UY23934A1 - IMIDAZODIAZEPINES, PROCEDURES FOR THEIR PREPARATION AND MEDICINES THAT CONTAIN THEM. - Google Patents
IMIDAZODIAZEPINES, PROCEDURES FOR THEIR PREPARATION AND MEDICINES THAT CONTAIN THEM.Info
- Publication number
- UY23934A1 UY23934A1 UY23934A UY23934A UY23934A1 UY 23934 A1 UY23934 A1 UY 23934A1 UY 23934 A UY23934 A UY 23934A UY 23934 A UY23934 A UY 23934A UY 23934 A1 UY23934 A1 UY 23934A1
- Authority
- UY
- Uruguay
- Prior art keywords
- imidazodiazepines
- preparation
- dimethylpiperidino
- radicals
- methyl
- Prior art date
Links
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Imidazodiazepinas de fórmula general (I) (figura 1), y sales de adicón de los mismos farmacéuticamente aceptables, donde: A y los átomos de carbono alfa y beta significan uno de los radicales de la figura 2; Q es uno de los radicales de la figura 3; R1 y R2 entre otras posibilidades, junto al átomo de Nitrógeno significan: 1-pirrolidinilo, 1-pirrolinilo, piperidino, 2,6-dimetilpiperidino, 3,3-dimetilpiperidino, morfolino, 4-metil-1-piperazinilo o isoindolin-2-ilo. Ejemplo no limitante: 3-(5-dipropilaminometil-1,2,4-oxadiazol-3-il)-8-fluoro-5-metil-5,6-dihidro-4H-imidazo(1,5-a) [1,4]benzodiazepin-6-ona. La invención también proporciona un procedimiento para la preparación de un compuesto según lo descrito. Los compuestos conforme a la invención son de utilidad para la producción de medicamentos ansiolíticos y/o anticonvulsivos y/o relantes musculaes y/osedativo-hiptónicos.Imidazodiazepines of general formula (I) (figure 1), and pharmaceutically acceptable addition salts thereof, where: A and the alpha and beta carbon atoms signify one of the radicals of figure 2; Q is one of the radicals in Figure 3; R1 and R2 among other possibilities, together with the Nitrogen atom mean: 1-pyrrolidinyl, 1-pyrrolinyl, piperidino, 2,6-dimethylpiperidino, 3,3-dimethylpiperidino, morpholino, 4-methyl-1-piperazinilo or isoindolin-2- ilo. Non-limiting example: 3- (5-dipropylaminomethyl-1,2,4-oxadiazol-3-yl) -8-fluoro-5-methyl-5,6-dihydro-4H-imidazo (1,5-a) [1 , 4] benzodiazepin-6-one. The invention also provides a process for the preparation of a compound as described. The compounds according to the invention are useful for the production of anxiolytic and / or anticonvulsant and / or muscle relaxant and / osdative-hyptonic drugs.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH78394 | 1994-03-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY23934A1 true UY23934A1 (en) | 1995-09-05 |
Family
ID=4195086
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY23934A UY23934A1 (en) | 1994-03-16 | 1995-03-15 | IMIDAZODIAZEPINES, PROCEDURES FOR THEIR PREPARATION AND MEDICINES THAT CONTAIN THEM. |
Country Status (9)
| Country | Link |
|---|---|
| BR (1) | BR9501104A (en) |
| HR (1) | HRP950125A2 (en) |
| PE (1) | PE2996A1 (en) |
| PL (1) | PL307711A1 (en) |
| SG (1) | SG24097A1 (en) |
| SV (1) | SV1995000014A (en) |
| UY (1) | UY23934A1 (en) |
| YU (1) | YU17695A (en) |
| ZA (1) | ZA951969B (en) |
-
1995
- 1995-03-09 PE PE26376795A patent/PE2996A1/en not_active Application Discontinuation
- 1995-03-09 ZA ZA951969A patent/ZA951969B/en unknown
- 1995-03-09 SG SG1995000082A patent/SG24097A1/en unknown
- 1995-03-14 SV SV1995000014A patent/SV1995000014A/en unknown
- 1995-03-15 PL PL30771195A patent/PL307711A1/en unknown
- 1995-03-15 UY UY23934A patent/UY23934A1/en unknown
- 1995-03-16 HR HRP950125 patent/HRP950125A2/en not_active Application Discontinuation
- 1995-03-16 BR BR9501104A patent/BR9501104A/en not_active IP Right Cessation
- 1995-03-16 YU YU17695A patent/YU17695A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PE2996A1 (en) | 1996-03-04 |
| YU17695A (en) | 1998-09-18 |
| PL307711A1 (en) | 1995-09-18 |
| SV1995000014A (en) | 1998-12-11 |
| ZA951969B (en) | 1995-09-18 |
| BR9501104A (en) | 1996-04-23 |
| SG24097A1 (en) | 1996-02-10 |
| HRP950125A2 (en) | 1997-10-31 |
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