UY39600A - Inhibidores del receptor del factor de crecimiento epidérmico - Google Patents

Inhibidores del receptor del factor de crecimiento epidérmico

Info

Publication number
UY39600A
UY39600A UY0001039600A UY39600A UY39600A UY 39600 A UY39600 A UY 39600A UY 0001039600 A UY0001039600 A UY 0001039600A UY 39600 A UY39600 A UY 39600A UY 39600 A UY39600 A UY 39600A
Authority
UY
Uruguay
Prior art keywords
growth factor
factor receptor
epidermal growth
receptor inhibitors
compounds
Prior art date
Application number
UY0001039600A
Other languages
English (en)
Inventor
Dmitry Valentinovich Morozov
Kirill Vadimovich Zavialov
Artsiom Evgenievich Shekhautsou
Ilia Alexeevich Smetanin
Georgii Viktorovich Iakobson
Shamil Dinarovich Kadyrov
Adel Ravilevich Khaidarov
Daria Dmitrievna Beketova
Daniel Evgenevich Polianczyk
Ramilia Rinadovna Starodubtseva
Polina Olegovna Suntsova
Dmitry Alekseevich Khalabudin
Original Assignee
Biocad Joint Stock Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from RU2021137120A external-priority patent/RU2021137120A/ru
Application filed by Biocad Joint Stock Co filed Critical Biocad Joint Stock Co
Publication of UY39600A publication Critical patent/UY39600A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/705Receptors; Cell surface antigens; Cell surface determinants
    • C07K14/71Receptors; Cell surface antigens; Cell surface determinants for growth factors; for growth regulators

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invención se refiere a nuevos compuestos de la fórmula I o sal, solvato o estereoisómero farmacéuticamente aceptables de los mismos, que tienen propiedades inhibidoras del EGFR, a las composiciones farmacéuticas que contienen dichos compuestos, a los métodos de tratamiento de enfermedades o trastornos y al uso de dichos compuestos como productos farmacéuticos para tratar enfermedades o trastornos.
UY0001039600A 2020-12-30 2021-12-30 Inhibidores del receptor del factor de crecimiento epidérmico UY39600A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
RU2020144141 2020-12-30
RU2021137120A RU2021137120A (ru) 2021-12-15 Ингибиторы рецептора эпидермального фактора роста

Publications (1)

Publication Number Publication Date
UY39600A true UY39600A (es) 2022-05-31

Family

ID=82259596

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001039600A UY39600A (es) 2020-12-30 2021-12-30 Inhibidores del receptor del factor de crecimiento epidérmico

Country Status (3)

Country Link
TW (1) TW202241890A (es)
UY (1) UY39600A (es)
WO (1) WO2022146201A1 (es)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110207736A1 (en) * 2009-12-23 2011-08-25 Gatekeeper Pharmaceuticals, Inc. Compounds that modulate egfr activity and methods for treating or preventing conditions therewith
US20130137709A1 (en) * 2010-05-05 2013-05-30 Nathanael S. Gray Compounds that modulate EGFR activity and methods for treating or preventing conditions therewith
CN104140418B (zh) * 2014-08-15 2016-08-24 常州润诺生物科技有限公司 2-(2,4,5-取代苯胺)嘧啶衍生物及其用途
RU2702631C2 (ru) * 2014-10-11 2019-10-09 Шанхай Хэнсох Биомедикал Ко., Лтд. Ингибитор egfr и его получение и применение

Also Published As

Publication number Publication date
WO2022146201A1 (en) 2022-07-07
TW202241890A (zh) 2022-11-01

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