WO2007138232A3 - Utilisation du granisetron pour le traitement de sous-types de la rosacée, et compositions pharmaceutiques le contenant - Google Patents

Utilisation du granisetron pour le traitement de sous-types de la rosacée, et compositions pharmaceutiques le contenant Download PDF

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Publication number
WO2007138232A3
WO2007138232A3 PCT/FR2007/051360 FR2007051360W WO2007138232A3 WO 2007138232 A3 WO2007138232 A3 WO 2007138232A3 FR 2007051360 W FR2007051360 W FR 2007051360W WO 2007138232 A3 WO2007138232 A3 WO 2007138232A3
Authority
WO
WIPO (PCT)
Prior art keywords
rosacea
granisetron
treatment
sub
types
Prior art date
Application number
PCT/FR2007/051360
Other languages
English (en)
Other versions
WO2007138232A2 (fr
Inventor
Jean-Dominique Pierret
Fabrizio Dolfi
Christian Loesche
Nadege Tremel
Original Assignee
Galderma Res & Dev
Jean-Dominique Pierret
Fabrizio Dolfi
Christian Loesche
Nadege Tremel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Galderma Res & Dev, Jean-Dominique Pierret, Fabrizio Dolfi, Christian Loesche, Nadege Tremel filed Critical Galderma Res & Dev
Publication of WO2007138232A2 publication Critical patent/WO2007138232A2/fr
Publication of WO2007138232A3 publication Critical patent/WO2007138232A3/fr

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4906Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
    • A61K8/4926Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having six membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Birds (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne l'utilisation du granisetron ou de ses sels en tant que principe actif dans une composition pharmaceutique, plus particulièrement dermatologique. De préférence, la composition est appliquée topiquement. Elle est destinée au traitement et/ou a la prévention de la rosacée papulopustuleuse, de la rosacée phymateuse et/ou de la rosacée oculaire.
PCT/FR2007/051360 2006-05-31 2007-05-31 Utilisation du granisetron pour le traitement de sous-types de la rosacée, et compositions pharmaceutiques le contenant WO2007138232A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0651983A FR2901702A1 (fr) 2006-05-31 2006-05-31 Utilisation de granisetron pour le traitement de sous-types de la rosacee, et compositions pharmaceutiques
FR0651983 2006-05-31

Publications (2)

Publication Number Publication Date
WO2007138232A2 WO2007138232A2 (fr) 2007-12-06
WO2007138232A3 true WO2007138232A3 (fr) 2008-03-27

Family

ID=37441246

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/FR2007/051360 WO2007138232A2 (fr) 2006-05-31 2007-05-31 Utilisation du granisetron pour le traitement de sous-types de la rosacée, et compositions pharmaceutiques le contenant

Country Status (2)

Country Link
FR (1) FR2901702A1 (fr)
WO (1) WO2007138232A2 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2960152A1 (fr) * 2010-01-27 2011-11-25 Galderma Res & Dev Utilisation de modulateur de recepteurs a l'histamine de type 2 pour le traitement de la rosacee et composition les contenant

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0834731A (ja) * 1994-07-26 1996-02-06 T T S Gijutsu Kenkyusho:Kk グラニセトロン含有経皮吸収型製剤
WO2004000358A1 (fr) * 2002-06-20 2003-12-31 Amnon Sintov Systeme d'administration transdermique de medicaments
US20040171561A1 (en) * 2002-09-03 2004-09-02 Popp Karl F. Topical formulations for treatment of rosacea
US20050042194A1 (en) * 2000-05-11 2005-02-24 A.P. Pharma, Inc. Semi-solid delivery vehicle and pharmaceutical compositions
WO2005058312A1 (fr) * 2003-12-10 2005-06-30 Galderma Research & Development, S.N.C. Utilisation d'ondansetron pour le traitement de l'inflammation et compositions pharmaceutiques a base d'ondansetron
US6916487B2 (en) * 1996-02-19 2005-07-12 Acrux Dds Pty Ltd Transdermal delivery of antiemetics

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0834731A (ja) * 1994-07-26 1996-02-06 T T S Gijutsu Kenkyusho:Kk グラニセトロン含有経皮吸収型製剤
US6916487B2 (en) * 1996-02-19 2005-07-12 Acrux Dds Pty Ltd Transdermal delivery of antiemetics
US20050042194A1 (en) * 2000-05-11 2005-02-24 A.P. Pharma, Inc. Semi-solid delivery vehicle and pharmaceutical compositions
WO2004000358A1 (fr) * 2002-06-20 2003-12-31 Amnon Sintov Systeme d'administration transdermique de medicaments
US20040171561A1 (en) * 2002-09-03 2004-09-02 Popp Karl F. Topical formulations for treatment of rosacea
WO2005058312A1 (fr) * 2003-12-10 2005-06-30 Galderma Research & Development, S.N.C. Utilisation d'ondansetron pour le traitement de l'inflammation et compositions pharmaceutiques a base d'ondansetron

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
JANSEN T: "Influence of the 5-HT3 receptor antagonist granisetron on erythema and flushing tendency in rosacea patients", KOSMETISCHE MEDIZIN 2005 GERMANY, vol. 26, no. 1, 2005, pages 22 - 24, XP009075700, ISSN: 1430-4031 *
WILKIN JONATHAN ET AL: "Standard grading system for rosacea: report of the National Rosacea Society Expert Committee on the classification and staging of rosacea.", JOURNAL OF THE AMERICAN ACADEMY OF DERMATOLOGY. JUN 2004, vol. 50, no. 6, June 2004 (2004-06-01), pages 907 - 912, XP002409907, ISSN: 0190-9622 *

Also Published As

Publication number Publication date
FR2901702A1 (fr) 2007-12-07
WO2007138232A2 (fr) 2007-12-06

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