TR200402307T2 - Beta-3 Adrenerjik reseptör agonistleri olarak aminoalkol türevleri. - Google Patents

Beta-3 Adrenerjik reseptör agonistleri olarak aminoalkol türevleri.

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Publication number
TR200402307T2
TR200402307T2 TR2004/02307T TR200402307T TR200402307T2 TR 200402307 T2 TR200402307 T2 TR 200402307T2 TR 2004/02307 T TR2004/02307 T TR 2004/02307T TR 200402307 T TR200402307 T TR 200402307T TR 200402307 T2 TR200402307 T2 TR 200402307T2
Authority
TR
Turkey
Prior art keywords
compound
beta
receptor agonists
adrenergic receptor
hydrogen
Prior art date
Application number
TR2004/02307T
Other languages
English (en)
Inventor
Hattori Kouji
Nakajima Yutaka
Imanishi Masashi
Tomishima Yasuyo
Original Assignee
Fujisawa Pharmaceutical Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AUPS1104A external-priority patent/AUPS110402A0/en
Priority claimed from AU2003900127A external-priority patent/AU2003900127A0/en
Application filed by Fujisawa Pharmaceutical Co., Ltd. filed Critical Fujisawa Pharmaceutical Co., Ltd.
Publication of TR200402307T2 publication Critical patent/TR200402307T2/tr

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    • C07C215/28—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
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Abstract

Mevcut buluş, R1 ve R5'ten her birinin bağımsız şekilde hidrojen, halojen, alt alkil, vb., R2'nin hidrojen veya amino koruyucu bir grup; x'in bir bağ, -o-o, -O-CH2, vb.; y'nin, Z'nin bağ, -O-(CH2)m- (ki buradaki m, 1 ila 4 arasındadır), vb. olduğu bir bileşik; R3'ün alt alkonil, karboksi, alt alkoksikarbonil, vb., ve R4'ün hidrojen, halojen, hidroksi, fenoksi, alt alkil, alt alkoksi, vb., ve n'nin 0,1 veya 2 olduğu bir formül[I] bileşiği veya bunun bir tuzu ile ilgilidir. Mevcut buluşa ait bileşik[I] ve bunun farmasötik açıdan kabul gören tuzları, polakiüri ve idrar tutamama hastalığının profilaktik ve/veya terapötik tedavisinde faydalıdır. Formül (I)
TR2004/02307T 2002-03-14 2003-03-10 Beta-3 Adrenerjik reseptör agonistleri olarak aminoalkol türevleri. TR200402307T2 (tr)

Applications Claiming Priority (3)

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AUPS1104A AUPS110402A0 (en) 2002-03-14 2002-03-14 Aminoalcohol derivatives
AU2003900127A AU2003900127A0 (en) 2003-01-10 2003-01-10 Aminoalcohol derivatives
PCT/JP2003/002821 WO2003076397A1 (en) 2002-03-14 2003-03-10 Aminoalcohol derivatives as beta-3 adrenergic receptor agonists

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TR200402307T2 true TR200402307T2 (tr) 2005-10-21

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EP (1) EP1483236A1 (tr)
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KR (1) KR20040095251A (tr)
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WO2005061433A2 (en) * 2003-12-23 2005-07-07 Astellas Pharma Inc. Aminoalcohol derivatives
US20120196901A1 (en) * 2009-10-29 2012-08-02 Merck Sharp & Dohme Corp. Tertiary amide orexin receptor antagonists

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GB9107827D0 (en) * 1991-04-12 1991-05-29 Fujisawa Pharmaceutical Co New ethanolamine derivatives,processes for the preparation thereof and pharmaceutical composition comprising the same
IL104567A (en) * 1992-02-03 1997-03-18 Fujisawa Pharmaceutical Co Ethanolamine derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same
WO1999051564A1 (en) * 1998-04-06 1999-10-14 Fujisawa Pharmaceutical Co., Ltd. Propanolamine derivatives

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CA2479065A1 (en) 2003-09-18
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TW200306805A (en) 2003-12-01
KR20040095251A (ko) 2004-11-12
NO20043554L (no) 2004-11-15
AR038980A1 (es) 2005-02-02
WO2003076397A1 (en) 2003-09-18
MXPA04008918A (es) 2004-11-26
RU2004130455A (ru) 2006-02-10
CN1653042A (zh) 2005-08-10
EP1483236A1 (en) 2004-12-08
US20050090669A1 (en) 2005-04-28
JP2005519951A (ja) 2005-07-07
BR0308534A (pt) 2005-02-01

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