WO2000020399A3 - Utilisation de 5-hydroxypyrazoles substitues, nouveaux 5-hydroxypyrazoles, procedes permettant de les preparer et agents les contenant - Google Patents

Utilisation de 5-hydroxypyrazoles substitues, nouveaux 5-hydroxypyrazoles, procedes permettant de les preparer et agents les contenant Download PDF

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Publication number
WO2000020399A3
WO2000020399A3 PCT/EP1999/007125 EP9907125W WO0020399A3 WO 2000020399 A3 WO2000020399 A3 WO 2000020399A3 EP 9907125 W EP9907125 W EP 9907125W WO 0020399 A3 WO0020399 A3 WO 0020399A3
Authority
WO
WIPO (PCT)
Prior art keywords
halide
alkyl
hydroxypyrazoles
alkynyl
alkenyl
Prior art date
Application number
PCT/EP1999/007125
Other languages
German (de)
English (en)
Other versions
WO2000020399A2 (fr
Inventor
Andreas Gypser
Reinhard Kirstgen
Hubert Sauter
Herbert Bayer
Oliver Cullmann
Markus Gewehr
Wassilios Grammenos
Bernd Mueller
Arne Ptock
I Blasco Jordi Tormo
Eberhard Ammermann
Thomas Grote
Gisela Lorenz
Siegfried Strathmann
Original Assignee
Basf Ag
Andreas Gypser
Reinhard Kirstgen
Hubert Sauter
Herbert Bayer
Oliver Cullmann
Markus Gewehr
Wassilios Grammenos
Bernd Mueller
Arne Ptock
I Blasco Jordi Tormo
Eberhard Ammermann
Thomas Grote
Gisela Lorenz
Siegfried Strathmann
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag, Andreas Gypser, Reinhard Kirstgen, Hubert Sauter, Herbert Bayer, Oliver Cullmann, Markus Gewehr, Wassilios Grammenos, Bernd Mueller, Arne Ptock, I Blasco Jordi Tormo, Eberhard Ammermann, Thomas Grote, Gisela Lorenz, Siegfried Strathmann filed Critical Basf Ag
Priority to AU61965/99A priority Critical patent/AU6196599A/en
Priority to JP2000574516A priority patent/JP2002526536A/ja
Priority to EP99948860A priority patent/EP1117650A2/fr
Publication of WO2000020399A2 publication Critical patent/WO2000020399A2/fr
Publication of WO2000020399A3 publication Critical patent/WO2000020399A3/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D231/08—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with oxygen or sulfur atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne l'utilisation pour lutter contre des champignons nuisibles, de 5-hydroxypyrazoles de la formule (I) dans laquelle les substituants ont la signification suivante: B désigne aryle ou hétaryle; A désigne C=O, C=S ou SO2; R1 désigne alkyle, halogénure d'alkyle, alkényle, halogénure d'alkényle, alkinyle ou halogénure d'alkinyle, cycloalkyle, cycloalkényle C¿3?-C10, cycloalkinyle, ou aryle, hétérocyclyle ou hétaryle; R?2¿ désigne hydrogène; R3 désigne hydrogène, nitro, cyano, N(R')¿2?, alkyle, halogénure d'alkyle, alcoxy, halogénure d'alcoxy, alkényle, halogénure d'alkényle, alkinyle ou halogénure d'alkinyle, les restes R' désignent indépendamment les uns des autres hydrogène ou alkyle; ou R?2 et R3¿ désignent conjointement un groupe =O, =S ou =N-O-R5, R5 désignant hydrogène, alkyle, halogénure d'alkyle, alkényle, halogénure d'alkényle, alkinyle ou halogénure d'alkynyle; R4 désigne hydrogène halogène, nitro, cyano, N(R')¿2?, alkyle, halogénure d'alkyle, COOR', hétaryle ou hétérocyclyle. L'invention concerne également des agents contenant lesdits composés, ainsi que de nouveaux 5-hydroxypyrazoles et des procédés permettant de les préparer.
PCT/EP1999/007125 1998-10-02 1999-09-24 Utilisation de 5-hydroxypyrazoles substitues, nouveaux 5-hydroxypyrazoles, procedes permettant de les preparer et agents les contenant WO2000020399A2 (fr)

Priority Applications (3)

Application Number Priority Date Filing Date Title
AU61965/99A AU6196599A (en) 1998-10-02 1999-09-24 Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for theproduction thereof and agents containing the same
JP2000574516A JP2002526536A (ja) 1998-10-02 1999-09-24 置換５−ヒドロキシピラゾールの使用、新規５−ヒドロキシピラゾール、それらの製造法、およびそれらを含有する組成物
EP99948860A EP1117650A2 (fr) 1998-10-02 1999-09-24 Utilisation de 5-hydroxypyrazoles substitues, nouveaux 5-hydroxypyrazoles, procedes permettant de les preparer et agents les contenant

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19845509 1998-10-02
DE19845509.7 1998-10-02

Publications (2)

Publication Number Publication Date
WO2000020399A2 WO2000020399A2 (fr) 2000-04-13
WO2000020399A3 true WO2000020399A3 (fr) 2000-07-27

Family

ID=7883246

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP1999/007125 WO2000020399A2 (fr) 1998-10-02 1999-09-24 Utilisation de 5-hydroxypyrazoles substitues, nouveaux 5-hydroxypyrazoles, procedes permettant de les preparer et agents les contenant

Country Status (4)

Country Link
EP (1) EP1117650A2 (fr)
JP (1) JP2002526536A (fr)
AU (1) AU6196599A (fr)
WO (1) WO2000020399A2 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101184393A (zh) * 2005-05-31 2008-05-21 巴斯福股份公司 双环5-羟基吡唑啉、其制备方法以及包含它们的试剂
EP1893018A1 (fr) * 2005-05-31 2008-03-05 Basf Se N-benzyl-5-hydroxy-5-phenylpyrazolines fongicides, procede de production de ces composes et agents contenant lesdits composes
CN101184736A (zh) * 2005-05-31 2008-05-21 巴斯福股份公司 杀真菌的5-羟基吡唑啉、其生产方法以及包含它们的试剂
BRPI0610964A2 (pt) * 2005-05-31 2016-08-30 Basf Ag uso de compostos, compostos, processo para preprarar os mesmos, agente fungicida, semente, processo para combater fungos nocivos fitopatogênicos, e, uso de compostos

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0556396A1 (fr) * 1990-11-09 1993-08-25 Nissan Chemical Industries, Limited Derive de pyrazol substitue et bactericide agrohorticole

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0556396A1 (fr) * 1990-11-09 1993-08-25 Nissan Chemical Industries, Limited Derive de pyrazol substitue et bactericide agrohorticole

Non-Patent Citations (12)

* Cited by examiner, † Cited by third party
Title
ANAL. CHIM. ACTA (1985), 170(2), 319-24 *
CHEMICAL ABSTRACTS, vol. 100, no. 3, 16 January 1984, Columbus, Ohio, US; abstract no. 22225, YAKIMOVICH, S.I. ET AL.: "Tautomerism of thiobenzoylhydrazones of aroylacetones and aroylacetaldehydes" XP002133646 *
CHEMICAL ABSTRACTS, vol. 103, no. 20, 18 November 1985, Columbus, Ohio, US; abstract no. 171065, UHLEMANN, E. ET AL: "Complex formation and liquid-liquid extraction of tin with potentially tridentate dianionic ligands" XP002133643 *
CHEMICAL ABSTRACTS, vol. 117, no. 24, 14 December 1992, Columbus, Ohio, US; abstract no. 244557, TOSHEV, M.T. ET AL.: "Structures of condensation products of .beta.-diketones with thiobenzoylhydrazine and their nickel(II) complexes" XP002133644 *
CHEMICAL ABSTRACTS, vol. 131, Columbus, Ohio, US; abstract no. 271830, KALLURAYA, BALAKRISHNA ET AL: "Reactions of aryl/aryloxyacet hydrazides with acetylenic ketones" XP002133647 *
CHEMICAL ABSTRACTS, vol. 96, no. 11, 15 March 1982, Columbus, Ohio, US; abstract no. 85477, KHRUSTALEV, V.A. ET AL.: "Ring-ring tautomerism in 1-thioacyl-5-hydroxy-2-pyrazoline 5-(2-oxoalkyl)-.Delta.21,3,4-thiadiazoline" XP002133645 *
D.M. EVANS ET AL.: "Thiadiazoles and Dihydrothiadiazoles. Part 5. Synthesis of 2,3-Dithydro-1,3,4-thiadiazoles by Reaction of Aldehydes or Ketones with Thioaroylhydrazines", JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS 1, no. 8, 1986, LETCHWORTH GB, pages 1499 - 1505, XP002133641 *
INDIAN J. HETEROCYCL. CHEM. (1999), 8(4), 309-314 *
YAKIMOVICH, S. I. ET AL: "Tautomerism in a series of products of condensation of fluorinated 1,3-diketones with aroylhydrazines", RUSS. J. ORG. CHEM. (1997), 33(3), 370-374, XP002133642 *
ZH. NEORG. KHIM., vol. 37, no. 5, 1992, pages 1052 - 1061 *
ZH. ORG. KHIM., vol. 17, no. 11, 1981, pages 2451 - 2452 *
ZH. ORG. KHIM., vol. 19, no. 9, 1983, pages 1875 - 1881 *

Also Published As

Publication number Publication date
AU6196599A (en) 2000-04-26
WO2000020399A2 (fr) 2000-04-13
JP2002526536A (ja) 2002-08-20
EP1117650A2 (fr) 2001-07-25

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