ZA200610264B - Glycopyrrolate for treating childhood asthma - Google Patents
Glycopyrrolate for treating childhood asthma Download PDFInfo
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- ZA200610264B ZA200610264B ZA200610264A ZA200610264A ZA200610264B ZA 200610264 B ZA200610264 B ZA 200610264B ZA 200610264 A ZA200610264 A ZA 200610264A ZA 200610264 A ZA200610264 A ZA 200610264A ZA 200610264 B ZA200610264 B ZA 200610264B
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- South Africa
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- glycopyrrolate
- use according
- microparticles
- medicament
- particles
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- ZQPPMHVWECSIRJ-KTKRTIGZSA-N oleic acid Chemical compound CCCCCCCC\C=C/CCCCCCCC(O)=O ZQPPMHVWECSIRJ-KTKRTIGZSA-N 0.000 description 1
- 239000013588 oral product Substances 0.000 description 1
- 229940023486 oral product Drugs 0.000 description 1
- 229950006841 oxitefonium bromide Drugs 0.000 description 1
- 229960005434 oxybutynin Drugs 0.000 description 1
- 238000002640 oxygen therapy Methods 0.000 description 1
- 229960002369 oxyphencyclimine Drugs 0.000 description 1
- UKLQXHUGTKWPSR-UHFFFAOYSA-M oxyphenonium bromide Chemical compound [Br-].C=1C=CC=CC=1C(O)(C(=O)OCC[N+](C)(CC)CC)C1CCCCC1 UKLQXHUGTKWPSR-UHFFFAOYSA-M 0.000 description 1
- 229960001125 oxyphenonium bromide Drugs 0.000 description 1
- SXGOKQARVJHRML-UHFFFAOYSA-M oxypyrronium bromide Chemical compound [Br-].C[N+]1(C)CCCC1COC(=O)C(O)(C=1C=CC=CC=1)C1CCCCC1 SXGOKQARVJHRML-UHFFFAOYSA-M 0.000 description 1
- 229950009905 oxypyrronium bromide Drugs 0.000 description 1
- 229960003293 penthienate Drugs 0.000 description 1
- NEMLPWNINZELKP-UHFFFAOYSA-N penthienate Chemical compound C=1C=CSC=1C(O)(C(=O)OCC[N+](C)(CC)CC)C1CCCC1 NEMLPWNINZELKP-UHFFFAOYSA-N 0.000 description 1
- 230000002093 peripheral effect Effects 0.000 description 1
- 239000002587 phosphodiesterase IV inhibitor Substances 0.000 description 1
- 229960001696 pipenzolate bromide Drugs 0.000 description 1
- 229960003033 piperidolate Drugs 0.000 description 1
- 230000036470 plasma concentration Effects 0.000 description 1
- 230000035935 pregnancy Effects 0.000 description 1
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 description 1
- 230000002294 pubertal effect Effects 0.000 description 1
- 230000000241 respiratory effect Effects 0.000 description 1
- 230000002441 reversible effect Effects 0.000 description 1
- 238000012552 review Methods 0.000 description 1
- 229960002052 salbutamol Drugs 0.000 description 1
- 229960004017 salmeterol Drugs 0.000 description 1
- 230000028327 secretion Effects 0.000 description 1
- 230000035945 sensitivity Effects 0.000 description 1
- 230000000391 smoking effect Effects 0.000 description 1
- 239000007787 solid Substances 0.000 description 1
- 239000002195 soluble material Substances 0.000 description 1
- 239000002904 solvent Substances 0.000 description 1
- 125000006850 spacer group Chemical group 0.000 description 1
- 229940046810 spiriva Drugs 0.000 description 1
- 238000013125 spirometry Methods 0.000 description 1
- 229910001220 stainless steel Inorganic materials 0.000 description 1
- 239000010935 stainless steel Substances 0.000 description 1
- 239000008117 stearic acid Substances 0.000 description 1
- 239000000725 suspension Substances 0.000 description 1
- 230000002459 sustained effect Effects 0.000 description 1
- 230000006794 tachycardia Effects 0.000 description 1
- 238000012360 testing method Methods 0.000 description 1
- LERNTVKEWCAPOY-DZZGSBJMSA-N tiotropium Chemical compound O([C@H]1C[C@@H]2[N+]([C@H](C1)[C@@H]1[C@H]2O1)(C)C)C(=O)C(O)(C=1SC=CC=1)C1=CC=CS1 LERNTVKEWCAPOY-DZZGSBJMSA-N 0.000 description 1
- 229940110309 tiotropium Drugs 0.000 description 1
- 230000001052 transient effect Effects 0.000 description 1
- 238000011269 treatment regimen Methods 0.000 description 1
- MDYZKJNTKZIUSK-UHFFFAOYSA-N tyloxapol Chemical compound O=C.C1CO1.CC(C)(C)CC(C)(C)C1=CC=C(O)C=C1 MDYZKJNTKZIUSK-UHFFFAOYSA-N 0.000 description 1
- 229960004224 tyloxapol Drugs 0.000 description 1
- 229920001664 tyloxapol Polymers 0.000 description 1
- 229920001285 xanthan gum Polymers 0.000 description 1
- XOOUIPVCVHRTMJ-UHFFFAOYSA-L zinc stearate Chemical class [Zn+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O XOOUIPVCVHRTMJ-UHFFFAOYSA-L 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/465—Nicotine; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0410399.0A GB0410399D0 (en) | 2004-05-10 | 2004-05-10 | The treatment of respiratory disease |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200610264B true ZA200610264B (en) | 2008-06-25 |
Family
ID=32526760
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200610264A ZA200610264B (en) | 2004-05-10 | 2005-05-10 | Glycopyrrolate for treating childhood asthma |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20070243260A1 (fr) |
| EP (1) | EP1750807A2 (fr) |
| JP (1) | JP2007536362A (fr) |
| KR (1) | KR20070042917A (fr) |
| CN (1) | CN1972730A (fr) |
| AU (1) | AU2005240406A1 (fr) |
| BR (1) | BRPI0510946A (fr) |
| CA (1) | CA2565170A1 (fr) |
| GB (1) | GB0410399D0 (fr) |
| IL (1) | IL178816A0 (fr) |
| MX (1) | MXPA06013040A (fr) |
| NO (1) | NO20065536L (fr) |
| NZ (1) | NZ550909A (fr) |
| WO (1) | WO2005107873A2 (fr) |
| ZA (1) | ZA200610264B (fr) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0008660D0 (en) * | 2000-04-07 | 2000-05-31 | Arakis Ltd | The treatment of respiratory diseases |
| GB0410398D0 (en) * | 2004-05-10 | 2004-06-16 | Arakis Ltd | The treatment of respiratory disease |
| GB0425758D0 (en) | 2004-11-23 | 2004-12-22 | Vectura Ltd | Preparation of pharmaceutical compositions |
| GB0613161D0 (en) | 2006-06-30 | 2006-08-09 | Novartis Ag | Organic Compounds |
| CN102573912B (zh) * | 2009-09-30 | 2014-01-01 | 三仪股份有限公司 | 难溶性物质的水溶性改善方法 |
| GB0918150D0 (en) * | 2009-10-16 | 2009-12-02 | Jagotec Ag | Improved formulations |
| SG181870A1 (en) | 2009-12-23 | 2012-07-30 | Chiesi Farma Spa | Aerosol formulation for copd |
| WO2011076840A2 (fr) | 2009-12-23 | 2011-06-30 | Chiesi Farmaceutici S.P.A. | Préparation aérosol pour bronchopneumopathie chronique obstructive |
| EP2515853B1 (fr) | 2009-12-23 | 2014-03-19 | Chiesi Farmaceutici S.p.A. | Polythérapie pour la COPD |
| NZ600790A (en) | 2009-12-23 | 2014-09-26 | Chiesi Farma Spa | Combination therapy for copd |
| JO3510B1 (ar) * | 2011-03-04 | 2020-07-05 | Heptares Therapeutics Ltd | استخدام جلايكوبيرولات لعلاج عدم انتظام دقات القلب |
| JP5909796B2 (ja) | 2012-03-02 | 2016-04-27 | 株式会社サンギ | 難溶性物質の水溶解性改善方法 |
| US20150038719A1 (en) * | 2012-03-14 | 2015-02-05 | Ltt Bio-Pharma Co., Ltd. | Agent for Ameliorating Chronic Obstructive Pulmonary Disease |
| WO2014062143A2 (fr) * | 2012-10-19 | 2014-04-24 | Mahmut Bilgic | Combinaisons d'agent anticholinergique |
| WO2014077787A1 (fr) * | 2012-11-16 | 2014-05-22 | Mahmut Bilgic | Combinaisons comprenant un bêta2-agoniste et glycopyrrolate |
| PL3089735T3 (pl) | 2013-12-30 | 2018-12-31 | Chiesi Farmaceutici S.P.A. | Trwała ciśnieniowa kompozycja roztworu aerozolowego kombinacji bromku glikopironium i formoterolu |
| MX2017003080A (es) * | 2014-09-09 | 2017-11-15 | Vectura Ltd | Formulacion que comprende glicopirrolato, metodo y aparato. |
| HUE056402T2 (hu) * | 2015-11-16 | 2022-02-28 | Chiesi Farm Spa | Eljárás antikolinerg szert, kortikoszteroidot és béta-adrenerg szert tartalmazó száraz porkészítmény elõállítására |
| US10098837B2 (en) | 2016-07-28 | 2018-10-16 | Chiesi Farmaceutici S.P.A. | Combination therapy for COPD |
| PE20221439A1 (es) | 2019-12-02 | 2022-09-21 | Chiesi Farm Spa | Lata de acero inoxidable para inhaladores dosificadores presurizados |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2347856C (fr) * | 1998-11-13 | 2009-02-17 | Jago Research Ag | Poudre seche pour inhalation |
| GB0008660D0 (en) * | 2000-04-07 | 2000-05-31 | Arakis Ltd | The treatment of respiratory diseases |
| ES2296831T3 (es) * | 2000-11-30 | 2008-05-01 | Vectura Limited | Metodo para preparar microparticulas para usar en composiciones farmaceuticas para inhalacion. |
-
2004
- 2004-05-10 GB GBGB0410399.0A patent/GB0410399D0/en not_active Ceased
-
2005
- 2005-05-10 MX MXPA06013040A patent/MXPA06013040A/es not_active Application Discontinuation
- 2005-05-10 EP EP05742199A patent/EP1750807A2/fr not_active Ceased
- 2005-05-10 NZ NZ550909A patent/NZ550909A/en unknown
- 2005-05-10 AU AU2005240406A patent/AU2005240406A1/en not_active Abandoned
- 2005-05-10 WO PCT/GB2005/001791 patent/WO2005107873A2/fr active Application Filing
- 2005-05-10 JP JP2007512333A patent/JP2007536362A/ja active Pending
- 2005-05-10 ZA ZA200610264A patent/ZA200610264B/en unknown
- 2005-05-10 US US11/579,096 patent/US20070243260A1/en not_active Abandoned
- 2005-05-10 KR KR1020067023268A patent/KR20070042917A/ko not_active Application Discontinuation
- 2005-05-10 CN CNA2005800149123A patent/CN1972730A/zh active Pending
- 2005-05-10 CA CA002565170A patent/CA2565170A1/fr not_active Abandoned
- 2005-05-10 BR BRPI0510946-9A patent/BRPI0510946A/pt not_active IP Right Cessation
-
2006
- 2006-10-23 IL IL178816A patent/IL178816A0/en unknown
- 2006-11-30 NO NO20065536A patent/NO20065536L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| IL178816A0 (en) | 2007-05-15 |
| GB0410399D0 (en) | 2004-06-16 |
| US20070243260A1 (en) | 2007-10-18 |
| MXPA06013040A (es) | 2007-02-12 |
| KR20070042917A (ko) | 2007-04-24 |
| JP2007536362A (ja) | 2007-12-13 |
| AU2005240406A1 (en) | 2005-11-17 |
| BRPI0510946A (pt) | 2007-11-20 |
| CA2565170A1 (fr) | 2005-11-17 |
| NO20065536L (no) | 2006-12-08 |
| WO2005107873A3 (fr) | 2006-03-16 |
| WO2005107873A2 (fr) | 2005-11-17 |
| CN1972730A (zh) | 2007-05-30 |
| NZ550909A (en) | 2011-02-25 |
| EP1750807A2 (fr) | 2007-02-14 |
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