WO2001023353A3 - Verfahren zur herstellung von indolderivaten an fester phase - Google Patents
Verfahren zur herstellung von indolderivaten an fester phase Download PDFInfo
- Publication number
- WO2001023353A3 WO2001023353A3 PCT/EP2000/008838 EP0008838W WO0123353A3 WO 2001023353 A3 WO2001023353 A3 WO 2001023353A3 EP 0008838 W EP0008838 W EP 0008838W WO 0123353 A3 WO0123353 A3 WO 0123353A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- solid phase
- indole derivatives
- producing indole
- indole
- producing
- Prior art date
Links
- 239000007790 solid phase Substances 0.000 title abstract 6
- 150000002475 indoles Chemical class 0.000 title abstract 4
- 229940054051 antipsychotic indole derivative Drugs 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- DCBDOYDVQJVXOH-UHFFFAOYSA-N azane;1h-indole Chemical compound N.C1=CC=C2NC=CC2=C1 DCBDOYDVQJVXOH-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D209/20—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/22—Tin compounds
- C07F7/2208—Compounds having tin linked only to carbon, hydrogen and/or halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA002386074A CA2386074A1 (en) | 1999-09-30 | 2000-09-11 | Method for producing indole derivatives on a solid phase |
EP00960641A EP1222167A2 (de) | 1999-09-30 | 2000-09-11 | Verfahren zur herstellung von indolderivaten an fester phase |
JP2001526507A JP2003510307A (ja) | 1999-09-30 | 2000-09-11 | 固相上でのインドール誘導体の製造法 |
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US15719799P | 1999-09-30 | 1999-09-30 | |
US60/157,197 | 1999-09-30 | ||
DE19955087A DE19955087A1 (de) | 1999-09-30 | 1999-11-17 | Verfahren zur Herstellung von Indolderivaten an fester Phase |
DE19955087.5 | 1999-11-17 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2001023353A2 WO2001023353A2 (de) | 2001-04-05 |
WO2001023353A3 true WO2001023353A3 (de) | 2002-05-02 |
Family
ID=26055552
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP2000/008838 WO2001023353A2 (de) | 1999-09-30 | 2000-09-11 | Verfahren zur herstellung von indolderivaten an fester phase |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP1222167A2 (de) |
JP (1) | JP2003510307A (de) |
CA (1) | CA2386074A1 (de) |
WO (1) | WO2001023353A2 (de) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7781478B2 (en) | 2004-07-14 | 2010-08-24 | Ptc Therapeutics, Inc. | Methods for treating hepatitis C |
US8039122B2 (en) | 2005-03-28 | 2011-10-18 | Semiconductor Energy Laboratory Co., Ltd. | Anthracene derivative, material for light emitting element, light emitting element, light emitting device, and electronic device |
CN101506163B (zh) | 2006-08-30 | 2012-05-02 | 株式会社半导体能源研究所 | 合成蒽衍生物的方法和蒽衍生物、发光元件、发光装置、电子装置 |
US7723722B2 (en) | 2007-03-23 | 2010-05-25 | Semiconductor Energy Laboratory Co., Ltd. | Organic compound, anthracene derivative, and light-emitting element, light-emitting device, and electronic device using anthracene derivative |
ATE517088T1 (de) | 2008-09-19 | 2011-08-15 | Semiconductor Energy Lab | Carbazolderivat und herstellungsverfahren dafür |
KR20170101128A (ko) | 2016-02-26 | 2017-09-05 | 가부시키가이샤 한도오따이 에네루기 켄큐쇼 | 유기 화합물, 발광 소자, 발광 장치, 전자 기기, 및 조명 장치 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0801083A2 (de) * | 1996-04-08 | 1997-10-15 | Pfizer Inc. | Funktionalisiertes Harz für die chemische Synthese |
-
2000
- 2000-09-11 JP JP2001526507A patent/JP2003510307A/ja active Pending
- 2000-09-11 WO PCT/EP2000/008838 patent/WO2001023353A2/de not_active Application Discontinuation
- 2000-09-11 EP EP00960641A patent/EP1222167A2/de not_active Withdrawn
- 2000-09-11 CA CA002386074A patent/CA2386074A1/en not_active Abandoned
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0801083A2 (de) * | 1996-04-08 | 1997-10-15 | Pfizer Inc. | Funktionalisiertes Harz für die chemische Synthese |
Non-Patent Citations (3)
Title |
---|
C C LEZNOFF AND J Y WONG: "The Use of Polymer Supports in Organic Synthesis. III: Selective Chemical Reactions on One Aldehyde Group of Symmetrical Dialdehydes", CANADIAN JOURNAL OF CHEMISTRY - JOURNAL CANADIEN DE CHIMIE,XX,XX, vol. 51, 1973, pages 3756 - 3764, XP002080845, ISSN: 0008-4042 * |
KRAXNER, JOHANNES ET AL: "Traceless linking of indoles. General methodology and application to solid phase supported Mannich and Stille reactions", SYNLETT (2000), (1), 125-127, XP002171484 * |
SMITH A L ET AL: "Traceless Solid Phase Synthesis of 2,3-Disubstituted Indoles", TETRAHEDRON LETTERS,NL,ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, vol. 39, no. 45, 5 November 1998 (1998-11-05), pages 8317 - 8320, XP004139405, ISSN: 0040-4039 * |
Also Published As
Publication number | Publication date |
---|---|
CA2386074A1 (en) | 2001-04-05 |
WO2001023353A2 (de) | 2001-04-05 |
JP2003510307A (ja) | 2003-03-18 |
EP1222167A2 (de) | 2002-07-17 |
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