UA84714C2 - Normal;heading 1;heading 2;IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION - Google Patents

Normal;heading 1;heading 2;IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION

Info

Publication number
UA84714C2
UA84714C2 UAA200603711A UAA200603711A UA84714C2 UA 84714 C2 UA84714 C2 UA 84714C2 UA A200603711 A UAA200603711 A UA A200603711A UA A200603711 A UAA200603711 A UA A200603711A UA 84714 C2 UA84714 C2 UA 84714C2
Authority
UA
Ukraine
Prior art keywords
heading
treatment
hiv
inflammation
normal
Prior art date
Application number
UAA200603711A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Пол Энтони Стаппл
Original Assignee
Пфайзер Инк
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Пфайзер Инк filed Critical Пфайзер Инк
Publication of UA84714C2 publication Critical patent/UA84714C2/en

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The present invention provides compounds of formula (I) wherein Rand Rare as defined hereinabove. The compounds of the present invention are modulators, especially antagonists, of the activity of chemokine CCR5 receptors. Modulators of the CCR5 receptor may be useful in the treatment of various inflammatory diseases and conditions, and in the treatment of infection by HIV and genetically related retroviruses.
UAA200603711A 2003-10-03 2004-09-28 Normal;heading 1;heading 2;IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION UA84714C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0323236.0A GB0323236D0 (en) 2003-10-03 2003-10-03 Chemical compounds

Publications (1)

Publication Number Publication Date
UA84714C2 true UA84714C2 (en) 2008-11-25

Family

ID=29415495

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200603711A UA84714C2 (en) 2003-10-03 2004-09-28 Normal;heading 1;heading 2;IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION

Country Status (5)

Country Link
CN (2) CN100526313C (en)
GB (1) GB0323236D0 (en)
GT (1) GT200400203A (en)
UA (1) UA84714C2 (en)
ZA (1) ZA200602096B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2010004493A (en) * 2007-10-25 2010-06-11 Exelixis Inc Tropane compounds.

Also Published As

Publication number Publication date
ZA200602096B (en) 2007-05-30
GB0323236D0 (en) 2003-11-05
CN100526313C (en) 2009-08-12
CN101632664A (en) 2010-01-27
GT200400203A (en) 2005-04-18
CN1863801A (en) 2006-11-15

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