UY37824A - CRYSTAL FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-TIAZOLIL) -2 - [[(3S) -2,2-DIMETIL-4-OXO-1- ( SULFOXI) -3-AZETIDINIL] AMINO] -2-OXOETILIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINE] METHYL] PHENOXY] -PROPANOIC - Google Patents

CRYSTAL FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-TIAZOLIL) -2 - [[(3S) -2,2-DIMETIL-4-OXO-1- ( SULFOXI) -3-AZETIDINIL] AMINO] -2-OXOETILIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINE] METHYL] PHENOXY] -PROPANOIC

Info

Publication number
UY37824A
UY37824A UY0001037824A UY37824A UY37824A UY 37824 A UY37824 A UY 37824A UY 0001037824 A UY0001037824 A UY 0001037824A UY 37824 A UY37824 A UY 37824A UY 37824 A UY37824 A UY 37824A
Authority
UY
Uruguay
Prior art keywords
amino
imino
phenoxy
oxo
methyl
Prior art date
Application number
UY0001037824A
Other languages
Spanish (es)
Inventor
Susanne Bonsmann
Wilfried Schwab Dr
Burkhard Klenke Dr
Original Assignee
Aicuris Anti Infective Cures Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aicuris Anti Infective Cures Gmbh filed Critical Aicuris Anti Infective Cures Gmbh
Publication of UY37824A publication Critical patent/UY37824A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención se refiere a la primera forma cristalina del ácido (2S)-2-[[(Z)-[1-(2-amino-4-tiazolil)-2-[[(3S)-2,2-dimetil-4-oxo-1-(sulfoxi)-3-azetidinil]amino]-2-oxoetiliden]amino]oxi]-3-[4-[imino[(3R)-3- piperidinilamino]metil]fenoxi]-propanoico, es decir, el compuesto de fórmula (I).The invention relates to the first crystalline form of (2S) -2 - [[((Z) - [1- (2-amino-4-thiazolyl) -2 - [[((3S) -2,2-dimethyl- 4-oxo-1- (sulfoxy) -3-azetidinyl] amino] -2-oxoethylidene] amino] oxy] -3- [4- [imino [(3R) -3-piperidinylamino] methyl] phenoxy] -propanoic acid, is ie, the compound of formula (I).

UY0001037824A 2017-07-28 2018-07-27 CRYSTAL FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-TIAZOLIL) -2 - [[(3S) -2,2-DIMETIL-4-OXO-1- ( SULFOXI) -3-AZETIDINIL] AMINO] -2-OXOETILIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINE] METHYL] PHENOXY] -PROPANOIC UY37824A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP17183862 2017-07-28

Publications (1)

Publication Number Publication Date
UY37824A true UY37824A (en) 2019-02-28

Family

ID=59485296

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001037824A UY37824A (en) 2017-07-28 2018-07-27 CRYSTAL FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-TIAZOLIL) -2 - [[(3S) -2,2-DIMETIL-4-OXO-1- ( SULFOXI) -3-AZETIDINIL] AMINO] -2-OXOETILIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINE] METHYL] PHENOXY] -PROPANOIC

Country Status (4)

Country Link
AR (1) AR112464A1 (en)
TW (1) TW201920163A (en)
UY (1) UY37824A (en)
WO (1) WO2019020810A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111592536B (en) * 2020-06-04 2023-11-03 宁夏农林科学院农业资源与环境研究所（宁夏土壤与植物营养重点实验室） Monocyclic beta-lactam compound, preparation method and application thereof
CN115210231B (en) * 2020-07-16 2024-10-08 宁夏农林科学院 Monocyclic lactams, process for their preparation and their use as antibacterial agents
US20230150996A1 (en) * 2020-08-06 2023-05-18 Ningxia Academy Of Agriculture And Forestry Sciences B-lactam compounds, their preparation and use as antibacterial agents
IL312841A (en) 2021-11-18 2024-07-01 Merck Sharp & Dohme Llc Chromane amidine monobactam antibiotics

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY34585A (en) 2012-01-24 2013-09-02 Aicuris Gmbh & Co Kg B-LACTAMIC COMPOUNDS REPLACED WITH AMIDINE, ITS PREPARATION AND USE

Also Published As

Publication number Publication date
AR112464A1 (en) 2019-10-30
TW201920163A (en) 2019-06-01
WO2019020810A1 (en) 2019-01-31

Similar Documents

Publication Publication Date Title
UY37824A (en) CRYSTAL FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-TIAZOLIL) -2 - [[(3S) -2,2-DIMETIL-4-OXO-1- ( SULFOXI) -3-AZETIDINIL] AMINO] -2-OXOETILIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINE] METHYL] PHENOXY] -PROPANOIC
CL2017000705A1 (en) New compounds
AR116394A2 (en) N- [5- (AMINOSULFONYL) -4-METHYL-1,3-THIAZOL-2-IL] -N-METHYL-2- [4- (2-PYRIDINYL) PHENYL] ACETAMIDE MONOHYDRATE MESILATE
CY1118435T1 (en) MORPHOLINE NUCLEAR ACID PRODUCER
EA201592305A1 (en) METHOD OF OBTAINING AND CRYSTAL FORMS OF MDM2 INHIBITOR
PE20170664A1 (en) APELINE RECEPTOR AGONISTS (APJ) AND USES OF THE SAME
AR098929A1 (en) CRYSTALLINE SOLID FORMS OF COMPOUND 2 - ((S) - (((2R, 3R, 4R, 5R) -5- (2,4-DIOXO-3,4-DIHYDROPIRIMIDIN-1 (2H) -IL) -4-FLUORO -3-HYDROXI-4-METHYLTHETRAHYDROFURAN-2-IL) METOXI) (PHENOXI) PHOSPHORILAMINE) PROPANOATE
PE20142403A1 (en) BETA-LACTAMASE INHIBITORS COMPOUNDS
PE20140849A1 (en) 3,5-DIAMINO-6-CHLORO-N- (N- (4- (4- (2- (HEXYL (2,3,4,5,6-PENTAHYDROXYHEXYL) AMINO) ETHOXY) PHENYL) BUTYL) CARBAMIMIDOYL) PYRAZINE -2-CARBOXAMIDE
ES2723277T3 (en) A solid form of (S) -3- (4 - ((4-morpholinomethyl) benzyl) oxy) -1-oxoisoindolin-2-yl) piperidine-2,6-dione hydrochloride
BR112015000160A2 (en) Manufacture of 2- (5-bromo-4- (4-cyclopropylhydronaphthalen-1-yl) -4h-1,2,4-triazol-3-yl-thio) acetic acid
AR078944A1 (en) N1-PIRAZOLOESPIROCETONA ACETIL-COA CARBOXYLASE INHIBITORS
MY172534A (en) Polymorphic forms of 2-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4h-1,2,4-triazol-3-ylthio)acetic acid and uses thereof
CO6210692A2 (en) HYDANTOIN DERIVATIVES USED AS MMP INHIBITORS
PE20090243A1 (en) IMIDAZOLE COMPOUNDS SUBSTITUTED AS RENIN INHIBITORS
WO2014188453A3 (en) Novel process for the preparation of 2-[4-(2-{4-[1-(2-ethoxyethyl)-1h-benzimidazol-2-yl]-1-piperidinyl}ethyl) phenyl]-2-methylpropanoic acid
CL2021000454A1 (en) Method for preparing 2 - [(3r) -3-methylmofolin-4-yl] -4- (1-methyl-1h-pyrazol-5-yl) -8- (1h-pyrazol-5-yl) -1 , 7-naphthyridine
PE20061421A1 (en) N-FORMIL-HYDROXYLAMINE COMPOUNDS AS PEPTIDYL-DEFORMYLASE INHIBITORS
CY1122506T1 (en) CRYSTAL FORM OF THE COMPOUND (S)-3-{4-[5-(2-CYCLOPENTYL-6-METHOXY- PYRIDIN-4- YL)-[1,2,4]OXADIAZOL-3- YL]-2- ETHYL- 6-METHYL- PHENOXY}-PROPANE-1,2-DIOL
ECSP11011081A (en) 3-AMINOCICLOPENTANCARBOXAMIDAS
CO6260137A2 (en) EPOXY COMPOUND AND METHOD TO MANUFACTURE THE SAME
CO6460700A2 (en) PIRAZOL COMPOUND
CO6700844A2 (en) New crystalline forms of (e) -3- (2- (1 - ((2- (5-bromo-pyrimidin-2-yl) -3- cyclopentyl-1 methyl-1h indole-6-carbonyl) -amino) -cyclobutyl-3-methyl-3h-bacimidazol-5 -) - acrylics as vhc inhibitors
MX365948B (en) Asymmetric synthesis of a substituted pyrrolidine-2-carboxamide.
NI200900154A (en) NEW PROCEDURE FOR OBTAINING THE CRYSTALLINE V FORM OF AGOMELATIN

Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20231110