TW337986B - Pyrazolo(1.5a) pyrimidines, their preparation and their use - Google Patents

Pyrazolo(1.5a) pyrimidines, their preparation and their use

Info

Publication number
TW337986B
TW337986B TW085105501A TW85105501A TW337986B TW 337986 B TW337986 B TW 337986B TW 085105501 A TW085105501 A TW 085105501A TW 85105501 A TW85105501 A TW 85105501A TW 337986 B TW337986 B TW 337986B
Authority
TW
Taiwan
Prior art keywords
noch3
alkyl
hydrogen
pyrazolo
h3co
Prior art date
Application number
TW085105501A
Other languages
English (en)
Inventor
Benoit Remy
Grote Thomas
Bayer Herbert
Muller Bernd
Oberdorff Klaus
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Application granted granted Critical
Publication of TW337986B publication Critical patent/TW337986B/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
TW085105501A 1995-05-09 1996-05-09 Pyrazolo(1.5a) pyrimidines, their preparation and their use TW337986B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19516843 1995-05-09
DE19602072 1996-01-20

Publications (1)

Publication Number Publication Date
TW337986B true TW337986B (en) 1998-08-11

Family

ID=26014970

Family Applications (1)

Application Number Title Priority Date Filing Date
TW085105501A TW337986B (en) 1995-05-09 1996-05-09 Pyrazolo(1.5a) pyrimidines, their preparation and their use

Country Status (14)

Country Link
US (1) US5902773A (zh)
EP (1) EP0824533B1 (zh)
JP (1) JPH11506428A (zh)
KR (1) KR19990008451A (zh)
CN (1) CN1183783A (zh)
AT (1) ATE208778T1 (zh)
AU (1) AU700001B2 (zh)
BR (1) BR9608100A (zh)
CA (1) CA2217778A1 (zh)
DE (1) DE59608203D1 (zh)
HU (1) HUP9801135A2 (zh)
IL (1) IL118167A0 (zh)
TW (1) TW337986B (zh)
WO (1) WO1996035690A1 (zh)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19731153A1 (de) 1997-07-21 1999-01-28 Basf Ag 2-(Pyrazolyl- und Triazolyl-3'-oxymethylen)-phenyl-isoxazolone und -triazolone, Verfahren zu ihrer Herstellung und ihre Verwendung
WO1999060858A1 (fr) * 1998-05-28 1999-12-02 Sumitomo Chemical Company, Limited Composes de pyrazolopyrimidine et leur utilisation
US6552026B2 (en) 1999-06-14 2003-04-22 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines
US20020061897A1 (en) 2000-03-30 2002-05-23 Elliott Richard L. Neuropeptide Y antagonists
US7067520B2 (en) * 2000-11-17 2006-06-27 Ishihara Sangyo Kaisha, Ltd. Preventive or therapeutic medicines for diabetes containing fused-heterocyclic compounds or their salts
AU2002359160A1 (en) * 2001-12-20 2003-07-09 Biovitrum Ab PIPAZOLO (1,5-a) PYRIMIDINE DERIVATIVES AS MODULATORS OF PPAR
WO2004082383A1 (en) * 2003-03-17 2004-09-30 Basf Aktiengesellschaft Use of triazolopyrimidines for combating nematode diseases of plants
DE10357569A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
WO2006128184A2 (en) * 2005-05-20 2006-11-30 Alantos-Pharmaceuticals, Inc. Pyrimidine or triazine fused bicyclic metalloprotease inhibitors
US20070155738A1 (en) * 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
WO2007075869A2 (en) 2005-12-23 2007-07-05 Ariad Pharmaceuticals, Inc. Bicyclic heteroaryl compounds
CN101967149B (zh) * 2009-07-28 2013-01-16 北京师范大学 18F取代硝基标记的吡唑并[1,5-a]嘧啶类化合物及制备和应用
US9309250B2 (en) 2011-06-22 2016-04-12 Vertex Pharmaceuticals Incorporated Substituted pyrrolo[2,3-b]pyrazines as ATR kinase inhibitors
HUE037371T2 (hu) 2012-12-07 2018-08-28 Vertex Pharma 2-Amino-6-fluor-N-(5-fluor-4-(4-(4-(oxetan-3-il)piperazin-1-karbonil)piperidin-1-il)piridin-3-il) pirazolo[1,5alfa]pirimidin-3-karboxamid mint ATR kináz inhibitor
JP2016512815A (ja) 2013-03-15 2016-05-09 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ Ａｔｒキナーゼの阻害剤として有用な縮合ピラゾロピリミジン誘導体
EP2970288A1 (en) 2013-03-15 2016-01-20 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
US8957078B2 (en) 2013-03-15 2015-02-17 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of ATR kinase
AU2014360380B2 (en) 2013-12-06 2019-03-21 Vertex Pharmaceuticals Incorporated 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as ATR kinase inhibitor, its preparation, different solid forms and radiolabelled derivatives thereof
SG11201610197XA (en) 2014-06-05 2017-01-27 Vertex Pharma Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, the preparation of said compound and different solid forms thereof
PL3157566T3 (pl) 2014-06-17 2019-10-31 Vertex Pharma Metoda leczenia nowotworu przy użyciu kombinacji inhibitorów chk1 i atr
WO2017059357A1 (en) 2015-09-30 2017-04-06 Vertex Pharmaceuticals Incorporated Method for treating cancer using a combination of dna damaging agents and atr inhibitors
KR102411150B1 (ko) 2016-08-31 2022-06-21 아지오스 파마슈티컬스 아이엔씨. 세포 대사 과정의 억제제

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8617648D0 (en) * 1986-07-18 1986-08-28 Ici Plc Fungicides
US4877738A (en) * 1986-07-25 1989-10-31 Wisconsin Alumni Research Foundation Biological control of damping off and root rot and inoculum preparation therefor
DE3889345T2 (de) * 1987-02-09 1994-09-01 Zeneca Ltd Schimmelbekämpfungsmittel.
DE3825043A1 (de) * 1988-07-20 1990-02-15 Schering Ag 3-methylsulfonyl-pyrazolo(1,5-a)pyrimidin-sulfonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung als mittel mit herbizider, pflanzenwuchsregulierender und fungizider wirkung
ATE145891T1 (de) * 1989-05-17 1996-12-15 Shionogi & Co Verfahren zur herstellung von alkoxyiminoacetamid-derivaten und ein zwischenproduckt dafür

Also Published As

Publication number Publication date
AU5648496A (en) 1996-11-29
EP0824533B1 (de) 2001-11-14
KR19990008451A (ko) 1999-01-25
CA2217778A1 (en) 1996-11-14
CN1183783A (zh) 1998-06-03
AU700001B2 (en) 1998-12-17
WO1996035690A1 (de) 1996-11-14
EP0824533A1 (de) 1998-02-25
IL118167A0 (en) 1996-09-12
DE59608203D1 (de) 2001-12-20
US5902773A (en) 1999-05-11
BR9608100A (pt) 1999-02-23
HUP9801135A2 (hu) 1998-08-28
JPH11506428A (ja) 1999-06-08
ATE208778T1 (de) 2001-11-15

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