UA96745C2 - PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS - Google Patents

PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS

Info

Publication number
UA96745C2
UA96745C2 UAA200808079A UAA200808079A UA96745C2 UA 96745 C2 UA96745 C2 UA 96745C2 UA A200808079 A UAA200808079 A UA A200808079A UA A200808079 A UAA200808079 A UA A200808079A UA 96745 C2 UA96745 C2 UA 96745C2
Authority
UA
Ukraine
Prior art keywords
pyrazo
pyrimido
pyrido
pyrimidine derivatives
mtor inhibitors
Prior art date
Application number
UAA200808079A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Марк Джеффри Хаммерсон
Сильви Гомез
Кейт Аллан Минер
Грейм Камерон Марри Смит
Карине Малагу
Хедер Мери Эллен Дагган
Сяо-Лин Фань Кокрофт
Гезине Йоханна Германн
Original Assignee
Кудос Фармасьютикалз Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Кудос Фармасьютикалз Лимитед filed Critical Кудос Фармасьютикалз Лимитед
Publication of UA96745C2 publication Critical patent/UA96745C2/en

Links

Abstract

, (I)There is provided compounds of formula (I), which are suitable for the treatment of cancer.
UAA200808079A 2005-11-22 2006-11-20 PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS UA96745C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73890205P 2005-11-22 2005-11-22

Publications (1)

Publication Number Publication Date
UA96745C2 true UA96745C2 (en) 2011-12-12

Family

ID=40332775

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200808079A UA96745C2 (en) 2005-11-22 2006-11-20 PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS

Country Status (3)

Country Link
CN (1) CN101360746B (en)
UA (1) UA96745C2 (en)
ZA (1) ZA200804104B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101914483B (en) * 2010-09-02 2013-07-31 福建新大陆生物技术股份有限公司 Liquid-based thin-layer cell preservation solution and use thereof
CN102887895B (en) * 2011-07-22 2016-08-24 山东轩竹医药科技有限公司 Pyridopyrimidine class mTOR inhibitors
CN103588792B (en) * 2013-03-04 2016-03-23 中国科学院上海药物研究所 Pyridopyrimidine or pyrimido-pyrimidine compounds, its preparation method, medical composition and its use
CN105669731B (en) * 2016-01-10 2017-06-30 沧州普瑞东方科技有限公司 A kind of synthetic method of 4 (4 alkyl epoxide) phenyl boric acids
BR112020008991A2 (en) 2017-11-06 2020-11-17 Medshine Discovery Inc. pyridopyrimidine compounds that act as dual inhibitors of mtorc 1/2
WO2023134266A1 (en) * 2022-01-17 2023-07-20 苏州浦合医药科技有限公司 2-piperidyl or 2-pyrazolyl substituted pyrimidine compound serving as egfr inhibitor

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2407593C (en) * 2000-04-27 2011-01-11 Yamanouchi Pharmaceutical Co. Ltd. Fused heteroaryl derivatives
DE60212487T2 (en) * 2001-04-13 2006-12-21 Pfizer Products Inc., Groton Bicyclic substituted 4-aminopyridopyrimidine derivatives
TW200418480A (en) * 2002-12-13 2004-10-01 Neurogen Corp 2-substituted quinazolin-4-ylamine analogues

Also Published As

Publication number Publication date
CN101360746A (en) 2009-02-04
CN101360746B (en) 2013-12-11
ZA200804104B (en) 2009-11-25

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