ZA200804104B - Pyrido-,pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors - Google Patents

Pyrido-,pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors

Info

Publication number
ZA200804104B
ZA200804104B ZA200804104A ZA200804104A ZA200804104B ZA 200804104 B ZA200804104 B ZA 200804104B ZA 200804104 A ZA200804104 A ZA 200804104A ZA 200804104 A ZA200804104 A ZA 200804104A ZA 200804104 B ZA200804104 B ZA 200804104B
Authority
ZA
South Africa
Prior art keywords
pyrazo
pyrimido
pyrido
pyrimidine derivatives
mtor inhibitors
Prior art date
Application number
ZA200804104A
Inventor
Marc Geoffrey Hummersone
Keith Allan Menear
Malagu Karine
Xiao-Ling Fan Cockroft
Gomez Sylvie
Smith Graeme Cameon Murray
Heather Mary Ellen Duggan
Gesine Johanna Hermann
Original Assignee
Kudos Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kudos Pharm Ltd filed Critical Kudos Pharm Ltd
Publication of ZA200804104B publication Critical patent/ZA200804104B/en

Links

ZA200804104A 2005-11-22 2008-05-13 Pyrido-,pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors ZA200804104B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73890205P 2005-11-22 2005-11-22

Publications (1)

Publication Number Publication Date
ZA200804104B true ZA200804104B (en) 2009-11-25

Family

ID=40332775

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200804104A ZA200804104B (en) 2005-11-22 2008-05-13 Pyrido-,pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors

Country Status (3)

Country Link
CN (1) CN101360746B (en)
UA (1) UA96745C2 (en)
ZA (1) ZA200804104B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101914483B (en) * 2010-09-02 2013-07-31 福建新大陆生物技术股份有限公司 Liquid-based thin-layer cell preservation solution and use thereof
CN102887895B (en) * 2011-07-22 2016-08-24 山东轩竹医药科技有限公司 Pyridopyrimidine class mTOR inhibitors
CN103588792B (en) * 2013-03-04 2016-03-23 中国科学院上海药物研究所 Pyridopyrimidine or pyrimido-pyrimidine compounds, its preparation method, medical composition and its use
CN105669731B (en) * 2016-01-10 2017-06-30 沧州普瑞东方科技有限公司 A kind of synthetic method of 4 (4 alkyl epoxide) phenyl boric acids
JP7340519B2 (en) * 2017-11-06 2023-09-07 メッドシャイン ディスカバリー インコーポレイテッド Pyridopyrimidine compounds as mTORC1/2 dual inhibitors
CN116478136A (en) * 2022-01-17 2023-07-25 苏州浦合医药科技有限公司 2-piperidinyl or 2-pyrazolyl substituted pyrimidine compounds as EGFR inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100345830C (en) * 2000-04-27 2007-10-31 安斯泰来制药有限公司 Condensed heteroaryl derivatives
DE60212487T2 (en) * 2001-04-13 2006-12-21 Pfizer Products Inc., Groton Bicyclic substituted 4-aminopyridopyrimidine derivatives
AU2003300898A1 (en) * 2002-12-13 2004-07-09 Neurogen Corporation Carboxylic acid, phosphate or phosphonate substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators

Also Published As

Publication number Publication date
CN101360746B (en) 2013-12-11
CN101360746A (en) 2009-02-04
UA96745C2 (en) 2011-12-12

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