TW201032818A - Novel vancomycin-aminoquinoline hybrid molecules their preparation and their application in therapeutics - Google Patents

Novel vancomycin-aminoquinoline hybrid molecules their preparation and their application in therapeutics Download PDF

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Publication number
TW201032818A
TW201032818A TW099103381A TW99103381A TW201032818A TW 201032818 A TW201032818 A TW 201032818A TW 099103381 A TW099103381 A TW 099103381A TW 99103381 A TW99103381 A TW 99103381A TW 201032818 A TW201032818 A TW 201032818A
Authority
TW
Taiwan
Prior art keywords
group
unsubstituted
vancomycin
formula
butyl
Prior art date
Application number
TW099103381A
Other languages
English (en)
Chinese (zh)
Inventor
Muriel Sanchez
Bernard Meunier
Original Assignee
Palumed Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Palumed Sa filed Critical Palumed Sa
Publication of TW201032818A publication Critical patent/TW201032818A/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
TW099103381A 2009-02-06 2010-02-04 Novel vancomycin-aminoquinoline hybrid molecules their preparation and their application in therapeutics TW201032818A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR0950753A FR2941955A1 (fr) 2009-02-06 2009-02-06 Nouvelles molecules hybrides vancomycine-aminoquinoleine denommees " vancomyquines", leur preparation et leur application en therapeutique
US15507009P 2009-02-24 2009-02-24
FR0952912A FR2941956A1 (fr) 2009-02-06 2009-04-30 NOUVELLES MOLECULES HYBRIDES VANCOMYCINE-AMINOQUINOLEINE DENOMMEES "VANCOMYQUINESr", LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
US17524909P 2009-05-04 2009-05-04

Publications (1)

Publication Number Publication Date
TW201032818A true TW201032818A (en) 2010-09-16

Family

ID=40999941

Family Applications (1)

Application Number Title Priority Date Filing Date
TW099103381A TW201032818A (en) 2009-02-06 2010-02-04 Novel vancomycin-aminoquinoline hybrid molecules their preparation and their application in therapeutics

Country Status (5)

Country Link
AR (1) AR075690A1 (fr)
FR (2) FR2941955A1 (fr)
TW (1) TW201032818A (fr)
UY (1) UY32418A (fr)
WO (1) WO2010089341A1 (fr)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2874922A1 (fr) 2004-07-30 2006-03-10 Palumed Sa Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien
WO2006024741A2 (fr) * 2004-07-30 2006-03-09 Palumed S.A. Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien

Also Published As

Publication number Publication date
FR2941956A1 (fr) 2010-08-13
FR2941955A1 (fr) 2010-08-13
UY32418A (es) 2010-03-26
WO2010089341A1 (fr) 2010-08-12
AR075690A1 (es) 2011-04-20

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