TWI838736B - 做為腺苷A2a受體拮抗劑之化合物及包含該化合物之醫藥組合物 - Google Patents

Info

Publication number

TWI838736B

TWI838736B TW111115277A TW111115277A TWI838736B TW I838736 B TWI838736 B TW I838736B TW 111115277 A TW111115277 A TW 111115277A TW 111115277 A TW111115277 A TW 111115277A TW I838736 B TWI838736 B TW I838736B

Authority

TW

Taiwan

Prior art keywords

compound

amino

triazolo

furan

trioxan

Prior art date

2021-04-23

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• 150000003839 salts Chemical class 0.000 claims abstract description 41
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• 125000000592 heterocycloalkyl group Chemical group 0.000 claims description 23
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• 150000002367 halogens Chemical class 0.000 claims description 21
• 102000007471 Adenosine A2A receptor Human genes 0.000 claims description 20
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• 229910052757 nitrogen Inorganic materials 0.000 claims description 16
• 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 10
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• 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 8
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