UY32412A - DERIVATIVES OF 4-AMINO-7,8-DIHYDROPIRIMIDO [4,3-d] PYRIMIDIN-5 (6H) -ONA - Google Patents

DERIVATIVES OF 4-AMINO-7,8-DIHYDROPIRIMIDO [4,3-d] PYRIMIDIN-5 (6H) -ONA

Info

Publication number
UY32412A
UY32412A UY0001032412A UY32412A UY32412A UY 32412 A UY32412 A UY 32412A UY 0001032412 A UY0001032412 A UY 0001032412A UY 32412 A UY32412 A UY 32412A UY 32412 A UY32412 A UY 32412A
Authority
UY
Uruguay
Prior art keywords
dihydropirimido
ona
pyrimidin
derivatives
amino
Prior art date
Application number
UY0001032412A
Other languages
Spanish (es)
Inventor
Robert Lee Dow
Michael Jhon Munchhhof
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of UY32412A publication Critical patent/UY32412A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La invención proporciona compuestos de fórmula (I a) o sales farmacéuticamente aceptables de los mismos, así como la preparación, composiciones y usos de los mismos, en la que R1, R2, R3 Y m se definen como se describe anteriormente.The invention provides compounds of formula (I a) or pharmaceutically acceptable salts thereof, as well as the preparation, compositions and uses thereof, wherein R1, R2, R3 and m are defined as described above.

UY0001032412A 2009-02-03 2010-02-02 DERIVATIVES OF 4-AMINO-7,8-DIHYDROPIRIMIDO [4,3-d] PYRIMIDIN-5 (6H) -ONA UY32412A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14952209P 2009-02-03 2009-02-03
US28525809P 2009-12-10 2009-12-10

Publications (1)

Publication Number Publication Date
UY32412A true UY32412A (en) 2010-09-30

Family

ID=42060744

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032412A UY32412A (en) 2009-02-03 2010-02-02 DERIVATIVES OF 4-AMINO-7,8-DIHYDROPIRIMIDO [4,3-d] PYRIMIDIN-5 (6H) -ONA

Country Status (4)

Country Link
AR (1) AR075208A1 (en)
TW (1) TW201040174A (en)
UY (1) UY32412A (en)
WO (1) WO2010089685A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014054053A1 (en) * 2012-10-03 2014-04-10 Advinus Therapeutics Limited Spirocyclic compounds, compositions and medicinal applications thereof
CN111018833B (en) * 2019-12-13 2021-01-01 宁波申泰生物科技有限公司 Apixaban intermediate and preparation method thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6100077A (en) 1998-10-01 2000-08-08 The Trustees Of Columbia University In The City Of New York Isolation of a gene encoding diacylglycerol acyltransferase
EP1383501B1 (en) 2001-02-28 2007-04-04 Merck & Co., Inc. Acylated piperidine derivatives as melanocortin-4 receptor agonists
MXPA05005425A (en) 2002-11-22 2005-11-23 Japan Tobacco Inc Fused bicyclic nitrogen-containing heterocycles.
CA2534643A1 (en) 2003-08-04 2005-02-24 Bayer Pharmaceuticals Corporation Methods for screening and identifying compounds
EP1718309A2 (en) * 2004-01-30 2006-11-08 Japan Tobacco, Inc. Anorectic compounds
JP4069159B2 (en) 2004-05-25 2008-04-02 ファイザー・プロダクツ・インク Tetraazabenzo [e] azulene derivatives and analogs thereof
PA8660701A1 (en) 2005-02-04 2006-09-22 Pfizer Prod Inc SMALL AGONISTS AND THEIR USES
US20090036425A1 (en) * 2007-08-02 2009-02-05 Pfizer Inc Substituted bicyclolactam compounds

Also Published As

Publication number Publication date
TW201040174A (en) 2010-11-16
AR075208A1 (en) 2011-03-16
WO2010089685A1 (en) 2010-08-12

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20181211