ZA200308004B - Utilization of galanthamine for the treatment of pathologies of the central nervous system owing to intoxications with psychotropic substances. - Google Patents
Utilization of galanthamine for the treatment of pathologies of the central nervous system owing to intoxications with psychotropic substances. Download PDFInfo
- Publication number
- ZA200308004B ZA200308004B ZA200308004A ZA200308004A ZA200308004B ZA 200308004 B ZA200308004 B ZA 200308004B ZA 200308004 A ZA200308004 A ZA 200308004A ZA 200308004 A ZA200308004 A ZA 200308004A ZA 200308004 B ZA200308004 B ZA 200308004B
- Authority
- ZA
- South Africa
- Prior art keywords
- galanthamine
- use according
- abuse
- medicament
- substances
- Prior art date
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- 229960003980 galantamine Drugs 0.000 title claims description 38
- ASUTZQLVASHGKV-UHFFFAOYSA-N galanthamine hydrochloride Natural products O1C(=C23)C(OC)=CC=C2CN(C)CCC23C1CC(O)C=C2 ASUTZQLVASHGKV-UHFFFAOYSA-N 0.000 title claims description 38
- HPOIPOPJGBKXIR-UHFFFAOYSA-N 3,6-dimethoxy-10-methyl-galantham-1-ene Natural products O1C(C(=CC=2)OC)=C3C=2CN(C)CCC23C1CC(OC)C=C2 HPOIPOPJGBKXIR-UHFFFAOYSA-N 0.000 title claims description 37
- LPCKPBWOSNVCEL-UHFFFAOYSA-N Chlidanthine Natural products O1C(C(=CC=2)O)=C3C=2CN(C)CCC23C1CC(OC)C=C2 LPCKPBWOSNVCEL-UHFFFAOYSA-N 0.000 title claims description 37
- BGLNUNCBNALFOZ-WMLDXEAASA-N galanthamine Natural products COc1ccc2CCCC[C@@]34C=CCC[C@@H]3Oc1c24 BGLNUNCBNALFOZ-WMLDXEAASA-N 0.000 title claims description 37
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
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- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10119862A DE10119862A1 (de) | 2001-04-24 | 2001-04-24 | Verwendung von Galanthamin zur Behandlung von Krankheitserscheinungen des zentralen Nervensystems aufgrund von Intoxikationen mit psychotropen Substanzen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200308004B true ZA200308004B (en) | 2004-02-11 |
Family
ID=7682409
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200308004A ZA200308004B (en) | 2001-04-24 | 2003-10-15 | Utilization of galanthamine for the treatment of pathologies of the central nervous system owing to intoxications with psychotropic substances. |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US8207159B2 (pl) |
| EP (1) | EP1383507B1 (pl) |
| JP (1) | JP2004531533A (pl) |
| KR (1) | KR20040005934A (pl) |
| CN (1) | CN100400043C (pl) |
| AR (1) | AR033468A1 (pl) |
| AT (1) | ATE378052T1 (pl) |
| AU (1) | AU2002308148B2 (pl) |
| BR (1) | BR0209126A (pl) |
| CA (1) | CA2444818C (pl) |
| CZ (1) | CZ20032789A3 (pl) |
| DE (2) | DE10119862A1 (pl) |
| DK (1) | DK1383507T3 (pl) |
| EA (1) | EA200301135A1 (pl) |
| ES (1) | ES2296990T3 (pl) |
| HK (1) | HK1062401A1 (pl) |
| HU (1) | HUP0401123A3 (pl) |
| IL (2) | IL158382A0 (pl) |
| MX (1) | MXPA03009765A (pl) |
| NO (1) | NO20034740L (pl) |
| NZ (1) | NZ529004A (pl) |
| PL (1) | PL207525B1 (pl) |
| PT (1) | PT1383507E (pl) |
| SK (1) | SK287235B6 (pl) |
| TW (1) | TWI329512B (pl) |
| WO (1) | WO2002085370A1 (pl) |
| ZA (1) | ZA200308004B (pl) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2004216360B2 (en) * | 2003-02-27 | 2009-09-17 | Eisai R & D Management Co., Ltd. | Pharmaceutical composition for treatment of drug dependence |
| DE10338544B4 (de) * | 2003-08-19 | 2017-08-31 | Janssen Pharmaceutica N.V. | Buccale Formulierungen des Galanthamins und deren Anwendungen |
| FR2930891B1 (fr) | 2008-05-06 | 2010-09-24 | Biocodex | Composes anti-amnesiants et compositions pharmaceutiques les comprenant |
| EP2586436A1 (en) | 2011-10-31 | 2013-05-01 | Commissariat à l'Énergie Atomique et aux Énergies Alternatives | Use of anti-connexin agents for enhancing the therapeutic effect of acetylcholinesterase inhibitor |
| US20180200259A1 (en) * | 2015-05-18 | 2018-07-19 | Synaptec Development Llc | GALANTAMINE CLEARANCE OF AMYLOID ß |
| US20230202978A1 (en) | 2022-03-04 | 2023-06-29 | Reset Pharmaceuticals, Inc. | Co-crystal or salt |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1193061B (de) | 1961-12-20 | 1965-05-20 | Vni Chimiko Pharmazewtitschesk | Verfahren zur Gewinnung von Galanthamin-hydrobromid aus Pflanzen der Familie der Amaryllidaceen |
| US3797494A (en) | 1969-04-01 | 1974-03-19 | Alza Corp | Bandage for the administration of drug by controlled metering through microporous materials |
| US3742951A (en) | 1971-08-09 | 1973-07-03 | Alza Corp | Bandage for controlled release of vasodilators |
| US3996934A (en) | 1971-08-09 | 1976-12-14 | Alza Corporation | Medical bandage |
| US4031894A (en) | 1975-12-08 | 1977-06-28 | Alza Corporation | Bandage for transdermally administering scopolamine to prevent nausea |
| DE3315272C2 (de) | 1983-04-27 | 1986-03-27 | Lohmann Gmbh & Co Kg, 5450 Neuwied | Pharmazeutisches Produkt und Verfahren zu seiner Herstellung |
| US4666829A (en) * | 1985-05-15 | 1987-05-19 | University Of California | Polypeptide marker for Alzheimer's disease and its use for diagnosis |
| US6150354A (en) * | 1987-01-15 | 2000-11-21 | Bonnie Davis | Compounds for the treatment of Alzheimer's disease |
| DE3843239C1 (pl) | 1988-12-22 | 1990-02-22 | Lohmann Therapie Syst Lts | |
| US5015645A (en) * | 1989-10-19 | 1991-05-14 | Ciba-Geigy Corporation | Tetracyclic pyrrole lactam derivatives |
| DE4010079A1 (de) * | 1990-03-29 | 1991-10-02 | Lohmann Therapie Syst Lts | Pharmazeutische formulierung zur behandlung des alkoholismus |
| US5519017A (en) * | 1990-03-29 | 1996-05-21 | Lts Lohmann Therapie-Systeme Gmbh + Co. Kg | Pharmaceutic formulation for the treatment of alcoholism |
| US5336675A (en) * | 1991-05-14 | 1994-08-09 | Ernir Snorrason | Method of treating mania in humans |
| DE4301782C1 (de) * | 1993-01-23 | 1994-08-25 | Lohmann Therapie Syst Lts | Verwendung von Galanthamin zur Behandlung der Nicotinabhängigkeit |
| DE19509663A1 (de) | 1995-03-17 | 1996-09-19 | Lohmann Therapie Syst Lts | Verfahren zur Isolierung von Galanthamin |
| US5965571A (en) * | 1996-08-22 | 1999-10-12 | New York University | Cholinesterase inhibitors for treatment of Parkinson's disease |
| US5932557A (en) * | 1997-08-12 | 1999-08-03 | Mustafa; S. Jamal | Adenosine A1 receptor antisense oligonucleotide treatment of alcohol and marijuana-induced psychomotor impairments |
| CN1240384C (zh) * | 1999-11-04 | 2006-02-08 | 美国爱科赛尔制药有限公司 | 石杉碱经皮给药制剂 |
| US20020151591A1 (en) * | 2000-10-17 | 2002-10-17 | Anabella Villalobos | Combination use of acetylcholinesterase inhibitors and GABAa inverse agonists for the treatment of cognitive disorders |
-
2001
- 2001-04-24 DE DE10119862A patent/DE10119862A1/de not_active Withdrawn
-
2002
- 2002-04-18 AT AT02764017T patent/ATE378052T1/de active
- 2002-04-18 SK SK1315-2003A patent/SK287235B6/sk not_active IP Right Cessation
- 2002-04-18 US US10/475,357 patent/US8207159B2/en not_active Expired - Fee Related
- 2002-04-18 WO PCT/EP2002/004277 patent/WO2002085370A1/de active IP Right Grant
- 2002-04-18 CN CNB028088905A patent/CN100400043C/zh not_active Expired - Lifetime
- 2002-04-18 MX MXPA03009765A patent/MXPA03009765A/es active IP Right Grant
- 2002-04-18 PT PT02764017T patent/PT1383507E/pt unknown
- 2002-04-18 JP JP2002582943A patent/JP2004531533A/ja active Pending
- 2002-04-18 ES ES02764017T patent/ES2296990T3/es not_active Expired - Lifetime
- 2002-04-18 EA EA200301135A patent/EA200301135A1/ru unknown
- 2002-04-18 IL IL15838202A patent/IL158382A0/xx unknown
- 2002-04-18 DE DE50211207T patent/DE50211207D1/de not_active Expired - Lifetime
- 2002-04-18 BR BR0209126-7A patent/BR0209126A/pt not_active Application Discontinuation
- 2002-04-18 NZ NZ529004A patent/NZ529004A/en unknown
- 2002-04-18 CA CA002444818A patent/CA2444818C/en not_active Expired - Lifetime
- 2002-04-18 DK DK02764017T patent/DK1383507T3/da active
- 2002-04-18 PL PL366840A patent/PL207525B1/pl not_active IP Right Cessation
- 2002-04-18 CZ CZ20032789A patent/CZ20032789A3/cs unknown
- 2002-04-18 EP EP02764017A patent/EP1383507B1/de not_active Expired - Lifetime
- 2002-04-18 HU HU0401123A patent/HUP0401123A3/hu unknown
- 2002-04-18 AU AU2002308148A patent/AU2002308148B2/en not_active Ceased
- 2002-04-18 KR KR10-2003-7013971A patent/KR20040005934A/ko active Search and Examination
- 2002-04-22 TW TW091108204A patent/TWI329512B/zh not_active IP Right Cessation
- 2002-04-24 AR ARP020101482A patent/AR033468A1/es unknown
-
2003
- 2003-10-13 IL IL158382A patent/IL158382A/en active IP Right Grant
- 2003-10-15 ZA ZA200308004A patent/ZA200308004B/en unknown
- 2003-10-23 NO NO20034740A patent/NO20034740L/no not_active Application Discontinuation
-
2004
- 2004-07-02 HK HK04104742A patent/HK1062401A1/xx not_active IP Right Cessation
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