ZA200805028B - Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor Xla inhibitors - Google Patents

Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor Xla inhibitors

Info

Publication number
ZA200805028B
ZA200805028B ZA200805028A ZA200805028A ZA200805028B ZA 200805028 B ZA200805028 B ZA 200805028B ZA 200805028 A ZA200805028 A ZA 200805028A ZA 200805028 A ZA200805028 A ZA 200805028A ZA 200805028 B ZA200805028 B ZA 200805028B
Authority
ZA
South Africa
Prior art keywords
arylpropynamide
arylmethylurea
arylpropionamide
arylacrylamide
analogs
Prior art date
Application number
ZA200805028A
Other languages
English (en)
Inventor
Donald J P Pinto
Joanne M Smallheer
James R Corte
Zilun Hu
Cullen L Cavallaro
Paul J Gilligan
Mimi L Quan
Il Leon M Smith
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ZA200805028B publication Critical patent/ZA200805028B/xx

Links

ZA200805028A 2005-12-14 2008-06-09 Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor Xla inhibitors ZA200805028B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US75013005P 2005-12-14 2005-12-14

Publications (1)

Publication Number Publication Date
ZA200805028B true ZA200805028B (en) 2009-12-30

Family

ID=40214768

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200805028A ZA200805028B (en) 2005-12-14 2008-06-09 Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor Xla inhibitors

Country Status (3)

Country Link
CN (1) CN101341129B (zh)
ES (1) ES2365815T3 (zh)
ZA (1) ZA200805028B (zh)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110097666A1 (en) * 2009-10-27 2011-04-28 Celin Savariar-Hauck Lithographic printing plate precursors
EA020528B1 (ru) 2010-02-11 2014-11-28 Бристол-Майерс Сквибб Компани Макроциклы в качестве ингибиторов фактора xia
GB2494851A (en) * 2011-07-07 2013-03-27 Kalvista Pharmaceuticals Ltd Plasma kallikrein inhibitors
ES2655669T3 (es) * 2011-12-21 2018-02-21 Ono Pharmaceutical Co., Ltd. Derivados de piridinona y pirimidinona como inhibidores del factor XIa
EP3024822B1 (de) * 2013-07-23 2017-05-03 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate und ihre verwendung als faktor xia und plasmakallikrein inhibitoren
CN112028877B (zh) * 2019-06-04 2021-11-26 江西济民可信集团有限公司 烷氧吡啶酮化合物及其制备方法和用途
JP7450024B2 (ja) * 2019-09-27 2024-03-14 シェンヅェン サルブリス ファーマシューティカルズ カンパニー リミテッド ＦＸＩａ阻害剤及びその調製方法と医薬用途
CN117480164B (zh) * 2020-12-11 2024-07-05 上海领泰生物医药科技有限公司 凝血因子XIa抑制剂及其制备方法和应用
WO2022194225A1 (zh) * 2021-03-18 2022-09-22 深圳信立泰药业股份有限公司 FXIa抑制剂化合物杂质及其制备方法和用途FXIa抑制剂化合物杂质及其制备方法和用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2263111C2 (ru) * 1998-06-12 2005-10-27 Сосьете Де Консей Де Решерш Э Д`Аппликасьон Сьентифик Сас Имидазольные производные
WO1999065942A1 (en) * 1998-06-16 1999-12-23 Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. Cyclic somatostatin analogs
CN1322001C (zh) * 2002-01-31 2007-06-20 莫弗凯姆联合化学股份公司 抑制因子Xa活性的新化合物
US7371743B2 (en) * 2004-02-28 2008-05-13 Boehringer Ingelheim International Gmbh Carboxylic acid amides, the preparation thereof and their use as medicaments
US7417063B2 (en) * 2004-04-13 2008-08-26 Bristol-Myers Squibb Company Bicyclic heterocycles useful as serine protease inhibitors

Also Published As

Publication number Publication date
CN101341129B (zh) 2011-12-14
CN101341129A (zh) 2009-01-07
ES2365815T3 (es) 2011-10-11

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