WO2005072082B1 - Composes de 2-guanidinylimidazolidinedione: procedes de preparation et d'utilisation - Google Patents
Composes de 2-guanidinylimidazolidinedione: procedes de preparation et d'utilisationInfo
- Publication number
- WO2005072082B1 WO2005072082B1 PCT/US2004/038909 US2004038909W WO2005072082B1 WO 2005072082 B1 WO2005072082 B1 WO 2005072082B1 US 2004038909 W US2004038909 W US 2004038909W WO 2005072082 B1 WO2005072082 B1 WO 2005072082B1
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- substituted
- unsubstituted
- compound
- acyl
- alkyl
- Prior art date
Links
- 0 C*C(*1*2)([C@@]12N=C(*)NC1=CC=IC=C1)N(C(C)C)C(C(N)=O)=O Chemical compound C*C(*1*2)([C@@]12N=C(*)NC1=CC=IC=C1)N(C(C)C)C(C(N)=O)=O 0.000 description 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/96—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP04821254A EP1686990B1 (fr) | 2003-11-21 | 2004-11-19 | Composes de 2-guanidinylimidazolidinedione: procedes de preparation et d'utilisation |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US52367003P | 2003-11-21 | 2003-11-21 | |
US60/523,670 | 2003-11-21 |
Publications (3)
Publication Number | Publication Date |
---|---|
WO2005072082A2 WO2005072082A2 (fr) | 2005-08-11 |
WO2005072082A3 WO2005072082A3 (fr) | 2005-12-22 |
WO2005072082B1 true WO2005072082B1 (fr) | 2006-05-11 |
Family
ID=34825868
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2004/038909 WO2005072082A2 (fr) | 2003-11-21 | 2004-11-19 | Composes de 2-guanidinylimidazolidinedione: procedes de preparation et d'utilisation |
Country Status (3)
Country | Link |
---|---|
US (1) | US7101902B2 (fr) |
EP (1) | EP1686990B1 (fr) |
WO (1) | WO2005072082A2 (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010051129A2 (fr) * | 2008-10-03 | 2010-05-06 | The United States Of America, As Represented By The Secretary Of The Army, On Behalf Of U.S. Army Medical Research And Materiel Command | Nouveaux dérivés d'imidazolidinedione comme agents antimalariques, leur préparation, et procédés d'utilisation |
WO2010144101A1 (fr) * | 2009-06-09 | 2010-12-16 | The United States Of America, As Represented By The Secretary Of The Army, On Behalf Of U.S. | Quinoléine méthanols de nouvelle génération |
WO2012149093A1 (fr) * | 2011-04-26 | 2012-11-01 | THE UNITED STATES OF AMERICA, as represented by THE SECRETARY OF ARMY | Dérivés de 2-guanidino-4-oxo-imidazoline en tant qu'agents antipaludiques, synthèse et procédés d'utilisation de ceux-ci |
WO2012149097A2 (fr) * | 2011-04-26 | 2012-11-01 | The United States Of America, As Represented By The Secretary Of Army, | Dérivés de guanidylimidazole et de guanidylimidazoline en tant qu'agents anti-malaria, leur synthèse et leurs procédés d'utilisation |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4957936A (en) * | 1989-02-01 | 1990-09-18 | Nippon Zoki Pharmaceutical Co., Ltd. | Glycocyamidine derivatives |
-
2004
- 2004-11-19 WO PCT/US2004/038909 patent/WO2005072082A2/fr active Application Filing
- 2004-11-19 EP EP04821254A patent/EP1686990B1/fr not_active Not-in-force
- 2004-11-19 US US10/992,363 patent/US7101902B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US20050148645A1 (en) | 2005-07-07 |
US7101902B2 (en) | 2006-09-05 |
EP1686990B1 (fr) | 2012-09-19 |
EP1686990A4 (fr) | 2009-06-03 |
EP1686990A2 (fr) | 2006-08-09 |
WO2005072082A3 (fr) | 2005-12-22 |
WO2005072082A2 (fr) | 2005-08-11 |
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