ZA200507258B - 4, 6-, or 7-hydroxyindoles having n-oxide groups and the use thereof as therapeutic agents - Google Patents
4, 6-, or 7-hydroxyindoles having n-oxide groups and the use thereof as therapeutic agents Download PDFInfo
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- ZA200507258B ZA200507258B ZA200507258A ZA200507258A ZA200507258B ZA 200507258 B ZA200507258 B ZA 200507258B ZA 200507258 A ZA200507258 A ZA 200507258A ZA 200507258 A ZA200507258 A ZA 200507258A ZA 200507258 B ZA200507258 B ZA 200507258B
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Classifications
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Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Immunology (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Diabetes (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Virology (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Dermatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Reproductive Health (AREA)
- AIDS & HIV (AREA)
- Molecular Biology (AREA)
- Vascular Medicine (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10318611A DE10318611A1 (de) | 2003-04-24 | 2003-04-24 | 4-, 6- oder 7-Hydroxyindole mit N-Oxidgruppen und deren Verwendung als Therapeutika |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200507258B true ZA200507258B (en) | 2006-06-28 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200507258A ZA200507258B (en) | 2003-04-24 | 2005-09-09 | 4, 6-, or 7-hydroxyindoles having n-oxide groups and the use thereof as therapeutic agents |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US7067536B2 (fr) |
| EP (1) | EP1615912A1 (fr) |
| JP (1) | JP2006524208A (fr) |
| KR (1) | KR20060021831A (fr) |
| CN (1) | CN1777600A (fr) |
| AR (1) | AR044081A1 (fr) |
| AU (1) | AU2004232482A1 (fr) |
| BR (1) | BRPI0409793A (fr) |
| CA (1) | CA2523048A1 (fr) |
| DE (1) | DE10318611A1 (fr) |
| MX (1) | MXPA05011437A (fr) |
| NO (1) | NO20055517L (fr) |
| RU (1) | RU2005136431A (fr) |
| TW (1) | TW200503693A (fr) |
| WO (1) | WO2004094405A1 (fr) |
| ZA (1) | ZA200507258B (fr) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200738677A (en) * | 2005-06-27 | 2007-10-16 | Elbion Ag | Nitro-substituted hydroxyindoles, their use as inhibitors of phosphodiesterase 4, and processes for preparing them |
| EP1956906A4 (fr) | 2005-11-09 | 2009-12-30 | Combinatorx Inc | Procedes, compositions et kits pour le traitement de pathologies |
| AU2007281747B2 (en) * | 2006-08-07 | 2013-11-07 | Ironwood Pharmaceuticals, Inc. | Indole compounds |
| NZ579645A (en) * | 2007-03-14 | 2012-01-12 | Ranbaxy Lab Ltd | Pyrazolo (3, 4-b) pyridine derivatives as phosphodiesterase inhibitors |
| AR084433A1 (es) | 2010-12-22 | 2013-05-15 | Ironwood Pharmaceuticals Inc | Inhibidores de la faah y composiciones farmaceuticas que los contienen |
| HRP20220331T1 (hr) | 2018-03-08 | 2022-05-13 | Incyte Corporation | Spojevi aminopirazin diola kao inhibitori pi3k-y |
| US11046658B2 (en) | 2018-07-02 | 2021-06-29 | Incyte Corporation | Aminopyrazine derivatives as PI3K-γ inhibitors |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19636150A1 (de) | 1996-09-06 | 1998-03-12 | Asta Medica Ag | N-substituierte Indol-3-glyoxylamide mit antiasthmatischer, antiallergischer und immunsuppressiver/immunmodulierender Wirkung |
| DE19814838C2 (de) | 1998-04-02 | 2001-01-18 | Asta Medica Ag | Indolyl-3-glyoxylsäure-Derivate mit Antitumorwirkung |
| ES2262072T3 (es) | 1998-04-28 | 2006-11-16 | Elbion Ag | Derivados de indol y su utilizacion como inhibidores de la fosfodiesterasa 4. |
| DE19962300A1 (de) * | 1999-12-23 | 2001-06-28 | Asta Medica Ag | Substituierte N-Benzyl-Indol-3-yl-glyoxylsäure-Derivate mit Antitumorwirkung |
| EP1432709B8 (fr) | 2001-09-13 | 2005-11-02 | Synta Pharmaceuticals Corporation | Indolizines de 1-glyoxylamide permettant de traiter le cancer |
| US20040116462A1 (en) | 2002-12-12 | 2004-06-17 | Mitsunori Ono | Indolizine compounds |
| DE10253426B4 (de) * | 2002-11-15 | 2005-09-22 | Elbion Ag | Neue Hydroxyindole, deren Verwendung als Inhibitoren der Phosphodiesterase 4 und Verfahren zu deren Herstellung |
| DE10318609A1 (de) * | 2003-04-24 | 2004-11-11 | Elbion Ag | 5-Hydroxyindole mit N-Oxidgruppen und deren Verwendung als Therapeutika |
-
2003
- 2003-04-24 DE DE10318611A patent/DE10318611A1/de not_active Withdrawn
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2004
- 2004-04-16 US US10/825,862 patent/US7067536B2/en not_active Expired - Fee Related
- 2004-04-21 TW TW093111114A patent/TW200503693A/zh unknown
- 2004-04-23 JP JP2006505245A patent/JP2006524208A/ja not_active Withdrawn
- 2004-04-23 EP EP04729109A patent/EP1615912A1/fr not_active Withdrawn
- 2004-04-23 AR ARP040101396A patent/AR044081A1/es not_active Application Discontinuation
- 2004-04-23 BR BRPI0409793-9A patent/BRPI0409793A/pt not_active Application Discontinuation
- 2004-04-23 CN CNA2004800110345A patent/CN1777600A/zh active Pending
- 2004-04-23 WO PCT/EP2004/004338 patent/WO2004094405A1/fr not_active Application Discontinuation
- 2004-04-23 RU RU2005136431/04A patent/RU2005136431A/ru not_active Application Discontinuation
- 2004-04-23 AU AU2004232482A patent/AU2004232482A1/en not_active Abandoned
- 2004-04-23 MX MXPA05011437A patent/MXPA05011437A/es unknown
- 2004-04-23 CA CA002523048A patent/CA2523048A1/fr not_active Abandoned
- 2004-04-23 KR KR1020057020097A patent/KR20060021831A/ko not_active Application Discontinuation
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2005
- 2005-09-09 ZA ZA200507258A patent/ZA200507258B/en unknown
- 2005-11-22 NO NO20055517A patent/NO20055517L/no not_active Application Discontinuation
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2006
- 2006-01-30 US US11/342,428 patent/US20060128758A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US7067536B2 (en) | 2006-06-27 |
| RU2005136431A (ru) | 2006-03-20 |
| CA2523048A1 (fr) | 2004-11-04 |
| NO20055517D0 (no) | 2005-11-22 |
| MXPA05011437A (es) | 2005-12-12 |
| AU2004232482A1 (en) | 2004-11-04 |
| CN1777600A (zh) | 2006-05-24 |
| NO20055517L (no) | 2006-01-18 |
| JP2006524208A (ja) | 2006-10-26 |
| AR044081A1 (es) | 2005-08-24 |
| WO2004094405A1 (fr) | 2004-11-04 |
| TW200503693A (en) | 2005-02-01 |
| BRPI0409793A (pt) | 2006-05-30 |
| DE10318611A1 (de) | 2004-11-11 |
| EP1615912A1 (fr) | 2006-01-18 |
| US20060128758A1 (en) | 2006-06-15 |
| KR20060021831A (ko) | 2006-03-08 |
| US20040242643A1 (en) | 2004-12-02 |
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