AR004696A1 - DERIVATIVES OF AMIDINE AND ISOTIOUREA, PROCEDURES FOR ITS PREPARATION, NEW INTERMEDIARIES USEFUL IN SUCH PROCEDURE, COMPOSITIONS THAT CONTAIN THEM, THEIR USE IN THERAPY AND TREATMENT METHODS THAT INCLUDE SUCH COMPOUND - Google Patents

DERIVATIVES OF AMIDINE AND ISOTIOUREA, PROCEDURES FOR ITS PREPARATION, NEW INTERMEDIARIES USEFUL IN SUCH PROCEDURE, COMPOSITIONS THAT CONTAIN THEM, THEIR USE IN THERAPY AND TREATMENT METHODS THAT INCLUDE SUCH COMPOUND

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Publication number
AR004696A1
AR004696A1 ARP960104929A ARP960104929A AR004696A1 AR 004696 A1 AR004696 A1 AR 004696A1 AR P960104929 A ARP960104929 A AR P960104929A AR P960104929 A ARP960104929 A AR P960104929A AR 004696 A1 AR004696 A1 AR 004696A1
Authority
AR
Argentina
Prior art keywords
therapy
procedures
preparation
isotiourea
amidine
Prior art date
Application number
ARP960104929A
Other languages
Spanish (es)
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE9600275A external-priority patent/SE9600275D0/en
Priority claimed from SE9603301A external-priority patent/SE9603301D0/en
Priority claimed from SE9603300A external-priority patent/SE9603300D0/en
Application filed by Astra Ab filed Critical Astra Ab
Publication of AR004696A1 publication Critical patent/AR004696A1/en

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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se presentan los novedosos compuestos de la fórmula I en los cuales X, R2, R3, R4 y R5 son tan como se los definiera en la memoria descriptiva y losisómeros ópticos y racematos de los mismos, y las sales farmacéuticamaente aceptables de losmis mos; junto con procedimientos para su preparación,composiciones que los contienen, su uso en terapia y compuestos intermediarios para su uso en el procedimiento de preparación de los compuestos de fórmula(I)The novel compounds of formula I in which X, R2, R3, R4 and R5 are as defined in the specification and the optical isomers and racemates thereof, and the pharmaceutically acceptable salts thereof are presented; together with procedures for their preparation, compositions containing them, their use in therapy and intermediates for their use in the process of preparing the compounds of formula (I)

ARP960104929A 1995-11-07 1996-10-25 DERIVATIVES OF AMIDINE AND ISOTIOUREA, PROCEDURES FOR ITS PREPARATION, NEW INTERMEDIARIES USEFUL IN SUCH PROCEDURE, COMPOSITIONS THAT CONTAIN THEM, THEIR USE IN THERAPY AND TREATMENT METHODS THAT INCLUDE SUCH COMPOUND AR004696A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US627695P 1995-11-07 1995-11-07
US625395P 1995-11-07 1995-11-07
SE9600275A SE9600275D0 (en) 1996-01-25 1996-01-25 Compounds
SE9603301A SE9603301D0 (en) 1996-09-11 1996-09-11 Compounds and compositions
SE9603300A SE9603300D0 (en) 1996-09-11 1996-09-11 Compounds

Publications (1)

Publication Number Publication Date
AR004696A1 true AR004696A1 (en) 1999-03-10

Family

ID=51929164

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP960104929A AR004696A1 (en) 1995-11-07 1996-10-25 DERIVATIVES OF AMIDINE AND ISOTIOUREA, PROCEDURES FOR ITS PREPARATION, NEW INTERMEDIARIES USEFUL IN SUCH PROCEDURE, COMPOSITIONS THAT CONTAIN THEM, THEIR USE IN THERAPY AND TREATMENT METHODS THAT INCLUDE SUCH COMPOUND

Country Status (1)

Country Link
AR (1) AR004696A1 (en)

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