hester
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of ZA722627B publication Critical patent/ZA722627B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ZA722627A 1971-05-11 1972-04-18 4h-5-triazolo(4,3-a)(1,4)benzodiazepines ZA722627B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US14241971A 1971-05-11 1971-05-11

Publications (1)

Publication Number Publication Date
ZA722627B true ZA722627B (en) 1973-02-28

Family

ID=22499772

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA722627A ZA722627B (en) 1971-05-11 1972-04-18 4h-5-triazolo(4,3-a)(1,4)benzodiazepines

Country Status (9)

Country Link
US (1) US3734922A (cs)
JP (1) JPS554110B1 (cs)
BE (1) BE783272A (cs)
CH (1) CH582179A5 (cs)
DE (1) DE2220623C2 (cs)
FR (1) FR2137714B1 (cs)
GB (1) GB1324318A (cs)
NL (1) NL7206301A (cs)
ZA (1) ZA722627B (cs)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904641A (en) * 1971-06-18 1975-09-09 Yoshitomi Pharmaceutical Triazolothienodiazepine compounds
US3886174A (en) * 1971-11-22 1975-05-27 Upjohn Co 1-Substituted-6-phenyl-4H-s-triazolo{8 4,3-a{9 {8 1,4{9 benzodiazepines
US3879406A (en) * 1972-07-13 1975-04-22 Hoffmann La Roche Preparation of triazolobenzodiazepines
US4155913A (en) * 1973-02-08 1979-05-22 Hoffmann-La Roche Inc. Thienotriazolodiazepine derivatives
FR2220257A1 (en) * 1973-03-09 1974-10-04 Lipha 5,6-Dihydro-(4H)-s-triazolo-(4,3-a) (1,5)benzodiazepines - as antiinflam-matory and analgesic agents without tranquillising effects
IE41197B1 (en) * 1973-05-29 1979-11-07 Squibb & Sons Inc 4h-s-triazolo (4,3-a)(1,5)benzodiazepin-5-ones
US3995043A (en) * 1974-05-13 1976-11-30 The Upjohn Company Composition and process
US4455307A (en) * 1982-01-04 1984-06-19 The Upjohn Company Antihypertensive use of triazolobenzodiazepines
JPS591395U (ja) * 1982-06-25 1984-01-06 株式会社東芝 縦形アイロン収納ケ−ス
FR2591596B1 (fr) * 1985-12-13 1988-09-09 Roussel Uclaf Nouvelles 4h-triazolo(4,3-a)(1,4)benzodiazepines, leur procede de preparation, leur application comme medicaments et les compositions les renfermant
ES2986407T3 (es) 2020-03-31 2024-11-11 Hoffmann La Roche Derivados de benzodiacepinas como PAM de GAMMA 1 GABA A
EP4408848A1 (en) 2021-09-29 2024-08-07 F. Hoffmann-La Roche AG New benzodiazepine derivatives as gaba a gamma1 pam
IL311377A (en) 2021-10-06 2024-05-01 Hoffmann La Roche Benzodiazepine derivatives as positive allosteric modulators of the GABA A GAMMA 1 receptor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
DE1955349C2 (de) * 1969-11-04 1982-01-28 Takeda Chemical Industries, Ltd., Osaka s-Triazolo [4,3-a] [1,4] benzodiazepine

Also Published As

Publication number Publication date
DE2220623A1 (de) 1972-11-16
FR2137714A1 (cs) 1972-12-29
NL7206301A (cs) 1972-11-14
BE783272A (fr) 1972-11-10
US3734922A (en) 1973-05-22
CH582179A5 (cs) 1976-11-30
GB1324318A (en) 1973-07-25
FR2137714B1 (cs) 1975-12-26
JPS554110B1 (cs) 1980-01-29
DE2220623C2 (de) 1985-04-25

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