TW201906608A - 口服固體製劑 - Google Patents
口服固體製劑 Download PDFInfo
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- TW201906608A TW201906608A TW107118464A TW107118464A TW201906608A TW 201906608 A TW201906608 A TW 201906608A TW 107118464 A TW107118464 A TW 107118464A TW 107118464 A TW107118464 A TW 107118464A TW 201906608 A TW201906608 A TW 201906608A
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- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/02—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements
- C07D295/027—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring
- C07D295/03—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring with the ring nitrogen atoms directly attached to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/02—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements
- C07D295/027—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring
- C07D295/033—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring with the ring nitrogen atoms directly attached to carbocyclic rings
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Organic Chemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Inorganic Chemistry (AREA)
- Hospice & Palliative Care (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HUP1700253 | 2017-06-13 | ||
| HUP1700253 HUP1700253A1 (hu) | 2017-06-13 | 2017-06-13 | Szilárd orális gyógyszerkészítmények |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW201906608A true TW201906608A (zh) | 2019-02-16 |
Family
ID=89992469
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW107118464A TW201906608A (zh) | 2017-06-13 | 2018-05-30 | 口服固體製劑 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20200222391A1 (enExample) |
| EP (1) | EP3638210A1 (enExample) |
| JP (1) | JP2020523335A (enExample) |
| KR (1) | KR20200016378A (enExample) |
| CN (1) | CN110769815A (enExample) |
| AR (1) | AR112137A1 (enExample) |
| AU (1) | AU2018284138A1 (enExample) |
| BR (1) | BR112019025214A2 (enExample) |
| CA (1) | CA3064694A1 (enExample) |
| CL (1) | CL2019003619A1 (enExample) |
| CO (1) | CO2020000168A2 (enExample) |
| EA (1) | EA202090029A1 (enExample) |
| HU (1) | HUP1700253A1 (enExample) |
| IL (1) | IL271108A (enExample) |
| MX (1) | MX2019015206A (enExample) |
| PE (1) | PE20200334A1 (enExample) |
| PH (1) | PH12019502566A1 (enExample) |
| TW (1) | TW201906608A (enExample) |
| WO (1) | WO2018229641A1 (enExample) |
| ZA (1) | ZA201908454B (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2009270823B2 (en) | 2008-07-16 | 2014-07-17 | Richter Gedeon Nyrt. | Pharmaceutical formulations containing dopamine receptor ligands |
| US11274087B2 (en) | 2016-07-08 | 2022-03-15 | Richter Gedeon Nyrt. | Industrial process for the preparation of cariprazine |
| US11547707B2 (en) | 2019-04-10 | 2023-01-10 | Richter Gedeon Nyrt. | Carbamoyl cyclohexane derivatives for treating autism spectrum disorder |
| US11344503B2 (en) | 2019-12-13 | 2022-05-31 | Halo Science LLC | Cariprazine release formulations |
| US20230355612A1 (en) * | 2020-08-26 | 2023-11-09 | Shanghai Bocimed Pharmaceutical Co., Ltd. | Pharmaceutically acceptable salt of cariprazine and crystal form thereof, and preparation method therefor and use thereof |
| CN114681406B (zh) * | 2020-12-25 | 2023-10-13 | 上海京新生物医药有限公司 | 一种卡利拉嗪长效缓释微球及其制备方法 |
| CN114748428B (zh) * | 2020-12-25 | 2023-05-23 | 上海京新生物医药有限公司 | 一种高载药量的盐酸卡利拉嗪长效缓释微球及其制备方法 |
| CN116675654B (zh) * | 2022-02-22 | 2025-06-13 | 上海云晟研新生物科技有限公司 | 卡利拉嗪药用盐及其晶型、药物组合物、制备方法和用途 |
| CA3244202A1 (en) | 2022-03-17 | 2023-09-21 | Mapi Pharma Ltd. | DEPOSIT SYSTEMS INCLUDING CARIPRAZINE OR SALTS THEREOF |
| HU231682B1 (hu) * | 2022-08-05 | 2025-10-28 | Richter Gedeon Nyrt. | Kariprazin tartalmú szájban diszpergálódó tabletta |
| TR2024011970A1 (tr) * | 2024-09-10 | 2026-03-23 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Kari̇prazi̇n hi̇droklorür i̇çeren kati bi̇r oral bi̇leşi̇m |
| TR2024011968A1 (tr) * | 2024-09-10 | 2026-03-23 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Kariprazin hidroklorür içeren kapsül formülasyonlari |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6248618A (ja) * | 1985-08-27 | 1987-03-03 | Zeria Shinyaku Kogyo Kk | 徐放性製剤およびその製造法 |
| US5910319A (en) | 1997-05-29 | 1999-06-08 | Eli Lilly And Company | Fluoxetine enteric pellets and methods for their preparation and use |
| HU227534B1 (en) | 2003-08-04 | 2011-08-29 | Richter Gedeon Nyrt | (thio)carbamoyl-cyclohexane derivatives, process for producing them and pharmaceutical compositions containing them |
| GB0618879D0 (en) | 2006-09-26 | 2006-11-01 | Zysis Ltd | Pharmaceutical compositions |
| ES2653852T3 (es) * | 2007-08-03 | 2018-02-09 | Richter Gedeon Nyrt. | Composiciones farmacéuticas que contienen ligandos del receptor de dopamina y procedimientos de tratamiento usando ligandos del receptor de dopamina |
| CA2715760C (en) | 2008-02-21 | 2017-06-13 | Mitsubishi Tanabe Pharma Corporation | Solid preparation for oral administration of cariprazine hydrochloride |
| AU2009270823B2 (en) | 2008-07-16 | 2014-07-17 | Richter Gedeon Nyrt. | Pharmaceutical formulations containing dopamine receptor ligands |
| MX2016010213A (es) * | 2014-02-07 | 2017-04-13 | Auspex Pharmaceuticals Inc | Formulaciones farmaceuticas novedosas. |
| CN106692149A (zh) * | 2015-11-13 | 2017-05-24 | 天津市汉康医药生物技术有限公司 | 一种卡利拉嗪药物口服制剂及其制备方法 |
-
2017
- 2017-06-13 HU HUP1700253 patent/HUP1700253A1/hu unknown
-
2018
- 2018-05-30 TW TW107118464A patent/TW201906608A/zh unknown
- 2018-06-12 EA EA202090029A patent/EA202090029A1/ru unknown
- 2018-06-12 CA CA3064694A patent/CA3064694A1/en not_active Abandoned
- 2018-06-12 AR ARP180101591A patent/AR112137A1/es unknown
- 2018-06-12 PE PE2019002491A patent/PE20200334A1/es unknown
- 2018-06-12 AU AU2018284138A patent/AU2018284138A1/en not_active Abandoned
- 2018-06-12 KR KR1020207001040A patent/KR20200016378A/ko not_active Ceased
- 2018-06-12 MX MX2019015206A patent/MX2019015206A/es unknown
- 2018-06-12 JP JP2019568138A patent/JP2020523335A/ja active Pending
- 2018-06-12 WO PCT/IB2018/054227 patent/WO2018229641A1/en not_active Ceased
- 2018-06-12 EP EP18734306.6A patent/EP3638210A1/en not_active Withdrawn
- 2018-06-12 CN CN201880040070.6A patent/CN110769815A/zh active Pending
- 2018-06-12 US US16/622,020 patent/US20200222391A1/en not_active Abandoned
- 2018-06-12 BR BR112019025214-2A patent/BR112019025214A2/pt not_active Application Discontinuation
-
2019
- 2019-11-15 PH PH12019502566A patent/PH12019502566A1/en unknown
- 2019-12-02 IL IL271108A patent/IL271108A/en unknown
- 2019-12-11 CL CL2019003619A patent/CL2019003619A1/es unknown
- 2019-12-18 ZA ZA2019/08454A patent/ZA201908454B/en unknown
-
2020
- 2020-01-09 CO CONC2020/0000168A patent/CO2020000168A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA201908454B (en) | 2021-10-27 |
| BR112019025214A2 (pt) | 2020-06-16 |
| AU2018284138A1 (en) | 2020-01-16 |
| MX2019015206A (es) | 2020-02-10 |
| JP2020523335A (ja) | 2020-08-06 |
| CO2020000168A2 (es) | 2021-06-21 |
| EP3638210A1 (en) | 2020-04-22 |
| PH12019502566A1 (en) | 2020-07-20 |
| CN110769815A (zh) | 2020-02-07 |
| US20200222391A1 (en) | 2020-07-16 |
| CL2019003619A1 (es) | 2020-05-15 |
| EA202090029A1 (ru) | 2020-03-26 |
| HUP1700253A1 (hu) | 2019-01-28 |
| KR20200016378A (ko) | 2020-02-14 |
| AR112137A1 (es) | 2019-09-25 |
| CA3064694A1 (en) | 2018-12-20 |
| WO2018229641A1 (en) | 2018-12-20 |
| IL271108A (en) | 2020-01-30 |
| PE20200334A1 (es) | 2020-02-14 |
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