UA94465C2 - Комбіновані препарати з вмістом біфепруноксу та l-dopa - Google Patents
Комбіновані препарати з вмістом біфепруноксу та l-dopaInfo
- Publication number
- UA94465C2 UA94465C2 UAA200900252A UAA200900252A UA94465C2 UA 94465 C2 UA94465 C2 UA 94465C2 UA A200900252 A UAA200900252 A UA A200900252A UA A200900252 A UAA200900252 A UA A200900252A UA 94465 C2 UA94465 C2 UA 94465C2
- Authority
- UA
- Ukraine
- Prior art keywords
- dopa
- bifeprunox
- combination preparations
- bifeprnnox
- simultaneous
- Prior art date
Links
- WTDRDQBEARUVNC-LURJTMIESA-N L-DOPA Chemical compound OC(=O)[C@@H](N)CC1=CC=C(O)C(O)=C1 WTDRDQBEARUVNC-LURJTMIESA-N 0.000 title abstract 2
- WTDRDQBEARUVNC-UHFFFAOYSA-N L-Dopa Natural products OC(=O)C(N)CC1=CC=C(O)C(O)=C1 WTDRDQBEARUVNC-UHFFFAOYSA-N 0.000 title abstract 2
- 238000002360 preparation method Methods 0.000 title abstract 2
- CYGODHVAJQTCBG-UHFFFAOYSA-N Bifeprunox Chemical compound C=12OC(=O)NC2=CC=CC=1N(CC1)CCN1CC(C=1)=CC=CC=1C1=CC=CC=C1 CYGODHVAJQTCBG-UHFFFAOYSA-N 0.000 title 1
- 229950009087 bifeprunox Drugs 0.000 title 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- 208000018737 Parkinson disease Diseases 0.000 abstract 1
- 208000005793 Restless legs syndrome Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 230000010249 dopaminergic function Effects 0.000 abstract 1
- 238000011084 recovery Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Винахід стосується застосування комбінованого препарату біфепруноксу або його N-оксиду чи фармакологічно прийнятних солей зазначених сполук та L-DOPA для одночасного, нарізного або послідовного застосування при лікуванні розладів, що потребують відновлення допамінергійної функції, зокрема, хвороби Паркінсона та синдрому неспокійних ніг.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP06115587 | 2006-06-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
UA94465C2 true UA94465C2 (uk) | 2011-05-10 |
Family
ID=37156018
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200900252A UA94465C2 (uk) | 2006-06-16 | 2007-06-15 | Комбіновані препарати з вмістом біфепруноксу та l-dopa |
Country Status (7)
Country | Link |
---|---|
CN (1) | CN101478990A (uk) |
AR (1) | AR061357A1 (uk) |
BR (1) | BRPI0713691A2 (uk) |
MX (1) | MX2008016226A (uk) |
SA (1) | SA07280316B1 (uk) |
TW (1) | TW200815031A (uk) |
UA (1) | UA94465C2 (uk) |
-
2007
- 2007-06-13 SA SA7280316A patent/SA07280316B1/ar unknown
- 2007-06-13 AR ARP070102582A patent/AR061357A1/es not_active Application Discontinuation
- 2007-06-13 TW TW096121306A patent/TW200815031A/zh unknown
- 2007-06-15 CN CNA2007800225408A patent/CN101478990A/zh active Pending
- 2007-06-15 BR BRPI0713691-9A patent/BRPI0713691A2/pt not_active IP Right Cessation
- 2007-06-15 MX MX2008016226A patent/MX2008016226A/es not_active Application Discontinuation
- 2007-06-15 UA UAA200900252A patent/UA94465C2/uk unknown
Also Published As
Publication number | Publication date |
---|---|
TW200815031A (en) | 2008-04-01 |
BRPI0713691A2 (pt) | 2012-10-30 |
SA07280316B1 (ar) | 2010-10-19 |
CN101478990A (zh) | 2009-07-08 |
MX2008016226A (es) | 2009-01-19 |
AR061357A1 (es) | 2008-08-20 |
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UA94465C2 (uk) | Комбіновані препарати з вмістом біфепруноксу та l-dopa |