WO2004091488A3 - Estrogen receptor modulators - Google Patents
Estrogen receptor modulators Download PDFInfo
- Publication number
- WO2004091488A3 WO2004091488A3 PCT/US2004/010853 US2004010853W WO2004091488A3 WO 2004091488 A3 WO2004091488 A3 WO 2004091488A3 US 2004010853 W US2004010853 W US 2004010853W WO 2004091488 A3 WO2004091488 A3 WO 2004091488A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- estrogen
- receptor modulators
- compounds
- estrogen receptor
- functioning
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
- C07D311/60—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4 with aryl radicals attached in position 2
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US46263503P | 2003-04-14 | 2003-04-14 | |
US60/462,635 | 2003-04-14 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2004091488A2 WO2004091488A2 (en) | 2004-10-28 |
WO2004091488A3 true WO2004091488A3 (en) | 2005-04-07 |
Family
ID=33299962
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2004/010853 WO2004091488A2 (en) | 2003-04-14 | 2004-04-09 | Estrogen receptor modulators |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2004091488A2 (en) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102695703A (en) * | 2009-08-19 | 2012-09-26 | 自由州大学 | Synthesis of C-3 coupled biflavonoids and C-3 coupled biflavonoid analogues |
CA2800673A1 (en) * | 2010-06-10 | 2011-12-15 | Aragon Pharmaceuticals, Inc. | Estrogen receptor modulators and uses thereof |
WO2011159769A2 (en) | 2010-06-17 | 2011-12-22 | Aragon Pharmaceuticals, Inc. | Indane estrogen receptor modulators and uses thereof |
US9187460B2 (en) | 2011-12-14 | 2015-11-17 | Seragon Pharmaceuticals, Inc. | Estrogen receptor modulators and uses thereof |
MX2014007198A (en) | 2011-12-16 | 2014-10-13 | Olema Pharmaceuticals Inc | Novel benzopyran compounds, compositions and uses thereof. |
CA2912853A1 (en) * | 2013-06-19 | 2014-12-24 | Seragon Pharmaceuticals, Inc. | Estrogen receptor modulator and uses thereof |
BR112015030595A2 (en) * | 2013-06-19 | 2017-07-25 | Seragon Pharmaceuticals Inc | azetidine estrogen receptor modulators and uses thereof |
WO2014203132A1 (en) | 2013-06-19 | 2014-12-24 | Olema Pharmaceuticals, Inc. | Substituted benzopyran compounds, compositions and uses thereof |
WO2014203129A1 (en) | 2013-06-19 | 2014-12-24 | Olema Pharmaceuticals, Inc. | Combinations of benzopyran compounds, compositions and uses thereof |
JP6768711B2 (en) | 2015-05-26 | 2020-10-14 | エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト | Heterocyclic estrogen receptor modulator and its use |
DK3368519T3 (en) * | 2015-10-27 | 2022-05-23 | Sun Pharma Advanced Res Co Ltd | Hitherto UNKNOWN, HETEROCYCLIC ANTIOSTROGENES |
KR102479822B1 (en) | 2016-02-05 | 2022-12-21 | 인벤티스바이오 엘엘씨 | Selective estrogen receptor degraders and their uses |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5395842A (en) * | 1988-10-31 | 1995-03-07 | Endorecherche Inc. | Anti-estrogenic compounds and compositions |
US20010025028A1 (en) * | 1998-03-13 | 2001-09-27 | Merck & Co., Inc. | Methods of inhibiting bone resorption |
-
2004
- 2004-04-09 WO PCT/US2004/010853 patent/WO2004091488A2/en active Application Filing
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5395842A (en) * | 1988-10-31 | 1995-03-07 | Endorecherche Inc. | Anti-estrogenic compounds and compositions |
US20010025028A1 (en) * | 1998-03-13 | 2001-09-27 | Merck & Co., Inc. | Methods of inhibiting bone resorption |
Also Published As
Publication number | Publication date |
---|---|
WO2004091488A2 (en) | 2004-10-28 |
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