WO2007047838A3 - Procede de preparation de l'olmesartan medoxomil - Google Patents
Procede de preparation de l'olmesartan medoxomil Download PDFInfo
- Publication number
- WO2007047838A3 WO2007047838A3 PCT/US2006/040883 US2006040883W WO2007047838A3 WO 2007047838 A3 WO2007047838 A3 WO 2007047838A3 US 2006040883 W US2006040883 W US 2006040883W WO 2007047838 A3 WO2007047838 A3 WO 2007047838A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- olmesartan medoxomil
- methylethyl
- carboxylate
- propyl
- hydroxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
L'invention porte sur un procédé de préparation de l'olmésartan médoxomil.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1517/CHE/2005 | 2005-10-20 | ||
IN1517CH2005 | 2005-10-20 | ||
US74567006P | 2006-04-26 | 2006-04-26 | |
US60/745,670 | 2006-04-26 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2007047838A2 WO2007047838A2 (fr) | 2007-04-26 |
WO2007047838A3 true WO2007047838A3 (fr) | 2007-12-06 |
Family
ID=37963278
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2006/040883 WO2007047838A2 (fr) | 2005-10-20 | 2006-10-18 | Procede de preparation de l'olmesartan medoxomil |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2007047838A2 (fr) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0710905D0 (en) * | 2007-06-07 | 2007-07-18 | Generics Uk Ltd | Amorphous olmesartan medoxomil |
CN102083823B (zh) | 2008-06-09 | 2015-10-07 | 第一三共株式会社 | 1-联苯甲基咪唑化合物的制备方法 |
SI2334668T1 (sl) * | 2008-09-05 | 2014-08-29 | Krka, Tovarna Zdravil D.D., Novo Mesto | Postopek priprave intermediata olmesartan medoksomila |
EP2426126B1 (fr) | 2009-04-28 | 2014-11-19 | Daiichi Sankyo Company, Limited | Procédé de production de l'olmésartan médoxomil |
EP2426127B1 (fr) * | 2009-04-28 | 2019-09-04 | Daiichi Sankyo Company, Limited | Nouveaux cristaux solvates |
WO2011007368A2 (fr) | 2009-07-14 | 2011-01-20 | Cadila Healthcare Limited | Procédé amélioré de préparation d'olmésartan |
WO2011021224A2 (fr) * | 2009-08-19 | 2011-02-24 | Msn Laboratories Limited | Procédé de préparation de (5-méthyl-2-oxo- 1,3-dioxolen-4-yl)méthyl-4-(1-hydroxy- 1 -méthyléthyl)-2-propyl- l-[4-[2-(tétrazol-5-yl)phényl]phényl]méthyl imidazole-5-carboxylate |
WO2011045760A2 (fr) | 2009-10-13 | 2011-04-21 | Ranbaxy Laboratories Limited | Compositions d'olmésartan médoxomil micronisé |
AR083523A1 (es) | 2010-10-29 | 2013-03-06 | Interquim Sa | Procedimiento de obtencion del olmesartan medoxomilo |
US20150225380A1 (en) | 2012-08-22 | 2015-08-13 | Lupin Limited | Novel Method to Obtain Olmesartan Medoxomil With Reduced Particle Size |
JP6382660B2 (ja) * | 2014-09-24 | 2018-08-29 | 株式会社トクヤマ | オルメサルタンメドキソミルの製造方法 |
CN106749195A (zh) * | 2016-12-30 | 2017-05-31 | 青岛黄海制药有限责任公司 | 一种奥美沙坦酯中间体杂质合成、鉴定的方法 |
CN112337419B (zh) * | 2020-10-27 | 2022-05-13 | 浙江花蝶染料化工有限公司 | 一种4-(1-羟基-1-甲基乙基)-2-丙基咪唑-5-羧酸乙酯的制备方法 |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5459148A (en) * | 1992-12-17 | 1995-10-17 | Sankyo Company, Limited | Biphenyl derivatives and their use for the treatment of hypertension and cardiac disease |
US5646171A (en) * | 1991-02-21 | 1997-07-08 | Sankyo Company, Limited | Angiotensin II antagonist 1-biphenylmethylimidazole compounds and their therapeutic use |
US5674879A (en) * | 1993-09-24 | 1997-10-07 | G.D. Searle & Co. | Compositions including and methods of using conformationally restricted angiotensin II antagonist |
US6878703B2 (en) * | 2000-11-21 | 2005-04-12 | Sankyo Company, Limited | Pharmaceutical composition |
-
2006
- 2006-10-18 WO PCT/US2006/040883 patent/WO2007047838A2/fr active Application Filing
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5646171A (en) * | 1991-02-21 | 1997-07-08 | Sankyo Company, Limited | Angiotensin II antagonist 1-biphenylmethylimidazole compounds and their therapeutic use |
US5459148A (en) * | 1992-12-17 | 1995-10-17 | Sankyo Company, Limited | Biphenyl derivatives and their use for the treatment of hypertension and cardiac disease |
US5674879A (en) * | 1993-09-24 | 1997-10-07 | G.D. Searle & Co. | Compositions including and methods of using conformationally restricted angiotensin II antagonist |
US6878703B2 (en) * | 2000-11-21 | 2005-04-12 | Sankyo Company, Limited | Pharmaceutical composition |
Also Published As
Publication number | Publication date |
---|---|
WO2007047838A2 (fr) | 2007-04-26 |
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