AR112464A1 - CRYSTALLINE FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-THIAZOLYL) -2 - [[(3S) -2,2-DIMETHYL-4-OXO-1- ( SULFOXI) -3-AZETIDINYL] AMINO] -2-OXOETHYLIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINO] METHYL] PHENOXY] -PROPANOICO - Google Patents

CRYSTALLINE FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-THIAZOLYL) -2 - [[(3S) -2,2-DIMETHYL-4-OXO-1- ( SULFOXI) -3-AZETIDINYL] AMINO] -2-OXOETHYLIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINO] METHYL] PHENOXY] -PROPANOICO

Info

Publication number
AR112464A1
AR112464A1 ARP180102116A AR112464A1 AR 112464 A1 AR112464 A1 AR 112464A1 AR P180102116 A ARP180102116 A AR P180102116A AR 112464 A1 AR112464 A1 AR 112464A1
Authority
AR
Argentina
Prior art keywords
amino
piperidinylamino
azetidinyl
imino
thiazolyl
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Susanne Bonsmann
Schwab Wilfried Dr
Klenke Burkhard Dr
Original Assignee
Aicuris Anti Infective Cures Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aicuris Anti Infective Cures Gmbh filed Critical Aicuris Anti Infective Cures Gmbh
Publication of AR112464A1 publication Critical patent/AR112464A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Se refiere a la primera forma cristalina del ácido (2S)-2-[[(Z)-[1-(2-amino-4-tiazolil)-2-[[(3S)-2,2-dimetil-4-oxo-1-(sulfoxi)-3-azetidinil]amino]-2-oxoetiliden]amino]oxi]-3-[4-[imino[(3R)-3-piperidinilamino]metil]fenoxi]-propanoico, es decir, el compuesto de fórmula (1).Refers to the first crystalline form of acid (2S) -2 - [[(Z) - [1- (2-amino-4-thiazolyl) -2 - [[(3S) -2,2-dimethyl-4- oxo-1- (sulfoxy) -3-azetidinyl] amino] -2-oxoethylidene] amino] oxy] -3- [4- [imino [(3R) -3-piperidinylamino] methyl] phenoxy] -propanoic, i.e. the compound of formula (1).

ARP180102116 2017-07-28 2018-07-27 CRYSTALLINE FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-THIAZOLYL) -2 - [[(3S) -2,2-DIMETHYL-4-OXO-1- ( SULFOXI) -3-AZETIDINYL] AMINO] -2-OXOETHYLIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINO] METHYL] PHENOXY] -PROPANOICO AR112464A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP17183862 2017-07-28

Publications (1)

Publication Number Publication Date
AR112464A1 true AR112464A1 (en) 2019-10-30

Family

ID=59485296

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP180102116 AR112464A1 (en) 2017-07-28 2018-07-27 CRYSTALLINE FORM OF ACID (2S) -2 - [[(Z) - [1- (2-AMINO-4-THIAZOLYL) -2 - [[(3S) -2,2-DIMETHYL-4-OXO-1- ( SULFOXI) -3-AZETIDINYL] AMINO] -2-OXOETHYLIDEN] AMINO] OXI] -3- [4- [IMINO [(3R) -3-PIPERIDINYLAMINO] METHYL] PHENOXY] -PROPANOICO

Country Status (4)

Country Link
AR (1) AR112464A1 (en)
TW (1) TW201920163A (en)
UY (1) UY37824A (en)
WO (1) WO2019020810A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111592536B (en) * 2020-06-04 2023-11-03 宁夏农林科学院农业资源与环境研究所（宁夏土壤与植物营养重点实验室） Monocyclic beta-lactam compound, preparation method and application thereof
WO2022011626A1 (en) * 2020-07-16 2022-01-20 Ningxia Academy Of Agriculture And Forestry Sciences Novel monobactam compounds, their preparation and use as antibacterial agents
CN114728953B (en) * 2020-08-06 2024-04-09 宁夏农林科学院 Beta-lactams, process for their preparation and their use as antibiotics
US11932637B2 (en) 2021-11-18 2024-03-19 Merck Sharp & Dohme Llc Chromane amidine monobactam compounds for the treatment of bacterial infections

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY34585A (en) 2012-01-24 2013-09-02 Aicuris Gmbh & Co Kg B-LACTAMIC COMPOUNDS REPLACED WITH AMIDINE, ITS PREPARATION AND USE

Also Published As

Publication number Publication date
UY37824A (en) 2019-02-28
WO2019020810A1 (en) 2019-01-31
TW201920163A (en) 2019-06-01

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