UY30424A1 - Derivados de quinolina, su preparacion, su uso y medicamentos que comprenden los mismos. - Google Patents

Derivados de quinolina, su preparacion, su uso y medicamentos que comprenden los mismos.

Info

Publication number
UY30424A1
UY30424A1 UY30424A UY30424A UY30424A1 UY 30424 A1 UY30424 A1 UY 30424A1 UY 30424 A UY30424 A UY 30424A UY 30424 A UY30424 A UY 30424A UY 30424 A1 UY30424 A1 UY 30424A1
Authority
UY
Uruguay
Prior art keywords
preparation
quinolina
medicines
derivatives
understand
Prior art date
Application number
UY30424A
Other languages
English (en)
Inventor
Knut Eis
Olaf Prien
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of UY30424A1 publication Critical patent/UY30424A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

Abstract

Un derivado de quinolina que responde a la formula general (A) : en la cual R1, R2, W, X, Y y Z tienen los valores que se definen en la memoria descriptiva y el uso de los compuestos de la formula general (A) para el tratamiento de diversos trastornos, y la preparacion de compuestos de la formula general (A).
UY30424A 2006-06-21 2007-06-20 Derivados de quinolina, su preparacion, su uso y medicamentos que comprenden los mismos. UY30424A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102006029446A DE102006029446A1 (de) 2006-06-21 2006-06-21 Neue 3-substituierte-Chinoline als Kinase-Inhibitoren

Publications (1)

Publication Number Publication Date
UY30424A1 true UY30424A1 (es) 2008-01-31

Family

ID=38578422

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30424A UY30424A1 (es) 2006-06-21 2007-06-20 Derivados de quinolina, su preparacion, su uso y medicamentos que comprenden los mismos.

Country Status (10)

Country Link
US (1) US20080056987A1 (es)
EP (1) EP2035434A1 (es)
JP (1) JP2009542585A (es)
AR (1) AR061536A1 (es)
CA (1) CA2654237A1 (es)
CL (1) CL2007001805A1 (es)
DE (1) DE102006029446A1 (es)
TW (1) TW200813058A (es)
UY (1) UY30424A1 (es)
WO (1) WO2007147578A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20171345A1 (es) 2010-04-02 2017-09-13 Senomyx Inc Modificador del sabor dulce
MX336378B (es) 2011-08-12 2016-01-15 Senomyx Inc Modificador del sabor dulce.
AU2015343463A1 (en) 2014-11-07 2017-06-15 Senomyx, Inc. Substituted 4-amino-5-(cyclohexyloxy)quinoline-3-carboxylic acids as sweet flavor modifiers
CN110577546B (zh) * 2018-06-08 2021-09-07 江苏威凯尔医药科技有限公司 Vegfr抑制剂及其制备方法和应用
WO2019233458A1 (zh) * 2018-06-08 2019-12-12 江苏威凯尔医药科技有限公司 Vegfr抑制剂及其制备方法和应用
US20230121233A1 (en) * 2020-01-02 2023-04-20 Accro Bioscience Inc. Heteroaryl compounds as inhibitors of programmed necrosis pathway, composition and method using the same
CN113061142A (zh) * 2020-01-02 2021-07-02 爱科诺生物医药股份有限公司 一类具有程序性细胞坏死通路抑制活性的杂环化合物及其应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3269743D1 (en) * 1981-12-14 1986-04-10 Norwich Eaton Pharma Use of the compound 9-(p-(n-methylacetamido)anilino)-7-methyl-1h-imidazo(4,5-f)quinoline hydrochloride (i) as antitumor agent
CA1263378A (en) * 1985-01-08 1989-11-28 Robert James Alaimo Imidazo¬4,5-f|quinolines useful as immunomodulating agents
US5506235A (en) * 1991-08-02 1996-04-09 Pfizer Inc. Quinoline derivatives as immunostimulants
NZ521117A (en) * 2000-03-13 2005-02-25 Wyeth Corp Method of treating or inhibiting colonic polyps
US7026484B2 (en) * 2001-02-23 2006-04-11 Ligand Pharmaceuticals Incorporated Tricyclic androgen receptor modulator compounds and methods

Also Published As

Publication number Publication date
AR061536A1 (es) 2008-09-03
CA2654237A1 (en) 2007-12-27
JP2009542585A (ja) 2009-12-03
EP2035434A1 (en) 2009-03-18
US20080056987A1 (en) 2008-03-06
TW200813058A (en) 2008-03-16
WO2007147578A1 (en) 2007-12-27
DE102006029446A1 (de) 2007-12-27
CL2007001805A1 (es) 2008-02-01

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20170711