TH79418A - The ligand of the nicotinic acetylcholine receptor - Google Patents
The ligand of the nicotinic acetylcholine receptorInfo
- Publication number
- TH79418A TH79418A TH401005075A TH0401005075A TH79418A TH 79418 A TH79418 A TH 79418A TH 401005075 A TH401005075 A TH 401005075A TH 0401005075 A TH0401005075 A TH 0401005075A TH 79418 A TH79418 A TH 79418A
- Authority
- TH
- Thailand
- Prior art keywords
- acetylcholine receptor
- methods
- ligand
- nicotinic acetylcholine
- formula
- Prior art date
Links
- 239000003446 ligand Substances 0.000 title abstract 3
- 102000019315 Nicotinic acetylcholine receptors Human genes 0.000 title 1
- 108050006807 Nicotinic acetylcholine receptors Proteins 0.000 title 1
- 239000000126 substance Substances 0.000 claims abstract 5
- 229940079593 drug Drugs 0.000 claims abstract 2
- 239000003814 drug Substances 0.000 claims abstract 2
- 125000001072 heteroaryl group Chemical group 0.000 claims 2
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 1
- 125000003118 aryl group Chemical group 0.000 claims 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 125000004122 cyclic group Chemical group 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 239000001301 oxygen Substances 0.000 claims 1
- 125000004430 oxygen atom Chemical group O* 0.000 claims 1
- 229910052717 sulfur Inorganic materials 0.000 claims 1
- 239000011593 sulfur Substances 0.000 claims 1
- 125000004434 sulfur atom Chemical group 0.000 claims 1
- 238000000034 method Methods 0.000 abstract 4
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 2
- 108010009685 Cholinergic Receptors Proteins 0.000 abstract 2
- 102000034337 acetylcholine receptors Human genes 0.000 abstract 2
- 238000004519 manufacturing process Methods 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
Abstract
DC60 (18/03/48) ลิแกนด์ของตัวรับอะเซทิลโคลีนที่สูตร I (สูตรเคมี) I ที่ซึ่ง D, Ar1, E และ Ar2 เป็นตามที่บรรยายไว้ในรายละเอียด, ไดอะสเตอรีโอเมอร์, อิแนนทิโอเมอร์, เกลือที่สามารถยอมรับได้ทางเภสัชกรรม, วิธีการผลิต, สารผสมทางเภสัชกรรมที่มี และวิธีการใช้สาร เดียวกันเหล่านี้ ลิแกนด์ของตัวรับอะเซทิลโคลีนที่สูตร I (สูตรเคมี) I ที่ซึ่ง D, Ar1, E และ Ar2 เป็นตามที่บรรยายไว้ในรายละเอียด, ไดอะสเตอรีโอเมอร์, อิแนนทิโอเมอร์, เกลือที่สามารถยอมรับได้ทางเภสัชกรรม, วิธีการผลิต, สารผสมทางเภสัชกรรมที่มี และวิธีการใช้สาร เดียวกันเหล่านี้ สิทธิบัตรยาDC60 (18/03/48) Acetylcholine receptor ligands of formula I (chemical formula) I, wherein D, Ar1, E and Ar2 are as described in detail, diastereomers, enantiomers, pharmaceutically acceptable salts, methods of manufacture, pharmaceutical mixtures containing and methods of using these same substances. Acetylcholine receptor ligands of formula I (chemical formula) I, wherein D, Ar1, E and Ar2 are as described in detail, diastereomers, enantiomers, pharmaceutically acceptable salts, methods of manufacture, pharmaceutical mixtures containing and methods of using these same substances. Patented drugs.
Claims (1)
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TH79418A true TH79418A (en) | 2006-08-24 |
Family
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