SK20242000A3 - Salts of paroxetine - Google Patents

Salts of paroxetine Download PDF

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SK20242000A3
SK20242000A3 SK2024-2000A SK20242000A SK20242000A3 SK 20242000 A3 SK20242000 A3 SK 20242000A3 SK 20242000 A SK20242000 A SK 20242000A SK 20242000 A3 SK20242000 A3 SK 20242000A3
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acid
benzoic
carboxylic
methyl
chloro
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SK2024-2000A
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Victor Witold Jacewicz
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Smithkline Beecham Plc
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
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  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Piperidine compounds, processes for preparing them, pharmaceutical compositions comprising them and their use in therapy are disclosed.

Description

Tento vynález sa týka solí paroxetínu, spôsobu ich prípravy a ich použitia pri liečení medicínskych porúch.The present invention relates to paroxetine salts, to a process for their preparation and to their use in the treatment of medical disorders.

Doterajší stav technikyBACKGROUND OF THE INVENTION

Farmaceutické produkty s antidepresívnymi a anti-Parkinsonovskými vlastnosťami sú opísané v US-A-3912743 a US-A-4007196. Zvlášť dôležitou látkou medzi opísanými látkami je paroxetín, (-)ŕrans izomér 4-(4’-fluórfenyl)-3-(3,,4,-metyléndioxy-fenoxymetyl)-piperidínu. Táto látka sa používa v terapii ako hydrochloridová soľ na liečenie a profylaxiu medzi iným depresie, obsedantno-kompulzívnej poruchy (OCD) a paniky.Pharmaceutical products with antidepressant and anti-Parkinsonian properties are described in US-A-3912743 and US-A-4007196. An especially important compound among those disclosed is paroxetine, the (-) trans isomer of 4- (4'-fluorophenyl) -3- (3, 4-methylenedioxy-phenoxymethyl) -piperidine. It is used in therapy as a hydrochloride salt for the treatment and prophylaxis of, inter alia, depression, obsessive-compulsive disorder (OCD) and panic.

Podstata vynálezuSUMMARY OF THE INVENTION

Podstatou vynálezu sú soli paroxetínu, ktoré sa môžu použiť ako alternatíva k bežne dostupnému hydrochloridu, alebo ako medziprodukt pri príprave hydrochloridu.The present invention provides salts of paroxetine, which may be used as an alternative to the commercially available hydrochloride, or as an intermediate in the preparation of the hydrochloride.

Podľa tohto vynálezu sa poskytuje soľ paroxetínu s kyselinou vybranou zo skupiny pozostávajúcej z:According to the present invention there is provided a salt of paroxetine with an acid selected from the group consisting of:

kyselina 2-metyl-3-fenylmaslová kyselina tricyklo(10.2.2.2(4,7))oktadeka-hexaén-9,10-dikarboxylová kyselina 1-pyrénoctová kyselina 2,4,6-trifluórškoricová kyselina 2-brómizomaslová kyselina cyklohexyljantárová kyselina 3,5-dichlór-2,6-dimetoxybenzoová kyselina 5-etoxy-2-hydroxybenzoová kyselina trans-11-eikozénová ·· ·· ···· ·· • · · · · · ··· · · · · ·2-methyl-3-phenylbutyric acid tricyclo (10.2.2.2 (4,7)) octadeca-hexaene-9,10-dicarboxylic acid 1-pyrene-acetic acid 2,4,6-trifluorocinnamic acid 2-bromoisobutyric acid cyclohexylsuccinic acid 3, 5-Dichloro-2,6-dimethoxybenzoic acid 5-ethoxy-2-hydroxybenzoic acid trans-11-eicosenoic acid ··· ················

-2kyselina 3-brómpropiónová kyselina 3-[5-(4-bróm-fenyl)-furán-2yl]-akrylová kyselina 2-fenylakrylová kyselina 21-dokozénová kyselina n-(p-amylcinamoyl)antranilová kyselina (2'-metyl-4,-amino)fenylazonaftylén-3,8-disulfónová kyselina 7,7-dimetyleikozadiénová kyselina 2,5-dibrómbenzénsulfónová kyselina 5,7-eikozadiynová kyselina nonadek-18-énová kyselina 3-metoxycyklohexánkarboxylová kyselina 5-chlór-2-tiofénkarboxylová beta-naftylfosfonát kyselina 2-(1,4-benzodioxán-2-yl)tiazol-4-karboxylová kyselina 2-metyl-1,6-naftyridín-3-karboxylová kyselina (10-ho-10-ph-4h-8-tia-7,10a-diaza-pentaleno( 1,2-a)riaftalén-9-yl)octová kyselina fmoc-izonipekotínová kyselina 4-(3-(2-fluór-5-nitrofenyl)ureido)benzoová kyselina n-etylmaleámová kyselina 7-metoxykumarín-4-octová kyselina ŕrans-4-n-pentylcyklohexánkarboxylová kyselina 2,4-dimetylcinamová kyselina (s)-3-metylpolargonová kyselina 3-maleimidobenzoová kyselina acetoxyvalérová kyselina 7,12-dimetylbenz(a)-antracén-5-karboxylová kyselina 4-chlórftalová kyselina 2-(karboxymetyl-amino)-6-chlórbenzoová kyselina 3'-metoxyftalanilová kyselina 1 -(+)-2-amino-6-fosfonohexánová kyselina (l)-2,3-diacetoxy-n-(1 -(1 -naftyl)etyl)jantárová kyselina 4-fluórfenoxydifluóroctová ·· ·· ···· ·· • · · · · · ··· · · · · · • ··· · · · · ·-2-3-bromopropionic acid 3- [5- (4-bromo-phenyl) -furan-2-yl] -acrylic acid 2-phenylacrylic acid 21-docosenoic acid n- (p-amylcinamoyl) anthranilic acid (2'-methyl-4 , -amino) phenylazonaphthylene-3,8-disulfonic acid 7,7-dimethyleicosadienoic acid 2,5-dibromobenzenesulfonic acid 5,7-eicosadiynic acid nonadec-18-enoic acid 3-methoxycyclohexanecarboxylic acid 5-chloro-2-thiophenecarboxylic acid beta-naphthyl 2- (1,4-benzodioxan-2-yl) thiazole-4-carboxylic acid 2-methyl-1,6-naphthyridine-3-carboxylic acid (10-ho-10-ph-4h-8-thia-7) 10α-Diaza-pentaleno (1,2-athiophthalen-9-yl) acetic acid fmoc-isonipecotinic acid 4- (3- (2-fluoro-5-nitrophenyl) ureido) benzoic acid n-ethylmaleamic acid 7-methoxycoumarin 4-acetic acid trans-4-n-pentylcyclohexanecarboxylic acid 2,4-dimethylcinnamic acid (s) -3-methylpolargonic acid 3-maleimidobenzoic acid acetoxyvaleric acid 7,12-dimethy 1-Benz (a) -anthracene-5-carboxylic acid 4-chlorophthalic acid 2- (carboxymethyl-amino) -6-chlorobenzoic acid 3'-methoxyphthalanic acid 1- (+) - 2-amino-6-phosphonohexanoic acid (1) - 2,3-diacetoxy-n- (1- (1-naphthyl) ethyl) succinic acid 4-fluorophenoxydifluoroacetic acid ··· ··· ··· ··· · · · · · · · · · · · ·

-3kyselina 3-(2-chlór-6-fluórfenyl)-5-metylizoxazol-4-karboxylová kyselina 3-(4-(2-karboxyetyl)-2,5-dimetoxyfenyl)propiónová kyselina 6-(6-hydroxy-3-oxo-3h-xantén-9-yl)-3-cyklohexén-1-karboxylová kyselina c/s-n-ŕerc-butylhexahydroftalámová kyselina 2,5-dihydroxyškoricová kyselina 3-bróm-2-(brómmetyl)propiónová kyselina 3-etyl-3-fenylglutárová kyselina alfa-(214-dimetoxy-6-metylbenzylidén)hipurová kyselina 5-fenylvalérová kyselina (+/-)-2-amino-3-[3-(karboxymetoxy)-5-metyl-izoxazol-4-yl]propiónová kyselina 4-aminonikotínová kyselina p-fluór-alfa-acetamidoškoricová kyselina 2,5-dihydroxybenzoová kyselina 10-( 1 -pyrén)-10-ketodekánová kyselina 2-chlór-3,5-dinitrobenzoová kyselina p-azoxybenzoová kyselina 2-etyltio-2,2-difenyloctová kyselina 4-(3-cinamoyl-2-tioureido)benzoová kyselina 2-hydroxydibenzofurán-3-karboxylová kyselina 2-(3,5-dinitro-tiofén-2-ylamino)-pentánová kyselina 2-benzoylamino-cyklohexánkarboxylová kyselina 3-hydroxyhomoftálová kyselina 2,5-dibrómbenzoová kyselina 4-(2-chlór-2-kyanoetyl)-benzoová kyselina 2-metylhydroškoricová kyselina 1,3-metylpentadekánová kyselina 3,4,5-trimetoxyfenyloctová kyselina dl-2-hydroxy-4-(metyltio)maslová kyselina 2-oxoadipová kyselina brómoctová kyselina 1-(4-izopropyl-3-metyl-fenyl)-5-oxo-pyrolidín-3-karboxylová kyselina perfluórazelaínová • 88 ·· ···· 88 ·· · · · · ·-3- (2-chloro-6-fluorophenyl) -5-methylisoxazole-4-carboxylic acid 3- (4- (2-carboxyethyl) -2,5-dimethoxyphenyl) propionic acid 6- (6-hydroxy-3- oxo-3h-xanthen-9-yl) -3-cyclohexene-1-carboxylic acid cis-tert-butylhexahydrophthalic acid 2,5-dihydroxycinnamic acid 3-bromo-2- (bromomethyl) propionic acid 3-ethyl-3- phenylglutaric acid alpha- (2 1 4-dimethoxy-6-methylbenzylidene) hippuric acid 5-phenylvaleric acid (+/-) - 2-amino-3- [3- (carboxymethoxy) -5-methyl-isoxazol-4-yl] propionic acid 4-aminonicotinic acid p-fluoro-alpha-acetamido cinnamic acid 2,5-dihydroxybenzoic acid 10- (1-pyrene) -10-ketodecanoic acid 2-chloro-3,5-dinitrobenzoic acid p-azoxybenzoic acid 2-ethylthio- 2,2-Diphenylacetic acid 4- (3-cinamoyl-2-thioureido) benzoic acid 2-hydroxydibenzofuran-3-carboxylic acid 2- (3,5-dinitro-thiophen-2-ylamino) -pentanoic acid 2-benzoylamino-cyclohexanecarboxylic acid 3-hydroxyhomophthaic acid 2,5-dibromobenzoic acid 4- (2-chloro-2-cyanoethyl) -benzoic acid 2-methylhydrocinnamic acid 1,3-methylpentadecanoic acid 3,4,5-trimethoxyphenylacetic acid dl-2-hydroxy-4- (methylthio) ) butyric acid 2-oxoadipic acid bromoacetic acid 1- (4-isopropyl-3-methylphenyl) -5-oxo-pyrrolidine-3-carboxylic acid perfluoroazelaic acid • 88 ·· ···· 88 ·· · · · · ·

888 8 · · · · • g 8 8888 88 8888 8 g 8 8888 88 8

888 88 88 88 88 888888 88 88 88 88 888

-4kyselina acetylsyringová kyselina 3’-acetylftalanilová kyselina alfa-brómfenyloctová kyselina 3-(3,4-diacetoxy-5-metyl-fenyl)-akrylová kyselina jódškoricová kyselina 4,4'-metylénbis(maleanilová) kyselina 3-(4-trifluórmetylsulfanyl-fenylkarbamoyl)-akrylová kyselina 3-[2-(pyrazín-2-yl)-1-[4-(trifluórmetyl)fenyl)etoxy]propánová kyselina 2-fenoxymaslová kyselina 2-[4-chlór(fenylsulfonyl)anilíno]octová kyselina boc-d/-beta-aminomaslová kyselina 3,5-dinitrobenzoová kyselina 4-íerc-butylcyklohexánkarboxylová kyselina (r)-2,2-dimetyl-3-formyl-4-tiazolidínkarboxylová kyselina (2s,4s)-(-)-azetidin-2,4-dikarboxylová kyselina 2-(4-nitro-fenyl)-3-fenyl-akrylová kyselina 3-nitrobenzoová kyselina 10,11-dihydro-dibenzo(b,f)oxepín-4,6-dikarboxylová kyselina (2-izopropyl-5-oxo-cyklohexyloxy)-octová kyseliny (s)-(-)-n-( 1 -fenyletyl)sukcínamová kyselina 6-(2-brómbenzoyl)hexánová kyselina (1alfa,3alfa,5beta)-1,3,5-trimetyl-1,3,5-cyklohexántrikarboxylová kyselina 2-metylpropántrikarboxylová kyselina 5-(4-hydroxymetyl-3-metoxyfenoxy)valérová kyselina n-(3,4-dikyano-fenyl)-ftalámová kyselina 5-fluórsalicylová kyselina itakónová kyselina 2,2-dimetyl-cyklobután-1,1,3,3-tetrakarboxylová kyselina 8-hydroxy-5-(4-sulfofenylazo)-2-naftalénsulfónová kyselina 3-(4-chlórfenyltio)maslová kyselina 1-benzylglutáramová kyselina 3-(2,5-dimetoxybenzoyl)propiónová-4-acetylsyringic acid 3'-acetylphthalanilic acid alpha-bromophenylacetic acid 3- (3,4-diacetoxy-5-methylphenyl) -acrylic acid iodicinic acid 4,4'-methylenebis (maleanilic acid) 3- (4-trifluoromethylsulfanyl- phenylcarbamoyl) acrylic acid 3- [2- (pyrazin-2-yl) -1- [4- (trifluoromethyl) phenyl] ethoxy] propanoic acid 2-phenoxybutyric acid 2- [4-chloro (phenylsulfonyl) anilino] acetic acid boc (R) -2,2-dimethyl-3-formyl-4-thiazolidinecarboxylic acid (2s, 4s) - (-) - azetidine- (N) -beta-aminobutyric acid 3,5-dinitrobenzoic acid 4-tert-butylcyclohexanecarboxylic acid 2,4-dicarboxylic acid 2- (4-nitro-phenyl) -3-phenyl-acrylic acid 3-nitrobenzoic acid 10,11-dihydro-dibenzo (b, f) oxepine-4,6-dicarboxylic acid (2-isopropyl -5-oxo-cyclohexyloxy) -acetic acid (s) - (-) - n- (1-phenylethyl) succinamic acid 6- (2-bromobenzoyl) hexanoic acid (1alpha, 3alpha, 5beta) -1,3,5- trimethyl-1,3,5-cyclohexanetricarboxylic acid 2-methylpropanetricarboxylic acid 5- (4-hydroxymethyl-3-methoxyphenoxy) valeric acid n- (3,4-dicyano-phenyl) -phthalic acid 5-fluoroalicylic acid itaconic acid 2,2-dimethyl-cyclobutane-1,1,3 3-tetracarboxylic acid 8-hydroxy-5- (4-sulfophenylazo) -2-naphthalenesulfonic acid 3- (4-chlorophenylthio) butyric acid 1-benzylglutaramic acid 3- (2,5-dimethoxybenzoyl) propionic acid

-5·· ···· kyselina 4-kyanoškoricová kyselina 2-(4-metoxy-fenyl)-1,3-dioxo-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina 2-hydroxyamino-pentándiová kyselina 6-metyl-1,3-benzodioxol-5-karboxylová kyselina 2-(4-hydroxyfenoxy Jpropiónová kyselina 7h-dodekafluórheptánová kyselina S'.S'-dimetylmaleanilová kyselina 2-butyl-5-ŕerc-butyl-izoftalová kyselina 4-chlór-2-ftalimidobenzoová kyselina 2-metyl-1,3-ditiolán-2-propiónová kyselina 4-chlór-2-nitrofenol-6-sulfónová kyselina n-metyl-1-glutámová kyselina 4,6,2’,4’-tetranitro-bifenyl-2-karboxylová kyselina (r)-(-)-2-amino-2-metylbutándiová kyselina 3-[2-(4-ŕerc-butylfenoxy)-5-nitrofenyl-akrylová kyselina 4-(trifluórmetyltio)fenyloctová kyselina ditiodiglykolová kyselina n,n-bis-(fosfonometyl)-glycín kyselina 3-( 10-(2-karboxy-etyl)-antracén-9-yl)-propiónová kyselina hydroškoricová kyselina 3,6-dichlór-5-hydroxy-o-anýzová kyselina 3,5-difluórfenyloctová kyselina 2,-(trifluórmetyl)sukcínanilová kyselina c/s-5,8,11,14,17-eikozapenténová kyselina 3,3'-(dimetylsilylén)bispropiónová kyselina 1-(3-chlór-5-trifluórmetyl-2-pyridyl)pyrol-2-karboxylová kyselina n-(4,6-dimetylpyrimidín-2-yl)-4-aminobenzoová kyselina 10,12-dokozadiíndiová kyselina 6,6-dimetyl-3-(metyltio)-4,5,6,7-tetrahydrobenzo[c]tiofén-4-ón-1-karboxylová kyselina gentisurová kyselina 2-fluór-4-heptyloxybenzoová ·· ···· • ·· · · · · · · · ··· ·· ·· ·· ·· ···-5 ·· ···· 4-Cyano cinnamic acid 2- (4-methoxyphenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid 2-hydroxyamino-pentanedioic acid 6-methyl-1,3-benzodioxole-5-carboxylic acid 2- (4-hydroxyphenoxy) propionic acid 7h-dodecafluoroheptanoic acid S'S'-dimethylmaleanilic acid 2-butyl-5-tert-butyl-isophthalic acid 4-chloro- 2-phthalimidobenzoic acid 2-methyl-1,3-dithiolane-2-propionic acid 4-chloro-2-nitrophenol-6-sulfonic acid n-methyl-1-glutamic acid 4,6,2 ', 4'-tetranitro- (r) - (-) - 2-Amino-2-methylbutanedioic acid biphenyl-2-carboxylic acid 3- [2- (4-tert-butylphenoxy) -5-nitrophenyl acrylic acid 4- (trifluoromethylthio) phenylacetic acid dithiodiglycolic acid n, n-bis- (phosphonomethyl) -glycine 3- (10- (2-carboxy-ethyl) -anthracen-9-yl) -propionic acid cinnamic acid 3,6-dichloro-5-hydroxy-o-anisic acid 3,5-Difluorophenylacetic acid 2 , - (trifluoromethyl) succinilo cis-5,8,11,14,17-eicosapentenoic acid 3,3 '- (dimethylsilylene) bispropionic acid 1- (3-chloro-5-trifluoromethyl-2-pyridyl) pyrrole-2-carboxylic acid n - (4,6-Dimethylpyrimidin-2-yl) -4-aminobenzoic acid 10,12-docosadinedioic acid 6,6-dimethyl-3- (methylthio) -4,5,6,7-tetrahydrobenzo [c] thiophene-4 -one-1-carboxylic acid gentisuric acid 2-fluoro-4-heptyloxybenzoic acid ···················

-6kyselina 2-(4-chlór-3-nitrobenzoyl)benzoová kyselina 3-(4-bróm-2-tienyl)akrylová kyselina 3,5-dimetoxyškoricová kyselina 3-((2-karboxy-etyl)-(1,3,4)tiadiazol-2-yl-amino)-propiónová kyselina 4-sulfo-antranilová kyselina d-pyroglutámová kyselina (2,5-xylyl)fosfónová kyselina 3-bróm-5-metoxy-benzo(b)tiofén-2-karboxylová kyselina 4,515,6,6,6-hexafluór-4-(trifluórmetyl)-2-hexénová kyselina 2,3-difluórfenyloctová kyselina 3,3,3 -trifluór-d/-mliečna kyselina 3-[4-(4-metylfenyltio)-3-nitrofenyl)akrylová kyselina 2,8-dimetoxy-dodekahydro-dibenzofurán-1 -karboxylová kyselina 4-cyklohexylbenzoová kyselina boc-d-1,2,3,4-tetrahydronorharmán-3-karboxylová kyselina 2-benzyl-cyklohexánkarboxylová kyselina 3-[(4-fliiór-fenyl)-(toluén-4-sulfonyl)-amino]-propiónová kyselina 3-(2,4,5-trimetyl-fenyl)-maslová kyselina 4-(1,3-dioxo-1,3-dihydro-izoindol-2-yl)-maslová kyselina chelidamová kyselina 4-(4-(1-metyl-1h-chinolín-4-ylidén)-but-2-enylidénamino)-benzoová kyselina 8-karbamoylnaftalén-1 -karboxylová kyselina n-(m-tolyl)sukcínamová kyselina n-(1-naftyl)ftalámová kyselina 3-(3,4-dihydro-naftalén-1 -yl)-propiónová kyselina 4-(2-fenylsulfanyl-acetylamino)-benzoová kyselina perfluórheptánová kyselina 4'-chlór-2'-metylftalanilová kyselina dietylfosfonopentánová kyselina 2-(3-metoxy-benzylidén)-pentándiová kyselina 4,4'-bifenyldikarboxylová kyselina 18-metylnonadekánová-6- 2- (4-chloro-3-nitrobenzoyl) benzoic acid 3- (4-bromo-2-thienyl) acrylic acid 3,5-dimethoxycinnamic acid 3 - ((2-carboxyethyl) - (1,3, 4) thiadiazol-2-yl-amino) -propionic acid 4-sulfo-anthranilic acid d-pyroglutamic acid (2,5-xylyl) phosphonic acid 3-bromo-5-methoxy-benzo (b) thiophene-2-carboxylic acid 4,5 1 5,6,6,6-hexafluoro-4- (trifluoromethyl) -2-hexenoic acid 2,3-difluorophenylacetic acid 3,3,3-trifluoro-d-lactic acid 3- [4- (4 -methylphenylthio) -3-nitrophenyl) acrylic acid 2,8-dimethoxy-dodecahydro-dibenzofuran-1-carboxylic acid 4-cyclohexylbenzoic acid boc-d-1,2,3,4-tetrahydronorharman-3-carboxylic acid 2-benzyl- 3 - [(4-Fluoro-phenyl) - (toluene-4-sulfonyl) -amino] -propionic acid cyclohexanecarboxylic acid 3- (2,4,5-trimethyl-phenyl) -butyric acid 4- (1,3-dioxo) -1,3-dihydro-isoindol-2-yl) butyric acid chelidamic acid 4- (4- (1-methyl-1H-quinolin-4-ylidene) -but-2-enylidenamino) -benzoic acid 8-carbamoylnaphthalene-1-carboxylic acid n- (m-tolyl) succinamic acid n- (1-naphthyl) phthalic acid 3- (3,4-dihydro-naphthalen-1-yl) -propionic acid 4- (2- phenylsulfanyl-acetylamino) -benzoic acid perfluoroheptanoic acid 4'-chloro-2'-methylphthalanilic acid diethylphosphonopentanoic acid 2- (3-methoxybenzylidene) -pentanedioic acid 4,4'-biphenyldicarboxylic acid 18-methylnonadecanoic acid

• ·· • · • BBB B B · • ·· • · • BBB B B · •B BBB· • B B • · 0 • · · B • BBB · • B B • · 0 • · · B • B B B • · • B B • B B B • · • B B B · B · ·· e· ·· e · • B ·♦ • B · ♦ • B • B • B • B

kyselina 4,-(n-metylacetamido)glutaranilová kyselina (+)-3-metyladipová kyselina 2-bróm-3-metoxytiofén-4-karboxylová kyselina (5-(4-chlór-fenyl)-pyrimidín-4-ylsulfanyl)-octová kyselina glycyl-d-asparágová kyselina 3-(/7-(3,4-dichlórfenyl)karbamoyl)-5-norbornén-2-karboxylová kyselina n-(3-bróm-2,4,6-trimetylfenylkarbamoylmetyl)iminodioctová kyselina 1,2,3,4,5,6-cyklohexánhexakarboxylová kyselina alfa-(fenyltio)fenyloctová kyselina geraniová kyselina 5-hydroxy-2-(1 -oktynyl)-3-oxo-1 -cyklopentén-1 -heptánová kyselina n-fmoc-2-aminoindan-2-karboxylová kyselina 3-(9,10-dioxo-9,10-dihydro-antracén-2-yl)-akrylová kyselina p-tolyloctová kyselina 4-(4-(4-tolyl)butyl)fenyloctová kyselina 2-metylcyklopropánkarboxylová kyselina 4-chlór-alfa,alfa-dimetylfenyloctová kyselina (2,4-dichlór-5-metylfenyltio)octová kyselina 3-(3,4-dichlórbenzyltio)tiofén-2-karboxylová kyselina (-)-3-metyl-2-fenylmaslová kyselina 3-cyklopenténkarboxylová kyselina n-tris(hydroxymetyl)metyl-2-amino-etánsulfónová kyselina (s)-5-oxotetrahydrofurán-2-karboxylová kyselina 5-benzoyltiofén-2-octová kyselina p-toluénsulfónová kyselina 3,6-dimetyl-cyklohex-4-én-1,2-dikarboxylová kyselina 3-(2-chlórfenyl)-5-metylizoxazol-4-karboxylová kyselina 1 -(4-acetylfenyl)izonipekotínová kyselina fenyl-o-tolyl-fosfinová kyselina 2-(1-(2-(3,4-dimetoxy-fenyl)-etyl)-5-etyl-2-oxo-piperidín-4-yl)-malónová kyselina n-(4-metoxyfenyl)malónová kyselina (+)-3-pinánkarboxylováacid 4 '- (N-methylacetamide) glutaranilová acid, (+) - 3-methyladipic acid 2-bromo-3-methoxy-thiophene-4-carboxylic acid (5- (4-chloro-phenyl) -pyrimidin-4-ylsulfanyl) -acetic acid glycyl-d-aspartic acid 3 - ([7- (3,4-dichlorophenyl) carbamoyl) -5-norbornene-2-carboxylic acid n- (3-bromo-2,4,6-trimethylphenylcarbamoylmethyl) iminodiacetic acid 1, 2,3,4,5,6-cyclohexanehexacarboxylic acid alpha- (phenylthio) phenylacetic acid geraniic acid 5-hydroxy-2- (1-octynyl) -3-oxo-1-cyclopentene-1-heptanoic acid n-fmoc-2 amino-indan-2-carboxylic acid 3- (9,10-dioxo-9,10-dihydro-anthracen-2-yl) -acrylic acid p-tolylacetic acid 4- (4- (4-tolyl) butyl) phenylacetic acid 2 4-chloro-alpha, alpha-dimethylphenylacetic acid (2,4-dichloro-5-methylphenylthio) acetic acid 3- (3,4-dichlorobenzylthio) thiophene-2-carboxylic acid (-) - 3-methyl-2-methylcyclopropanecarboxylic acid Phenylbutyric acid 3-cyclopentenecarboxylic acid n-tris (hydroxymet yl) methyl-2-amino-ethanesulfonic acid (s) -5-oxotetrahydrofuran-2-carboxylic acid 5-benzoylthiophene-2-acetic acid p-toluenesulfonic acid 3,6-dimethyl-cyclohex-4-ene-1,2- 3- (2-chlorophenyl) -5-methylisoxazole-4-carboxylic acid dicarboxylic acid 1- (4-acetylphenyl) isonipecotinic acid phenyl-o-tolylphosphinic acid 2- (1- (2- (3,4-dimethoxy- phenyl) -ethyl) -5-ethyl-2-oxo-piperidin-4-yl) malonic acid n- (4-methoxyphenyl) malonic acid (+) - 3-pinanecarboxylic acid

• ·· • · Φ ··· • ·· • · Φ ··· ·· · · • · · · • • • · · · • • ·· · · ·· · · • • • • • • • • • • • • • • • • • · · • · · • · • · ·· ·· ·· ·· ·· · · ·· · · ·· · · • · • ·

kyselina 2-(2,4,5-trichlórfenoxy)-propiónová kyselina 10-hydroxydekánová kyselina 5-(3-chlór-fenyl)-pentánová kyselina 4-[[4-[(dimetylpyrimidín-2-yl)tio]fenyl]amino]-4-oxo-(2z)-buténová kyselina 2-acetamido-3-(4’-chlórfenyl)-akrylová kyselina 2-hydroxy-6-[3-(trifluórmetyl)fenyl)-3,5-pyridíndikarboxylová kyselina 9-hydroxylimino-9h-fluorén-4-karboxylová kyselina mukochlorečná kyselina 4-metyl-1-naftoová kyselina 2-naftyl-akrylová kyselina 4-hexyl-cyklohexánkarboxylová kyselina 4-(3,5-dimetyl-naftalén-2-yl)-3-metyl-pentánová kyselina n,n,n’,n-etyléndiamíntetra(metylénfosfónová) kyselina 6-heptínová kyselina 2-(4-metoxybenzylidén)jantárová kyselina (r)-(+)-2-chlórpentánová kyselina 2-(3-chlór-4-metoxy-fenylamino)-benzoová kyselina 3,5-bis(trifluórmetyl)škoricová kyselina 4-hexyloxybifenyl-4'-karboxylová kyselina (+/-)-10-gáforsulfónová kyselina 4,4'-oxybisbutánová kyselina 2-metyldekánová kyselina 4-bifenylkarboxylová kyselina 3-chlór-n-maslová kyselina 3-antracén-2-yl-akrylová kyselina (s,s)-(+)-2,3-difenyljantárová kyselina 10-metyldodekánová kyselina 4'-fluórsukcínanilová kyselina 2-bróm-3-metylbenzoová kyselina n-(4-trifluórmetoxyfenyl)malonámová kyselina 3-(2-tienyl)akrylová kyselina 3-(3-metoxyfenoxy)propiónová ·· ·· ···· ·· • · · · · · · ··· * · · · ·2- (2,4,5-Trichlorophenoxy) -propionic acid 10-Hydroxydecanoic acid 5- (3-chloro-phenyl) -pentanoic acid 4 - [[4 - [(dimethylpyrimidin-2-yl) thio] phenyl] amino 4-Oxo- (2z) -butenoic acid 2-Acetamido-3- (4'-chlorophenyl) -acrylic acid 2-hydroxy-6- [3- (trifluoromethyl) phenyl) -3,5-pyridinedicarboxylic acid 9- hydroxylimino-9h-fluorene-4-carboxylic acid mucochloric acid 4-methyl-1-naphthoic acid 2-naphthyl-acrylic acid 4-hexyl-cyclohexanecarboxylic acid 4- (3,5-dimethyl-naphthalen-2-yl) -3- methylpentanoic acid n, n, n ', n-ethylenediaminetetra (methylenephosphonic acid) 6-heptic acid 2- (4-methoxybenzylidene) succinic acid (r) - (+) - 2-chloropentanoic acid 2- (3-chloro- 4-methoxy-phenylamino) -benzoic acid 3,5-bis (trifluoromethyl) cinnamic acid 4-hexyloxybiphenyl-4'-carboxylic acid (+/-) - 10-camphorsulfonic acid 4,4'-oxybisbutanoic acid 2-methyldecanoic acid 4 -biphenylcarboxylic acid 3-ch lor-n-butyric acid 3-anthracen-2-yl-acrylic acid (s, s) - (+) - 2,3-diphenylsuccinic acid 10-methyldodecanoic acid 4'-fluorosuccinic acid 2-bromo-3-methylbenzoic acid n - (4-Trifluoromethoxyphenyl) malonamic acid 3- (2-thienyl) acrylic acid 3- (3-methoxyphenoxy) propionic acid · · · · · · · · · ·

-9kyselina 2,3,6-trifluórškoricová kyselina 3-chlóradamantán-1 -karboxylová kyselina 2,5-dichlór-alfa-metyl-3-tiofénakrylová kyselina 2-ho-10-metánsulfonyl-9-oxa-tricyklo(6.2.1.0(1,5))undekán-4-karboxylová kyselina 2,2-dichlóroktánová kyselina 7-chlór-6-f I uór-1 -etyl-4-oxochinolín-3-karboxylová kyselina acetoxy-dekánová kyselina 5-brómvalérová kyselina mezo-2,3-bis(benzylamino)jantárová kyselina 3,6-dimetyl-4,5-difenyl-cyklohexa-3,5-dién-1,2-dikarboxylová kyselina dodekafluór-2-metyl-3-oxahexánová kyselina d/-2-(4-metoxyfenyl)maslová kyselina 3-(n,n-dietylkarbamoyl)-5-norbôrnén-2-karboxylová o-karboxyfenylfosfát kyselina n-boc-2-aminoindán-2-karboxylová kyselina 9-hydroxynonánová kyselina 3-(2,5-dimetoxy-fenyl)-propiónová kyselina 4-((2-hydroxy-3-nitro-benzylidén)-amino)-benzoová kyselina fmoc-10-aminodekánová kyselina tiofén-2,5-dikarboxylová kyselina 2-brómfenyloctová kyselina 3-(3,4-metyléndioxyfenyl)propiónová kyselina (z)-styrylsulfonylpropiónová kyselina 2'-karboxymaleanilová kyselina gama-oxo-1 -naftalénmaslová kyselina 11 -((5-dimetylaminonaftalén-1 -sulfonyl)amino)undekánová kyselina 2-[[(4-chlórfenyl)sulfonyl]-3-(trifluórmetyl)anilíno]octová kyselina 2-nonénová kyselina 2-formylfenoxyoctová kyselina 2,4-pyridíndikarboxylová kyselina 2-fluór-6-(trifluórmetyl)fenyloctová kyselina acenaftén-3-karboxylová-9-2,3,6-Trifluoric cinnamic acid 3-chloro-adamantane-1-carboxylic acid 2,5-dichloro-alpha-methyl-3-thiophenacrylic acid 2-ho-10-methanesulfonyl-9-oxa-tricyclo (6.2.1.0 ( 1,5)) undecane-4-carboxylic acid 2,2-dichlorooctanoic acid 7-chloro-6-fluoro-1-ethyl-4-oxoquinoline-3-carboxylic acid acetoxy decanoic acid 5-bromovaleric acid meso-2 3-bis (benzylamino) succinic acid 3,6-dimethyl-4,5-diphenyl-cyclohexa-3,5-diene-1,2-dicarboxylic acid dodecafluoro-2-methyl-3-oxahexanoic acid d / -2- (4-Methoxyphenyl) butyric acid 3- (n, n-Diethylcarbamoyl) -5-norbornene-2-carboxylic o-Carboxyphenyl phosphate n-boc-2-aminoindan-2-carboxylic acid 9-hydroxynonanoic acid 3- (2,5 -dimethoxy-phenyl) -propionic acid 4 - ((2-hydroxy-3-nitro-benzylidene) -amino) -benzoic acid fmoc-10-aminodecanoic acid thiophene-2,5-dicarboxylic acid 2-bromophenylacetic acid 3- (3 (4-methylenedioxyphenyl) propionic acid (z) -styr ylsulfonylpropionic acid 2'-carboxymaleanilic acid gamma-oxo-1-naphthalenebutyric acid 11 - ((5-dimethylaminonaphthalene-1-sulfonyl) amino) undecanoic acid 2 - [[(4-chlorophenyl) sulfonyl] -3- (trifluoromethyl) anilino] acetic acid 2-nonenoic acid 2-formylphenoxyacetic acid 2,4-pyridinedicarboxylic acid 2-fluoro-6- (trifluoromethyl) phenylacetic acid acenaphthene-3-carboxylic acid

• ·· • · • ··· • ·· • · • ··· 99 9 9 99 9 9 9 • 9 • ···· • • ···· • • 99 99 9 9 9 9 • • • • 9 · 9 9 · 9 9 9 • 9 • 9 99 99 99 99 99 99 99 99 ·· · ·

kyselina 2-fluór-6-hydroxybenzoová kyselina 4-((pyridín-3-ylmetylén)-amino)-benzoová kyselina 4-izobutylbenzoová kyselina diheptyl-fosfínová kyselina 3-chlórpivalová kyselina 2-(2-nitro-4-(trifluórmetyl)fenyl)octová kyselina 2,5-dichlórbenzoová kyselina 4-metoxy-3-metylbenzoová kyselina 2-fluór-5-metoxybenzoová kyselina 14(s), 15(r)-epoxy-(5z,8z, 11 z)-eikozatriénová kyselina (2-( 1 -fenyl-etyl)-fenoxy)-octová kyselina 4-(benzénsulfonamido)-salicylová kyselina 4-hydroxy-3-jód-5-nitro-fenyloctová kyselina 2,6-dihydroxy-3,5-dimetyl-benzoová kyselina 2,4-dimetoxy-6-metyl-benzoová kyselina n-(2-tiazolyl)sukcínamová kyselina 7-(3,3-dimetyl-2,3-2h-benzo(b)tiofén-5-yl)-3-metyl-okta-2,4,6-tnénová kyselina r-4-nitromandlová kyselina (1 r)-(-)-10-gáforsulfónová kyselina 2-fluór-4-(trifluórmetyl)škoricová kyselina 3-(4-íerc-buty]-fenylsulfanyl)-propiónová kyselina 2-(3,5-dinitro-tiofén-2-ylamino)-jantárová kyselina (2-((3,4-dimetoxy-fenyl)-acetyl)-5-metoxy-fenyl)-octová kyselina 3,5-dijódosalicylová kyselina 2-(3-chlórfenoxy)propiónová kyselina erytro-9,10-dihydroxystearová kyselina dusitá kyselina shikimová kyselina 2'-me-1,3,ľ,3'-tetraoxo-1,3I2,,3,-4h-ľh-(2,5')biizoindolyl-5-karboxylová kyselina alfa3-chlór-5,7-dimetyl-1,3-adamantándioctová kyselina 4-(4-pentyl-cyklohexyl)-benzoová kyselina 3-metyl-2-(toluén-4-sulfonylamino)-maslová2-fluoro-6-hydroxybenzoic acid 4 - ((pyridin-3-ylmethylene) -amino) -benzoic acid 4-isobutylbenzoic acid diheptylphosphinic acid 3-chloropivalic acid 2- (2-nitro-4- (trifluoromethyl) phenyl ) acetic acid 2,5-dichlorobenzoic acid 4-methoxy-3-methylbenzoic acid 2-fluoro-5-methoxybenzoic acid 14 (s), 15 (r) -epoxy- (5z, 8z, 11z) -eicosatrienoic acid (2 - (1-Phenyl-ethyl) -phenoxy) -acetic acid 4- (benzenesulfonamido) -salicylic acid 4-hydroxy-3-iodo-5-nitro-phenylacetic acid 2,6-dihydroxy-3,5-dimethyl-benzoic acid 2,4- Dimethoxy-6-methyl-benzoic acid n- (2-thiazolyl) succinamic acid 7- (3,3-dimethyl-2,3-2h-benzo (b) thiophen-5-yl) -3-methyl -octa-2,4,6-tenoic acid r-4-nitromanedioic acid (1R) - (-) - 10-camphorsulfonic acid 2-fluoro-4- (trifluoromethyl) cinnamic acid 3- (4-tert-butyl) -phenylsulfanyl) -propionic acid 2- (3,5-dinitro-thiophen-2-ylamino) -succinic acid (2 - ((3,4-dimethoxy-phenyl) -acetyl) -5-mee 3,5-diiodosalicylic acid 2- (3-chlorophenoxy) propionic acid erythro-9,10-dihydroxystearic acid nitrous acid shikimic acid 2'-me-1,3,1 ', 3'-tetraoxo- 1.3 L of 2, 3, -4-H- (2.5) biizoindolyl-5-carboxylic acid The a3 subunit-chloro-5,7-dimethyl-1,3-adamantándioctová 4- (4-pentyl-cyclohexyl 3-Methyl-2- (toluene-4-sulfonylamino) butyric acid

BB ·· e···BB ·· e ···

B BBB B B · · · • B BBB B B B ·B • •B · · · · ·BB BBB B B BBB B B B B

BBB ·· ·· ····BBB ·· ·· ····

-11 kyselina (s)-1 -amino-(3-metylbután)fosfónová kyselina 5-benzyloxy-4-metoxy-2-metyl-benzoová kyselina 4'-bróm-2,-chlórhexahydroftalanilová kyselina 2-pentínová kyselina 2-benzofuránkarboxylová kyselina 3-(p-tolyltio)propiónová kyselina 2-kyano-3-etoxyakrylová kyselina 2-[3-(/?-oktanoyl-hydrazíno)-3-oxo-propionylamino)-benzoová kyselina 4-hydroxy-3-nitrozo-1 -naftalénsulfónová kyselina 3-jód-4-(izopropylsulfonyl)-5-(metyltio)tiofén-2-karboxylová kyselina n-boc-1-1,2,3,4-tetrahydroizochinolín-3-karboxylová kyselina 3-(1-naftyltio)propiónová kyselina 2,4,6-trimetylbenzoová kyselina bicyklo(2.2.1)heptán-3 4-dikarboxylová kyselina 1 ,ľ-etylénbis(5-oxo-3-pyrolidínkarboxylová) kyselina rodanín-3-octová kyselina nitranilová kyselina (r)-(-)-2-hydroxy-2-fenylpropiónová kyselina metyltiohydantoín-dl-asparágová kyselina 6-metyl-2-pyridín-3-yl-chinolín-4-karboxylová kyselina citrakónová kyselina n-(acetoacetyl)antranilová kyselina n-(3-etoxyfenyl)maleámová kyselina 2',4'-difluórftalanilová kyselina 2,4-dimetoxyškoricová kyselina 12-me-tricyklo(8.2.2.2(4,7))hexadeka-hexaén-5-karboxylová kyselina [2-(propán-2-sulfonyl)-acetylamino]-octová kyselina 2-hydroxydekánová kyselina c/s-n-benzylhexahydroftalámová kyselina 1,4-fenyléndiakrylová kyselina (2-(4-metoxy-fenyl)-6-oxo-cyklohex-1 -enyl)-octová kyselina 2-(5-fluór-1-naftoyl)benzoová(11) (s) -1-amino- (3-methylbutane) phosphonic acid 5-benzyloxy-4-methoxy-2-methyl-benzoic acid 4'-bromo-2 , -chlorohexahydrophthalanilic acid 2-pentanoic acid 2-benzofuranecarboxylic acid 3- (p-tolylthio) propionic acid 2-cyano-3-ethoxyacrylic acid 2- [3- (R-octanoyl-hydrazino) -3-oxo-propionylamino) -benzoic acid 4-hydroxy-3-nitroso-1- 3-Iodo-4- (isopropylsulfonyl) -5- (methylthio) thiophene-2-carboxylic acid naphthalenesulfonic acid n-boc-1-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid 3- (1-naphthylthio) propionic acid 2,4,6-trimethylbenzoic acid bicyclo (2.2.1) heptane-3 4-dicarboxylic acid 1,1'-ethylenebis (5-oxo-3-pyrrolidinecarboxylic acid) rodanine-3-acetic acid nitranilic acid (r) - (-) - 2-hydroxy-2-phenylpropionic acid methylthiohydantoin-dl-aspartic acid 6-methyl-2-pyridin-3-yl-quinoline-4-carboxylic acid citraconic acid n- (acetoacetyl) anthranilic acid n- (3- ethoxyphenyl l) maleic acid 2 ', 4'-difluorophthalanic acid 2,4-dimethoxycinnamic acid 12-methicyclo (8.2.2.2 (4,7)) hexadeca-hexaene-5-carboxylic acid [2- (propane-2-sulfonyl) (acetylamino) -acetic acid 2-hydroxydecanoic acid cis -benzylhexahydrophthalic acid 1,4-phenylenediacrylic acid (2- (4-methoxyphenyl) -6-oxo-cyclohex-1-phenyl) -acetic acid 2- ( 5-fluoro-1-naphthoyl) benzoic acid

• ·· • · • ··· • · · • ·· • · • ··· • · · ·· ···· 9 9 · 9 9 9 9 9 9 9 ·· ···· 9 9 · 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 99 99 ·· ·· ·· ·· 99 99 99 99 9 9 9 9 99 99

kyselina (2,2,2-trichlór-1-(3-(4-metoxykarbonyl-ph)-tioureido)-etyl)-karbámová kyselina 2-[3-(n-benzoyl-hydrazíno)-3-oxo-propionylamino]-benzoová kyselina ď/-p-aminobenzyljantárová kyselina 2-izopropyl-2-fenyloctová kyselina fmoc-(3s,4s,5s)-4-amino-3-hydroxy-5-metyl-heptánová kyselina 2-chlórizonikotínová kyselina 3,4,4-trichlór-but-3-énová kyselina 1 -(4-chlórfenyl)-1 -cyklobutánkarboxylová kyselina 4-(4-(4-chlór-fenoxy)-benzénsulfonyl)-benzoová kyselina (4-acetylamino-benzénsulfonylsulfanyl)-octová kyselina n-(4-aminobenzoyl)-1 -glutámová kyselina 4-(3-fenylureido)maslová kyselina 2,-fluór-3,4,5,6-tetrachlórftalanilová kyselina 4-sulfobenzoová askorbylpatmitan kyselina [4-chlór-6-(2,3-xylidino)-2-pyrimidinyltio]octová kyselina 2-amino-4-fenyltiazol-5-karboxylová kyselina 4-hydroxy-5-metoxy-1 -fenyl-naftalén-2-karboxylová kyselina 3,4,5-trimetyl-1 h-pyrole-2-karboxylová kyselina S.S'^^’-benzofenóntetrakarboxylová kyselina 4’-chlór-2,,5'-dimetoxyhexahydroftalanilová kyselina 3-(4-etoxybenzoylJpropiónová kyselina 4-chlór-2,6-dimetyl-nikotínová kyselina 3-[2-(4-butoxy-benzylamino)-3-(4-metoxy-fenyl)-akryloylamino]-propiónová kyselina 2-metyltiobenzimidazolsulfónová kyselina fenaceturová alfa, beta-dibrómškoricová kyselina o-trifluórmetyl-alfa-acetamidoškoricová kyselina boc-d-alfa-amino-gama-(4-metylbenzylmerapto)-maslová kyselina n-alfa-(benzyloxykarbonyl)-d-asparágová kyselina 2-fluór-4-pentyloxybenzoová kyselina boc-(3s,4s)-4-amino-3-hydroxy-5-fenyl-pentánová ·· ·· ···· ·· • · · · · · · ··· · · · · ·(2,2,2-Trichloro-1- (3- (4-methoxycarbonyl-ph) -thioureido) -ethyl) -carbamic acid 2- [3- (n-benzoyl-hydrazino) -3-oxo-propionylamino] 2-isopropyl-2-phenylacetic acid fmoc- (3s, 4s, 5s) -4-amino-3-hydroxy-5-methyl-heptanoic acid 3,4-p-aminobenzylsuccinic acid 2-chloro-isonicotinic acid 3,4, 4-Trichloro-but-3-enoic acid 1- (4-chlorophenyl) -1-cyclobutanecarboxylic acid 4- (4- (4-chloro-phenoxy) -benzenesulfonyl) -benzoic acid (4-acetylamino-benzenesulfonylsulfanyl) -acetic acid n- (4-aminobenzoyl) -1-glutamic acid 4- (3-phenylureido) butyric acid 2 , -fluoro-3,4,5,6-tetrachlorophthalanic acid 4-sulfobenzoic acid ascorbylpatmitate [4-chloro-6- (2) 3-xylidino) -2-pyrimidinylthio] acetic acid 2-amino-4-phenylthiazole-5-carboxylic acid 4-hydroxy-5-methoxy-1-phenyl-naphthalene-2-carboxylic acid 3,4,5-trimethyl- 1H-pyrrole-2-carboxylic acid S, S '^^' - benzophenonetetracarboxylic acid, 4'-chloro-2 ', 5'-dimethyl 3- (4-ethoxybenzoyl) propionic acid 4-chloro-2,6-dimethyl-nicotinic acid 3- [2- (4-butoxybenzylamino) -3- (4-methoxyphenyl) -acryloylamino] -propionic acid 2-ethoxyhexahydrophthalanilic acid -methylthiobenzimidazolesulfonic acid phenaceturic alpha, beta-dibromocinnamic acid o-trifluoromethyl-alpha-acetamidocinnamic acid boc-d-alpha-amino-gamma- (4-methylbenzylmerapto) -butyric acid n-alpha- (benzyloxycarbonyl) -d-aspartic acid 2- Fluoro-4-pentyloxybenzoic acid boc- (3s, 4s) -4-amino-3-hydroxy-5-phenylpentanoic acid ··· ············· · ·

-13kyselina pyrohroznová kyselina 4-(2-chlórfenoxy)-3-nitroškoricová kyselina 3-(aminokarbonylmetyltio)tiofén-2-karboxylová kyselina chlórbenzoyl(4-) benzoová kyselina 3-fenyl-2-p-tolyl-propiónová kyselina 7-hydroxykumarín-4-octová kyselina 2,3,4-trifluórbenzoová kyselina 3-acetyl-2-fenyl-4-tiazolidínkarboxylová kyselina 2-(3-(2,2I2-trichlór-1-((furán-2-karbonyl)-amino)-et)-tioureido)-benzoová kyselina 2-(3-chlór-benzoyl)-benzoová kyselina n-ftaloyl-gly-d/-alfa-amino-n-maslová kyselina 7-naftoová kyselina cyklooktán-1,2-dikarboxylová-13 pyruvic acid 4- (2-chlorophenoxy) -3-nitrocinnamic acid 3- (aminocarbonylmethylthio) thiophene-2-carboxylic acid chlorobenzoyl (4-) benzoic acid 3-phenyl-2-p-tolyl-propionic acid 7-hydroxycoumarin- 4-acetic acid, 2,3,4-trifluorobenzoic acid, 3-acetyl-2-phenyl-4-thiazolidinecarboxylic acid, 2- (3- (2.2 L 2-trichloro-1 - ((furan-2-carbonyl) -amino (Ethyl-thioureido) -benzoic acid 2- (3-chloro-benzoyl) -benzoic acid n-phthaloyl-gly-d-alpha-amino-n-butyric acid 7-naphthoic acid cyclooctane-1,2-dicarboxylic acid

A.A'-dikarboxydifenylsuifón kyselina 3-(4-n-heptyloxybenzoyl)propiónová kyselina n-(4-metoxyfenyl)maleámová kyselina 3-((2-karboxy-etyl)-(6-metyl-benzotiazol-2-yl)-amino)-propiónová kyselina 3,6-difenyl-cyklohex-4-én-1,2-dikarboxylová kyselina 5-(3-brómbenzoyl)pentánová kyselina diizooktylditiofosfínová kyselina 5-bróm-2-furoová kyselina 1,2,3,4-tetrahydro-fenantrén-1,2-dikarboxylová kyselina 9-etyl-3-karbazolfosforná kyselina 4-(2-hydroxy-6-(trimetylsilyl)-1 -naftylazo)benzoová kyselina etylmalónová kyselina cyklobutylfenylglykolová kyselina 3-brómfenyloctová kyselina n-(2-karboxyetyl)iminodioctová kyselina 4-(ŕerc-butyl)benzamidooctová kyselina fmoc-11-aminoundekánová kyselina fmoc-1 -oktahydroindol-2-karboxylová kyselina 2-(3-(4-(4,4-dikarboxy-butyl)-fenyl)-propyl)-malónová • ·· ·· ···· ·· ··· · · · · · · • ··· · · · · ·N - (4-Methoxyphenyl) maleic acid 3- (4-n-heptyloxybenzoyl) propionic acid 3 - ((2-carboxyethyl) - (6-methylbenzothiazol-2-yl) - amino) -propionic acid 3,6-diphenyl-cyclohex-4-ene-1,2-dicarboxylic acid 5- (3-bromobenzoyl) pentanoic acid diisooctyldithiophosphinic acid 5-bromo-2-furoic acid 1,2,3,4- tetrahydro-phenanthrene-1,2-dicarboxylic acid 9-ethyl-3-carbazolphosphoric acid 4- (2-hydroxy-6- (trimethylsilyl) -1-naphthylazo) benzoic acid ethyl malonic acid cyclobutylphenylglycolic acid 3-bromophenylacetic acid n- (2- carboxyethyl) iminodiacetic acid 4- (tert-butyl) benzamidoacetic acid fmoc-11-aminoundecanoic acid fmoc-1-octahydroindole-2-carboxylic acid 2- (3- (4- (4,4-dicarboxybutyl) phenyl) - propyl) -malonic acid

-14··· ···· ·· · ··· ·· ·· ·· ·· ··· kyselina 3-(4-metylbenzamido)benzoová kyselina 1 -(2-benzo[1,3]dioxol-5-yl-et)-2-(2-karboxy-et)-oxo-pyrolidín-karboxylová kyselina 4-hydroxy-3,5-diizopropyl-benzoová kyselina 3-((2-karboxy-etyl)-fenyl-amino)-propiónová kyselina p-fenylazomaleanilová kyselina 2-brómakrylová kyselina 2,3-bis-(4-chlór-benzylidén)-jantárová kyselina n-(4-metyl-3-nitrofenyl)glutarámová kyselina 3-bróm-5-metoxy-2-propyl-benzoová kyselina oxámová kyselina 2-(2-naftoyl)benzoová kyselina 2-(2-formamidotiazol-4-yl)-2-metoxylminooctová kyselina (r)-tetrahydrofurán-2-karboxylová kyselina 4-merkaptobenzoová kyselina (s)-2-fluór-2-metylpentánová kyselina 4-nitrofenoxyoctová kyselina ac-d-ala-d-mliečna kyselina 2-(4-hydroxymetyl-3-metoxyfenoxy)maslová kyselina 4-(3-nitrofenyl)-1,3-butadién-1-karboxylová kyselina 4-bróm-4,4-difluórmaslová kyselina 3-(4-chlór-2-nitro-fenyl)-2-oxo-propiónová kyselina 20,20,20-trifluórarachidónová kyselina dibrómfluóroctová kyselina 2-brómlaurová kyselina bis(4-chlórfenoxy)octová kyselina 4,4'-trimetylénbis(fenyloctová) kyselina 4-hydroxy-pyridín-3,5-dikarboxylová kyselina 2-etoxy-1-naftoová kyselina 3-(4,5-difenyl-2-oxazolyl)propiónová kyselina tetrachlórftalová kyselina chloristá kyselina [3-(metoxykarbonyl)-2-metyl-5-oxo-2-pyrolín-4-yl]octová-14 3- (4-Methylbenzamido) benzoic acid 1- (2-benzo [1,3] dioxol-5) -yl-ethyl-2- (2-carboxy-ethyl) -oxo-pyrrolidine-carboxylic acid 4-hydroxy-3,5-diisopropyl-benzoic acid 3 - ((2-carboxy-ethyl) -phenylamino) - propionic acid p-phenylazomaleanilic acid 2-bromoacrylic acid 2,3-bis- (4-chlorobenzylidene) -succinic acid n- (4-methyl-3-nitrophenyl) glutaramic acid 3-bromo-5-methoxy-2-propyl -benzoic acid oxamic acid 2- (2-naphthoyl) benzoic acid 2- (2-formamidothiazol-4-yl) -2-methoxy-aminoacetic acid (R) -tetrahydrofuran-2-carboxylic acid 4-mercaptobenzoic acid (s) -2- Fluoro-2-methylpentanoic acid 4-nitrophenoxyacetic acid ac-d-ala-d-lactic acid 2- (4-hydroxymethyl-3-methoxyphenoxy) butyric acid 4- (3-nitrophenyl) -1,3-butadiene-1-carboxylic acid 4-Bromo-4,4-difluorobutyric acid 3- (4-chloro-2-nitro-phenyl) -2-oxo-propionic acid hidonic acid dibromofluoroacetic acid 2-bromolauric acid bis (4-chlorophenoxy) acetic acid 4,4'-trimethylenebis (phenylacetic) 4-hydroxy-pyridine-3,5-dicarboxylic acid 2-ethoxy-1-naphthoic acid 3- (4 5-diphenyl-2-oxazolyl) propionic acid tetrachlorophthalic acid perchloric acid [3- (methoxycarbonyl) -2-methyl-5-oxo-2-pyrrolin-4-yl] acetic acid

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · ···· • 9 ···· • 9 99 9 9 9 9 99 9 9 9 9 9 9 9 9 ·· ·· ·· ·· ·· · · 99 99 99 99 9 · 9 ·

kyselina 3-(3-(1-butyrylamino-2,2,2-trichlór-etyl)-tioureido)-benzoová kyselina 3,4,9,10-peryléntetrakarboxylová kyselina 3-fluór-4-hydroxybenzoová kyselina d/-alfa-hydroxyizovalérová kyselina 3-(2-chlór-etánsulfonyl)-propiónová kyselina fmoc-1-pipekolínová kyselina 2-metyl-1,1-dioxo-2,3-dihydro-l h-benzo(b)tiofén-2-karboxylová kyselina 3-acetyl-tiazolidiη-2-karboxylová kyselina 1 -metyl-1 -cyklohexánkarboxylová kyselina 2-(3-benzyloxy-4-metoxy-benzyl)-2-fenyl-malónová kyselina n-(3-(trietoxysilyl)propyl]ftalámová kyselina 2,2,5,5-tetrametyl-3-pyrolin-1 -oxyl-3-karboxylová kyselina fmoc-8-aminokaprylová kyselina 3-metyltianaftén-2-octová kyselina 3-brómškoricová kyselina 1-oxalyl-1,4-fenyléndiamín-2-sulfónová kyselina sukcínamová kyselina 4-[(d/-n-propylamino)sulfonyl]benzoová kyselina alfa-fluórškoricová kyselina 2,3-difenyl-2-cyklopropén-1 -karboxylová kyselina 3,4-pyridíndikarboxylová kyselina p-pentyloxybenzoová kyselina 3-(1,3-dioxo-1 h,3h-benzo(de)izochinolín-2-yl)-benzoová kyselina 3-tricyklo(8.2.2.2(4,7))hexadeka-hexén-2-yl-akrylová kyselina 2-(1 -metyl-2-(4-nitro-fenyl)-propoxy)-benzoová kyselina 2,4,5-trifluórfenyloctová kyselina 3-chlór-3-p-tolylkarbamoyl-akrylová kyselina 3,7-dihydroxy-2-naftoová kyselina 3-metoxyfenyloctová kyselina 2-benzoylamino-3-(4-hydroxy-3-metoxy-fenyl)-propiónová kyselina 3-(4-metylbenzoyl)-akrylová kyselina n-cyklododecylmaleámová ·· ·· ···· ·· • · · · · · · ··· · · · · ·3- (3- (1-butyrylamino-2,2,2-trichloro-ethyl) -thioureido) -benzoic acid 3,4,9,10-perylenetetracarboxylic acid 3-fluoro-4-hydroxybenzoic acid d-alpha- 3- (2-chloro-ethanesulfonyl) -propionic acid hydroxymovaleric acid fmoc-1-pipecolinic acid 2-methyl-1,1-dioxo-2,3-dihydro-1H-benzo (b) thiophene-2-carboxylic acid 3 Acetyl-thiazolidine-2-carboxylic acid 1-methyl-1-cyclohexanecarboxylic acid 2- (3-benzyloxy-4-methoxy-benzyl) -2-phenyl-malonic acid n- (3- (triethoxysilyl) propyl] phthalic acid 2 2,5,5-tetramethyl-3-pyrolin-1-oxyl-3-carboxylic acid fmoc-8-aminocaprylic acid 3-methylthianaphthene-2-acetic acid 3-bromocinnamic acid 1-oxalyl-1,4-phenylenediamine-2 sulfonic acid succinic acid 4 - [(d-n-propylamino) sulfonyl] benzoic acid alpha-fluorocinnamic acid 2,3-diphenyl-2-cyclopropene-1-carboxylic acid 3,4-pyridinedicarboxylic acid p-pentyloxybenzoic acid 3- (1,3-dioxo-1 h, 3h-Benzo (de) isoquinolin-2-yl) -benzoic acid 3-tricyclo (8.2.2.2 (4,7)) hexadeca-hexen-2-yl-acrylic acid 2- (1-methyl-2- ( 4-nitro-phenyl) -propoxy) -benzoic acid 2,4,5-trifluorophenylacetic acid 3-chloro-3-p-tolylcarbamoyl-acrylic acid 3,7-dihydroxy-2-naphthoic acid 3-methoxyphenylacetic acid 2-benzoylamino- 3- (4-hydroxy-3-methoxy-phenyl) -propionic acid 3- (4-methylbenzoyl) -acrylic acid n-cyclododecylmaleamic acid ··· ·················· · · · ·

-16kyselina 11-hydroxyundekánová kyselina 3-bróm-2-metylbenzoová kyselina n-(2,3-dichlórfenyl)maleámová kyselina 2-fluór-5-nitrobenzoová kyselina hydroxy-(2,3,5I6-tetrametyl-fenyl)-octová kyselina 2-izopropyl-2-fenylglykolová kyselina 1 -hydroxy-4-(4-nitrofenoxy)-2-naftoová kyselina 2-hydroxy-6-(3,4I5-trimetoxyfenyl)-3,5-pyridíndikarboxylová kyselina (1 -amino-1 -fosfóno-etyl)-fosfónová kyselina n-(2,4-dichlórfenyl)maleámová kyselina n,/ť-tereftalylidén-bis(4-aminosalicylová) kyselina írans-akonitová kyselina 5’-chlór-2',4'-dimetoxyftalanilová kyselina (ij-2-brómmaslová kyselina 4-azido-2,3,5,6-tetrafluórbenzoová kyselina n-(3-metoxyfenyl)tetrachlórftalámová kyselina 5-fluór-2-(trifluórmetyl)benzoová kyselina 2,2-dimetyl-4-penténová kyselina heptadekánová kyselina 3,5-pyridíndikarboxylová kyselina beta.beta-dimetyl-1-pyrolpropánová kyselina 2-chlór-3-(trifluórmetyl)benzoová kyselina 2,3-dihydro-benzo(b)azepín-1-karboxylová kyselina 4-( 1 -metyl-butyl)-benzoová kyselina p-(beta-brómetyl)benzoová kyselina 2,2-dichlórpentánová kyselina 7-(dimetylaminosulfonyl)-2,3-dihydro-gama-oxo-1-(1h)-indolbutánová kyselina 13(s)-hydroxyoktadeka-9z,11e-diénová kyselina 4-brómfenyloctová kyselina (s)-(+)-o-acetylmandlová kyselina 3-chlór-2-fluórbenzoová kyselina gáforchinón-10-sulfónová-16kyselina 11-hydroxyundekánová acid 3-bromo-2-methylbenzoic acid, N- (2,3-dichlorophenyl) maleamic acid 2-fluoro-5-nitrobenzoic acid hydroxy- (2,3,5-I, 6-tetramethyl-phenyl) -acetic acid acid 2-isopropyl-2-mandelic acid, 1-hydroxy-4- (4-nitrophenoxy) -2-naphthoic acid, 2-hydroxy-6- (3,4 I 5-trimethoxyphenyl) -3,5-pyridinedicarboxylic acid (1 - amino-1-phosphono-ethyl) -phosphonic acid N- (2,4-dichlorophenyl) maleic acid N, N-terephthalylidene-bis (4-aminosalicyl) trans-aconitic acid 5'-chloro-2 ', 4' -dimethoxyphthalanic acid (ij-2-bromobutyric acid 4-azido-2,3,5,6-tetrafluorobenzoic acid n- (3-methoxyphenyl) tetrachlorophthalic acid 5-fluoro-2- (trifluoromethyl) benzoic acid 2,2-dimethyl- 4-Pentenoic heptadecanoic acid 3,5-pyridinedicarboxylic acid beta-beta-dimethyl-1-pyrrolepropanoic acid 2-chloro-3- (trifluoromethyl) benzoic acid 2,3-dihydro-benzo (b) azepine-1-carboxylic acid 4- (1-methyl-butyl) -benzoic acid p- (beta-bromomethyl) benzoic acid 2,2-dichloropentanoic acid 7- (dimethylaminosulfonyl) -2,3-dihydro-gamma-oxo-1- (1h) -indolbutanoic acid 13 (s) -hydroxyoctadeca-9z, 11e-dienoic acid 4-bromophenylacetic acid (s) - (+) - o-acetylmandelic acid 3-chloro-2-fluorobenzoic acid Camphorquinone-10-sulfonic acid

• 99 • · • ··· • 99 • · • ··· • • • • ·· • • · · • • ···· • • ···· • • • · • · ·· · · • • • • • • • • • · · • · · • · • · ·· ·· ·· ·· ·· · · ·· · · ·· · · 99 99

kyselina 3-nonénová kyselina 9-oxo-bicyklo(3.3.1 )non-6-én-3-karboxylová kyselina 3’-chlór-2,3-dibróm-4'-metylsukcínanilová kyselina 4-bróm-2-fluórbenzoová kyselina 17-jódheptadekánová kyselina I^.S^.ej.e-heptachlór-tricyklo^^.O.OÍS.ejlokM-én^J-dikarboxylová kyselina n-cbz-1-glutámová karboxyfenylgama-kyselina kyselina 4-benzyloxy-3,5-dimetoxy-benzoová kyselina 4-krezidín-6-sulfónová kyselina 2-(2,5-dichlórfenoxy)propiónová kyselina (2-bróm-4,5-dimetoxy-fenyl)-octová kyselina 2'-hydroxy-2-bifenylkarboxylová kyselina 4,4,4-trifluór-3-(trifluórmetyl)krotónová kyselina 16-hydroxyhexadekánová kyselina 4-nitro-3-(oktanoyloxy)-benzoová kyselina 1,3-diaminopropán-n,n,n’,n-tetraoctová kyselina 4-fluór-2-(trifluórmetyl)škoricová kyselina 2,3-dichlórizomaslová kyselina 3,4-difluórškoricová kyselina 3-(3-adamantán-1-yl-ureido)-propiónová kyselina 1,1-dimetyl-indán-4-karboxylová kyselina d(-)-2-amino-5-fosfonopentánová kyselina fmoc-5-aminovalérová kyselina 3-metoxy-9-oxo-6,7,8,9-tetrahydro-5h-benzocykloheptén-6-karboxylová kyselina 4,4-dichlór-4-fluórbutánová kyselina (4-(4-karboxymetylsulfanyl-benzyl)-fenylsulfanyl)-octová kyselina ŕrans-2-(2-tiofénkarbonyl)-1 -cyklohexánkarboxylová kyselina 3,5-dimetoxy-4-hydroxyfenyloctová kyselina 1-pyrénmaslová kyselina n-(2,6-dimetylfenylkarbamoylmetyl)iminodioctová kyselina 4-nitrofenyloxámová ·· ·· ····3-nonenoic acid 9-oxo-bicyclo (3.3.1) non-6-ene-3-carboxylic acid 3'-chloro-2,3-dibromo-4'-methylsuccinilic acid 4-bromo-2-fluorobenzoic acid 17 4-Benzyloxy-3,5- [iodo-heptadecanoic acid] -S-E-heptachloro-tricyclo [1.0.0.0 < 2,7 > -ocenoic acid] n-cbz-1-glutamic carboxyphenyl-gamma-acid dimethoxybenzoic acid 4-cresidine-6-sulfonic acid 2- (2,5-dichlorophenoxy) propionic acid (2-bromo-4,5-dimethoxyphenyl) acetic acid 2'-hydroxy-2-biphenylcarboxylic acid 4, 4,4-trifluoro-3- (trifluoromethyl) crotonic acid 16-hydroxyhexadecanoic acid 4-nitro-3- (octanoyloxy) benzoic acid 1,3-diaminopropane-n, n, n ', n-tetraacetic acid 4-fluoro- 2- (Trifluoromethyl) cinnamic acid 2,3-dichloroisobutyric acid 3,4-Difluorocinnamic acid 3- (3-adamantan-1-yl-ureido) -propionic acid 1,1-dimethyl-indane-4-carboxylic acid d (- -2-Amino-5-phosphonopentanoic acid fmoc-5-amine 3-methoxy-9-oxo-6,7,8,9-tetrahydro-5h-benzocycloheptene-6-carboxylic acid ovaleric acid 4,4-dichloro-4-fluorobutanoic acid (4- (4-carboxymethylsulfanyl-benzyl) -phenylsulfanyl) trans-2- (2-Thiophenecarbonyl) -1-cyclohexanecarboxylic acid 3,5-dimethoxy-4-hydroxyphenylacetic acid 1-pyrene-butyric acid 4- (2,6-dimethylphenylcarbamoylmethyl) iminodiacetic acid 4-nitrophenyloxamic acid ·· ··· ····

-18kyselina 3-etyl-cyklohex-4-én-1,2-dikarboxylová kyselina (l)-mentylkarboxylová kyselina 3,3,3-trimetylpyrohroznová kyselina 1 -metyl-2-fenyl-cyklopent-2-énkarboxylová kyselina hexahydrcM'-sulfamoylftalanilová kyselina 2-metoxyfenyloctová-18-3-ethyl-cyclohex-4-ene-1,2-dicarboxylic acid (1) -mentylcarboxylic acid 3,3,3-trimethylpyruvic acid 1-methyl-2-phenyl-cyclopent-2-enecarboxylic acid hexahydric-4'-sulfamoyl-phthalanilic acid 2-methoxyphenylacetic acid

3-karboxybenzaldehyd kyselina n-fenetylmaleámová citrinín kyselina 3-nitrofenoxyoctová kyselina 8-hydroxyoktánová kyselina bis-(3-chlór-fenyl)-fosfínová kyselina 2-(2-karboxy-etyl)-6,6-dimetyl-3-oxo-cyklohex-1-énkarboxylová kyselina c/s-8-metylnon-6-énová kyselina o-(karbometoxy)-salicylová kyselina 3-benzoyl-2-(3-chlórfenyl)propiónová kyselina (2-[2-(5-me-[1,3,4]tiadiazol-2-ylsulfanyl)-ac-amino]-tiazol-4-yl)-octová kyselina oktahydro-3-metyl-1 -pentalénkarboxylová kyselina p-fenylhipurová kyselina n-(2,2-dichlóracetyl)-5-jódantranilová3-carboxybenzaldehyde n-phenethylmaleamic acid citrinine 3-nitrophenoxyacetic acid 8-hydroxyoctanoic acid bis- (3-chlorophenyl) phosphinic acid 2- (2-carboxyethyl) -6,6-dimethyl-3-oxo-cyclohex 1-enecarboxylic acid cis-8-methylnon-6-enoic acid o- (carbomethoxy) -salicylic acid 3-benzoyl-2- (3-chlorophenyl) propionic acid (2- [2- (5-me- [ 1,3,4] Thiadiazol-2-ylsulfanyl) -ac-amino] -thiazol-4-yl) -acetic acid octahydro-3-methyl-1-pentalenecarboxylic acid p-phenylhipuric acid n- (2,2-dichloroacetyl) 5-iodoanthranilic

2-fluór-4-nonyloxybenzoová kyselina 3,5-dimetyl-p-anízová kyselina etyléndiaminetetrapropiónová kyselina 2-amino-3,6-dimetyl-5-nitro-benzoová kyselina 4-(4-metoxybenzoyl)maslová kyselina metoxyoctová kyselina 5-benzo(1,3)dioxol-5-yl-8-hydroxy-nafto(2,3-d)(1,3)dioxol-6-karboxylová kyselina 4-oxohexánová kyselina 2-(p-hydroxybenzoyl)benzoová kyselina 2-hydroxyeikozánová kyselina (r)-3-hydroxy-3-fenylpropánová kyselina 4-oxo-6-fenyl-5-hexénová ** · · · * · · ·· • · · · · ··· · · · ·2-fluoro-4-nonyloxybenzoic acid 3,5-dimethyl-p-anisic acid ethylenediaminetetrapropionic acid 2-amino-3,6-dimethyl-5-nitro-benzoic acid 4- (4-methoxybenzoyl) butyric acid 5-benzoic acid (1,3) dioxol-5-yl-8-hydroxy-naphtho (2,3-d) (1,3) dioxole-6-carboxylic acid 4-oxohexanoic acid 2- (p-hydroxybenzoyl) benzoic acid 2-hydroxyeicosanoic acid (r) -3-Hydroxy-3-phenylpropanoic acid 4-oxo-6-phenyl-5-hexenoic acid ** · · · · ··· · · · · ··· · · · ·

-19d-destiobiotín kyselina 7-oxo-6-oxa-bicyklo[3.2.1 ]oktán-3-karboxylová kyselina 2-hydroxy-3,5-dimetyl-benzoová kyselina (+)-c/s-2-benzamidocyklohexánkarboxylová kyselina antracén-1,5-dikarboxylová kyselina fenyl-n-propylfosfínová kyselina 3-hydroxyundekánová kyselina (2-naftalén-2-yl-acetylamino)-octová kyselina (5-kyano-6-hydroxy-4-metyl-2-oxo-2h-pyridín-1-yl)-octová kyselina 2-benzoylamino-3,3-dichlór-akrylová kyselina 3-metylundekánová kyselina 4,4-bis-(3,5-dichlór-4-hydroxyfenyl)-valérová kyselina fmoc-d/-2-aminohexánová kyselina 4-hexénová kyselina cyklobutánkarboxylová kyselina 4,4,5,5,6,6,6-heptafluórhexánová kyselina n,n-dimetylsukcínamová kyselina 2’-karboxysukcínanilová kyselina 2,5-dimetylbenzénsulfónová kyselina 4-metyl-4-cyklohexén-1,2-dikarboxylová kyselina (2-se/r-butyl-3-chlór-fenoxy)-octová kyselina 3',4'-dichlór-1,2,3,6-tetrahydroftalanilová kyselina (r)-(-)-( 1 -aminoetyl)fosfónová kyselina (s)-(+)-2-oxo-4-fenyl-3-oxazolidínoctová kyselina 4-hydroxymetylbenzoová kyselina 3-hydroxy-4-metoxymandlová kyselina 3-brómanízová kyselina (2-nitro-benzénsulfonyl)-octová kyselina 3,3,3-trifluór-2,2-dihydroxy-propiónová kyselina n-alfa-(benzyloxykarbonyl)-gama-(ŕerc-butylester)-d-glutárnová kyselina l-(+)-2-amino-5-fosfonovalérová kyselina 2-fluórbenzoová-19d-destiobiotin 7-oxo-6-oxa-bicyclo [3.2.1] octane-3-carboxylic acid 2-hydroxy-3,5-dimethyl-benzoic acid (+) - cis-2-benzamidocyclohexanecarboxylic acid anthracene -1,5-dicarboxylic acid phenyl-n-propylphosphinic acid 3-hydroxyundecanoic acid (2-naphthalen-2-yl-acetylamino) -acetic acid (5-cyano-6-hydroxy-4-methyl-2-oxo-2h- pyridin-1-yl) -acetic acid 2-benzoylamino-3,3-dichloro-acrylic acid 3-methylenedecanoic acid 4,4-bis- (3,5-dichloro-4-hydroxyphenyl) -valeric acid fmoc-d] - 2-aminohexanoic acid 4-hexenoic acid cyclobutanecarboxylic acid 4,4,5,5,6,6,6-heptafluorohexanoic acid n, n-dimethylsuccinamic acid 2'-carboxysuccinilic acid 2,5-dimethylbenzenesulfonic acid 4-methyl-4-cyclohexene -1,2-Dicarboxylic acid (2-sec-tert-butyl-3-chloro-phenoxy) -acetic acid 3 ', 4'-dichloro-1,2,3,6-tetrahydrophthalanic acid (r) - (-) - (1-Aminoethyl) phosphonic acid (s) - (+) - 2-oxo-4-phenyl-3-o xazolidinacetic acid 4-hydroxymethylbenzoic acid 3-hydroxy-4-methoxymandelic acid 3-bromoanonic acid (2-nitro-benzenesulfonyl) -acetic acid 3,3,3-trifluoro-2,2-dihydroxypropionic acid n-alpha- (benzyloxycarbonyl) 1-(+) - 2-Amino-5-phosphonovaleric acid 2-fluorobenzoic acid-gamma- (tert-butyl ester) -d-glutaric acid

-20·· ···· • · · • · · • · · · · • · · ·-20 ·· ···· · · · · · · · · · · · · · · · ·

9999

kyselina n-(3,3,5-trimetylcyklohexyl)-ditiokarbámová kyselina l-(+)-mandlová kyselina 5-fluór-2-(trifluórmetyl)škoricová kyselina 2,6-dimetylbenzoová kyselina (2-chlór-2-fenyl-vinyl)-fosfónová kyselina 3-benzoyl-2-benzylidénpropiónová kyselina auríntrikarboxylová kyselina 4-(2-naftyl)maslová kyselina c/s-10-pentadecénová (c15:1) kyselina 2-butínová kyselina 2,3-dibróm-n-( 1 -naftyl)sukcínamová kyselina p-chlórfenoxyoctová kyselina (r)-3-fenylmaslová kyselina (o-tolyl)fosfónová kyselina 4’-bróm-3'-metylftalanilová kyselina 15-ketoeikoza-6e,8z, 11 z, 13e-tetránová kyselina homoizocitrónová kyselina para-(4-oxo-2-tioxotiazolidino)-benzoová kyselina ŕrans-5-acetoxy-1,3-oxatiolán-2-karboxylová kyselina 3-formyl-2,4,6-trimetyl-benzoová kyselina d-3-fenylmliečna kyselina 4-etylftalanilová kyselina 2-[2-[3-chlór-5-(trifluórmetyl)-2-pyridyl]karbohydazonyl]-benzoová kyselina 2'-metylglutaranilová kyselina 4-nitropikolínová kyselina 4-chlór-3,5-dinitrobenzénsulfónová kyselina 2-brómškoricová kyselina 3-butoxy-4-nitrobenzoová kyselina fosforná kyselina butylmalónová kyselina 4-metoxyškoricová kyselina tiofén-2-octováN- (3,3,5-trimethylcyclohexyl) -dithiocarbamic acid 1- (+) - mandelic acid 5-fluoro-2- (trifluoromethyl) cinnamic acid 2,6-dimethylbenzoic acid (2-chloro-2-phenyl-vinyl) ) Phosphonic acid 3-benzoyl-2-benzylidenepropionic acid aurin tricarboxylic acid 4- (2-naphthyl) butyric cis-10-pentadecenoic acid (c15: 1) 2-butyric acid 2,3-dibromo-n- (1) (naphthyl) succinamic acid p-chlorophenoxyacetic acid (r) -3-phenylbutyric acid (o-tolyl) phosphonic acid 4'-bromo-3'-methylphthalanilic acid 15-ketoeicoza-6e, 8z, 11z, 13e-tetrano homoisocitric acid para- (4-oxo-2-thioxothiazolidino) -benzoic acid trans-5-acetoxy-1,3-oxathiolane-2-carboxylic acid 3-formyl-2,4,6-trimethyl-benzoic acid d-3-phenyl-lactic acid 4-ethylphthalanic acid 2- [2- [3-chloro-5- (trifluoromethyl) -2-pyridyl] carbohydazonyl] -benzoic acid 2'-methylglutaranilic acid 4-nitropicolinic acid 4-chloro-3,5-d initrobenzenesulfonic acid 2-bromocinnamic acid 3-butoxy-4-nitrobenzoic acid phosphoric acid butyl malonic acid 4-methoxycinnamic acid thiophene-2-acetic acid

-21 ·· ·· ···· ·· • · · · · · · ··· · · · · · kyselina cykloundekánkarboxylová kyselina 3’-hydroxyftalanilová kyselina (4-ŕerc-butyl-fenoxy)-octová kyselina 3-(4-n-pentylbenzoyl)propiónová kyselina 5-(3,5-dichlórfenoxy)furán-2-karboxylová kyselina 2-[(4,6-dimetoxypyrimidín-2-yl)oxy]-6-metoxybenzoová kyselina hydroxy-fenyl-p-tolyl-octová kyselina 2-norbornén-2,3-dikarboxylová kyselina (fenyltio)octová kyselina 5-keto-d-glukónová kyselina 7-ho-1,3-dimetyl-2,4-dioxo-1 ^.S^^h-pyridoíS^-djpyrimidín-e-karboxylová kyselina m-hydroxymandlová kyselina oxanilová kyselina alfa-etylškoricová kyselina 3-[5-(4-metoxy-fenyl)-furán-2-yl]-akrylová kyselina 2,5-dimetoxyfenyloctová kyselina hroznová kyselina 2-hydroxyimino-propiónová kyselina 1,2,3-benzéntrikarboxylová kyselina 2,4-dimetylglutárová kyselina 4-metylcyklohexánoctová kyselina 3-(2-chlórfenyl)-2-kyanopropiónová fmoc-1-norleucín kyselina 1,4-benzodioxán-2-karboxylová kyselina 3-(4-chlór-2-oxo-benzotiazol-3-yl)-propiónová kyselina 4,5,5,5-tetrafluór-4-(trifluórmetoxy)pentánová kyselina 2,3-dimetylglutárová kyselina heptafluórmaslová kyselina 2-benzénsulfonyloxy-3-metoxy-benzoová-21 Cycloundecanecarboxylic acid 3'-hydroxyphthalanilic acid (4-tert-butyl-phenoxy) -acetic acid 3- ( 4-n-Pentylbenzoyl) propionic acid 5- (3,5-dichlorophenoxy) furan-2-carboxylic acid 2 - [(4,6-dimethoxypyrimidin-2-yl) oxy] -6-methoxybenzoic acid hydroxyphenyl-p- tolyl-acetic acid 2-norborene-2,3-dicarboxylic acid (phenylthio) acetic acid 5-keto-d-gluconic acid 7-ho-1,3-dimethyl-2,4-dioxo-1,1'S m -hydroxymandelic acid oxanilic acid alpha-ethylcinnamic acid 3- [5- (4-methoxyphenyl) -furan-2-yl] -acrylic acid 2,5-dimethoxyphenylacetic acid 2-hydroxyimino-propionic acid 1,2,3-benzenetricarboxylic acid 2,4-dimethylglutaric acid 4-methylcyclohexaneacetic acid 3- (2-chlorophenyl) -2-cyanopropionic acid fmoc-1-norleucine 1,4-benzodioxane-2-carboxylic acid kysel 3- (4-chloro-2-oxo-benzothiazol-3-yl) -propionic acid 4,5,5,5-tetrafluoro-4- (trifluoromethoxy) pentanoic acid 2,3-dimethylglutaric acid heptafluorobutyric acid 2-benzenesulfonyloxy- 3-methoxy-benzoic acid

2’-karboxy-2-hydroxy-4-metoxy-benzofenón kyselina 7-metyl-2-fenylimidazo[1,2-a]pyridín-3-karboxylová kyselina 5-hexénová • · ·· ···· ·· · · e · · · ··· · · B · ·2'-carboxy-2-hydroxy-4-methoxy-benzophenone 7-methyl-2-phenylimidazo [1,2-a] pyridine-3-carboxylic acid 5-hexenoic acid • · ·· ······· e · · · ··· · · ·

-22kyselina S'-chlór^.S-dibrómsukcínanilová kyselina 2,2-dichlórhexánová kyselina 4-((pyridín-4-karbonyl)-amino)-maslová kyselina 3,3-dichlórpivalová kyselina 2-imidazolidón-4-karboxylová beta-oxalylamino-ď-alanín kyselina 4,-etoxy-3,4,5,6-tetrachlórftalanilová kyselina (2-benzotiazolyltio)octová kyselina 4-benzyloxyindol-2-karboxylová kyselina 2-ŕrans-benzoyl-5-ŕrans-fenyl-1 -cyklohexánkarboxylová kyselina 12-nitro-tricyklo(8.2.2.2(4,7))hexadeka-hexaén-5-karboxylová kyselina 2-acetyl-3-tiofénkarboxylová kyselina 4'-nitrosukcínanilová kyselina 2-hydroxyizomaslová kyselina 2,3-dimetylbenzoová kyselina propyléndifosfónová kyselina 2-cyklopentén-1-octová kyselina 4-pyridín-2-yl-acetyl)-benzoová kyselina 4-(3-(3-chlór-4-fluórfenyl)ureido)benzoová kyselina 4-nitrofenylglyoxylová kyselina pth-glutámová kyselina (8r, 15s)-dihydroxy-(5z,9e, 11 z,13e)-eikozatetraénová kyselina 5-nitro-2-furoová kyselina 2-butyloktánová kyselina n-formyl-4-nitroantranilová kyselina 2-metoxy-alfa-metylškoricová kyselina 2-(2-etoxykarbonyl-acetylamino)-benzoová kyselina 2,3-dimetylfenoxyoctová kyselina 3,5-dimetoxy-4-hydroxyškoricová kyselina 3-chlór-4-nitrobenzénsulfónová kyselina d/-alfa-aminopimelová kyselina alfa-kyano-4-hydroxyškoricová2-imidazolidone-4-carboxylic acid beta-oxalylamino-2,2'-dibromosuccinilic acid 2,2-dichlorohexanoic acid 4 - ((pyridine-4-carbonyl) -amino) -butyric acid 3,3-dichloropivalic acid -D-alanine acid 4-ethoxy-3,4,5,6-tetrachlórftalanilová acid (2-benzothiazolylthio) acetic acid 4-benzyloxy-indole-2-carboxylic acid 2-benzoyl-trans-5-trans-1-phenyl-cyclohexanecarboxylic 12-nitro-tricyclo (8.2.2.2 (4,7)) hexadeca-hexaene-5-carboxylic acid 2-acetyl-3-thiophenecarboxylic acid 4'-nitrosuccinilic acid 2-hydroxyisobutyric acid 2,3-dimethylbenzoic acid propylenediphosphonic acid 2 -cyclopentene-1-acetic acid 4-pyridin-2-yl-acetyl) -benzoic acid 4- (3- (3-chloro-4-fluorophenyl) ureido) benzoic acid 4-nitrophenylglyoxylic acid pth-glutamic acid (8r, 15s ) -dihydroxy- (5z, 9e, 11z, 13e) -eicosatetraenoic acid 5-nitro-2-furoic acid 2-butyloctanoic acid n-formyl-4-nitro 2-methoxy-alpha-methyl cinnamic acid 2- (2-ethoxycarbonyl-acetylamino) -benzoic acid 2,3-dimethylphenoxyacetic acid 3,5-dimethoxy-4-hydroxycinnamic acid 3-chloro-4-nitrobenzenesulfonic acid d-alpha -aminopimelic acid alpha-cyano-4-hydroxy cinnamic acid

• ·· • · • ··· • · · • ·· • · • ··· • · · ·· ···· • · · • · · · ·· ···· • · · • · · · • · • · • · • · * • · • · • · • · * • · • · ·· ·· ·· ·· ·· ·· ·· ·· ·· · · ·· · ·

kyselina 3-((5-bróm-1,3-dioxo-1,3-dihydro-izoindol-2-ylmetyl)-amino)-benzoová kyselina n-etyl-1-asparágová kyselina n-alfa-fmoc-n-beta-boc-d-diaminopropiónová kyselina n-ŕerc-boc-(2s,3r)-amino-2-hydroxy-4-(4-nitrofenyl)maslová kyselina 2,6-pyridíndikarboxylová kyselina 3-dibenzo(a,c)fenazín-11-yl-akrylová kyselina valerénová kyselina nikotínová, n-oxid kyselina 4-chlórfenyl-cyklohexánkarboxylová kyselina 4-(p-chlórfenoxy)maslová kyselina n-tris[hydroxymetyl]metyl-4-aminobutánsulfónová kyselina s-4-nitromandlová kyselina 4,5-dichlór-2-fluórbenzoová kyselina n-(2,3-xylyl)glutarámová kyselina 4,5,5-trifluór-4-penténová kyselina 5-fluór-2,6-dihydroxy-pyrimidín-4-karboxylová kyselina 3-fenylsalicylová kyselina 2-(2-hydroxy-5-metyl-benzoyl)-benzoová kyselina c/s-4-cyklohexén-1,2-dikarboxylová kyselina 2-brómstearová kyselina /-ŕrans-pyrolidín-2,4-dikarboxylová kyselina 2-chlórbenzoová kyselina 5-sulfónová kyselina 3-tiofénkarboxylová kyselina 2-((3-metoxy-fenyl)-fenyl-metylén)-jantárová kyselina 3-chlórškoricová kyselina 4-fenylškoricová kyselina 3-(3,5-dinitro-4-hydroxyfenyl)propiónová kyselina 7-acetoxykumarín-3-karboxylová kyselina d-alfa-galakturónová kyselina 3-bróm-2,5,6-trimetoxybenzoová kyselina 3-ŕerc-butyladipová3 - ((5-bromo-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl) -amino) -benzoic acid n-ethyl-1-aspartic acid n-alpha-fmoc-n-beta -boc-d-diaminopropionic acid n-tert-boc- (2s, 3r) -amino-2-hydroxy-4- (4-nitrophenyl) butyric acid 2,6-pyridinedicarboxylic acid 3-dibenzo (a, c) phenazine- 11-yl-acrylic acid valerenic acid nicotinic acid, n-oxide 4-chlorophenyl-cyclohexanecarboxylic acid 4- (p-chlorophenoxy) butyric acid n-tris [hydroxymethyl] methyl-4-aminobutanesulfonic acid s-4-nitromanedioic acid 4,5 -dichloro-2-fluorobenzoic acid n- (2,3-xylyl) glutaramic acid 4,5,5-trifluoro-4-pentenoic acid 5-fluoro-2,6-dihydroxy-pyrimidine-4-carboxylic acid 3-phenylsalicylic acid 2- (2-hydroxy-5-methyl-benzoyl) -benzoic acid cis-4-cyclohexene-1,2-dicarboxylic acid 2-bromostearic acid / trans -pyrrolidine-2,4-dicarboxylic acid 2-chlorobenzoic acid 5-sulfonic acid of 3-thiophenecarboxylic acid and 2 - ((3-methoxy-phenyl) -phenyl-methylene) -succinic acid 3-chlorocinnamic acid 4-phenylcinnamic acid 3- (3,5-dinitro-4-hydroxyphenyl) propionic acid 7-acetoxycoumarin-3-carboxylic acid d-alpha-galacturonic acid 3-bromo-2,5,6-trimethoxybenzoic acid 3-tert-butyladipic acid

• ·· • · • ··· • ·· • · • ··· ·· • · • · · · • · • · ···· • • ···· • • ·· · • · ·· • · · ·· · • · ·· • · · ·· ·· ·· ·· «· «· ·· · · ·· ·· ·· ··

kyselina 2-metylnonánová kyselina 3-hydroxy-4-metyl-2-nitrobenzoová kyselina 2,6-dihydroxy-4-metyl-benzoová kyselina 7-(3,3-dimetyl-2,3-benzofurán-5-yl)-3-metyl-okta-2,4,6-triénová kyselina 5-metoxy-2-propyl-izoftalová kyselina 3-(3-benzyloxy-4,5-dimetoxy-fenyl)-propiónová kyselina (1 s,2s )-(+)-1,2-cyklohexándikarboxylová kyselina 2-(amidínotio)etánsulfónová kyselina d-(-)-s-benzoyl-b-merkaptoizomaslová kyselina 3-fluór-5-(trifluórmetyl)benzoová kyselina 2-(9h-fluorén-9-ylmetoxykarbonylamino)-3-hydroxy-maslová kyselina 2-bróm-4-nitro-benzoová kyselina (s)-2-etyldekánová kyselina 11-fenoxyundekánová kyselina 2-nitro-6-(2,4-pentadién-1-yloxy)benzoová kyselina 5-(metánsulfonyl)tiofén-2-karboxylová kyselina 2-(4-fluórbenzoyl)benzoová kyselina 2-benzoyl-3,6-dimetylbenzoová kyselina 2-karboetoxysyringová kyselina 3,3’4,4’,5,6-hexachlórftalanilová kyselina 3-metyltiopropiónová kyselina (+/-)-abscisová (([R/S]-5-[1 -hydroxy-2,6,6-trimetyl-4-oxocyklohex-2-en-1 -yI]-2-methylnonanoic acid 3-hydroxy-4-methyl-2-nitrobenzoic acid 2,6-dihydroxy-4-methylbenzoic acid 7- (3,3-dimethyl-2,3-benzofuran-5-yl) -3 -methyl-octa-2,4,6-trienoic acid 5-methoxy-2-propyl-isophthalic acid 3- (3-benzyloxy-4,5-dimethoxy-phenyl) -propionic acid (1 s, 2s) - (+ ) -1,2-Cyclohexanedicarboxylic acid 2- (amidinothio) ethanesulfonic acid d - (-) - s-benzoyl-b-mercaptoisobutyric acid 3-fluoro-5- (trifluoromethyl) benzoic acid 2- (9h-fluoren-9-ylmethoxycarbonylamino) ) -3-Hydroxy-butyric acid 2-bromo-4-nitro-benzoic acid (s) -2-ethyldecanoic acid 11-phenoxyundecanoic acid 2-nitro-6- (2,4-pentadien-1-yloxy) benzoic acid 5 - (methanesulfonyl) thiophene-2-carboxylic acid 2- (4-fluorobenzoyl) benzoic acid 2-benzoyl-3,6-dimethylbenzoic acid 2-carboethoxysyring acid 3,3'4,4 ', 5,6-hexachlorophthalanic acid 3- methylthiopropionic acid (+/-) - abscisic acid (([R / S] -5- [1-hydroxy-2,6,6-trimethyl-4-oxocycle) lohex-2-en-1-yl] -

3-metyl-[2z,4e]-pentándiénová kyselina 4-chlór-3-nitrofenyloctová kyselina 2-oktínová kyselina 3-(4-azidofenyl)propiónová kyselina 9,10-dihydro-9,10-etanoantracén-11-karboxylová kyselina (2-hydroxyimino-propionylamino)-octová kyselina n-(4-etoxykarbonylfenyl)ftalámová kyselina d/-2-amino-3-fosfonopropiónová kyselina 2-(2-dibenzo(a,d)cykloheptén-5-ylidén-etyl)malónová kyselina 7-fenylheptánová3-methyl- [2z, 4e] -pentanedienoic acid 4-chloro-3-nitrophenylacetic acid 2-octanoic acid 3- (4-azidophenyl) propionic acid 9,10-dihydro-9,10-ethanoanthracene-11-carboxylic acid ( 2-hydroxyimino-propionylamino) -acetic acid N- (4-ethoxycarbonylphenyl) phthalic acid d -2-amino-3-phosphonopropionic acid 2- (2-dibenzo (a, d) cyclohepten-5-ylidene-ethyl) malonic acid 7-phenylheptanoic

• ·· • · • ··· • · · • ·· • · • ··· • · · ·· ···· • · · • · · • · · · · ·· ···· • · · • · · • · · · · ·· • · • t • 9 ·· • · • t • 9 99 99 • · ·· • · ·· ·· ·· ·· ·· 99 99 99 99

kyselina 5-bróm-4,4,5,5-tetrafluórpentánová kyselina 8-benzoyloktánová kyselina 3-hydroxy-5-( 1 -hydroxy-1 -metyl-etyl)-cyklohexánkarboxylová kyselina 3-dodecénová kyselina n-(1 -naftyO-SAS.e-tetrachlórftalámová kyselina 4-(trifluórmetyl)fenyloctová kyselina 5-acetamidometyl-3-merkaptopropiónová kyselina dihydroantracén-9,10-dikarboxylová kyselina mezo-2,5-dibrómadipová kyselina 2,3-dibróm-2’-metoxy-5’-metylsukcínanilová kyselina 3-chlór-4-(izopropylsulfonyl)-5-(metyltio)tiofén-2-karboxylová kyselina 4-n-propylbenzoová kyselina 2,3-dibróm-3-(2-(metoxykarbonyl)fenylkarbamoyl)propiónová kyselina 10-heptadecénová kyselina 3-metoxyfenoxyoctová kyselina 4,4'-dimetylénbisfenyloctová kyselina 4-chlór-3,5-dinitrobenzoová kyselina dietylfosfónoctová kyselina (1 r)-(-)-(1 -aminopropyl)fosfónová kyselina (r)-3-(4-fluórfenyl)butánová kyselina fenazín-1,6-dikarboxylová kyselina [1 r-(exo,exo)]-3-(benzoyloxy)-8-azabicyklo[3.2.1 ]oktán-2beta-karboxylová kyselina 2'-fliiórftalanilová kyselina 4-bróm-3-metylbenzoová kyselina 3-(morfolín-4-karbotioylsulfanyl)-propiónová kyselina (6-jód-benzo(1,3)dioxol-5-yl)-octová kyselina 3'-fluórhexahydroftalanilová kyselina 1 -fenylsulfonyl-4,4-piperidíndikarboxylová kyselina 2-(3,5-xylyl)octová kyselina beta-chlórmliečna kyselina 10,12-heptakozadiínová kyselina n-acetyl-1-tiazolidín-4-karboxylová5-Bromo-4,4,5,5-tetrafluoropentanoic acid 8-Benzoyloctanoic acid 3-Hydroxy-5- (1-hydroxy-1-methyl-ethyl) -cyclohexanecarboxylic acid 3-Dodecenoic acid n- (1-naphthyl-) SAS.e-tetrachlorophthalic acid 4- (trifluoromethyl) phenylacetic acid 5-acetamidomethyl-3-mercaptopropionic acid dihydroanthracene-9,10-dicarboxylic acid meso-2,5-dibromadipic acid 2,3-dibromo-2'-methoxy-5 ' 3-chloro-4- (isopropylsulfonyl) -5- (methylthio) thiophene-2-carboxylic acid 4-n-propylbenzoic acid 2,3-dibromo-3- (2- (methoxycarbonyl) phenylcarbamoyl) propionic acid 10- heptadecenic acid 3-methoxyphenoxyacetic acid 4,4'-dimethylenebisphenylacetic acid 4-chloro-3,5-dinitrobenzoic acid diethylphosphonic acid (1 r) - (-) - (1-aminopropyl) phosphonic acid (r) -3- (4-) fluorophenyl) butanoic acid phenazine-1,6-dicarboxylic acid [1 '- (exo, exo)] - 3- (benzoyloxy) -8-azabicyclo [3.2.1] octane-2-beta-carboxy 2'-Fluoro-phthalanic acid 4-bromo-3-methyl-benzoic acid 3- (morpholine-4-carbothioylsulfanyl) -propionic acid (6-iodo-benzo (1,3) dioxol-5-yl) -acetic acid 3'- 1-Phenylsulfonyl-4,4-piperidinedicarboxylic acid 2- (3,5-xylyl) acetic acid beta-chloro-lactic acid 10,12-heptacosadioic acid n-acetyl-1-thiazolidine-4-carboxylic acid

-26* ·· ·· ···· ·· •·· ·· ···· • ··· · · · · · • · · · · · ··· · *·· ·· ·· ·· ·· · kyselina 6-hydroxy-2,5,7,8-tetrametylchroman-2-karboxylová kyselina trans-15-oktadecénová kyselina 2,-(hydroxymetyl)-2-bifenylkarboxylová kyselina kumalínová kyselina n-(2,4,6-trimetylfenylkarbamoylmetyl)iminodioctová kyselina 2-(3,4-dimetoxy-fenyl)-3-(2-nitro-fenyl)-akrylová kyselina korková kyselina heptadekándiová kyselina 2’,4,,6,-trimetylmaleanilová kyselina uramil-n,n-dioctová kyselina (2,3-xylyl)fosfónová kyselina 6-chlórkynurénová kyselina 8-jód-1-naftoová-26 * ·· ······································· 6-hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acid trans-15-octadecenic acid 2 , - (hydroxymethyl) -2-biphenylcarboxylic acid cumalic acid n- (2,4,6- trimethyl phenylcarbamoylmethyl) iminodiacetic acid 2- (3,4-dimethoxy-phenyl) -3- (2-nitro-phenyl) -acrylic acid, suberic acid heptadecanedioic acid 2 ', 4, 6, -trimetylmaleanilová Urama acid-n, n-diacetic acid (2,3-xylyl) phosphonic acid 6-Chloro-kenyenic acid 8-iodo-1-naphthoic acid

4-(1,1,2,2-tetrafluóretoxy)benzoová kyselina 3-n-(4-metylfenyl)karbamoyl)-5-norbornén-2-karboxylová kyselina elaidová kyselina n,n,n’,n -1,4-fenyléndiamintetraoctová kyselina 3-(3,4-dichlórbenzoyl)-2-(4-metylfenyl)propiónová kyselina 3-fenyl-pyrolo(2,1,5-cd)indolizín-1,2-dikarboxylová kyselina fenylglycín-o-karboxylová kyselina 2,4-dimetyl-6-(2'-metylpropyl)benzén-1,2’-dikarboxylová kyselina 4-benzoylmaslová kyselina n-alfa-n-beta-d/-z-1 -diaminopropiónová kyselina 4-((6-fenyl)-1,3,5-hexatrienyl)benzoová kyselina 4-(2-chlóretyl)benzoová kyselina (2,2-difluór-adamantan-1 -yl)-octová kyselina ŕrans-2-okténová kyselina cis,c/s-2,5-dimetylmukonová kyselina 4-(fluórsulfonyl)benzoová kyselina 2-[[(4-chlórfenyl)sulfonyl]-(2-pyridyl)amino]octová beta-n-oxalylamino-1 -alanín kyselina oktánová * ·· ·· ···· ·· ·· · · · ···· • ··· · · · · ·4- (1,1,2,2-tetrafluoroethoxy) benzoic acid 3-N- (4-methylphenyl) carbamoyl) -5-norbornene-2-carboxylic acid elaidic acid n, n, n ', n -1,4- Phenylenediaminetetraacetic acid 3- (3,4-dichlorobenzoyl) -2- (4-methylphenyl) propionic acid 3-phenyl-pyrrolo (2,1,5-cd) indolizine-1,2-dicarboxylic acid phenylglycine-o-carboxylic acid 2 4-Dimethyl-6- (2'-methylpropyl) benzene-1,2'-dicarboxylic acid 4-Benzoylbutyric acid n-alpha-n-beta-d-z-1-diaminopropionic acid 4 - ((6-phenyl) (-1,3,5-hexatrienyl) benzoic acid 4- (2-chloroethyl) benzoic acid (2,2-difluoro-adamantan-1-yl) -acetic acid trans-2-octenoic acid cis, cis-2 5-dimethylmuconic acid 4- (fluorosulfonyl) benzoic acid 2 - [[(4-chlorophenyl) sulfonyl] - (2-pyridyl) amino] acetic acid beta-n-oxalylamino-1-alanine octanoic acid * ·· ·· ··· ·················

-27kyselina 1-dihydroorotová (orotová = tetrahydro-4-pyrimidínkarboxylová) kyselina 14-hydroxy-10,12-tetradekadiínová kyselina 4-(2,5-dimetylfenyl)maslová kyselina 2,2-difluór-2-fenoxyoctová kyselina n-[3-(trifluórmetyl)fenyl)maleámová kyselina n-karbamyl-d/-alfa-amino-n-maslová-27 1-dihydroorotic acid (orotic acid = tetrahydro-4-pyrimidinecarboxylic acid) 14-hydroxy-10,12-tetradecadioic acid 4- (2,5-dimethylphenyl) butyric acid 2,2-difluoro-2-phenoxyacetic acid n- [3 - (trifluoromethyl) phenyl) maleic acid n-carbamyl-N-alpha-amino-n-butyric acid

1-(m-sulfofenyl)-3-metyl-5-pyrazolón kyselina acenaftén-5-yl-octová kyselina c/s-15-oktadecénová kyselina benzo(c)fenantrén-6-karboxylová kyselina 2-chlór-5-jódbenzoová kyselina 1 -(4-fluórfenyl)cyklopentánkarboxylová kyselina 3-hepténová kyselina chromon-3-karboxylová kyselina (s)-(-)-2-chlórpentánová kyselina 3-(2,5-dimetyl-fenyl)-3-metyl-maslová kyselina (s)-(+)-2-bróm-3-fenylpropiónová kyselina cyklohexylfenyloctová kyselina 3,3’,3”-nitrilotripropiónová kyselina 2-bifenylkarboxylová kyselina (4-chlór-3,5-dimetyl-fenoxy)-octová kyselina 4-(2-amino-5-bróm-3-etyl-fenyl)-4-oxo-maslová kyselina 3,4-metyléndioxyškoricová kyselina 5-(2-nitrofenyl)-2-furoová kyselina 4’-bróm-3,-metylsukcínanilová kyselina 2,3-dihydrobenzofurán-7-karboxylová kyselina 4-(2,4-d/-terc-pentyl-fenoxy)-maslová kyselina 4-(3,4-dimetoxyfenyl)maslová kyselina 2[(5-chlór-4,6-dimetoxypyrimidín-2-yl)oxy]benzoová kyselina 9-antracénkarboxylová kyselina (r)-3-(4-ferc-butoxyfenyl)butánová kyselina 5,5'-metyléndisalicylová ·· ·· 999t 99 • 9 9 9 9 91- (m-sulfophenyl) -3-methyl-5-pyrazolone acenaphthen-5-yl-acetic acid cis-15-octadecenic acid benzo (c) phenanthrene-6-carboxylic acid 2-chloro-5-iodobenzoic acid 1- (4-fluorophenyl) cyclopentanecarboxylic acid 3-heptenoic acid chromone-3-carboxylic acid (s) - (-) - 2-chloropentanoic acid 3- (2,5-dimethylphenyl) -3-methylbutyric acid ( s) - (+) - 2-bromo-3-phenylpropionic acid cyclohexylphenylacetic acid 3,3 ', 3'-nitrilotripropionic acid 2-biphenylcarboxylic acid (4-chloro-3,5-dimethyl-phenoxy) -acetic acid 4- ( 2-amino-5-bromo-3-ethyl-phenyl) -4-oxo-butyric acid 3,4-methylenedioxycinnamic acid 5- (2-nitrophenyl) -2-furoic acid 4'-bromo-3 , -methylsuccinilic acid 2 4- (2,4-di-tert-pentyl-phenoxy) -butyric acid 3-dihydrobenzofuran-7-carboxylic acid 4- (3,4-dimethoxyphenyl) butyric acid 2 [(5-chloro-4,6- dimethoxypyrimidin-2-yl) oxy] benzoic acid 9-anthracenecarboxylic acid (r) -3- (4-tert-but oxyphenyl) butanoic acid 5,5'-methylenedisalicylic acid ·· ·· 999t 99 • 9 9 9 9 9

999 9 9 9 9 9999 9 9 9 9 9

-28kyselina 4-metylnonánová kyselina 2-fluór-6-jódbenzoová kyselina 1 -(+)-s-acetyl-beta-meraptoizomaslová kyselina r(+)-2-(2,4-dichlórfenoxy) propiónová kyselina (+/-)-5,6-epoxyeikoza-8z,11z,14z-triénová kyselina 1,6-naftaléndikarboxylová kyselina 3-izobutyrylamino-3-fenyl-propiónová kyselina (z)-(3)-jódakrylová-28 4-methylnonanoic acid 2-fluoro-6-iodobenzoic acid 1- (+) - s-acetyl-beta-mercaptoisobutyric acid r (+) - 2- (2,4-dichlorophenoxy) propionic acid (+/-) - 5,6-epoxyeicoza-8z, 11z, 14z-trienoic acid 1,6-naphthalenedicarboxylic acid 3-isobutyrylamino-3-phenyl-propionic acid (z) - (3) -iodo-acrylic acid

1-(4’-sulfofenyl)-3-karboxy-5-pyrazolón kyselina 4-(3-fenyl-2-tioureido)hipurová kyselina 4-(2-(2-hydroxy-fenoxy)-acetylamino)-benzoová kyselina 1-etyl-4-oxo-1,4-dihydrochinolín-3-karboxylová kyselina 6-(trifluórmetyl)nikotínová kyselina 5-norbornén-2-endo-3-exo-dikarboxylová kyselina 4’-bróm-2'-chlórsukcínanilová kyselina 2-acetoxy-3-metylbenzoová kyselina 4-chlór-3-nitroškoricová kyselina 2-(benzénsulfonyl)etyltio-octová kyselina 11-(metoxykarbonylmetyltio)-undekánová kyselina c/s-3',5'-dimetylhexahydroftalanilová kyselina 2,6-dichlórfenoxyoctová kyselina 3-chlór-4-hydroxyfenyloctová kyselina 7-[(4-amino-3-sulfofenyl)amino]-4-hydroxy-2-naftalénsulfónová kyselina n-alfa-(benzyloxykarbonyl)-alfa-(terc-butylester)-1-glutámová kyselina 6-ketoundekán-1,11-diová kyselina 6-amino-2-(2-ho-et)-1,3-dioxo-2,3-2h-1 h-benzo(de)izochinolín-5-sulfónová kyselina 3-nitrofenyloctová kyselina 5-metyl-2-tiofénkarboxylová kyselina 2-[3-dodekanoyl-hydrazíno)-3-oxo-propionylamino]-benzoová kyselina 4'-nitroftalanilová kyselina 3-nitro-4-fenoxybenzénsulfónová kyselina 1,2,3,4-butántetrakarboxylová1- (4'-Sulfophenyl) -3-carboxy-5-pyrazolone 4- (3-phenyl-2-thioureido) hipuric acid 4- (2- (2-hydroxy-phenoxy) -acetylamino) -benzoic acid 1- ethyl 4-oxo-1,4-dihydroquinoline-3-carboxylic acid 6- (trifluoromethyl) nicotinic acid 5-norbornene-2-endo-3-exo-dicarboxylic acid 4'-bromo-2'-chlorosuccinilic acid 2-acetoxy 3-methylbenzoic acid 4-chloro-3-nitrocinnamic acid 2- (benzenesulfonyl) ethylthioacetic acid 11- (methoxycarbonylmethylthio) -undecanoic acid cis-3 ', 5'-dimethylhexahydrophthalanic acid 2,6-dichlorophenoxyacetic acid 3- chloro-4-hydroxyphenylacetic acid 7 - [(4-amino-3-sulfophenyl) amino] -4-hydroxy-2-naphthalenesulfonic acid n-alpha- (benzyloxycarbonyl) -alpha- (tert-butyl ester) -1-glutamic acid 6 6-amino-2- (2-ho-et) -1,3-dioxo-2,3-2h-lh-benzo (de) isoquinoline-5-sulfonic acid-ketoundecane-1,11-dioic acid 3- nitrophenylacetic acid 5-methyl-2-thiophenecarboxylic acid 2- [3-dodecanoyl-hydrazino) -3- oxo-propionylamino] -benzoic acid 4'-nitropthalanilic acid 3-nitro-4-phenoxybenzenesulfonic acid 1,2,3,4-butanetetracarboxylic acid

• ·· • · 9 999 9 9 9 • ·· • · 9 999 9 9 9 99 9999 9 9 9 9 9 9 9 9 9 9 99 9999 9 9 9 9 9 9 9 • · • · 9 9 9 9 9 • · • · 9 9 9 9 9 99 99 99 99 99 99 99 99 99 99 99 99 99 99

kyselina (1s)-(+)-(1-aminohexyl)fosfónová kyselina (s)-3-fenylmaslová kyselina dietyléntriamínpentaoctová kyselina boc-d-2-aminomaslová kyselina 3-bróm-4-chlórpentafluórmaslová kyselina 2,4,6-trinitrobenzoová kyselina 2-nitrofenoxyoctová kyselina dl-homocysteínová kyselina (4-etylfenyl)fosfónová kyselina 4-(4-nitrofenyl)maslová kyselina c/s-cyklobután-1,2-dikarboxylová kyselina tieno(3,2-b)tiofén-2-karboxylová kyselina mezo-bután-1,2,3,4-tetrakarboxylová kyselina pentafluórbenzénsulfónová kyselina o-jódhipurová kyselina 4,5,6,7-tetrafluór-3-indoloctová kyselina 2-(fenetyltio)-octová kyselina 1-hydroxyetán-1,1-difosfónová kyselina 1,2-aminoadipová kyselina 6-oxoheptánová kyselina 2-formamido-3-tiofénkarboxylová kyselina 14-metylpentadekánová kyselina bis-(4-bróm-fenyl)-hydroxy-octová kyselina 3-jódpropiónová kyselina 2,6-dioxo-4-piperidínkarboxylová kyselina d-alfa-aminoadipová kyselina 3-bróm-5-chlór-2,6-dimetoxybenzoová kyselina orotová (tetrahydro-4-pyrimidínkarboxylová) kyselina 6-[2-acetylamino-3-(4-metoxy-fenyl)-akryloylamino]-hexánová kyselina 3-(4-chlórbenzénsulfonyl) maslová kyselina 2-brómizoftalová kyselina 3-amino-4-izopropenyl-benzoová(1s) - (+) - (1-Aminohexyl) phosphonic acid (s) -3-phenylbutyric acid diethylenetriaminepentaacetic acid boc-d-2-aminobutyric acid 3-bromo-4-chloropentafluorobutyric acid 2,4,6-trinitrobenzoic acid 2-nitrophenoxyacetic acid dl-homocysteic acid (4-ethylphenyl) phosphonic acid 4- (4-nitrophenyl) butyric cis -cyclobutane-1,2-dicarboxylic acid thieno (3,2-b) thiophene-2-carboxylic acid meso-butane-1,2,3,4-tetracarboxylic acid pentafluorobenzenesulfonic acid o-iodo-tonic acid 4,5,6,7-tetrafluoro-3-indole acetic acid 2- (phenethylthio) -acetic acid 1-hydroxyethane-1,1- diphosphonic acid 1,2-aminoadipic acid 6-oxoheptanoic acid 2-formamido-3-thiophenecarboxylic acid 14-methylpentadecanoic acid bis- (4-bromo-phenyl) -hydroxy-acetic acid 3-iodopropionic acid 2,6-dioxo-4- piperidinecarboxylic acid d-alpha-aminoadipic acid 3-bromo-5-chloro-2,6-dimethoxybenzoic acid or Acetic (tetrahydro-4-pyrimidinecarboxylic acid) 6- [2-acetylamino-3- (4-methoxyphenyl) -acryloylamino] -hexanoic acid 3- (4-chlorobenzenesulfonyl) butyric acid 2-bromoisophthalic acid 3-amino-4- isopropenyl-benzoic acid

-30kyselina 3-fenoxypropiónová kyselina n-(2-chlórfenyl)glutarámová kyselina 4-[(e)-2-(5,6,7,8-tetrahydro-5,5,8,8-tetrametyl-2-nafl:alenyl)-1-propenyl]benzoová kyselina 3-chlór-2-metylbenzoová kyselina 3-(3-etoxyfenyl)propiónová kyselina 2,-chlór-6,-metylftalanilová kyselina 4-[[2-fluór-5-(metylsulfonyl)fenyl]amino]-4-oxobutánová kyselina 3,6-dimetylsalicylová kyselina 3-(2,6-dichlórbenzyltio)-2-tiofénkarboxylová (s)-(-)-2-guanidínoglutárová kyselina 3,4-dinitrobenzoová kyselina alfa-trifenylmetyl-2-naftalénpropiónová kyselina 3,4-dichlórfenyloctová fenylbenzén-omega-fosfono-alfa-amino-kyselina kyselina n-metylhipurová kyselina hydrochinón-o.o-dioctová kyselina 3-(4-n-oktylbenzoyl)propiónová kyselina 11-metyltridekánová kyselina 3-cyklohexylpropiónová kyselina 3,5-d/-ferc-butyl-4-hydroxybenzoová kyselina (3-kyano-6-(4-metoxy-fenyl)-3-metyl-2-oxo-cyklohexyl)-octová kyselina 4-hydroxyizoftalová kyselina di(cyklohexyl)-fosforečná kyselina 3-aminoadipová kyselina (4-nitrobenzyl)fosfónová kyselina 4-(4-metoxy-fenyl)-4-metyl-pentánová kyselina 4-(2-hydroxybenzylidénamino)salicylová kyselina n-hexadecylfosfónová kyselina 4'-metoxyftalanilová kyselina 1-ho-8-imino-5-oxo-4-(4-sulfo-fenylamino)-5,8-2h-naftalén-2-sulfonová kyselina kainová (2-karboxy-3-karboxymetyl-4-izopropenylpyrolidín)3-Phenoxypropionic acid n- (2-chlorophenyl) glutaramic acid 4 - [(e) -2- (5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenenyl) -1-propenyl] benzoic acid 3-chloro-2-methylbenzoic acid 3- (3-ethoxyphenyl) propionic acid 2 , -chloro-6 , methylphthalanilic acid 4 - [[2-fluoro-5- (methylsulfonyl) phenyl] amino] -4-oxobutanoic acid 3,6-dimethylsalicylic acid 3- (2,6-dichlorobenzylthio) -2-thiophenecarboxylic acid (s) - (-) - 2-guanidinoglutaric acid 3,4-dinitrobenzoic acid alpha-triphenylmethyl-2- naphthalenepropionic acid 3,4-dichlorophenylacetic phenylbenzene-omega-phosphono-alpha-amino-acid n-methylhipuric acid hydroquinone-oo-diacetic acid 3- (4-n-octylbenzoyl) propionic acid 11-methyltridecanoic acid 3-cyclohexylpropionic acid 3, 5-tert-Butyl-4-hydroxybenzoic acid (3-cyano-6- (4-methoxyphenyl) -3-methyl-2-oxo-cyclohexyl) -acetic acid 4-hydroxyisophthalic acid di (cyclohexyl) - phosphoric acid 3-am inoadipic acid (4-nitrobenzyl) phosphonic acid 4- (4-methoxyphenyl) -4-methylpentanoic acid 4- (2-hydroxybenzylideneamino) salicylic acid n-hexadecylphosphonic acid 4'-methoxyphthalanilic acid 1-ho-8-imino -5-oxo-4- (4-sulfo-phenylamino) -5,8-2h-naphthalene-2-sulfonic acid kainic acid (2-carboxy-3-carboxymethyl-4-isopropenylpyrrolidine)

• · • · • · • ··· • · • ··· ·· • · • e ·· • · • e ···· • • ···· • • • · · • · ·· • · e • · · · ··· • · e ·· · ·· · ·· · · ·· · · ·· · · ·· ··· ·· ···

kyselina tetrahydrofurán-2,3,4,5-tetrakarboxylová kyselina 4-metyl-5-oxohexánová kyselina 12-oxo-12-(1 -pyrenyl)dodekánová kyselina alfa-izoatropová kyselina 4-(2-tienylmetylénamino)salicylová kyselina jodičná kyselina 2-fluórfenyloctová kyselina (benzoyl-benzyl-amino)-octová kyselina c/s-3-chlórakrylová kyselina 3-pyrimidín-2-yl-propiónová kyselina 2-(2-(3,4-dimetyl-fenoxy)-acetylamino)-benzoová kyselina malonámová kyselina (s)-(+)-(1-aminoetyl)fosfónová kyselina 6-metyl-2-pyridín-4-yl-chinolín-4-karboxylová kyselina 4,6-dimetyl-izoftalová d/-n-propylfosfát kyselina benzotiazol-2-yl-2-(2-aminotiazole-4-yl)-octová kyselina 5-(4-fluórbenzoyl)tiofén-2-octová kyselina 2-acetylamino-but-2-énová kyselina 4-fluór-2-(trifluórmetyl)benzoová kyselina 8,11-eikozadiínová kyselina n-(4-metylfenyl)tetrachlórftalámová kyselina 4'-butylhexahydroftalanilová kyselina etylxantogénoctová kyselina alfa-fenylcyklopentánoctová kyselina n-metyl-1-asparágová kyselina 3-bróm-5-metoxy-2-metyl-benzoová kyselina izo-oktyl-fosforečná kyselina 2-(2,2-dimetyl-propionylamino)-4,5,617-4h-benzo[b]tiofén-3-karboxylová kyselina 4-chlór-3-nitrobenzoylbenzoová kyselina n-(2-karboxyfenyl)malonámová kyselina 2,5-norbornadién-2,3-dikarboxylovátetrahydrofuran-2,3,4,5-tetracarboxylic acid 4-methyl-5-oxohexanoic acid 12-oxo-12- (1-pyrenyl) dodecanoic acid alpha-isoatropic acid 4- (2-thienylmethyleneamino) salicylic acid iodic acid 2 -fluorophenylacetic acid (benzoyl-benzyl-amino) -acetic acid cis-3-chloroacrylic acid 3-pyrimidin-2-yl-propionic acid 2- (2- (3,4-dimethyl-phenoxy) -acetylamino) -benzoic acid Malonic acid (s) - (+) - (1-aminoethyl) phosphonic acid 6-methyl-2-pyridin-4-yl-quinoline-4-carboxylic acid 4,6-dimethyl-isophthalic d-n-propylphosphate acid benzothiazol-2-yl-2- (2-aminothiazole-4-yl) -acetic acid 5- (4-fluorobenzoyl) -thiophene-2-acetic acid 2-acetylamino-but-2-enoic acid 4-fluoro-2- ( trifluoromethyl) benzoic acid 8,11-eicosadioic acid n- (4-methylphenyl) tetrachlorophthalic acid 4'-butylhexahydrophthalanic acid ethylxanthogenetic acid alpha-phenylcyclopentaneacetic acid n-methyl-1-aspartic acid yselina 3-bromo-5-methoxy-2-methyl-benzoic acid, iso-octyl-2-phosphoric acid (2,2-dimethyl-propionylamino) -4,5,6-1 7-4h [b] thiophene-3 4-chloro-3-nitrobenzoylbenzoic acid-2- (2-carboxyphenyl) malonamic acid 2,5-norbornadiene-2,3-dicarboxylic acid

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · ···· • • ···· • • ·· · • · ·· • · · ·· · • · ·· • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 3-benzyloxy-4,5-dimetoxy-benzoová kyselina 4-(2-izopropylsulfanyl-acetylamino)-benzoová kyselina 5-fluór-6-hydroxy-pyrimidín-4-karboxylová kyselina 2-(3-nitro-benzylidén)-pent-4-énová kyselina n-karbamoylmaleámová kyselina 4-(4-hydroxyfenoxy)benzoová kyselina tetrakozándiová kyselina 2-bróm-5-metoxybenzoová kyselina 4-formylškoricová kyselina (metyltio)octová kyselina 4-oxo-4-(4-(4-(etoxykarbonyl)butyl)fenyl)maslová kyselina 2,4-dichlórfenoxyoctová kyselina 4-((1,3-dioxo-1,3-dihydro-izoindol-2-ylmetyl)-amino)-benzoová kyselina 3,4-dimetoxyfenylpyrohroznová kyselina (s)-2-fluór-2-metylheptánová kyselina 2-benzoylamino-3-(4-benzyloxy-3-metoxy-fenyl)-akrylová kyselina 3-naftalén-1 -yl-propínová kyselina 4,4-dinitroheptándiová kyselina 3-benzo(1,3)dioxol-5-yl-propínová kyselina tetraacetyl-slizová kyselina c/s-hexahydro-n-(4-etoxyfenyl)ftalámová kyselina 3-[(3,5-dimetoxyfenyl)-(toluén-4-sulfonyl)-amino]-propiónová kyselina 3-(4-n-pentyloxybenzoyl)propiónová kyselina 2-chlórškoricová kyselina n-cyklohexylglutarámová kyselina (-)-c/s-2-benzamidocyklohexánkarboxylová kyselina d/-citrajablčná (ο-2-metyl-jablčná) kyselina 1 h-pyrazol-3,4-dikarboxylová kyselina 2-fluór-4-hexyloxybenzoová kyselina n-(3-chlór-2-metylfenyl)glutarámová kyselina trans-1,2-diaminocyklohexán-n,n,n’,n’-tetraoctová kyselina 2,2-dichlóroktadekánová monohydrát3-Benzyloxy-4,5-dimethoxy-benzoic acid 4- (2-isopropylsulfanyl-acetylamino) -benzoic acid 5-fluoro-6-hydroxy-pyrimidine-4-carboxylic acid 2- (3-nitro-benzylidene) -pent 4-enoic acid n-carbamoylmaleamic acid 4- (4-hydroxyphenoxy) benzoic acid tetracosanedioic acid 2-bromo-5-methoxybenzoic acid 4-formylcinnamic acid (methylthio) acetic acid 4-oxo-4- (4- (4- (4- ( ethoxycarbonyl) butyl) phenyl) butyric acid 2,4-dichlorophenoxyacetic acid 4 - ((1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl) amino) benzoic acid 3,4-dimethoxyphenylpyruvic acid (s -2-fluoro-2-methylheptanoic acid 2-benzoylamino-3- (4-benzyloxy-3-methoxyphenyl) -acrylic acid 3-naphthalen-1-yl-propionic acid 4,4-dinitroheptanedioic acid 3-benzo ( 1,3) dioxol-5-yl-propionic acid tetraacetyl-mucic acid cis-hexahydro-1- (4-ethoxyphenyl) phthalic acid 3 - [(3,5-dimethoxyphenyl) - (toluene-4-sulfonyl) - amino] -propionic acid 3- (4-n-pentyloxybe) nzoyl) propionic acid 2-chlorocinnamic acid n-cyclohexylglutaramic acid (-) - cis-2-benzamidocyclohexanecarboxylic acid d-citric acid (ο-2-methyl-malic acid) 1 h-pyrazole-3,4-dicarboxylic acid 2 -fluoro-4-hexyloxybenzoic acid n- (3-chloro-2-methylphenyl) glutaramic acid trans-1,2-diaminocyclohexane-n, n, n ', n'-tetraacetic acid 2,2-dichlorooctadecanoic monohydrate

• ·· • ·· ·· ···· ·· ···· • · • · ·· · ·· · • · · • · · • · • · ·· · · • ··· • ··· • · · • · · • · • · • · · • · · ♦ · · · · ♦ · · · · • · • · ·· · ·· ·· · ·· ·· ·· ·· ·· ·· · · ·· · ·

kyselina 2-fluór-6-(trifluórmetyl)škoricová kyselina boc-cA7-hyclroxy-1,2,3,4-tetrahydrOizochinolín-3-karboxylová kyselina 5-(3-metoxy-fenyl)-hexa-2,4-diénová kyselina 5-(4-hydroxy-3-metoxy-fenyl)-pentánová kyselina 5-(alfa,alfa-dimetyl-4-hydroxybenzyl)salicylová kyselina 3-decénová kyselina n-benzyliminodioctová kyselina n-alfa-(benzyloxykarbonyl)-1 -glycyl-1 -glycín kyselina (4-etoxyfenyl)fenylfosfínová kyselina (4'-karboxymetylsulfanyl-bifenyl-4-ylsulfanyl)-octová kyselina 1-metylorotová kyselina 3-(3,5-ď/-ŕerc-butyl-benzoylamino)-benzoová kyselina 4-(2,5-dioxo-2,5-dihydro-pyrol-1 -yl)-benzoová kyselina 2,,5'-dimetoxymaleanilová kyselina boc-alfa-aminomaslová kyselina (3-nitro-fenyl)-fosfónová kyselina 4-(2-acetylamino-3-fenyl-akryloylamino)-maslová kyselina 2,2-bis-(4-chlórfenyl)-octová kyselina 1 -alfa-glutamyl-1 -alfa-glutamyl-1 -glutámová kyselina 4-(trifluórmetoxy)fenoxyoctová kyselina 2-én-valproová (2-propyl-pentánová) kyselina n-(o-tolyl)ftalimidová kyselina n-(2-etylfenyl)glutarámová kyselina 2,4,6-trihydroxybenzoová kyselina c/s-2-hydroxy-1 -cyklopentánkarboxylová kyselina difenylfosfínová kyselina 4-(4-metoxyfenyl)tiofén-2-karboxylová kyselina 4-(4-metylbenzylidénamino)salicylová kyselina (2,2l2-trichlór-1-(3-p-tolyl-tioureido)-etyl)-karbámová kyselina (s)-(+)-alfa-hydroxy-1,3-dioxo-2-izoindolínmaslová kyselina 2,2’-(1,2-etándiyl)bis[5-aminobenzénsulfónová] kyselina 4'-nitromaleanilová • ·· ·· ···· ·· ·· · · · ···· • ··· · · · · ·2-fluoro-6- (trifluoromethyl) cinnamic acid boc-A7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid 5- (3-methoxyphenyl) -hexa-2,4-dienoic acid 5- (4-hydroxy-3-methoxyphenyl) -pentanoic acid 5- (alpha, alpha-dimethyl-4-hydroxybenzyl) salicylic acid 3-decenoic acid n-benzyliminodiacetic acid n-alpha- (benzyloxycarbonyl) -1-glycyl -1-Glycine (4-ethoxyphenyl) phenylphosphinic acid (4'-carboxymethylsulfanyl-biphenyl-4-ylsulfanyl) -acetic acid 1-methylorotic acid 3- (3,5-tert-butyl-benzoylamino) -benzoic acid 4- (2,5-dioxo-2,5-dihydro-pyrrol-1-yl) -benzoic acid 2,5 ' , 5'-dimethoxymaleanilic acid boc-alpha-aminobutyric acid (3-nitro-phenyl) -phosphonic acid 4- (2-Acetylamino-3-phenyl-acryloylamino) -butyric acid 2,2-Bis- (4-chlorophenyl) -acetic acid 1-alpha-glutamyl-1-alpha-glutamyl-1-glutamic acid 4- (trifluoromethoxy) phenoxyacetic acid 2-en-valproic acid (2-propyl-pentanoic acid) n- (o-tol yl) phthalimic acid n- (2-ethylphenyl) glutaramic acid 2,4,6-trihydroxybenzoic acid cis-2-hydroxy-1-cyclopentanecarboxylic acid diphenylphosphinic acid 4- (4-methoxyphenyl) thiophene-2-carboxylic acid 4- (4-methylbenzylidenamino) salicylic acid (2,2 L 2-trichloro-1- (3-p-tolyl-thioureido) ethyl) -carbamic acid (s) - (+) - alpha-hydroxy-1,3-dioxo -2'-isoindolinebutyric acid 2,2 '- (1,2-ethanediyl) bis [5-aminobenzenesulfonic acid] 4'-nitromaleanilic acid • ··········· ·· · · · · ·

-34kyselina 3,5-diizopropoxybenzoová kyselina n-(4-(4-chlór-fenoxy)-fenyl)-ftalámová kyselina benzoylamino-fenyl-octová kyselina 4-chlór-3-nitrobenzoová kyselina 4-metylftalová kysel ina beta-(2-acetoxyfenyI)propiónová kyselina (3-fluórfenyl)fosfónová kyselina (r,r)-(-)-2,3-difenyljantárová kyselina 2-(4-chlórfenyl)-1-(2-(3,4-dimetoxyfenyl)etyl)-6-oxo-3-piperidínkarboxylová kyselina etoxyoctová kyselina 3-(3-(2,4,5-trichlórfenyl)ureido)benzoová kyselina 2-[3-oxo-3-(n’-tetradekanoyl-hydrazíno)-propionylamino]benzoová kyselina 2-(2-(2-chlórfenyl)-4-fenyltiazol-5-yl)octová kyselina 4-(benzylidénamino)benzoová kyselina heneikozánová kyselina c/s-hexahydro-n-(3-nitrofenyl)ftalámová kyselina 3-(n-cyklohexylkarbamoyl)-5-norbornén-2-karboxylová kyselina cyklohexánkarboxylová kyselina 3-(2-hydroxyfenyl)propiónová kyselina 3’-fluórglutaranilová kyselina tetrafluórtereftalová kyselina 4-acetamido-3-fluórbenzoová kyselina dihydroxyfumárová kyselina 4-butoxyfenyloctová kyselina d/-beta-hydroxypalmitová kyselina 13-keto-oktadeka-9z,11e-diénová kyselina 1 -propionyl-pyrolidín-2-karboxylová kyselina 3',5'-dichlór-2'-hydroxy-4’-metylmaleanilová kyselina 3-(trifenylsilyl)propiónová kyselina 2-metyl-2-penténová kyselina (3-chlórfenyl)fosfónová kyselina 3-(tiofén-3-ylsulfanyl)-tiofén-2-karboxylová-34-3,5-diisopropoxybenzoic acid n- (4- (4-chloro-phenoxy) -phenyl) -phthalic acid benzoylamino-phenyl-acetic acid 4-chloro-3-nitrobenzoic acid 4-methylphthalic acid beta- (2- acetoxyphenyl) propionic acid (3-fluorophenyl) phosphonic acid (R, R) - (-) - 2,3-diphenylsuccinic acid 2- (4-chlorophenyl) -1- (2- (3,4-dimethoxyphenyl) ethyl) - 6-oxo-3-piperidinecarboxylic acid ethoxyacetic acid 3- (3- (2,4,5-trichlorophenyl) ureido) benzoic acid 2- [3-oxo-3- (n'-tetradecanoyl-hydrazino) -propionylamino] benzoic acid 2- (2- (2-chlorophenyl) -4-phenylthiazol-5-yl) acetic acid 4- (benzylideneamino) benzoic acid heneicosanoic acid cis-hexahydro-1- (3-nitrophenyl) phthalic acid 3- (n- cyclohexylcarbamoyl) -5-norbornene-2-carboxylic acid cyclohexanecarboxylic acid 3- (2-hydroxyphenyl) propionic acid 3'-fluoroglutaranilic acid tetrafluoro-terephthalic acid 4-acetamido-3-fluorobenzoic acid dihydroxyfumaric acid 4-butoxyphenylacetic acid d-beta-hydroxypalmitic acid 13-keto-octadeca-9z, 11e-dienoic acid 1-propionyl-pyrrolidine-2-carboxylic acid 3 ', 5'-dichloro-2'-hydroxy-4'-methylmaleanilic acid 3- (triphenylsilyl) propionic acid 2-methyl-2-pentenoic acid (3-chlorophenyl) phosphonic acid 3- (thiophen-3-ylsulfanyl) -thiophene-2-carboxylic acid

• · · • · • ··· • · · • ··· ·· • · 0 0 · · • · 0 0 • · · · • • • · · · • • · · • · ·· • · · • · · · ··· • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 3-fluór-4-metoxybenzoová kyselina 3-(4-bifenylyloxy)propiónová kyselina boc-gama-aminomaslová kyselina 4,5-dimetoxy-2-nitrofenyloctová kyselina 3-(2,4-dihydroxyfenyl)propiónová kyselina 2-hexadecylkarbamoyl-4-nitrobenzoová kyselina 3-fluór-4-hydroxyfenyloctová kyselina 4-(trifluórmetoxy)fenyloctová kyselina benzoylmravčia kyselina gáfrová kyselina 5-benzo(1,3 )dioxol-5-yl-penta-2,4-diénová kyselina 2,3,4-trimetoxyfenyloctová kyselina 2-(315-dinitro-tiofén-2-ylamino)-3-metyl-maslová kyselina 3-(4-metoxy-fenyl)-2-(1-fenyl-etylidénamino)-akrylová kyselina L-askorbová kyselina metyljantárová kyselina (-)-izoborneol-3-octová kyselina 1,1,2-cyklopropántrikarboxylová kyselina indol-6-karboxylová kyselina 4-(hexadecyltio)benzénsulfonová kyselina hexahydro-n-(2,3-xylyl)ftalámová kyselina (r)-(+)-n-(1-fenyletyl)sukcínamová kyselina 2,6-naftaléndikarboxylová kyselina 5-chlór-2-jódbenzoová kyselina 2-(4-brómbenzoyl)-akrylová kyselina 2-fluór-3-(trifluórmetyl)škoricová kyselina 8,8’-diapokaroténdiová kyselina 5,6-dichlórvanilová kyselina 3-hydroxytridekánová kyselina 2-([2-[3-chlór-5-(trifluórmetyl)-2-pyridyl-hydrazíno-karbonyl)benzoová kyselina 2-metoxy-9-oxo-8,9-dihydro-7h-benzocykloheptén-5-karboxylová kyselina c/s-5,8,11-eikozatriénová • ·· ·· ···· ·· ·· · ·· ···· • ··· · · · · ·3-fluoro-4-methoxybenzoic acid 3- (4-biphenylyloxy) propionic acid boc-gamma-aminobutyric acid 4,5-dimethoxy-2-nitrophenylacetic acid 3- (2,4-dihydroxyphenyl) propionic acid 2-hexadecylcarbamoyl-4 -nitrobenzoic acid 3-fluoro-4-hydroxyphenylacetic acid 4- (trifluoromethoxy) phenylacetic acid benzoyl formic acid camphoric acid 5-benzo (1,3) dioxol-5-yl-penta-2,4-dienoic acid 2,3,4- trimethoxyphenylacetic acid 2- (3 1 5-dinitro-thiophen-2-ylamino) -3-methyl-butyric acid 3- (4-methoxy-phenyl) -2- (1-phenyl-ethylideneamino) -acrylic acid, L-ascorbic acid methylsuccinic acid (-) - isoborneol-3-acetic acid 1,1,2-cyclopropanetricarboxylic acid indole-6-carboxylic acid 4- (hexadecylthio) benzenesulfonic acid hexahydro- (2,3-xylyl) phthalic acid (r) - (+) - n- (1-phenylethyl) succinamic acid 2,6-naphthalenedicarboxylic acid 5-chloro-2-iodobenzoic acid 2- (4-bromobenzoyl) -acrylic acid 2-fluoro-3 - (trifluoromethyl) cinnamic acid 8,8'-diapocarotenedioic acid 5,6-dichloro-vanoic acid 3-hydroxytridecanoic acid 2 - ([2- [3-chloro-5- (trifluoromethyl) -2-pyridyl-hydrazino-carbonyl) benzoic acid 2-Methoxy-9-oxo-8,9-dihydro-7H-benzocycloheptene-5-carboxylic acid cis-5,8,11-eicosatrienoic acid · · · · · · · · · ··· • ··· · · · · ·

-36kyselina 3-hydroxymaslová kyselina 2-nitro-4-(trifluórmetyl)fenyltioglykolová kyselina 2,4-bis(trifluórmetyl)fenyloctová kyselina 4-hydroxy-alfa-merkapto-3-metoxyškoricová kyselina 4-chlór-nitrobenzénsulfónová3-hydroxy-butyric acid 2-nitro-4- (trifluoromethyl) phenylthioglycolic acid 2,4-bis (trifluoromethyl) phenylacetic acid 4-hydroxy-alpha-mercapto-3-methoxycinnamic acid 4-chloro-nitrobenzenesulfonic acid

4-metylumbeliferyl-fosfát kyselina 2,,5,-dimetylftalanilová kyselina 3-(naftalén-2-sulfonyl)-propiónová kyselina 2',6’-diizopropylglutaranilová kyselina 2-(3,4-dimetoxystyryl)glyoxylová kyselina 6-(4-(3-karboxy-propyl)-fenyl)-hexánová kyselina metavínna kyselina dodekafluórkorková kyselina fenolsulfónová kyselina 5-bróm-2,4-dihydroxybenzoová kyselina 2-(9h-fluóren-9-ylmetoxykarbonylamino)-3-fenyl-propiónová kyselina 4-butyloxybifenyl-4’-karboxylová kyselina p-fenylazobenzénsulfónová kyselina 4-metylsulfonylfenyloctová kyselina 3-benzyloxy-4-metoxy-2-nitro-benzoová kyselina 4,5-dihydro-4I5-dioxo-1h-pyrolo[2,3-f]chinolíne-2,7,9-trikarboxylová kyselina 2'-(trifluórmetyl)maleanilová kyselina 2-benzoylbenzoová kyselina 4-chlór-2-(2-tienyletyl)benzoová kyselina r-(-)-hexahydromandlová kyselina 2,5-dichlór-4-metoxy-benzoová kyselina benzyloxykarbonyl-d-pyroglutámová kyselina n-(2-kyanoacetamido)-3,4,5I6-tetrachlórftalámová kyselina (r,s)-fmoc-1,3-dihydro-2h-izoindolkarboxylová kyselina c/s-1 -amino-3-(2-fosfonoacetyl)cyklobután-1 -karboxylová kyselina alfa-(2,4-dimetoxy-3-metylbenzylidén)hipurová kyselina 5-fluór-2-metylbenzoová ·· ·· ······ ···· ··· ···· ·· ··· ·· ·· ·· ··4-methylumbelliferyl-phosphate acid, 2, 5, -dimetylftalanilová 3- (naphthalene-2-sulfonyl) -propionic acid 2 ', 6'-diizopropylglutaranilová 2- (3,4-dimethoxystyryl) glyoxylic acid 6- (4- (3-carboxy-propyl) -phenyl) -hexanoic acid dodecafluorocorkic acid phenolsulfonic acid 5-bromo-2,4-dihydroxybenzoic acid 2- (9h-fluoro-9-ylmethoxycarbonylamino) -3-phenyl-propionic acid 4-butyloxybiphenyl 4'-carboxylic acid p-fenylazobenzénsulfónová; 4-methylsulfonylphenylacetic acid 3-benzyloxy-4-methoxy-2-nitro-benzoic acid, 4,5-dihydro-4 I 5-dioxo-1 H -pyrrolo [2,3-f] quinoline-2,7,9-tricarboxylic acid 2 '- (trifluoromethyl) maleanilic acid 2-benzoylbenzoic acid 4-chloro-2- (2-thienylethyl) benzoic acid r - (-) - hexahydromanedioic acid 2,5-dichloro-4 methoxy-benzoic acid benzyloxycarbonyl-d-pyroglutamic acid n- (2-cyanoacetamide) -3,4,5-I 6 tetrachlórftalámová acid (r, s) -Fmoc-1, 3-Dihydro-2H-isoindolecarboxylic acid cis-1-amino-3- (2-phosphonoacetyl) cyclobutane-1-carboxylic acid alpha- (2,4-dimethoxy-3-methylbenzylidene) hippuric acid 5-fluoro-2- methylbenzoic acid ···············································

-37kyselina 1,3,3a,4,7,7a-hexahydro-2-metyl-3-fenyl-1 -oxo-3a-izoindolkarboxylová kyselina 5(s), 12(s)-dihydroxyeikoza-6e,8z, 10e, 14z-tetraénová kyselina 5(s), 14(r), 15(s)-trihydroxyikoza-6-ŕrans-8-c/s-10-trans-12-ŕrans-tetraénová kyselina 4-(3-[2I2,2-tri-cl-1-(cyklopentánkarbonyl-amino)-et]-tioureido)-benzoová kyselina dodecenyljantárová, zmes kyselina alfa-fluórfenyloctová kyselina (4-amino-(3-chlór-fenyl)-pyrimidín-2-ylsulfanyl)-octová kyselina 3-(3,4,5-trimetoxyfenyl)-2-tiopyrohroznová kyselina n-fmoc-(3s,4s)-4-amino-3-hydroxy-5-cyklohexylpentánová kyselina n-acetyl-d/-glutámová kyselina 2-(hexadecyloxy)benzoová kyselina 3-(2,2-dimetyl-propionylamino)-3-fenyl-propiónová kyselina 4-(4'-n-heptylfenyl)benzoová kyselina 3-(4-n-hexyloxybenzoyl)propiónová kyselina (+/-)-1 -amino-c/s-3-fosfóncyklopentánkarboxylová kyselina d/-pyroglutámová kyselina 4-(2-karboxy-acetylamino)-benzoová kyselina 8,11,14-eikozatriínová kyselina 2,2-bis(hydroxymetyl)maslová kyselina 1,10-fenantrolín-2,9-dikarboxylová kyselina 2-karboxy-metoxy-3-metoxy-benzoová kyselina (s)-(+)-2,2-dimetyl-5-oxo-1,3-dioxolán-4-octová kyselina 1,2-difenyl-cyklopropánkarboxylová kyselina d-glutámová kyselina (4-izopropyl-2-metoxy-fenoxy)-octová kyselina (4-dimetylamino-6-metyl-pyrimidín-2-ylsulfanyl)-octová kyselina d/-glycerová kyselina 1 -beta-p-nitrofenylmliečna kyselina 5-bróm-6-hydroxy-pyrimidín-4-karboxylová kyselina 2-(2-chlórfenyl)-4-metyltiazol-5-karboxylová kyselina 2-benzamido-3-metylkrotónová kyselina 2-amino-4-trifluórmetyltiazol-5-karboxylová • ·· ·· ···· ·· ·· · · · ···· • ··· · · · · ·-37 acid 1,3,3a, 4,7,7a-hexahydro-2-methyl-3-phenyl-1-oxo-3α-isoindolecarboxylic acid 5 (s), 12 (s) -dihydroxyeicose-6e, 8z, 10e, 14z-Tetraenoic acid 5 (s), 14 (r), 15 (s) -trihydroxyicoza-6-trans-8-cis-10-trans-12-trans-tetraenoic acid 4- (3- [2 I 2 2-tri-cl-1- (cyclopentanecarbonyl-amino) -et] thioureido) -benzoic acid dodecenylsuccinic acid, alpha-fluorophenylacetic acid mixture (4-amino- (3-chloro-phenyl) -pyrimidin-2-ylsulfanyl) -acetic acid 3- (3,4,5-trimethoxyphenyl) -2-thiopyruvic acid n-fmoc- (3s, 4s) -4-amino-3-hydroxy-5-cyclohexylpentanoic acid n-acetyl-d-glutamic acid 2- (hexadecyloxy) benzoic acid 3- (2,2-dimethyl-propionylamino) -3-phenyl-propionic acid 4- (4'-n-heptylphenyl) benzoic acid 3- (4-n-hexyloxybenzoyl) propionic acid (+ (-) - 1-amino-cis-3-phosphonocyclopentanecarboxylic acid d-pyroglutamic acid 4- (2-carboxy-acetylamino) -benzoic acid 8,11,14-eicosatriic acid 2,2-bis (hydroxymethyl) butyric acid 1,10-phenanthroline-2,9-dicarboxylic acid 2-carboxymethoxy-3-methoxybenzoic acid (s) - (+) - 2,2-dimethyl-5-oxo-1,3-dioxolane- 4-acetic acid 1,2-diphenyl-cyclopropanecarboxylic acid d-glutamic acid (4-isopropyl-2-methoxy-phenoxy) -acetic acid (4-dimethylamino-6-methyl-pyrimidin-2-ylsulfanyl) -acetic acid d / 5-Bromo-6-hydroxy-pyrimidine-4-carboxylic acid 1-beta-p-nitrophenyl-lactic acid 2- (2-chloro-phenyl) -4-methyl-thiazole-5-carboxylic acid 2-benzamido-3-methyl-crotonic acid 2 -amino-4-trifluoromethylthiazole-5-carboxylic acid

-38kyselina 4,5,10,1 l-tetrametyl-tetradeka-2,4,10,12-tetraén-6,8-diíndiová kyselina 3-hydroxy-4,4,4-trifluórmaslová kyselina 4’-fluór-3'-nitroglutáranilová kyselina (3,5-dimetoxyfenyl)octová kyselina 4-fenylftalová kyselina 2’-chlór-hexahydro-5,-(trifluórmetyl)ftalanilová kyselina n-(4,6-dimetylpyriľnidín-2-yl)-3-aminobenzoová kyselina 4-(hexadecyloxy)-3-nitrobenzénsulfónová kyselina (r)-(+)-2-brómpentánová kyselina s-trans,ŕrans-farnesyltiosalicylová kyselina (4-(5,5-dimetyl-hexyl)-fenoxy)-octová kyselina 4-(2,4,5-trichlórfenoxy)-maslová kyselina (+/-) 12-hydroxyeikoza-5z,8z,10e,14z-tetraénová kyselina 4-(oktadecyloxy)benzoová kyselina 4’-fluór-3,-nitrohexahydroftalanilová kyselina 4-brómftalová kyselina hydantoín-5-octová kyselina n-terc-butylftalámová kyselina d-(-)-o-formyloxy-2-fenyloctová kyselina 2,3-dichlórpropiónová kyselina 2-dodecéndiová kyselina izo-butylakrylová kyselina 3-(4-fluórtiofénoxy)propiónová kyselina 4-(2-benzoylacetamido)benzoová kyselina 4-oxo-4-fenylamino-2-buténová kyselina 4-oxo-hepta-2,5-diéndiová kyselina acetodifosfónová kyselina 3,5,5-trimetylhexánová kyselina 3-etyl-2-hexénová kyselina 3’-chlór-2'-metyl-1,2,3,6-tetrahydroftalanilová kyselina 3,4-diacetoxyfenyloctová kyselina trans-1,4-cyklohexándikarboxylová * ·· ······ ·· ·· · · · ···· • ··· · · · · ·-38 acid 4,5,10,1 1-tetramethyl-tetradeca-2,4,10,12-tetraene-6,8-diindioic acid 3-hydroxy-4,4,4-trifluorobutyric acid 4'-fluoro-3 ' (3,5-dimethoxyphenyl) acetic acid 4-phenylphthalic acid 2'-chloro-hexahydro-5 ' - (trifluoromethyl) phthalic acid n- (4,6-dimethylpyrimidin-2-yl) -3-aminobenzoic acid 4 - (hexadecyloxy) -3-nitrobenzenesulfonic acid (R) - (+) - 2-bromopentanoic acid s-trans, trans-farnesylthiosalicylic acid (4- (5,5-dimethyl-hexyl) -phenoxy) -acetic acid 4- ( 2,4,5-Trichlorophenoxy) butyric acid (+/-) 12-hydroxyeicoza-5z, 8z, 10e, 14z-tetraenoic acid 4- (octadecyloxy) benzoic acid 4'-fluoro-3 , -nitrohexahydrophthalanilic acid 4-bromophthalic acid hydantoin-5-acetic acid n-tert-butylphthalic acid d - (-) - o-formyloxy-2-phenylacetic acid 2,3-dichloropropionic acid 2-dodecenedioic acid isobutyl acrylic acid 3- (4-fluorothiophenoxy) propionic acid 4- (2-benz oylacetamido) benzoic acid 4-oxo-4-phenylamino-2-butenoic acid 4-oxo-hepta-2,5-dienedioic acid acetodiphosphonic acid 3,5,5-trimethylhexanoic acid 3-ethyl-2-hexenoic acid 3'-chloro -2'-Methyl-1,2,3,6-tetrahydrophthalanic acid 3,4-diacetoxyphenylacetic acid trans-1,4-cyclohexanedicarboxylic acid * ·················· ··· · · · · ·

-39kyselina 3-(3-hydroxy-fenyl)-2-metyl-akrylová boc-1 -4-tiazolylalanín kyselina n-(5-chlór-2,4-dimetoxyfenyl)glutarámová kyselina 16-metyloktadekánová kyselina 4-n-hexyloxybenzoová kyselina 3-(n-(3,4-dimetylfenyl)karbamoyl)-5-norbornén-2-karboxylová kyselina 2-dodekanoylamino-benzoová kyselina 2-izopropoxybenzoová kyselina 3-(2-karboxy-etyl)-6-chlór-1 h-indol-2-karboxylová kyselina beta-fenylškoricová kyselina 3-(n-(4-chlórfenyl)karbamoyl)-5-norbornén-2-karboxylová kyselina 2-(3,4-dimetoxy-fenyl)-3-fenyl-akrylová kyselina 1,2,3,4-tetrahydro-2-naftalénpropiónová kyselina 3-(3,5-dimetoxy-4-hydroxyfenyl)-propiónová kyselina 3-bróm-4-metoxyfenyloctová kyselina 1 -acetoxy-2-naftoová kyselina 4-hydroxy-3-(p-diazofenylfosforylcholín)-fenyloctová kyselina 6-nitrokaprónová kyselina 3-nitro-4-(4-chlórfenoxy)škoricová kyselina oktadec-9-índiová kyselina n-(2-chlórfenyl)malonámová kyselina 4’-etoxyglutaran ílová kyselina 2,4,6-trihydroxybenzoová kyselina n-fmoc-1 -homofenylalanín kyselina n-(4-acetamido-3-metoxyfenyl)ftalámová kyselina n-(4-piperidón)glutarámová kyselina 4-(1-(n-(2-chlór-5-nitrofenyl)karbamoyl)-3,3-dimetyl-2-oxobutoxy)benzoová kyselina 1-naftoxyoctová kyselina benzyloxykarbonyl-1 -pyroglutámová kyselina 2-chlórizoftalová kyselina 2-amino-3-bróm-5-jódbenzoová kyselina 2,4,6-trifluórfenyloctová-39 3- (3-Hydroxy-phenyl) -2-methyl-acrylic acid boc-1-4-thiazolylalanine n- (5-chloro-2,4-dimethoxyphenyl) glutaramic acid 16-methyloctadecanoic acid 4-n-hexyloxybenzoic acid 3- (n- (3,4-dimethylphenyl) carbamoyl) -5-norbornene-2-carboxylic acid 2-dodecanoylamino-benzoic acid 2-isopropoxybenzoic acid 3- (2-carboxyethyl) -6-chloro-1 h- Indole-2-carboxylic acid beta-phenyl cinnamic acid 3- (n- (4-chlorophenyl) carbamoyl) -5-norborene-2-carboxylic acid 2- (3,4-dimethoxyphenyl) -3-phenyl-acrylic acid 1 2,3,4-tetrahydro-2-naphthalenepropionic acid 3- (3,5-dimethoxy-4-hydroxyphenyl) -propionic acid 3-bromo-4-methoxyphenylacetic acid 1-acetoxy-2-naphthoic acid 4-hydroxy-3 - (p-diazophenylphosphorylcholine) -phenylacetic acid 6-nitrocaproic acid 3-nitro-4- (4-chlorophenoxy) cinnamic acid octadec-9-indioic acid n- (2-chlorophenyl) malonamic acid 4'-ethoxyglutaranic acid 2,4 6-trihydroxybenzoic acid n-fmoc-1-homophenylalanine n- (4-acetamido-3-methoxyphenyl) phthalic acid n- (4-piperidone) glutaramic acid 4- (1- (n- (2-chloro-5-nitrophenyl) carbamoyl)) -3,3-dimethyl-2-oxobutoxy) benzoic acid 1-naphthoxyacetic acid benzyloxycarbonyl-1-pyroglutamic acid 2-chloroisophthalic acid 2-amino-3-bromo-5-iodobenzoic acid 2,4,6-trifluorophenylacetic acid

• BB • · • ··· • BB • · • ··· ·· • · • B ·· • · • B BBBB • B BBBB • B BB B B B · BB B B B · B B B B B · ·· B · ·· BB BB BB BB BB BB BB BB

kyselina fmoc-(3s,4s)-4-amino-5-cyklohexyl-3-hydroxypentánová kyselina S-S'AS.S'.e-hexachlórftalanilová kyselina 2,4,5-trifluórškoricová kyselina 2-bróm-5-fluórškoricová kyselina 3-hydroxy-alfa-merkapto-beta-metylškoricová kyselina 3-benzoyl-2-(4-chlórfenyl)propiónová kyselina 1-homocysteínová kyselina 4-(3-(2,6-xylyl)ureido)benzoová kyselina n-4-ŕerc-butylbenzoyl-n-fenylantranilová kyselina benzotiazol-2-sulfónová kyselina 4-metyl-dec-4-én-8-inová kyselina 4-metoxy-3-nitrobenzoová kyselina 4-(3-(5-chlór-2-metoxyfenyl)ureido)benzoová kyselina 3-bróm-2-metylakrylová kyselina d-kamfolová kyselina fmoc-(3s,4s)-4-amino-3-hydroxy-6-metyltiohexánová kyselina 10,12-heptadekadiínová kyselina 4-(((4-chlór-benzénsulfonylimino)fenyl-metyl)-amino-benzoová kyselina 13-c/s-retinová kyselina 2-(karboxymetoxy)benzoová kyselina c/s-hexahydro-n-(4-metyl-3-nitrofenyl)ftalámová kyselina 6-hydroxy-5-nitrózo-2-naftalénsulfónová kyselina 3-chlórtiofén-2-karboxylová kyselina 3-benzyladipová kyselina 2,,5’-dimetylsukcínanilová kyselina bis(2-etylhexyl)pyrofosforečná kyselina 4-oxo-3-fenyl-2-tioxo-1 -imidazolidínoctová kyselina (1r,2s)-1-hydroxy-1,2,3,4-tetrahydro-2-naftoová kyselina 5-(4-fluórfenyl)-2,3-dihydro-1h-pyrolizín-6,7-dikarboxylová kyselina 3-(n,-(2,4-dinitro-fenyl)-hydrazínokarbonyl)-akrylová kyselina n-chlóracetyl-d/-alfa-amino-maslová kyselina 2-(2-hydroxy-benzoyl)-benzoováfmoc- (3s, 4s) -4-amino-5-cyclohexyl-3-hydroxypentanoic acid S-S'AS.S'e-hexachlorophthalanic acid 2,4,5-trifluorcinnamic acid 2-bromo-5-fluorocinnamic acid 3-hydroxy-alpha-mercapto-beta-methyl cinnamic acid 3-benzoyl-2- (4-chlorophenyl) propionic acid 1-homocysteic acid 4- (3- (2,6-xylyl) ureido) benzoic acid n-4-tert -butylbenzoyl-n-phenylanthranilic acid benzothiazole-2-sulfonic acid 4-methyl-dec-4-en-8-ynoic acid 4-methoxy-3-nitrobenzoic acid 4- (3- (5-chloro-2-methoxyphenyl) ureido benzoic acid 3-bromo-2-methylacrylic acid d-campholic acid fmoc- (3s, 4s) -4-amino-3-hydroxy-6-methylthiohexanoic acid 10,12-heptadecadiic acid 4 - ((((4-chloro- Benzenesulfonylimino) phenyl-methyl) -amino-benzoic acid 13-cis-retinoic acid 2- (carboxymethoxy) benzoic acid cis-hexahydro-1- (4-methyl-3-nitrophenyl) phthalic acid 6-hydroxy-5 -nitroso-2-naphthalenesulfonic acid 3-chlorothiophene-2-carboxy 3-Benzyladipic acid 2 , 5'-dimethylsuccinilic acid bis (2-ethylhexyl) pyrophosphoric acid 4-oxo-3-phenyl-2-thioxo-1-imidazolidineacetic acid (1r, 2s) -1-hydroxy-1, 2,3,4-tetrahydro-2-naphthoic acid 5- (4-fluorophenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid 3- (n , - (2,4-dinitrophenyl) (Hydrazinocarbonyl) -acrylic acid n-chloroacetyl-1H-alpha-amino-butyric acid 2- (2-hydroxy-benzoyl) -benzoic acid

0 · • ··· 0 · • ··· • · • · • f • · • · • f ···· • • ···· • • ·· · • · ·· • · · ·· · • · ·· • · · • · • · ·· · · e · ·· · · ·· ·· ·· ··

kyselina 3-benzoylamino-3-fenyl-propiónová kyselina 4-heptyloxybifenyl-4'-karboxylová kyselina 4-nitrohipurová kyselina 4’-jódsukcínanilová kyselina 2-acetamidoizoftalová kyselina 15-fenyl-3-metyl-pentadekánová kyselina ŕrans-4-propylcyklohexánkarboxylová dibutylfosfát kyselina 4’,4-sulfonyldimaleanilová kyselina ŕra/?s,ŕrans-mukonová kyselina 2-(3,4-dimetoxyfenyltio)octová kyselina 4-((5-bróm-2-hydroxy-benzylidén)-amino)-benzoová kyselina (s)-(+)-3-(benzyloxykarbonyl)-5-oxo-4-oxazolidínoctová kyselina fmoc-(3s,4s)-4-amino-3-hydroxy-6-metylheptánová kyselina 3-(n-benzylkarbamoyl)-5-norbornén-2-karboxylová kyselina (s)-(+)-2-(benzyloxykarbonyl)-1,2,3,4-tetrahydro-3-izochinolínkarboxylová kyselina (2-fenoxyetyltio)octová kyselina 1 -nitroantrachinón-2-karboxylová kyselina d-homocysteínsulfínová kyselina 3-metoxymaslová kyselina 2-jódbenzoová kyselina alfa,3-dibróm-1 -adamantánoctová kyselina 4-(2-hydroxyetoxy)benzoová kyselina 4-benzénsulfonyl-4-kyano-heptándiová kyselina n-ftalyl-d/-asparágová kyselina 2-( 1 -cyklohexenyl)-maslová kyselina 3-(4-chlórbenzyloxy)tiofén-2-karboxylová kyselina 4-(2-hydroxy-etylamino)-3-nitro-benzoová kyselina 2,3-dichlór-6-fluórbenzoová kyselina 6-(2-karboxy-etyl)-2,3-dimetoxy-benzoová kyselina 4,5-dibróm-2-fluórbenzoová kyselina etylchromotropová ·· ·· ···· ·· • · · · · · · ··· B B B B ·3-benzoylamino-3-phenyl-propionic acid 4-heptyloxybiphenyl-4'-carboxylic acid 4-nitrohipuric acid 4'-iodosuccinilic acid 2-acetamidoisophthalic acid 15-phenyl-3-methylpentadecanoic acid trans-4-propylcyclohexanecarboxylic dibutylphosphate acid 4 ', 4-sulfonyldimaleanilic acid trans, muconic acid 2- (3,4-dimethoxyphenylthio) acetic acid 4 - ((5-bromo-2-hydroxy-benzylidene) -amino) -benzoic acid (s) - (+) - 3- (Benzyloxycarbonyl) -5-oxo-4-oxazolidineacetic acid fmoc- (3s, 4s) -4-amino-3-hydroxy-6-methylheptanoic acid 3- (n-benzylcarbamoyl) -5-norbornene -2-carboxylic acid (s) - (+) - 2- (benzyloxycarbonyl) -1,2,3,4-tetrahydro-3-isoquinolinecarboxylic acid (2-phenoxyethylthio) acetic acid 1-nitroanthraquinone-2-carboxylic acid d- homocysteine sulfinic acid 3-methoxybutyric acid 2-iodobenzoic acid alpha, 3-dibromo-1-adamantane acetic acid 4- (2-hydroxyethoxy) benzoic acid 4-benzenesulfo n-4-cyano-heptanedioic acid n-phthalyl-d-aspartic acid 2- (1-cyclohexenyl) butyric acid 3- (4-chlorobenzyloxy) thiophene-2-carboxylic acid 4- (2-hydroxy-ethylamino) - 3-nitro-benzoic acid 2,3-dichloro-6-fluorobenzoic acid 6- (2-carboxyethyl) -2,3-dimethoxybenzoic acid 4,5-dibromo-2-fluorobenzoic acid ethylchromotropic acid ·· ·· · ··· ··· · BBBB ·

-42• ·· ·· ·· ·· · kyselina 4-butylbenzoová edta, izotiokyanobenzylkyselina 5,6-diamino-1,3-naftaléndisulfónová kyselina 11-(butyltio)-undekánová kyselina 3-(2-etylsulfanyl-benzotiazol-6-ylkarbamoyl)-akrylová kyselina 5-nitrobenzofurán-2-karboxylová kyselina (etylénditio)dioctová kyselina o-izopropylbenzoová kyselina 3-(3-(4-acetoxy-fenyl)-2-benzoylamino-akryloylamino)-propiónová kyselina 2,3,5,6-tetrametyl-benzoová kyselina 3,4-metyléndioxyfenyloctová kyselina 2-hydroxyamino-3-metyl-maslová kyselina trans, ŕrans-2,4-hexadiénová kyselina 3-(trifluórmetyl)benzoová kyselina 1 -naftylamín-3,5,7-trisulfónová kyselina 4-aminofenyljantárová kyselina 3-[benzyl-(toluén-4-sulfonyl)-amino]-propiónová kyselina 11-metyldodekánová kyselina 3,5-difluórmandlová kyselina 2’,4,,5,-trichlórsukcínanilová kyselina (+/-)-jasmonová kyselina (+/-)-2-(6-metoxy-2-naftyl)propiónová kyselina nitrilotrioctová kyselina 2-metoxy-3-metylbenzoová kyselina 2-(4-chlór-benzoylamino)-3-hydroxy-propiónová kyselina 3-benzoyl-2-naftoová kyselina 4’-(trifluórmetyl)-2-bifenylkarboxylová kyselina 4-(dodecyltio)maslová kyselina 4-(trifluórmetyl)mandlová kyselina n-alfa-boc-n-gama-fmoc-cŕ-diaminomaslová kyselina 4-formamidobenzoová kyselina boc-11-aminoundekánová * ·♦ ·· ···· ·· ··· · · · β·· • ··· 9 · 9 · ·4-Butylbenzoic acid edta, isothiocyanobenzyl acid 5,6-diamino-1,3-naphthalenedisulfonic acid 11- (butylthio) -undecanoic acid 3- (2-ethylsulfanyl-benzothiazole-6- ylcarbamoyl) -acrylic acid 5-nitrobenzofuran-2-carboxylic acid (ethylenedithio) diacetic acid o-isopropylbenzoic acid 3- (3- (4-acetoxyphenyl) -2-benzoylamino-acryloylamino) -propionic acid 2,3,5, 6-tetramethyl-benzoic acid 3,4-methylenedioxyphenylacetic acid 2-hydroxyamino-3-methylbutyric acid trans, trans-2,4-hexadienoic acid 3- (trifluoromethyl) benzoic acid 1-naphthylamine-3,5,7-trisulfonic acid acid 4-aminofenyljantárová 3- [benzyl- (toluene-4-sulfonyl) amino] propionic acid, 11-metyldodekánová 3,5-difluoromandelic acid 2 ', 4, 5, -trichlórsukcínanilová of (+/-) - jasmonic acid (+/-) - 2- (6-methoxy-2-naphthyl) propionic acid nitrilotriacetic acid 2-methoxy-3-methylbenzoic acid 2- (4 3-Benzoyl-2-naphthoic acid 4 '- (trifluoromethyl) -2-biphenylcarboxylic acid 4- (dodecylthio) butyric acid 4- (trifluoromethyl) mandelic acid n-alpha-boc -n-gamma-fmoc-α-diaminobutyric acid 4-formamidobenzoic acid boc-11-aminoundecanoic acid 9 · 9 · · · · · ·

-43kyselina 4-fluór-2-metylfenoxyoctová kyselina 7-amino-1,3-naftaléndisulfónová kyselina 2,3-dibróm-3-(3,4-dimetoxyfenyl)propiónová kyselina 3-[[(4-chlórfenyl)sulfonyl]metyl]-4-nitrobenzoová kyselina m-anízová kyselina 2’,4’-dimetyl-3,4,516-tetrachlórftalanilová kyselina 3-brómtiofén-2-karboxylová kyselina 2-(tiobenzoyl)tioloctová edta, aminobenzyl kyselina 2,3-dibróm-2'-metyl-4'-nitrosukcínanilová kyselina (1 -karboxymetyl-3,3-dimetyl-cyklohexyl)-octová kyselina 4'-etyl-3,4,5,6-tetrachlórftalanilová kyselina c/s-1,2-cyklohexándikarboxylová kyselina 4-ureidobenzoová kyselina 2-fenyl-5-(trifluórmetyl)-oxazol-4-karboxylová kyselina 5-chlór-2-hydroxy-benzénsulfónová kyselina 3-etoxy-4-hydroxyfenyloctová kyselina 3-(decyloxy)benzoová n-acetyl-d/-etionín kyselina eikoza-5,8-diénová kyselina 2,5-dihydroxybenzén-1,4-disulfónová kyselina 2-brómbenzoová kyselina 2-chlórmandlová kyselina r-4-metoxymandlová kyselina 3-chlór-3'-metyl-bifenyl-2,2'-dikarboxylová kyselina p-nitroškoricová kyselina 6-bróm-2-pyridín-4-yl-chinolín-4-karboxylová kyselina 4-fluórglutámová kyselina benzo(c)fenantrén-5,6-dikarboxylová kyselina 3-benzyloxytiofén-2-karboxylová kyselina 2-(4-metylbenzoyl)benzoová kyselina n-(fenyletyl)sukcínamová4-Fluoro-2-methylphenoxyacetic acid 7-amino-1,3-naphthalenedisulfonic acid 2,3-dibromo-3- (3,4-dimethoxyphenyl) propionic acid 3 - [[(4-chlorophenyl) sulfonyl] methyl] 4-nitrobenzoic acid m-anisic acid 2 ', 4'-dimethyl-3,4,5 1 6-tetrachlorophthalanic acid 3-bromothiophene-2-carboxylic acid 2- (thiobenzoyl) thiol acetic acid, aminobenzyl acid 2,3-dibromo 2'-methyl-4'-nitrosuccinilic acid (1-carboxymethyl-3,3-dimethyl-cyclohexyl) -acetic acid 4'-ethyl-3,4,5,6-tetrachlorophthalanilic acid cis-1,2- cyclohexanedicarboxylic acid 4-ureidobenzoic acid 2-phenyl-5- (trifluoromethyl) oxazole-4-carboxylic acid 5-chloro-2-hydroxy-benzenesulfonic acid 3-ethoxy-4-hydroxyphenylacetic acid 3- (decyloxy) benzoic n-acetyl- d -ethionine eicoza-5,8-dienoic acid 2,5-dihydroxybenzene-1,4-disulfonic acid 2-bromobenzoic acid 2-chloro-mandelic acid r-4-methoxy-butyric acid 3-chloro-3'-methyl-biphenyl- 2,2-a p-nitrocinnamic acid 6-bromo-2-pyridin-4-yl-quinoline-4-carboxylic acid 4-fluoroglutamic acid benzo (c) phenanthrene-5,6-dicarboxylic acid 3-benzyloxy-thiophene-2-carboxylic acid 2- (4-methylbenzoyl) benzoic acid n- (phenylethyl) succinamic acid

• ·* • · * • · • · ···· ···· • · · • · · • 4 • 4 • · • · • · ·· • · ·· • ··· • ··· • · • · • · · • · · ·· «· ·· «· • · • · • · • · ·· · · ·· · ·

kyselina cyklohexán-1,1-bis-(3-merkaptopropiónová) kyselina 2-jód-5-metylbenzoová kyselina 1 -(4-fluórfenyl)cyklohexánkarboxylová kyselina (adamantán-1 -yloxy)-octová gama-ŕerc-butylester kyseliny fmoc-d-glutámovej kyselina 4-(ŕerc-butoxykarbonylamino-metyl)-benzoová kyselina 9,10-dihydro-12-etoxy-9,10-etanoantracén-11-karboxylová kyselina 3-fluórftalová kyselina c/s-hexahydro-n-(2-metoxy-5-metylfenyl)ftalámová kyselina 2-bróm-5-jódbenzoová kyselina alfa-metyl-levulínová kyselina 2,6-dibróm-benzoová kyselina n-(2,4-dichlórfenyl)malonámová kyselina (+/-)-beta-p-chlórfenylglutámová kyselina 3-brómbenzoová kyselina (+)-alfa-metyl-4-karboxyfenylglycín gama-ŕerc-butylester kyseliny boc-1-glutámovej kyselina 4-(2-benzoylamino-3-metyl-but*2-enoylamino)maslová kyselina 3-(n-(2,4,6-trimetylfenyl)karbamoyl)-5-norbornén-2-karboxylová kyselina 1 -(4-metoxyfenyl)-1 -cyklopentánkarboxylová kyselina n-alfa-(ŕerc-butyloxykarbonyl)-beta-(1 -adamantyl ester)-1 -asparágová kyselina 3,4-difluórfenyloctová kyselina chlorečná kyselina n-((r)-1-(1-naftyl)etyl)ftalámová kyselina hydroxy-2-naftalényl-metylfosfónová kyselina 3-(4-izopropyl-benzoyl)akrylová kyselina (3-metoxyfenyl)fosfónová kyselina 2,4-difluórbenzoová kyselina 2-(2,4,6-trimetylbenzoyl)benzoová kyselina (3-chlór-1,4-dioxo-1,4-dihydro-naftalén-2-ylamino)octová kyselina 2-etyl-2-hydroxymaslová kyselina iminobis(metylfosfónová) ·· ·· ···· ·· • · · · · · · ··· · · · · ·cyclohexane-1,1-bis- (3-mercaptopropionic acid) 2-iodo-5-methylbenzoic acid 1- (4-fluorophenyl) cyclohexanecarboxylic acid (adamantan-1-yloxy) -acetic acid gamma-tert-butyl ester fmoc-d -glutamic acid 4- (tert-butoxycarbonylamino-methyl) -benzoic acid 9,10-dihydro-12-ethoxy-9,10-ethanoanthracene-11-carboxylic acid 3-fluorophthalic acid cis-hexahydro-n- (2- methoxy-5-methylphenyl) phthalic acid 2-bromo-5-iodobenzoic acid alpha-methyl-levulinic acid 2,6-dibromo-benzoic acid n- (2,4-dichlorophenyl) malonamic acid (+/-) - beta-p 3-bromobenzoic acid (+) - alpha-methyl-4-carboxyphenylglycine boc-1-glutamic acid gamma-tert-butyl ester 4- (2-benzoylamino-3-methyl-but-2-enoylamino) butyric acid 3-chlorophenylglutamic acid 3 - (n- (2,4,6-trimethylphenyl) carbamoyl) -5-norbornene-2-carboxylic acid 1- (4-methoxyphenyl) -1-cyclopentanecarboxylic acid n-alpha- (tert-butyloxycarbonyl) -beta- (1) -adamantyl ester) -1 aspartic acid 3,4-difluorophenylacetic acid chloric acid n - ((r) -1- (1-naphthyl) ethyl) phthalic acid hydroxy-2-naphthalenylmethylphosphonic acid 3- (4-isopropylbenzoyl) acrylic acid (3 Methoxyphenyl) phosphonic acid 2,4-difluorobenzoic acid 2- (2,4,6-trimethylbenzoyl) benzoic acid (3-chloro-1,4-dioxo-1,4-dihydro-naphthalen-2-ylamino) acetic acid 2 -ethyl-2-hydroxybutyric acid iminobis (methylphosphonic) ·· ··············

-45* ·· 99 99 99 9 kyselina 1 -(aminokarbonyl)-l -cyklopropánkarboxylová kyselina (r)-(+)-3-hydroxy-1 -cyklopentén-1 -heptánová kyselina 2,3-dimetyljantárová kyselina d/-n-propylmalónová kyselina 4-dibenzo(a,d)cykloheptén-5-ylidén-maslová kyselina 15(s)-hydroxyeikoza-8z, 11 z, 13e-triénová kyselina 4-fosfono-benzoová kyselina c/s-2’,5'-dimetylhexahydroftalámová kyselina c/s-n-(2,3-dichlórfenyl)hexahydroftalámová kyselina 3-(2-metoxy-benzoylamino)-benzoová kyselina (+/-)-1-aminocyklohexán-ŕrans-1,2-dikarboxylová kyselina n-benzoyl-d-asparágová kyselina 2-(2-fenoxy-acetylamino)-3-fenyl-propiónová kyselina ŕra/?s-2-(p-metylbenzoyl)-1 -cyklohexán-karboxylová kyselina n-alfa-(benzyloxykarbonyl)-gama-(benzylester)-1-glutámová kyselina 4-brómmaslová kyselina beta-(3-acetoxyfenyl)propiónová kyselina alfa-chlór-3,5-dimetyl-1 -adamantánoctová kyselina 11-dodecénová (s)-cbz-oxaprolín kyselina mezitylglyoxylová kyselina cyklopentyloctová kyselina 3-chlórsalicylová kyselina 2-metylglutárová kyselina n-alfa-(9-fluórenylmetyloxykarbonyl)-1 -norvalín kyselina 1 -alfa-glutamyl-1 -asparágová kyselina n-(4,6-dimetylpyrimidín-2-yl)-2-aminobenzoová kyselina 6-heptadecyloxy-1 -hydroxy-naftalén-2-karboxylová kyselina 1,3-fenyléndipropiónová kyselina 4’-metyl-3’-nitromaleanilová kyselina trikoza-10,12-diíndiová kyselina d/-2-[4-(trifluórmetoxy)fenoxy]propiónová-45 * ·· 99 99 99 9 1- (Aminocarbonyl) -1-cyclopropanecarboxylic acid (R) - (+) - 3-hydroxy-1-cyclopentene-1-heptanoic acid 2,3-dimethylsuccinic acid d / -n -propylmalonic acid 4-dibenzo (a, d) cyclohepten-5-ylidene-butyric acid 15 (s) -hydroxyeicose-8z, 11 z, 13e-trienoic acid 4-phosphonobenzoic acid cis-2 ', 5' -dimethylhexahydrophthalic acid cis- (2,3-dichlorophenyl) hexahydrophthalic acid 3- (2-methoxy-benzoylamino) -benzoic acid (+/-) - 1-aminocyclohexane-trans-1,2-dicarboxylic acid n-benzoyl- d-Aspartic acid 2- (2-phenoxy-acetylamino) -3-phenyl-propionic acid trans-2- (p-methylbenzoyl) -1-cyclohexanecarboxylic acid n-alpha- (benzyloxycarbonyl) -gamma- ( benzyl ester) -1-glutamic acid 4-bromobutyric acid beta- (3-acetoxyphenyl) propionic acid alpha-chloro-3,5-dimethyl-1-adamantaneacetic acid 11-dodecenoic (s) -cbz-oxaproline mesitylglyoxylic acid cyclopentylacetic acid 3 - chlorosalicylic acid 2-methylglutaric acid n-alpha- (9-fluorenylmethyloxycarbonyl) -1 -norvaline 1-alpha-glutamyl-1-aspartic acid n- (4,6-dimethylpyrimidin-2-yl) -2-aminobenzoic acid 6- heptadecyloxy-1-hydroxy-naphthalene-2-carboxylic acid 1,3-phenylenedipropionic acid 4'-methyl-3'-nitromaleanilic acid tricose-10,12-diindioic acid d] -2- [4- (trifluoromethoxy) phenoxy] propionic acid

• · · • · • ··· • · · • · • ··· ·· ···· ♦ · · • · · ·· ···· ♦ · · · · · e · • · e · • · • · • · • · • · ·· · · ·· ·· ·· ·· • · • · • · • ·

kyselina n-(difenylmetyl)glutarámová kyselina 2-benzoylpyridín-4-karboxylová kyselina 2,4,6-trichlórbenzoová kyselina 2-(2,4-dimetyl-benzyl)-benzoová kyselina 2,4-henikozadiínová kysel ina 3-metyl-2-(orto-tolyl )-maslová kyselina 2,3,4,5,6-pentachlórbenzoová kyselina 3,4-dichlórpentafluórmaslová kyselina 3,4,4-trichlór-2-nitro-but-3-énová kyselina 1,2,4-benzéntrikarboxylová kyselina 5-merkapto-tetrazol-1 -propiónová kyselina laurová kyselina 4-jódmaslová kyselina c/s-8,11,14-eikozatriénován- (diphenylmethyl) glutaramic acid 2-benzoylpyridine-4-carboxylic acid 2,4,6-trichlorobenzoic acid 2- (2,4-dimethylbenzyl) -benzoic acid 2,4-henosadioic acid 3-methyl-2 - (ortho-tolyl) butyric acid 2,3,4,5,6-pentachlorobenzoic acid 3,4-dichloropentafluorobutyric acid 3,4,4-trichloro-2-nitro-but-3-enoic acid 1,2,4 -benzenetricarboxylic acid 5-mercapto-tetrazole-1-propionic acid lauric acid 4-iodobutyric acid cis-8,11,14-eicosatrienoic acid

3-karboxy-4-hydroxy-5-sulfoanilin kyselina 2-furyltio-pyrohroznová kyselina 2-chlór-5-nitrobenzénsulfínová kyselina n-alfa-(ŕerc-butyloxykarbonyl)beta-(2-adamantylester)-1-asparágová kyselina 1 -c/s-pyrolidín-2,4-dikarboxylová kyselina 2-amino-5-kyano-3-etyl-benzoová kyselina 1 -acetoxynaftalén-6-sulfónová kyselina 5(s)-hydroxyeikoza-6e,8z,11z,14z-tetraénová fmoc-d-norvalín kyselina 4-(n-(3-chlórfenyl)karbamoyl)maslová kyselina 3-metyl-1,1-cyklohexándioctová kyselina 6-nitro-1 -diazo-2-naftol-4-sulfónová kyselina 2-(4-metoxyfenoxy)-5-nitrobenzoová kyselina 4,4’-diaminodifenylamín-2,2-disulfónová kyselina 2-metyloktadekánová kyselina 2,6-difluórškoricová kyselina 20-hydroxy-(5z,8z,11z,14z)-eikozatetraénová kyselina 4-toluénsulfonyloctová ·· ·· ···· 993-carboxy-4-hydroxy-5-sulfoaniline 2-furylthiopyruvic acid 2-chloro-5-nitrobenzenesulfonic acid n-alpha- (tert-butyloxycarbonyl) beta- (2-adamantylester) -1-aspartic acid 1-c (S) -pyrrolidine-2,4-dicarboxylic acid 2-Amino-5-cyano-3-ethyl-benzoic acid 1-Acetoxynaphthalene-6-sulfonic acid 5 (s) -Hydroxyicose-6e, 8z, 11z, 14z-tetraenoic fmoc -d-norvaline 4- (n- (3-chlorophenyl) carbamoyl) butyric acid 3-methyl-1,1-cyclohexanediacetic acid 6-nitro-1-diazo-2-naphthol-4-sulfonic acid 2- (4- methoxy-phenoxy) -5-nitrobenzoic acid 4,4'-diaminodiphenylamine-2,2-disulfonic acid 2-methyloctadecanoic acid 2,6-difluoro cinnamic acid 20-hydroxy- (5z, 8z, 11z, 14z) -eicosatetraenoic acid 4-toluenesulfonylacetic acid · · ·· ··· 99

9 9 9 9 9 9 ··· · 9 · · ·9 9 9 9 9 9 ··· · 9 · · ·

-479 99 9 9 9 9 9 9 9 kyselina 5-bróm-3-metylsalicylová kyselina 5-chlórvalérová kyselina 5-benzyl-3,6-dioxo-2-piperazínoctová kyselina 5-hydroxy-cyklohexán-1,3-dikarboxylová kyselina 3-bróm-2-metoxy-5-metyl-benzoová kyselina 2-furoová kyselina 5-(2,5-dichlórfenylazo)-4-metylsalicylová kyselina 4-((benzénsulfonylimino-fenyl-metyl)-amino)benzoová kyselina 1-naftyloctová kyselina 3-((furán-2-karbonyl)-amino)-benzoová kyselina trans-2,4-pentadiénová kyselina 3-(3-(2-chlór-6-metylfenyl)ureido)benzoová kyselina 2-(3-(2,2,2-trichlór-1-(2,2-d-me-propionylamino)-et]-tioureido)benzoová kyselina 5,5'-ditiobis(2-nitrobenzoová) kyselina c/s-hexahydro-n-(3-chlór-4-metylfenyl)ftalámová kyselina (z)-(2-formamido)tiazol-4-yl)(metoxyimino)octová kyselina pyridín-2-sulfónová kyselina 4-(tetradecyloxy)benzoová kyselina 4-cyklopentyl-naftalén-1 -karboxylová kyselina 4-(4-(1-metyl-1h-chinolín-2-ylidén)-but-2-enylidénamino)-benzoová kyselina 3-amino-2-naftol-1,8-disulfónová kyselina 5-nitroorotová kyselina 4’-(2-furoylamino)-3'-hydroxymalonanilová kyselina (2-fenyl-cyklohexyl)-octová kyselina 4-dodecyloxybenzoová kyselina 15-metylhexadekánová kyselina (r)-(+)-2-chlórbutánová kyselina 3-amino-1,5-naftaléndisulfónová kyselina izoindolín-1 -όη-2-octová kyselina 2-(3-[n’-(3-metyl-butyryl)-hydrazíno]-3-oxo-propionylamino)-benzoová kyselina (3,3-dimetyl-1 -fenyl-1,3-dihydro-izobenzofurán-1 -yl)-octová kyselina 2-metyl-4-naftalén-1 -yl-maslová ·· Μ 888-479 99 9 9 9 9 9 9 9 5-Bromo-3-methylsalicylic acid 5-Chlorovaleric acid 5-Benzyl-3,6-dioxo-2-piperazinecacetic acid 5-Hydroxy-cyclohexane-1,3-dicarboxylic acid 3 -bromo-2-methoxy-5-methyl-benzoic acid 2-furoic acid 5- (2,5-dichlorophenylazo) -4-methylsalicylic acid 4 - ((benzenesulfonylimino-phenyl-methyl) -amino) benzoic acid 1-naphthylacetic acid 3 - ((furan-2-carbonyl) -amino) -benzoic acid trans-2,4-pentadienoic acid 3- (3- (2-chloro-6-methylphenyl) ureido) benzoic acid 2- (3- (2, 2-chloro-6-methylphenyl) ureido) 2,2'-trichloro-1- (2,2-d-metropionylamino) -ethyl] thioureido) benzoic acid 5,5'-dithiobis (2-nitrobenzoic acid) cis-hexahydro-n- (3- chloro-4-methylphenyl) phthalic acid (z) - (2-formamido) thiazol-4-yl) (methoxyimino) acetic acid pyridine-2-sulfonic acid 4- (tetradecyloxy) benzoic acid 4-cyclopentyl-naphthalene-1-carboxylic acid 4- (4- (1-Methyl-1H-quinolin-2-ylidene) -but-2-enylidenamino) -benzoic acid 3-amino-2-naphthol-1,8-disulphuric acid phonic acid 5-nitroorotic acid 4 '- (2-furoylamino) -3'-hydroxymalonanilic acid (2-phenyl-cyclohexyl) -acetic acid 4-dodecyloxybenzoic acid 15-methylhexadecanoic acid (r) - (+) - 2-chlorobutanoic acid 3-Amino-1,5-naphthalenedisulfonic acid Isoindoline-1-chloro-2-acetic acid 2- (3- [n '- (3-methyl-butyryl) -hydrazino] -3-oxo-propionylamino) -benzoic acid ( 3,3-Dimethyl-1-phenyl-1,3-dihydro-isobenzofuran-1-yl) -acetic acid 2-methyl-4-naphthalen-1-yl-butyric acid ·· Μ 888

8 88 8

8·· 8 8 8 8 88 ·· 8 8 8 8 8

-4888 kyselina 4-(chlórsulfonyl)benzoová kyselina 3-karboxy-2-furánoctová kyselina 3-[4-(4-brómfenyltio)-3-nitrofenyl]akrylová kyselina bicyklo(2.2.1 )heptán-1-karboxylová kyselina 2'-etoxymaleanilová kyselina 2-nitro-5-(trifluórmetyl)benzoová kyselina p-(benzylsulfónamido)benzoová kyselina 3-(1-naftyl)akrylová kyselina n-acetyl-8-hydroxy-2-naftylamín-6-sulfónová kyselina [bifenyl-2-yl-(toluén-4-sulfonyl)-amino]-octová kyselina n-acetylglycyl-d-glutámová kyselina 3-etylheptánová kyselina 7-chlórbenzofurán-2-karboxylová kyselina 3,5-difluórškoricová kyselina 3-(3,4-dimetyl-fenyl)-3-metyl-maslová kyselina 5,8,11,14,17-eikozapenténová kyselina 2,4,6-trinitrobenzénsulfónová kyselina nervonová (c/s-15-tetrakozénová) kyselina 5-metyl-2-fenyltiazol-4-yl-octová kyselina (5,6-dimetoxy-3-oxo-1,3-dihydro-izobenzofurán-1 -yl)-octová kyselina 1 -metylcyklopropán-1 -karboxylová kyselina dodecylbenzén-sulfónová kyselina 3-etylhexánová kyselina 1 -n-(1-karboxy-5-amino-pentyl)-iminodioctová kyselina 4-hydroxy-3-nitrobenzoová kyselina d/-n-butylfosfínová kyselina 4’-oktyloxy-4-bifenylkarboxylová kyselina 2-diazo-1 -naftol-5-sulfónová kyselina 4'-brómftalanilová kyselina 2,6-dinitrotoluén-4-sulfónová kyselina n-acetyl-6-chlór-antranilová kyselina 4-(2-acetylamino-4,5-dimetylfenyl)-4-oxo-maslová • ·· ·· ···· ·· ··· ·· ···· • ··· · · · · ·-4888 4- (chlorosulfonyl) benzoic acid 3-carboxy-2-furanacetic acid 3- [4- (4-bromophenylthio) -3-nitrophenyl] acrylic acid bicyclo (2.2.1) heptane-1-carboxylic acid 2'- ethoxymaleanilic acid 2-nitro-5- (trifluoromethyl) benzoic acid p- (benzylsulfonamido) benzoic acid 3- (1-naphthyl) acrylic acid n-acetyl-8-hydroxy-2-naphthylamine-6-sulfonic acid [biphenyl-2- yl- (toluene-4-sulfonyl) -amino] -acetic acid n-acetylglycyl-d-glutamic acid 3-ethylheptanoic acid 7-chlorobenzofuran-2-carboxylic acid 3,5-difluoro cinnamic acid 3- (3,4-dimethyl- phenyl) -3-methylbutyric acid 5,8,11,14,17-eicosapentenoic acid 2,4,6-trinitrobenzenesulfonic acid nervonic acid (cis-15-tetracosenoic) 5-methyl-2-phenylthiazole-4- yl-acetic acid (5,6-dimethoxy-3-oxo-1,3-dihydro-isobenzofuran-1-yl) -acetic acid 1-methylcyclopropane-1-carboxylic acid dodecylbenzenesulfonic acid 3-ethylhexanoic acid 1-n- (1-a 4-hydroxy-3-nitrobenzoic acid 4-hydroxy-3-nitrobenzoic acid di-n-butylphosphinic acid 4'-octyloxy-4-biphenylcarboxylic acid 2-diazo-1-naphthol-5-sulfonic acid 4'- Bromophthalanilic acid 2,6-dinitrotoluene-4-sulfonic acid n-acetyl-6-chloro-anthranilic acid 4- (2-acetylamino-4,5-dimethylphenyl) -4-oxo-butyric acid · ·· ·· ···· ····················

-49kyselina 2,4-dinitrobenzénsulfónová kyselina 3-(2-chlór-3,4-dimetoxyfenyl)-akrylová kyselina p-heptyloxybenzoová kyselina 4-chlór-3-hydroxybenzoová kyselina 3-(ac-(5-nitro-1,3-dioxo-1,3-dihydroizoindol-2-ylmetyl)-amino)benzoová kyselina 12-hydroxydodekánová kyselina trichlórakrylová kyselina piperonylová kyselina 4-metoxy-alfa-metylškoricová kyselina 5-benzyloxy-2-nitrofenylpyrohroznová kyselina 2-(2-hydroxy-1 -naftylmetylénamino)benzoová kyselina 7-metoxy-2,2-difenyl-benzo(1,3)dioxol-5-karboxylová kyselina I 3-oxotetrakoza nová kyselina dipropyl-fosfínová kyselina gibberová (C18H20O3) kyselina 3’-chlór-4’-metylsukcínanilová kyselina 1-hexadecenyljantárová kyselina 3-bróm-4-hydroxy-5-metoxy-fenyloctová kyselina n-(2,4-dichlórbenzyl)-1,2,3,6-tetrahydroftalámová kyselina 2,4-heptadekadiínová kyselina (+)-4’-metyltartranilová kyselina 3,5-dimetyl-4-formyl-2-pyrolkarboxylová kyselina 11 (r)-hydroxy-(5z,8z, 12e, 14z)-eikozatetraénová kyselina n-formyl-4-(metylamino)benzoová kyselina jantárová kyselina 2-(/7-heptoxy)-maslová kyselina 2,3,4-trifluórškoricová kyselina 3-(4-metoxy-2-metyl-fenyl)-propiónová kyselina gama-d-glutamyltaurin-4-chlór-3-fluórškoricová kyselina 4-(5-indanylmetylénamino)benzoová kyselina 2,4-difluórmandlová kyselina 5-oxoazelainová • ·· ·· ···· ·· • B · ·· ···· • ··· · · · B B-49-2,4-dinitrobenzenesulfonic acid 3- (2-chloro-3,4-dimethoxyphenyl) -acrylic acid p-heptyloxybenzoic acid 4-chloro-3-hydroxybenzoic acid 3- (ac- (5-nitro-1,3-) dioxo-1,3-dihydroisoindol-2-ylmethyl) amino) benzoic acid 12-hydroxydodecanoic acid trichloroacrylic acid piperonyl acid 4-methoxy-alpha-methylcinnamic acid 5-benzyloxy-2-nitrophenylpyruvic acid 2- (2-hydroxy-1- 7-methoxy-2,2-diphenyl-benzo (1,3) dioxole-5-carboxylic acid 3-oxotetracosoic dipropyl-phosphinic acid, gibberic acid (C18H20O3) 3'-chloro-4'-methylsuccinilic acid 1-hexadecenylsuccinic acid 3-bromo-4-hydroxy-5-methoxy-phenylacetic acid n- (2,4-dichlorobenzyl) -1,2,3,6-tetrahydrophthalic acid 2,4-heptadecadioic acid (+) - 4 3,5-Dimethyl-4-formyl-2-pyrrolecarboxylic acid 11'-methyltartranilic acid 11 (r) -hydroxy- (5z, 8z, 12e, 14z) -eicosatetraenoic acid n-formyl-4- (methylamino) benzoic acid succinic acid 2- (7-heptoxy) butyric acid 2,3,4-trifluorcinnamic acid 3- (4-methoxy-2-methylphenyl) -propionic acid gamma- d-glutamyltaurine-4-chloro-3-fluorocinnamic acid 4- (5-indanylmethyleneamino) benzoic acid 2,4-difluoromandelic acid 5-oxoazelaic acid · B · ······ BB

-50kysel ina 3-[3-chlór-5-(trifl uórmetyl )-2-pyridyl]propánová kyselina ŕrans-3-(4-metoxybenzoyl)akrylová kyselina n-alfa-(ŕerc-butyloxykarbonyl)-1-oktahydroindol-2-karboxylová kyselina (s)-(+)-hexahydromandlová kyselina n-(3-chlórfenyl)ftalámová kyselina n-(1-naftyl)-maleámová kyselina 2-(4-ŕerc-butylfenoxy)-2,2-difluóroctová kyselina 2-etylnonánová kyselina 3-(5-bróm-2-etoxyfenyl)akrylová kyselina fmoc-6-aminohexánová kyselina chlórjantárová kyselina gama-d-glutamylaminoetylfosfónová kyselina 3-hydroxy-4,4,4-trichlórmaslová kyselina acetyl-d-aminoenantová kyselina 3-(metoxykarbonylmetyltio)tiofén-2-karboxylová kyselina n-O.I-bisíhydroxymetyOetyO-SAS.e-tetrahydroftalámová kyselina 1,1-cyklopropándikarboxylová kyselina 4-amino-acetanilide-2-sulfónová kyselina 2-(4-hexyl-benzoylamino)-benzoová kyselina 4,4'-(karbonyldiimino)bis-benzoová kyselina 3-izobutyrylamino-3-(4-metoxy-fenyl)-propiónová kyselina bifenyl-3,5-dikarboxylová kyselina 3,3-dimetyl-4-oxovalérová kyselina pinónová (c/s-3-acetyl-2,2-dimetyl-cyklobutánoctová) kyselina 3-chlór-pentándiová kyselina giberelová (C19H22O6) kyselina 3-(nonylamido)benzoová kyselina 4-(trifluórmetyl)benzoová kyselina 3-(alylsulfanyl)-2-tiofénkarboxylová kyselina S'^'-dibrómftalanilová kyselina 3-hydroxynonánová kyselina 3-(4-oxo-3,4,5,6,718-6h-benzo[4,5]tieno[2,3-d]pyrimidín-2-yl)-propiónová-50-3- [3-chloro-5- (trifluoromethyl) -2-pyridyl] propanoic acid trans-3- (4-methoxybenzoyl) acrylic acid n-alpha- (tert-butyloxycarbonyl) -1-octahydroindole-2- (s) - (+) - hexahydromanedioic acid n- (3-chlorophenyl) phthalic acid 2- (4-tert-butylphenoxy) -2,2-difluoroacetic acid 2-ethylnonanoic acid 3- (5-bromo-2-ethoxyphenyl) acrylic acid fmoc-6-aminohexanoic acid chlorosuccinic acid gamma-d-glutamylaminoethylphosphonic acid 3-hydroxy-4,4,4-trichlorobutyric acid acetyl-d-aminoenantic acid 3- (methoxycarbonylmethylthio) 1-Cyclopropanedicarboxylic acid 4-Amino-acetanilide-2-sulfonic acid 2- (4-hexyl-benzoylamino) -benzoic acid 4,4-thiophene-2-carboxylic acid n-1,1-bis-hydroxymethyl-ethyl-SAS 3-isobutyrylamino-3- (4-methoxyphenyl) propionic acid biphenyl-3,5-dicarboxylic acid 3,3-di- (carbonyldiimino) bis-benzoic acid methyl 4-oxovaleric pinonic acid (cis-3-acetyl-2,2-dimethylcyclobutaneacetic) 3-chloropentanedioic acid Gibberellic acid (C19H22O6) 3- (nonylamido) benzoic acid 4- (trifluoromethyl) benzoic acid of 3- (allylsulfanyl) -2-thiophenecarboxylic acid, S '' - dibrómftalanilová acid, 3-hydroxynonanoic acid, 3- (4-oxo-3,4,5,6,7 1 8-6h-benzo [4,5] thieno [ 2,3-d] pyrimidin-2-yl) -propionic acid

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · ···· • • ···· • • ·· · • · ·· • · · ·· · • · ·· • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 4-(4-fenoxy-benzoyl)-benzoová kyselina 2,5-dijódbenzoová kyselina 3-(n-(2,4-difluórfenyl)karbamoyl)-5-norbomén-2-karboxylová kyselina benzo(c)fenantrén-3-karboxylová kyselina 2-metyl-2-(7-metylindán-4-yloxy)propiónová kyselina exo-2-bróm-5-5-etyléndioxy-bicyklo[2,2,1]heptán-syn-7-karboxylová kyselina 3-metoxy-2,4,5-trifluórbenzoová kyselina (+)-2-(1-naftoxy)propiónová kyselina 2,2-dichlór-1 -metyl-cyklopropánkarboxylová kyselina 2-fluór-4-(trifluórmetyl)fenyloctová kyselina (+/-)-azetidín-2-ón-4-karboxylová kyselina 4-(3-(3,5-d/-íerc-butyl-4-hydroxy-fenyl)-3-oxo-properiyl)benzoová kyselina levulová dimetyl-fosfát kyselina 2,4-dinitrofenyloctová kyselina 3,4-dichlórbenzénsulfónová kyselina boc-3-aminobenzoová kyselina 3,4-dimetylbenzoová kyselina 2-fluór-5-metylbenzoová kyselina n-alfa-(9-fluórenylmetyloxykarbonyl)-1-2-amino-5-ureido-n-valérová kyselina o-nitrobenzoová kyselina 2,3-dibrómjantárová kyselina beta-s-(4-metoxybenzylmerkapto)-izovalérová kyselina 4-bróm-7-oxo-6-oxa-bicyklo(3,2,1 )oktán-2-karboxylová kyselina 1-pentánsulfónová kyselina 5-hydroxyizoftalová kyselina s-4-chlórmandlová kyselina 1-hydroxy-2-oxo-1,2-dihydro-pyridín-3-karboxylová kyselina 3-acetamido-3-metylmaslová kyselina 3’-(trifluórmetyl)sukcínanilová kyselina 2-meo-4-metyl-6-(2,2,2-trichlór-1-hydroxy-etyl)-cyklohexánkarboxylová kyselina 4-etoxyškoricová4- (4-Phenoxy-benzoyl) -benzoic acid 2,5-diiodobenzoic acid 3- (n- (2,4-difluorophenyl) carbamoyl) -5-norbomene-2-carboxylic acid benzo (c) phenanthrene-3- 2-methyl-2- (7-methylindan-4-yloxy) propionic acid exo-2-bromo-5-5-ethylenedioxy-bicyclo [2.2.1] heptane-syn-7-carboxylic acid carboxylic acid 3-methoxy -2,4,5-trifluorobenzoic acid (+) - 2- (1-naphthoxy) propionic acid 2,2-dichloro-1-methyl-cyclopropanecarboxylic acid 2-fluoro-4- (trifluoromethyl) phenylacetic acid (+/-) -azetidin-2-one-4-carboxylic acid 4- (3- (3,5-tert-butyl-4-hydroxyphenyl) -3-oxo-properyl) benzoic acid levulinic dimethyl phosphate acid 2, 4-dinitrophenylacetic acid 3,4-dichlorobenzenesulfonic acid boc-3-aminobenzoic acid 3,4-dimethylbenzoic acid 2-fluoro-5-methylbenzoic acid n-alpha- (9-fluorenylmethyloxycarbonyl) -1-2-amino-5-ureido- n-valeric acid o-nitrobenzoic acid 2,3-dibromosuccinic acid beta-s- (4-methoxybenzylme) 4-Bromo-7-oxo-6-oxa-bicyclo (3,2,1) octane-2-carboxylic acid 1-pentanesulfonic acid 5-hydroxyisophthalic acid s-4-chloro-butyric acid 1-hydroxy-2 -oxo-1,2-dihydro-pyridine-3-carboxylic acid 3-acetamido-3-methylbutyric acid 3 '- (trifluoromethyl) succinilic acid 2-meo-4-methyl-6- (2,2,2-trichloro- 1-hydroxy-ethyl) -cyclohexanecarboxylic acid 4-ethoxycinnamic acid

• ·· • · • ··· • ·· • · • ··· • e • · • · • e • · • · ···· • • ···· • • • · • · • · • · • · • · • · • · • · ·· • · ·· ·· · · ·· · · ·· · · ·· · ·

kyselina 5-bróm-izoftalová kyselina 2'-chlór-5'-nitroftalanilová kyselina 2-metyl-3-p-tolyl-akrylová kyselina S.S.e.ej.y.ľ-heptafluór-M-bisítrifluórmetylJ^-hepténová kyselina 2,,4,-dimetylmaleanilová kyselina 4-acetoxybenzoová kyselina 3,6-disulfo-naftalén-1,8-dikarboxylová kyselina (r)-(-)-citra-jablčná (ο-2-metyl-jablčná) kyselina 1-oktánsulfónová kyselina 2-metyl-2-fenyl-hexándiová kyselina 3-noradamantánkarboxylová kyselina 2-kyano-3-(3,4-dihydroxy-5-metoxyfenyl)-akrylová kyselina 3,5-dinitro-4-hydroxyfenyloctová kyselina 2-chlór-3,4-dimetoxybenzoová kyselina 5-(trifluórmetyl)tieno[3,2-b]pyridín-6-karboxylová kyselina 9,9-dihydroxy-5-oxo-nonánová kyselina diizooktylfosfínová kyselina boc-nipekotínová kyselina 3,4-dichlór-2-tiofénkarboxylová kyselina n-alfa-fmoc-n-gama-aloc-1 -diaminomaslová kyselina c/s-2-(ŕerc-butoxykarbonylamino)-1-cyklopentánkarboxylová kyselina boc-4-aminobenzoová kyselina fosfatidová kyselina c/s-S'^'-dimetylhexahydroftalanilová kyselina 1,2,3-triazol-4,5-dikarboxylová kyselina /?-(3-nitrofenyl)-1,2,5,6-tetrahydroftalámová kyselina 3-((2-karboxy-etyl)-(4-metyl-tiazol-2-yl)-amino)-propiónová kyselina 2,3,4-trimetyl-cyklobutánkarboxylová kyselina 5-(2,-(3,-chlór-5’-trifluórmetyl)pyridylamino)metyl-3,4-dihydroizoxazol-2-3(n-etyltiokarbamoyltio)-propiónová kyselina n-alfa-boc-n-beta-brómacetyl-1-diamino-propiónová kyselina trans-Ί ,2-cyklohexándioctová • ·· ·· ···· ·· ··· · · ···· • ··· · · · · ·5-bromo-isophthalic acid 2'-chloro-5'-nitroftalanilová 2-methyl-3-p-tolyl-acrylic acid SSeej.y.ľ-heptafluoro-N-heptenoic acid bisítrifluórmetylJ ^ 2,, 4, - 4-acetoxybenzoic acid, 3,6-disulfonaphthalene-1,8-dicarboxylic acid (r) - (-) - citric acid (ο-2-methyl-malic acid) 1-octanesulfonic acid 2-methyl-2 -phenyl-hexanedioic acid 3-noradamantanecarboxylic acid 2-cyano-3- (3,4-dihydroxy-5-methoxyphenyl) -acrylic acid 3,5-dinitro-4-hydroxyphenylacetic acid 2-chloro-3,4-dimethoxybenzoic acid 5 - (trifluoromethyl) thieno [3,2-b] pyridine-6-carboxylic acid 9,9-dihydroxy-5-oxo-nonanoic acid diisoctylphosphinic acid boc-nipecotinic acid 3,4-dichloro-2-thiophenecarboxylic acid n-alpha- fmoc-n-gamma-aloc-1-diaminobutyric acid cis-2- (tert-butoxycarbonylamino) -1-cyclopentanecarboxylic acid boc-4-aminobenzoic acid phosphatidic acid cis-S 1 '- dimethyl 1,2,3-triazole-4,5-dicarboxylic acid R - (3-nitrophenyl) -1,2,5,6-tetrahydrophthalic acid 3 - ((2-carboxyethyl) - (4-methyl) -thiazol-2-yl) -amino) 2,3,4-trimethyl-cyclobutanecarboxylic acid 5- (2 - (3-chloro-5'-trifluoromethyl) pyridylamino) methyl-3,4-dihydroisoxazol 2-3 (n-ethylthiocarbamoylthio) -propionic acid n-alpha-boc-n-beta-bromoacetyl-1-diamino-propionic acid trans-Ί, 2-cyclohexanediacetic acid • ·· ·· ···· ·· ··· · · ···· · ··· · · · · ·

-53kyselina 2,6-difluórmandlová kyselina c/s-n-(2-chlórfenyl)hexahydroftalámová kyselina 2,6-dichlórpyridín-4-karboxylová kyselina n-(1-naftyl)-1,2,3,6-tetrahydroftalámová kyselina 3-(trifluórmetyltio)benzoová kyselina n-(2-brómfenyl)maleámová kyselina beta-glutámová kyselina 6-hydroxy-1-naftoová kyselina 4-(2-tienylmetylénamino)benzoová kyselina n-(2,4-dimetoxy-fenyl)-ftalámová kyselina heptafluór-2-hexénová kyselina (4-benzyloxy-5-metoxy-2-nitro-fenyl)-octová kyselina 3-(4-chlórfenyl)propiónová kyselina boc-1-beta-aminomaslová kyselina (4-fluórfenyltio)octová kyselina (2-izopropylsulfanyl-acetylamino)-octová kyselina 2-(3,5-dinitro-tiofén-2-ylamino)-pentándiová kyselina 3,3'-dichlórpivalová kyselina (2-butyryl-fenoxy)-octová kyselina styrénfosfónová kyselina 1 -(2-fluórfenyl)cyklopentánkarboxylová kyselina 2-(2,3-dimetoxystyryl)glyoxylová kyselina 3,5-ď/-ŕerc-butylsalicylová kyselina 2-(pentametylbenzoyl)benzoová kyselina 4-etyl-2-pyridínkarboxylová kyselina n,/?-dodekametylénbis(glutarámová) kyselina n-cbz-(2r,3r)-3-amino-2-hydroxy-4-fenyl-maslová kyselina karboxymetánsulfonylmetánsulfonyl-octová kyselina 3-(2,3,4-trimetoxyfenyl)propiónová kyselina 17-(p-toluénsulfonyloxy)-heptadekánová kyselina 4-((2-hydroxy-5-nitro-benzylidén)-amino)-benzoová kyselina 4-((naftalén-1 -ylmetylén)-amino)-benzoová2,6-Difluoromandelic acid cis- (2-chlorophenyl) hexahydrophthalic acid 2,6-dichloropyridine-4-carboxylic acid n- (1-naphthyl) -1,2,3,6-tetrahydrophthalic acid 3- ( trifluoromethylthio) benzoic acid n- (2-bromophenyl) maleic acid beta-glutamic acid 6-hydroxy-1-naphthoic acid 4- (2-thienylmethyleneamino) benzoic acid n- (2,4-dimethoxyphenyl) -phthalic acid heptafluoro- 2-hexenoic acid (4-benzyloxy-5-methoxy-2-nitro-phenyl) -acetic acid 3- (4-chlorophenyl) propionic acid boc-1-beta-aminobutyric acid (4-fluorophenylthio) acetic acid (2-isopropylsulfanyl) -acetylamino) -acetic acid 2- (3,5-dinitro-thiophen-2-ylamino) -pentanedioic acid 3,3'-dichloropivalic acid (2-butyryl-phenoxy) -acetic acid styrene phosphonic acid 1- (2-fluorophenyl) cyclopentanecarboxylic acid 2- (2,3-dimethoxystyryl) glyoxylic acid 3,5-tert-butylsalicylic acid 2- (pentamethylbenzoyl) benzoic acid 4-ethyl-2-pyr N, R-dodecamethylenebis (glutaramic acid) n-cbz- (2r, 3r) -3-amino-2-hydroxy-4-phenylbutyric acid carboxymethanesulfonylmethanesulfonyl acetic acid 3- (2,3,4-trimethoxyphenyl) ) Propionic acid 17- (p-toluenesulfonyloxy) -heptadecanoic acid 4 - ((2-hydroxy-5-nitro-benzylidene) -amino) -benzoic acid 4 - ((Naphthalen-1-ylmethylene) -amino) -benzoic acid

• ·· • · • ··· • ·· • · • ··· • · • · • · • · • · • · ···· • • ···· • • ·· • · • · ·· • · • · • · • · ·· ·· ·· ·· ·· · · ·· · · ·· · · • e • e

kyselina 3-benzoyl-3-benzylidénpropiónová valerylsalicylát kyselina 3,4-difenyl-cyklobután-1,2-dikarboxylová kyselina 2-chlór-5-(trifluórmetyl)benzoová kyselina 3-pyridínpropiónová kyselina 4-(2,5-bis-(2,2-dimetyl-propyl)-fenoxy)-maslová kyselina 3-(oktadecyloxy)benzoová kyselina (r)-(+)-2-brómpropiónová kyselina 3,4-dihydro-6-metoxy-1 -naftoová kyselina 2-nitro-4-(2,2,2-trif luór-1 -hydroxy-1 -trifluórmetyl-etylj-benzoová kyselina glykolová kyselina 2-izochinolin-1 -ylmetyl-benzoová kyselina 3,4,4-trichlór-2-dichlórmetylén-but-3-énová kyselina 4-metyl-2-fenyl-1,2,3-triazol-5-karboxylová kyselina 3-bróm-4-fluórškoricová kyselina 8-nitro-chinolín-4-karboxylová kyselina 3-(3-me-5-oxo-4,5-dihydro-pyrazol-1-yl)-2-fenylkarbamoyl-benzénsulfónová kyselina 4-(trifluórmetyltio)benzoová kyselina 4-(3-(2-etylfenyl)ureido)salicylová kyselina 2-etylmaleanilová kyselina p-xylén-2-sulfónová kyselina 2,3,4,4,5,5,5-heptafluór-2-penténová kyselina 4-jód-3-nitrobenzoová kyselina 2-benzoylamino-3-(dietoxy-fosforyl)-3-fenyl-akrylová kyselina 4,4,-dinitrostilbén-2,2’-disulfónová kyselina ŕrans-4-/?-butylcyklohexánkarboxylová kyselina 3,4-difluór-5-(trifluórmetyl)fenyloctová kyselina 2-nitro-alfa,alfa,alfa-trifluór-p-toluylová kyselina 2,4-dichlórpyridín-5-karboxylová kyselina 2-(morfolin-4-karbotioylsulfanyl)-propiónová kyselina alfa-metyl-4-nitroškoricová kyselina 6-metyl-2-fenylimidazo[1,2-a]pyridín-3-karboxylová3-benzoyl-3-benzylidenepropionic acid valerylsalicylate 3,4-diphenyl-cyclobutane-1,2-dicarboxylic acid 2-chloro-5- (trifluoromethyl) benzoic acid 3-pyridinepropionic acid 4- (2,5-bis- (2 (2-Dimethyl-propyl) -phenoxy) -butyric acid 3- (octadecyloxy) -benzoic acid (R) - (+) - 2-bromopropionic acid 3,4-dihydro-6-methoxy-1-naphthoic acid 2-nitro- 4- (2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl) -benzoic acid glycolic acid 2-isoquinolin-1-ylmethyl-benzoic acid 3,4,4-trichloro-2-dichloromethylene-but- 3-enoic acid 4-methyl-2-phenyl-1,2,3-triazole-5-carboxylic acid 3-bromo-4-fluorocinnamic acid 8-nitroquinoline-4-carboxylic acid 3- (3-me-5 -oxo-4,5-dihydro-pyrazol-1-yl) -2-phenylcarbamoyl-benzenesulfonic acid 4- (trifluoromethylthio) benzoic acid 4- (3- (2-ethylphenyl) ureido) salicylic acid 2-ethylmaleanilic acid p-xylene -2-sulfonic acid 2,3,4,4,5,5,5-heptafluoro-2-pentenoic acid 4-iodo-3 nitrobenzoic acid 2-benzoylamino-3- (diethoxy-phosphoryl) -3-phenyl-acrylic acid 4,4, 2,2 -dinitrostilbén-disulfonic acid trans-4 - /? - Butylcyclohexanecarboxylic 3,4-difluoro- 5- (trifluoromethyl) phenylacetic acid 2-nitro-alpha, alpha, alpha-trifluoro-p-toluic acid 2,4-dichloropyridine-5-carboxylic acid 2- (morpholine-4-carbothioylsulfanyl) -propionic acid alpha-methyl-4 6-methyl-2-phenylimidazo [1,2-a] pyridine-3-carboxylic acid

• · • · · • ·• • •

-55• ·· ·· ·· kyselina (1-(2-(3,4-dimetoxy-fenyl)-etyl)-5-etyl-2-oxo-piperidín-4-yl)-octová kyselina 5-karboxyvanilová kyselina 3-benzyl-chinolín-4-karboxylová kyselina 3-(4-metyltiobenzoyl)propiónová kyselina n-(2-benzylsulfanyl-benzotiazol-6-yl)-sukcinamová kyselina 3-(8-benzyl-9-oxo-6,7,8,9-tetrahydro-5h-benzocykloheptén-8-yl)propiónová kyselina sukcínanilová kyselina n-toluénsulfonyl-3-pyrolkarboxylová kyselina 2-etyl-3-(4-metoxy-fenyl)-akrylová kyselina maslová kyselina (1 alfa,2alfa,3beta,4beta)-2,4-bis(4-hydroxyfenyl)-1,3-cyklobutándikarboxylová kyselina 3,4-difluór-5-(trifluórmetyl)benzoová kyselina 2,3,5,6-tetrafluór-p-toluylová kyselina 2-bróm-4,5-dimetoxybenzoová kyselina 3-(2-benzoylamino-3-(4-metoxy-fenyl)-akryloylamino)-propiónová kyselina 5-nitro-1,2,3,4-tetrahydro-1,4-etenonaftalén-2,3-dikarboxylová kyselina 3-(4-n-heptylbenzoyl)propiónová kyselina (1 -oxo-dekahydro-naftalen-2-yl)-octová kyselina 2-(karboxy-hydroxy-metyl)-6-hydroxy-4-metyl-cyklohexánkarboxylová kyselina n-furfurylftalámová kyselina 3-(2-furyl)-2-oximino-propiónová kyselina 10,11-dihydroxy-undekánová kyselina 2-tioorotová kyselina 2,-chlór-5'-nitroglutaranilová kyselina 8-nonínová kyselina (rs)-1-aminoindán-1,5-dikarboxylová kyselina 4-(3,5-diizopropyl-benzoylamino)-benzoová kyselina 2-butyl-3-(2-metoxy-fenyl)-akrylová kyselina n-fmoc-1 -amino-cyklopropán-1 -karboxylová kyselina iminodioctová bis(p-nitrofenyl)fosfát * ·· ·· ···· ·· ··· ·· · · · · • ··· · · · e · ······ ···· • · · ···· t · ··· ·· ·· ·· ·· ·-55 • ····· 1- (2- (3,4-Dimethoxy-phenyl) -ethyl) -5-ethyl-2-oxo-piperidin-4-yl) -acetic acid 5-carboxyvanilic acid 3-Benzyl-quinoline-4-carboxylic acid 3- (4-methylthiobenzoyl) propionic acid N- (2-benzylsulfanyl-benzothiazol-6-yl) -succinamic acid 3- (8-benzyl-9-oxo-6,7, 8,9-tetrahydro-5h-benzocyclohepten-8-yl) propionic acid succinilic acid n-toluenesulfonyl-3-pyrrolecarboxylic acid 2-ethyl-3- (4-methoxyphenyl) -acrylic acid butyric acid (1 alpha, 2alpha, 3beta, 4beta) -2,4-bis (4-hydroxyphenyl) -1,3-cyclobutanedicarboxylic acid 3,4-difluoro-5- (trifluoromethyl) benzoic acid 2,3,5,6-tetrafluoro-p-toluylic acid 2 -bromo-4,5-dimethoxybenzoic acid 3- (2-benzoylamino-3- (4-methoxyphenyl) -acryloylamino) -propionic acid 5-nitro-1,2,3,4-tetrahydro-1,4-etenonaphthalene -2,3-dicarboxylic acid 3- (4-n-heptylbenzoyl) propionic acid (1-oxo-decahydro-naphthalen-2-yl) -acetic acid 2- (carboxy-hydroxymethyl) -6-hydro xy-4-methyl-cyclohexanecarboxylic acid n-furfuryl-phthalic acid 3- (2-furyl) -2-oximino-propionic acid 10,11-dihydroxy-undecanoic acid 2-thioorotic acid 2 , -chloro-5'-nitroglutaranilic acid 8- (rs) -1-aminoindan-1,5-dicarboxylic acid 4- (3,5-diisopropyl-benzoylamino) -benzoic acid 2-butyl-3- (2-methoxy-phenyl) -acrylic acid n-fmoc- 1-Amino-cyclopropane-1-carboxylic acid iminodiacetic acid bis (p-nitrophenyl) phosphate * ·· ·············· · · · · ··· ··· ···· · · ··· t · ··· ·· ·· ·· ·· ·

-56kyselina 2-benzoylamino-3-(3,4-dimetoxy-fenyl)-propiónová kyselina 3-(3,5-dimetyl-naftalén-2-yl)-2-metyl-maslová kyselina 2-etoxy-4-metoxybenzoová kyselina ď/-2-hydroxy-n-maslová kyselina (2-karbamoylfenoxy)octová kyselina 5-acetylsalicylová kyselina n-benzylftalámová kyselina n-(4-metylfenyl)maleámová kyselina 1-leucyl-1-glutámová kyselina (4-(3-metyl-ureido)-benzoylamino)-octová kyselina arabinová kyselina 9-metylundekánová kyselina 2-(metyltio)benzoová kyselina arachidónová kyselina 2,4-dichlórfenyloctová kyselina 2-dibenzotiofénpropiónová kyselina 3-(3,4-etyléndioxybenzoyl)propiónová kyselina 2-metyl-2-(4-metyl-3-oxocyklohexyl)malónová kyselina 8-kyano-naftalén-1 -sulfónová kyselina 5-(metyltio)tiofén-2-karboxylová kyselina 2-brómdekánová kyselina 2-izopropylidénaminooxy-maslová kyselina alylmalónová kyselina 3,5-dimetoxy-4-metylbenzoová kyselina alfa-(4-metoxy-1-naftyl)-o-toluylová kyselina 3-(4-etoxyfenyl)propiónová kyselina 3-(2-nitro-4-trifluórmetylfenoxy)-2-tiofénkarboxylová kyselina 3-(2,6-dichlór-fenyl)-2-metyl-akrylová kyselina 4-(4-kyano-fenoxy)-benzoová kyselina (lAS.ejJ-hexachlór-S-norbornén^.S-dikarboxylová) kyselina 12-formyl-tricyklo(8,2,2,2(4,7))hexadeka-hexaén-5-karboxylová kyselina n-(2,6-dimetylfenyl)-1,2,3,6-tetrahydroftalámová ·· ···· ·Ι· ···· ·· · ·*· ·· ·· ·· ·· ···2-Benzoylamino-3- (3,4-dimethoxy-phenyl) -propionic acid 3- (3,5-dimethyl-naphthalen-2-yl) -2-methyl-butyric acid 2-Ethoxy-4-methoxy-benzoic acid 1 '-2-hydroxy-n-butyric acid (2-carbamoylphenoxy) acetic acid 5-acetylsalicylic acid n-benzylphthalic acid n- (4-methylphenyl) maleic acid 1-leucyl-1-glutamic acid (4- (3-methyl) -ureido-benzoylamino) -acetic acid arabinic acid 9-methylundecanoic acid 2- (methylthio) benzoic acid arachidonic acid 2,4-dichlorophenylacetic acid 2-dibenzothiophenepropionic acid 3- (3,4-ethylenedioxybenzoyl) propionic acid 2-methyl-2 - (4-Methyl-3-oxocyclohexyl) malonic acid 8-Cyano-naphthalene-1-sulfonic acid 5- (methylthio) thiophene-2-carboxylic acid 2-Bromodecanoic acid 2-Isopropylideneamininooxybutyric acid Allyl malonic acid 3,5-Dimethoxy 4-Methylbenzoic acid alpha- (4-methoxy-1-naphthyl) -o-toluic acid 3- (4-ethoxyphenyl) propionic acid 3- (2 -nitro-4-trifluoromethylphenoxy) -2-thiophenecarboxylic acid 3- (2,6-dichloro-phenyl) -2-methyl-acrylic acid 4- (4-cyano-phenoxy) -benzoic acid (10E) -hexachloro-S 12-formyl-tricyclo (8,2,2,2 (4,7)) hexadeca-hexaene-5-carboxylic acid n- (2,6-dimethylphenyl) -1,2-non-boronene (5-dicarboxylic acid) 3,6-tetrahydrophthalama ·······································

-57kyselina poly-1-glutámová kyselina (s)-(+)-ketopinová kyselina 3,4,5-trimetoxy-2-nitro-benzoová kyselina homovanilová kyselina 8-chlór-4-dibenzofuránkarboxylová kyselina 5I6a,7I7a-tetrahydro-4h-cyklopropa(e)acenaftylén-7-karboxylová kyselina 3-(n-(2,6-xylyl)karbamoyl)propiónová kyselina (4-metoxyfenyl)fenylfosfínová kyselina 4-acetamidomaslová kyselina ŕrans-norpinová kyselina fmoc-(3r,4s)-4-amino-3-hydroxy-6-metylheptánová kyselina 3,4,5,6-tetrachlór-pyridín-2-karboxylová kyselina 2'-metoxy-5'-metylmaleanilová kyselina 3-(oktán-1 -sulfonyl)-propiónová kyselina 2-chlórpropiónová kyselina 4-(4-(1,3-dioxo-1,3-dihydro-izobenzofurán-5-karbonyl)-fenoxy)-benzoová kyselina 12-metyltetradekánová kyselina trifenyloctová kyselina 3-metyl-1 -oxo-izochroman-5-karboxylová kyselina (4-fenyl-5-fenylamino-4h-(1,2I4)triazol-3-ylsulfanyl)-octová kyselina 9-hydroxyimino-9,10-dihydro-antracén-1 -karboxylová kyselina 7-metoxy-1 -metyl-4-oxo-2,3,4,5-tetrahydro-1 h-benzo[d]azepín-2-karboxylová kyselina 2,5-dichlórfenyltioglykolová kyselina 1 -kyanocyklopropánkarboxylová kyselina 2,6-dinitromezitylén-4-sulfónová kyselina 3-(4-hydroxy-3-metoxy-fenyl)-2-metyl-akrylová kyselina 3-(4-cyklohexylbenzoyl)akrylová kyselina 2-kyano-2-metyl-3-fenyl-propiónová kyselina 2,3-dimetoxyfenyloctová kyselina n-alfa-(benzyloxykarbonyl)-gama-(benzylester)-ď-glutámová kyselina n-(4-metoxyfenyl)tetrachlórftalámová-57 poly-1-glutamic acid (s) - (+) - ketopinic acid 3,4,5-trimethoxy-2-nitro-benzoic acid homovanilic acid 8-chloro-4-dibenzofuranecarboxylic acid 5 L 6a, 7 L 7a- tetrahydro-4h-cyclopropa (e) acenaphthylene-7-carboxylic acid 3- (n- (2,6-xylyl) carbamoyl) propionic acid (4-methoxyphenyl) phenylphosphinic acid 4-acetamidobutyric acid trans-norpinic acid fmoc- (3r, 4s) -4-amino-3-hydroxy-6-methylheptanoic acid 3,4,5,6-tetrachloro-pyridine-2-carboxylic acid 2'-methoxy-5'-methylmaleanilic acid 3- (octane-1-sulfonyl) -propionic acid 2-chloropropionic acid 4- (4- (1,3-dioxo-1,3-dihydro-isobenzofuran-5-carbonyl) -phenoxy) -benzoic acid 12-methyltetradecanoic acid triphenylacetic acid 3-methyl-1-oxo -isochroman-5-carboxylic acid (4-phenyl-5-phenylamino-4h- (1,2 L ) triazol-3-ylsulfanyl) -acetic acid 9-hydroxyimino-9,10-dihydro-anthracene-1-carboxylic acid 7-Methoxy-1-methyl-4-oxo-2,3,4,5-tetrahydro- 1 H -benzo [d] azepine-2-carboxylic acid 2,5-dichlorophenylthioglycolic acid 1-cyanocyclopropanecarboxylic acid 2,6-dinithromezitylene-4-sulfonic acid 3- (4-hydroxy-3-methoxyphenyl) -2-methyl -acrylic acid 3- (4-cyclohexylbenzoyl) acrylic acid 2-cyano-2-methyl-3-phenyl-propionic acid 2,3-dimethoxyphenylacetic acid n-alpha- (benzyloxycarbonyl) -gamma- (benzyl ester) -β-glutamic acid n- (4-methoxyphenyl) tetrachlórftalámová

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-58kyselina 4-fenylmaslová kyselina 3-nitrobenzaldehyd-4-sulfónová kyselina n-oktadecyljantárová kyselina pyridín-4-sulfónová kyselina 2-hydroxy-2-trifluórmetylmaslová kyselina 2,6-dimetyl-tereftalová kyselina tereftalová kyselina 3,5-d/-ŕerc-butyl-4-hydroxyškoricová kyselina 3-etoxypropiónová kyselina 4-alyl-2-metoxyfenoxyoctová kyselina d-(-)-diizopropyl-d-vínna kyselina 4-brómmetyl-naftalén-1 -karboxylová kyselina 2,-chlór-6'-metylsukcínanilová kyselina 2',4'-dimetoxyhexahydroftalanilová kyselina 2,7-difluór-9-oxo-4-fluorénkarboxylová kyselina 2-metoxy-6-(2,2-dimetylpropionamido)cyklohexánkarboxylová kyselina 3-hydroxyfenyloctová kyselina 6-jódhexánová kyselina 3-bróm-2,6-dimetoxybenzoová kyselina 3-(4-chlórfenyl)-2-fenyl-propiónová kyselina (s)-(-)-2-chlór-3-metylpentánová kyselina alfa-chlór-3-(trifluórmetyl)-hydroškoricová kyselina 3-(hexadekán-1 -sulfonyl)-propiónová kyselina 12(s)-hydroxy-(5z,8e, 10e)-heptadekatriénová kyselina 1,3,5-cyklohexántrikarboxylová kyselina 3-hydroxy-4,5-dimetoxy-benzoová kyselina 4-bróm-1,2,3,4-tetrachlór-l ,3-butadién-1-karboxylová kyselina (2,4-xylyl)fosfónová kyselina 4-bróm-3-metoxy-naftalén-2-karboxylová kyselina (+/-)-treo-4-metylglutámová oxím kyseliny levulovej kyselina c/s-13-oktadecénová • ·· ·· ···· ·· · «· · · 4 · · · ·· • 4·· · · · · ·· ······ f·** í • · · · · · I · ·· ··· ·3 ·4 ·Φ ·····4-Phenylbutyric acid 3-nitrobenzaldehyde-4-sulfonic acid n-octadecylsuccinic acid pyridine-4-sulfonic acid 2-hydroxy-2-trifluoromethylbutyric acid 2,6-dimethyl-terephthalic acid terephthalic acid 3,5-d-tert -butyl-4-hydroxycinnamic acid 3-ethoxypropionic acid 4-allyl-2-methoxyphenoxyacetic acid d - (-) - diisopropyl-d-tartaric acid 4-bromomethyl-naphthalene-1-carboxylic acid 2 , -chloro-6'-methylsuccinilic acid 2 ', 4'-dimethoxyhexahydrophthalanic acid 2,7-difluoro-9-oxo-4-fluorenecarboxylic acid 2-methoxy-6- (2,2-dimethylpropionamido) cyclohexanecarboxylic acid 3-hydroxyphenylacetic acid 6-iodohexanoic acid 3-bromo- 2,6-Dimethoxybenzoic acid 3- (4-chlorophenyl) -2-phenylpropionic acid (s) - (-) - 2-chloro-3-methylpentanoic acid alpha-chloro-3- (trifluoromethyl) hydrocinnamic acid 3- (Hexadecane-1-sulfonyl) -propionic acid 12 (s) -Hydroxy- (5z, 8e, 10e) -heptadecatrienoic acid 1,3,5-cyclohexanetricarboxylic acid 3-hydroxy-4,5-dimethoxybenzoic acid 4-bromo-1,2,3,4-tetrachloro-1,3-butadiene-1-carboxylic acid (2,4- xylyl) phosphonic acid 4-bromo-3-methoxy-naphthalene-2-carboxylic acid (+/-) - threo-4-methylglutamic acid oxime levisic acid cis-13-octadecenic acid · ·· ·· ···· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · Φ ·····

-59kyselina 4-(metylsulfonyl)benzoová kyselina (3-metoxy-4-fenoxy-fenyl)-octová kyselina karboxypyrazolón-2,5-disulfónová kyselina 5-metoxy-1 -indanón-3-octová kyselina tnp-1 -glutámová kyselina 4-chlórmaslová kyselina 1 -naftylamín-2,4,7-trisulfónová kyselina 6-hydroxy-3-oxo-7a-propionyl-oktahydro-indén-1-karboxylová kyselina furán-2,5-dikarboxylová kyselina alfa-(4-chlórfenyl)-4-nitroškoricová kyselina 2-brómvalérová kyselina 2,2-dietylmaslová kyselina d/-glutámová kyselina 4-(4-hydroxybenzylidénamino)salicylová kyselina (s)-(+)-2-metylmasiová kyselina n-alfa-n-beta-bis-boc-1 -diaminopropiónová kyselina 2,2-difenylpropiónová kyselina 1 -hydroxycyklohexánkarboxylová kyselina stearová kyselina 2-(2-karboxy-etylamino)-jantárová kyselina kumarín-3-karboxylová kyselina 4-(2-(4-íerc-oktylfenoxy)etoxy)benzoová kyselina 2-(2-chlór-4-fluórfenyltio)octová kyselina 5-bróm-2-metyl-benzoová kyselina myristová kyselina c/s-10-nonadecénová kyselina 2-bróm-4-fluórškoricová kyselina 1 -(4-metylbenzénsulfonyl)indol-3-akrylová kyselina 1-et-6-fluór-7-hydroxy-4-oxo-1,4-dihydro-(1,8)naftyridín-3-karboxylová kyselina 3,4-dietoxyfenyloctová kyselina 12(r)-hydroxy-16-heptadecínová kyselina 4-chlórbenzénsulfínová-59 4- (methylsulfonyl) benzoic acid (3-methoxy-4-phenoxy-phenyl) -acetic acid carboxypyrazolone-2,5-disulfonic acid 5-methoxy-1-indanone-3-acetic acid tp-1-glutamic acid 4 1-naphthylamine-2,4,7-trisulfonic acid 6-hydroxy-3-oxo-7α-propionyl-octahydro-indene-1-carboxylic acid furan-2,5-dicarboxylic acid alpha- (4-chlorophenyl) 4-nitrocinnamic acid 2-bromovaleric acid 2,2-diethylbutyric acid d-glutamic acid 4- (4-hydroxybenzylideneamino) salicylic acid (s) - (+) - 2-methylbutyric acid n-alpha-n-beta-bis -boc-1-diaminopropionic acid 2,2-diphenylpropionic acid 1-hydroxycyclohexanecarboxylic acid stearic acid 2- (2-carboxy-ethylamino) -succinic acid Coumarin-3-carboxylic acid 4- (2- (4-tert-octylphenoxy) ethoxy ) Benzoic acid 2- (2-chloro-4-fluorophenylthio) acetic acid 5-bromo-2-methyl-benzoic acid myristic acid cis-10-nonadecenic acid 2-Bromo-4-fluorocinnamic acid 1- (4-methylbenzenesulfonyl) indole-3-acrylic acid 1-Et-6-fluoro-7-hydroxy-4-oxo-1,4-dihydro- (1,8) naphthyridine- 3-Carboxylic acid 3,4-diethoxyphenylacetic acid 12 (R) -hydroxy-16-heptadecinic acid 4-chlorobenzenesulfonic acid

-60kyselina 11-bróm-undec-10-ínová kyselina 3-[(4,6-dimetoxypyrimidín-2-yl)oxy]pyridín-2-karboxylová kyselina 3,4,5-trimetoxybenzoová kyselina 2-fluór-4-oktyloxybenzoová kyselina 4-metyl-2-tioxo-2,3-dihydro-tiazol-5-karboxylová kyselina 4-metyl-2-penténová kyselina 2-karboxymetyl-2-metyl-cyklohexánkarboxylová kyselina 7-hydroxy-4-metyl-kumarón-1 -yl-octová kyselina 15-pentánbisfosfónová kyselina ŕrans-3-furánakrylová kyselina 3-acetamido-p-toluylová kyselina 3-[4-(metylsulfonyl)fenyl]-(2e)-propénová kyselina 4-fluór-2,3,5,6-tetrametyl-benzoová kyselina 4-tricyklo(4.3.1.1 (3,8)undekánkarboxylová kyselina 2-metoxy-4-nitrobenzoová kyselina vanilová kyselina n-(4-acetylfenyl)-maleanilová kyselina taurín-n,n-dioctová kyselina 4,5,515-tetrafluór-4-(heptafluórpropoxy)pentánová kyselina dietylmalónová kyselina 3-(3-(3-(trifluórmetyl)fenyl)ureido)benzoová kyselina 5-bróm-2-nitrobenzoová kyselina 2-(4-cinamoylfenoxy)octová kyselina adrenová kyselina tetrakozánová kyselina 3-(trifluórmetyl)antranilová kyselina 3-(2-o-tolyloxy-acetylamino)-benzoová kyselina n-(2,4,6-trimetylfenyl)glutarámová kyselina 2,,4'-dichlórsukcínanilová kyselina 2,3-dihydrobenzo[b]furán-5-karboxylová kyselina 3-(2-chlórfenyl)propiónová kyselina 2-fluórpalmitová11-Bromo-undec-10-ynoic acid 3 - [(4,6-dimethoxypyrimidin-2-yl) oxy] pyridine-2-carboxylic acid 3,4,5-trimethoxybenzoic acid 2-fluoro-4-octyloxybenzoic acid 4-methyl-2-thioxo-2,3-dihydro-thiazole-5-carboxylic acid 4-methyl-2-pentenoic acid 2-carboxymethyl-2-methyl-cyclohexanecarboxylic acid 7-hydroxy-4-methyl-coumarone-1- Acetic acid 15-pentanebisphosphonic acid trans-3-furanacrylic acid 3-acetamido-p-toluic acid 3- [4- (methylsulfonyl) phenyl] - (2e) -propenoic acid 4-fluoro-2,3,5,6 -tetramethyl-benzoic acid 4-tricyclo (4.3.1.1 (3,8) undecanecarboxylic acid 2-methoxy-4-nitrobenzoic acid vanilic acid n- (4-acetylphenyl) -maleeanilic acid taurine-n, n-diacetic acid 4,5 5 1 5-Tetrafluoro-4- (heptafluoropropoxy) pentanoic acid Diethyl malonic acid 3- (3- (3- (trifluoromethyl) phenyl) ureido) benzoic acid 5-Bromo-2-nitrobenzoic acid 2- (4-cinamoylphenoxy) acetic acid adrenic acid and octadecanoic acid 3- (trifluoromethyl) anthranilic acid 3- (2-o-tolyloxy-acetylamino) -benzoic acid N- (2,4,6-trimethylphenyl) glutaramic acid 2 ', 4'-dichlórsukcínanilová 2,3-dihydro-benzo [b] furan-5-carboxylic acid 3- (2-chlorophenyl) propionic acid 2-fluoropalmitic acid

-61 8888 •8 88 88*8 ·· •-61 8888 • 8 88 88 * 8

888888

8 8 β 8 kyselina 5-(4-metoxyfenyl)-2,3-dihydro-1h-pyrolizín-6,7-dikarboxylová kyselina (5-kyano-2-(4-metoxy-fenyl)-6-oxo-cyklohex-1-enyl)-octová kyselina glutatiónsulfónová kyselina 4-(4-acetamidofenylimino)-2,3-dichlór-2-buténová kyselina (4-benzyloxy-3-metoxy-fenyl)-octová kyselina 2-fenyl-hexándiová kyselina 4-metyl-2-oxovalérová kyselina 2'-benzoyl-4'-chlórmaleanilová kyselina 5,6-acenafténdikarboxylová kyselina 5-(2-chlór-5-(trifluórmetyl)fenyl)-2-furoová kyselina 3-(2,4-dimetylbenzoyl)propiónová kyselina 2-fluór-3-(trifluórmetyl)fenyloctová kyselina 4,5-dihydro-1 -(metyltio)benzo[c]tiofén-3-karboxylová kyselina (2-karboxymetyl-cyklopropyl)-octová kyselina 2-(butylkarbamoyl)benzoová kyselina 3-alyloxypropiónová kyselina 2'-karbamoyl-bifenyl-2-karboxylová kyselina 6-(1,3-dioxo-1 h,3h-benzo(de)izochinolín-2-yl)-hexánová kyselina 3,5-diizopropylsalicylová kyselina 4-etylbenzénsulfónová kyselina boc-1-pipekolínová kyselina 2,6-dichlór-4-(trifluórmetyl)fenyloctová kyselina 3-tiofénmalónová kyselina 3-hydroxy-2,2-dimetyl-3-fenylpropiónová kyselina 3-(9-metyl-9h-fluorén-9-yl)-rnaslová kyselina 2-(1,2,3I4I5-pentahydroxy-pentyl)-tiazolidín-4-karboxylová kyselina d/-atromliečna (2-hydroxy-2-fenylpropiónová) kyselina n-ŕerc-boc-(2r,3r)-3-amino-2-hydroxy-5-metylhexánová kyselina 2-(1-naftoyl)benzoová kyselina 1 -(2-(3-chlór-5-trifluórmetylpyridyl)indol-3-propénová kyselina 4*-butylmaleanilová kyselina 4-fluór-3,5-dimetyl-benzoová8 8 β 8 5- (4-Methoxy-phenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid (5-cyano-2- (4-methoxy-phenyl) -6-oxo-cyclohex- 1-enyl) -acetic acid glutathione sulfonic acid 4- (4-acetamidophenylimino) -2,3-dichloro-2-butenoic acid (4-benzyloxy-3-methoxyphenyl) -acetic acid 2-phenyl-hexanedioic acid 4-methyl 2-Oxovaleric acid 2'-benzoyl-4'-chloraleanilic acid 5,6-acenaphthenedicarboxylic acid 5- (2-chloro-5- (trifluoromethyl) phenyl) -2-furoic acid 3- (2,4-dimethylbenzoyl) propionic acid 2-fluoro-3- (trifluoromethyl) phenylacetic acid 4,5-dihydro-1- (methylthio) benzo [c] thiophene-3-carboxylic acid (2-carboxymethyl-cyclopropyl) -acetic acid 2- (butylcarbamoyl) benzoic acid 3-Allyloxypropionic acid 2'-carbamoyl-biphenyl-2-carboxylic acid 6- (1,3-dioxo-1h, 3h-benzo (de) isoquinolin-2-yl) -hexanoic acid 3,5-diisopropylsalicylic acid 4- ethylbenzenesulfonic acid boc-1-pipecolinic acid 2,6-dichloro-4- (tri fluoromethyl) phenylacetic acid 3-thiophenemalonic acid 3-hydroxy-2,2-dimethyl-3-phenylpropionic acid 3- (9-methyl-9h-fluoren-9-yl) butyric acid 2- (1,2,3 L 4 I, 5-pentahydroxy-pentyl) -thiazolidine-4-carboxylic acid, d / -atromliečna (2-hydroxy-2-phenyl-propionic acid) of n-t-Boc- (2R, 3R) -3-amino-2-hydroxy-5- 2- (1-naphthoyl) benzoic acid methylhexanoic acid 1- (2- (3-chloro-5-trifluoromethylpyridyl) indole-3-propenoic acid) 4-fluoro-3,5-dimethylbenzoic acid

-62• · ··· • · · • · • ·· ·· ···· kyselina 4-chlór-3-fluórbenzoová kyselina n-alfa-fmoc-n-gama-boc-d-diaminomaslová kyselina cyklohexa-2I4-dienyl-(2,3,5,6-tetrametyl-fenyl)-octová kyselina 8-(4-metoxy-fenyl)-6-metyl-8h-[1,3]dioxolo[4,5-g]chromén-7-karboxylová kyselina 11-(4-chlór-fenylsulfanyl)-undekánová kyselina 1,3-dioxo-2-p-tolyl-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina c/s-2-(p-metylbenzoyl)-1 -cyklohexán-karboxylová kyselina slizová kyselina 4'-(metyltio)sukcínanilová kyselina 3-etoxy-2-buténová kyselina acetoxyoctová kyselina 5-metyl-2-nitrobenzoová kyselina 4-chlór-2-fluórbenzoová kyselina 2,5-dimetoxyškoricová kyselina (+/-)-beta-fenylglutámová kyselina 3-metyl-2-oxomaslová kyselina 1-heptánsulfónová kyselina 4-metyl-3-nitrobenzoová kyselina 2-karboxyškoricová kyselina alfa-metylškoricová kyselina 4-(3-hexadecyl-2-tioureido)-benzoová kyselina dehydroabietová kyselina (2-nitro-benzénsulfonylamino)-octová kyselina (3-benzyloxy-4-metoxy-fenyl)-octová kyselina 5-bróm-2-jódbenzoová kyselina 1,1,3-trimetyl-3-fenylindán-4',5-dikarboxylová kyselina oxaloctová kyselina 2-aminotereftalová kyselina perfluórhexánová kyselina 2,6-dichlórfenyloctová kyselina 6-bróm-2-pyridin-3-yl-chinolín-4-karboxylová kyselina 4-(chlórmetyl)benzoová-62 4-chloro-3-fluorobenzoic acid n-alpha-fmoc-n-gamma-boc-d-diaminobutyric acid cyclohexa-2 I 4-Dienyl- (2,3,5,6-tetramethyl-phenyl) -acetic acid 8- (4-methoxy-phenyl) -6-methyl-8h- [1,3] dioxolo [4,5-g] chromene -7-carboxylic acid 11- (4-chloro-phenylsulfanyl) -undecanoic acid 1,3-dioxo-2-p-tolyl-2,3-dihydro-1H-isoindole-5-carboxylic acid cis-2- (p-methylbenzoyl) -1-cyclohexanecarboxylic acid mucic acid 4 '- (methylthio) succinilic acid 3-ethoxy-2-butenoic acid acetoxyacetic acid 5-methyl-2-nitrobenzoic acid 4-chloro-2-fluorobenzoic acid 2, 5-dimethoxycinnamic acid (+/-) - beta-phenylglutamic acid 3-methyl-2-oxobutyric acid 1-heptanesulfonic acid 4-methyl-3-nitrobenzoic acid 2-carboxycinnamic acid alpha-methylcinnamic acid 4- (3-hexadecyl-2) -thioureido) -benzoic acid dehydroabietic acid (2-nitro-benzenesulfonylamino) -acetic acid (3-benzyloxy-4-methoxy-phenyl) -acetic acid 5-bromo-2-iodobenzoic acid 1,1,3-trimethyl-3-phenylindan-4 ', 5-dicarboxylic acid oxaleacetic acid 2-aminoterephthalic acid perfluorohexanoic acid 6-Bromo-2-pyridin-3-yl-quinoline-4-carboxylic acid 2,6-dichloro-phenylacetic acid 4- (chloromethyl) -benzoic acid

-63kyselina 2-(4-izopropylbenzoyl)akrylová kyselina 5-jódferulová kyselina 3-(1,2,3,4-tetrahydro-naftalén-1-yl)-propiónová kyselina 2-[3-oxo-3-(n-tridekanoyl-hydrazíno)-propionylamino]-benzoová kyselina 2'-karbamoyl-3,4,5,6-tetrachlórftalanilová kyselina 4-(2,6-dibróm-1 h-indol-3-yl)-maslová kyselina (4-bróm-benzoylamino)-octová kyselina dietylfosfonobutánová kyselina 4-amino-benzyl-sulfónová kyselina n-benzoyl-8-hydroxy-2-naftylamín-6-sulfónová kyselina 2,6-dimetylfenoxyoctová kyselina p-hydroxyhipurová n-(3-(trifluórmetyl )benzoy I )glycí n kyselina (2-fenoxy-acetylamino)-octová kyselina 8-metylnonánová kyselina 3-(3-metoxy-fenyl)-2-metyl-akrylová kyselina 2-(2,4-dibrómfenoxy)-propiónová kyselina 4-nitrosalicylová kyselina 4-(3-(4-acetyl-fenyl)-propyl)-benzoová kyselina (s)-(-)-2-acetoxypropiónová kyselina 5-(fenylazo)salicylová kyselina 5-karboxydehydrooctová kyselina dimetyldianilinotereftalová kyselina fenyl-cyklohexyl-oxyoctová kyselina 3,4-dichlórfenoxyoctová kyselina n-(2,6-diizopropylfenyl-karbamoylmetyl)iminodioctová kyselina 3-(4-n-propylbenzoyl)propiónová kyselina ŕrans-3-hexénová kyselina l-beta-amino-adipová kyselina 3-(4-chlórbenzyltio)tiofén-2-karboxylová kyselina 3-(1,1,2,2-tetrafluóretoxy)benzoová kyselina 5-acetyl-4-hydroxy-3-metoxy-furán-2-karboxylová-63- 2- (4-Isopropylbenzoyl) acrylic acid 5-Iodferulic acid 3- (1,2,3,4-tetrahydro-naphthalen-1-yl) -propionic acid 2- [3-oxo-3- (n-tridecanoyl) -hydrazino) -propionylamino] -benzoic acid 2'-carbamoyl-3,4,5,6-tetrachlorophthalanilic acid 4- (2,6-dibromo-1H-indol-3-yl) butyric acid (4-bromo- benzoylamino) -acetic acid diethylphosphonobutanoic acid 4-amino-benzylsulfonic acid n-benzoyl-8-hydroxy-2-naphthylamine-6-sulfonic acid 2,6-dimethylphenoxyacetic acid p-hydroxyhipuric acid n- (3- (trifluoromethyl) benzoyl) ) glycine (2-phenoxy-acetylamino) -acetic acid 8-methylnonanoic acid 3- (3-methoxy-phenyl) -2-methyl-acrylic acid 2- (2,4-dibromophenoxy) -propionic acid 4-nitrosalicylic acid 4- (3- (4-acetyl-phenyl) -propyl) -benzoic acid (s) - (-) - 2-acetoxypropionic acid 5- (phenylazo) salicylic acid 5-carboxydehydroacetic acid dimethyldianilinoterephthalic acid phenyl-cyclohexyl-oxyacetic acid 3 4 -dichlorophenoxyacetic acid n- (2,6-diisopropylphenylcarbamoylmethyl) iminodiacetic acid 3- (4-n-propylbenzoyl) propionic acid trans-3-hexenoic acid 1-beta-amino-adipic acid 3- (4-chlorobenzylthio) thiophene- 2-Carboxylic acid 3- (1,1,2,2-tetrafluoroethoxy) benzoic acid 5-acetyl-4-hydroxy-3-methoxy-furan-2-carboxylic acid

999999999999

9 9 999

9 · ·· • Í 9 999 · ·· • 9 99

9999

9999 ·· ····9999 ·· ····

-64kyselina 2,4-dihydroxy-5-(izobutyltio)-benzénsulfónová kyselina 3-acetoxyškoricová kyselina 1 -amino-2-(3-indolyl)etán-fosfónová kyselina 2-fluór-4-propoxybenzoová kyselina 3-(4-chlórbenzoyl)-2-(4-izopropylfenyl)propiónová kyselina 2-acetyl-3,6-dinr>etylbenzoová kyselina 2',5'-dichlórsukcínanilová kyselina 2-hydroxy-3(s)-(n-ŕerc-boc-amino)-heptánová kyselina (-)n-(fenylsulfonyl)glutámová kyselina (z-styryltio)octová kyselina gama-d-glutamylaminometylsulfónová kyselina dodecyloxy-octová kyselina 4’-(metyltio)-3I4,5,6-tetrachlórftalanilová kyselina alfa-metyl-2-(metyltio)-5-nitroškoricová kyselina 1 -(p-toly I)-1 -cyklopropánkarboxylová kyselina 3-(hexadecylsulfónamido)-propiónová kyselina (2s)-alfa-etykglutámová etylénglykol-bis(4-karboxyfenyl)éter kyselina (+)-n-benzoylglutámová kyselina alfa-ketovalérová kyselina 2,3-diacetoxy-n-(1 -naftalén-1 -yl-etyl)-sukcínamová kyselina 5-metyl-1h-(1,2,3)triazol-4-karboxylová kyselina dipivaloyl-d-vínna kyselina 3-(4-benzyloxy-3-metoxy-fenyl)-propínová kyselina 1 -(4-brómbenzoyl)piperazín-2,3-dikarboxylová kyselina d/-cyklopentylmandlová-64 2,4-dihydroxy-5- (isobutylthio) -benzenesulfonic acid 3-acetoxycinnamic acid 1-amino-2- (3-indolyl) ethanephosphonic acid 2-fluoro-4-propoxybenzoic acid 3- (4-chlorobenzoyl) 2- (4-isopropylphenyl) propionic acid 2-acetyl-3,6-dinobutylbenzoic acid 2 ', 5'-dichlorosuccinilic acid 2-hydroxy-3 (s) - (n-tert-boc-amino) -heptanoic acid acid (-) -N- (phenylsulfonyl) glutamic acid (from-styryltio) -acetic acid gamma-d-dodecyloxy-glutamylaminometylsulfónová acetic acid 4 '- (methylthio) -3-4,5,6 tetrachlórftalanilová I, alpha-methyl-2 - (methylthio) -5-nitrocinnamic acid 1- (p-tolyl) -1-cyclopropanecarboxylic acid 3- (hexadecylsulfonamido) -propionic acid (2s) -alpha-ethylglutamic ethylene glycol bis (4-carboxyphenyl) ether acid (+) -n-benzoylglutamic acid alpha-ketovaleric acid 2,3-diacetoxy-1- (1-naphthalen-1-yl-ethyl) -succinamic acid 5-methyl-1H- (1,2,3) triazole-4-carboxylic acid dipivaloyl- d-Tartaric acid 3- (4-benzyloxy-3-methoxyphenyl) -propionic acid 1- (4-bromobenzoyl) piperazine-2,3-dicarboxylic acid d -cyclopentylmandelic acid

1-(4’-sulfofenyl)-3-metyl-5-pyrazolón kyselina 2,,5'-dichlórglutaranilová kyselina perfluórpentánová kyselina 4-hydroxymetyl-3-pyridínkarboxylová kyselina n-boc-aminoheptánová kyselina 2,3,5-trichlórbenzoová1- (4'-sulfophenyl) -3-methyl-5-pyrazolone 2 , 5'-dichloroglutaranilic acid perfluoropentanoic acid 4-hydroxymethyl-3-pyridinecarboxylic acid n-boc-aminoheptanoic acid 2,3,5-trichlorobenzoic acid

ΦΦ ···· • φφφ φφφ φ · • φ φ φ φ φ φφφφΦΦ · · · φ · · • • • • φ φ

Φ·« φφφφ φ» φφφ ΦΦ ΦΦ 99 99 9 Φ · «φφφφ φ» φφφ ΦΦ 99 99 99 9

-65kyselina 2,2-dimetyljantárová kyselina benzoová kyselina d-izoaskorbová kyselina d/-fenylmerkapturová beta-benzyl-ester kyseliny n-fmoc-1-asparágovej kyselina 2-chlór-4,5-difluórbenzoová kyselina glyoxylová kyselina 9-metyl-9h-fluorén-2-karboxylová kyselina (2,3I4,5I6-pentahydroxy-hexanoylamino)-octová kyselina 4-(hexadecyltio)benzoová kyselina 3-(5-hydroxy-4-metoxy-2-nitro-fenyl)-akrylová kyselina trifluórtioloctová kyselina n-formyl-d/-2-amino-n-maslová kyselina 4-ketopimelová kyselina 3,4,5-trimetoxyškoricová kyselina 2,5-dibróm-3,6-dichlór-tereftalová kyselina 1-fluorénkarboxylová kyselina 2-(2-chlór-1,1,2-trifluóretyltio)-benzoová kyselina 11-(5-azido-1-naftoxy)undekánová kyselina 2-(2,5-dimetoxy-benzyl)-benzoová kyselina 3,8-dioxa-tricyklo(5.1.0.0(2,4))oktán-5,6-dikarboxylová kyselina 2-cyklopentylhexánová kyselina 2-(4-(2,2-dikarboxy-etyl)2,5-dimetoxy-benzyl)malónová kyselina 2-metyl-non-2-énová kyselina (4,4-dimetyl-3-oxo-cyklohexyl)-octová kyselina 2-karboxymetyl-5-metoxy-benzoová kyselina ŕrans-4-hydroxy-4-(4-nitrofenyl)-2-buténová kyselina 3-(2,6-dietyl-fenylkarbamoyl)-akrylová kyselina 2-[2-(3-metoxy-fenyl)-acetylamino]-3-metyl-maslová kyselina 11,12-epoxy-(5z,8z, 14z)-eikozatriénová kyselina 2-brómmaslová kyselina ftalyl-d/-glutámová ·« ····-65-2,2-dimethylsuccinic acid benzoic acid d-isoascorbic acid d-phenylmercapturic beta-benzyl ester n-fmoc-1-aspartic acid 2-chloro-4,5-difluorobenzoic acid glyoxylic acid 9-methyl-9h- Fluorene-2-carboxylic acid (2,3 L 4,5 L 6-pentahydroxy-hexanoylamino) -acetic acid 4- (hexadecylthio) benzoic acid 3- (5-hydroxy-4-methoxy-2-nitro-phenyl) -acrylic acid trifluorothiol acetic acid n-formyl-η-2-amino-n-butyric acid 4-ketopimelic acid 3,4,5-trimethoxycinnamic acid 2,5-dibromo-3,6-dichloro-terephthalic acid 1-fluorenecarboxylic acid 2- (2-Chloro-1,1,2-trifluoroethylthio) -benzoic acid 11- (5-azido-1-naphthoxy) undecanoic acid 2- (2,5-dimethoxy-benzyl) -benzoic acid 3,8-dioxa-tricyclo (5.1.0.0 (2,4)) octane-5,6-dicarboxylic acid 2-cyclopentylhexanoic acid 2- (4- (2,2-dicarboxyethyl) 2,5-dimethoxybenzyl) malonic acid 2-methyl- Non-2-enoic acid (4,4-dimethyl-3-oxo-cyclohexy l) -Acetic acid 2-carboxymethyl-5-methoxybenzoic acid trans-4-hydroxy-4- (4-nitrophenyl) -2-butenoic acid 3- (2,6-diethylphenylcarbamoyl) -acrylic acid 2- [ 2- (3-Methoxy-phenyl) -acetylamino] -3-methyl-butyric acid 11,12-epoxy- (5z, 8z, 14z) -eicosatrienoic acid 2-bromobutyric acid phthalyl-d-glutamic acid · «··· ·

-66e··· kyselina 4-nitro-2-(3-nitrofenoxy)benzoová kyselina 4-metoxycyklohexánkarboxylová kyselina 3-metyl-3-(3,4,5-trimetyl-fenyl)-maslová kyselina 2-(difluórmetoxy)benzoová kyselina n-(3,4-dichlórfenyl)malonámová kyselina tiodijantárová kyselina 4-chlórfenyloctová kyselina 5-chlórbenzo[b]tiofén-3-octová kyselina 4-benzyloxy-3-metoxyškoricová kyselina 2-propylnonánová kyselina indazol-3-karboxylová kyselina antrachinón-2-karboxylová kyselina boc-6-aminokaprónová kyselina fmoc-nipekotínová kyselina 4-((2-hydroxy-5-metoxy-benzylidén)-amino)-benzoová kyselina hydroferulová kyselina pth-d/-cysteínová kyselina (+/-)-c/s-1 -amino-1 -karboxycyklopentán-3-octová kyselina 1 -naftol-3,6,8-trisulfónová kyselina 3-(4-chlórbenzoyl)-2-(4-fluórfenyl)propiónová n-karbamyl-d/-alan í n kyselina c/s-hexahydro-n-(2-fenetyl)ftalámová imobilizovaná kyselina iminodioctová kyselina ŕra/?s-2-(4-fluórbenzoyl)-1 -cyklohexán-karboxylová kyselina 2-pyridylakrylová kyselina 4-ferc-butyl-3-nitrobenzoová kyselina 3-(4-metyl-3-nitrofenylureido)benzoová kyselina 2-benzhydrylidén-jantárová kyselina 3-pentánová kyselina 2-(1-indenylidén)glykolová kyselina 1 h, 1 h,2h,2h-perfluórdekánová kyselina 4-(3-chlór-1,4-dioxo-1 -4-dihydro-naftalén-2-ylamino)-maslová φ-66e ··· 4-nitro-2- (3-nitrophenoxy) benzoic acid 4-methoxycyclohexanecarboxylic acid 3-methyl-3- (3,4,5-trimethylphenyl) butyric acid 2- (difluoromethoxy) benzoic acid n- (3,4-dichlorophenyl) malonamic acid thiodisuccinic acid 4-chlorophenylacetic acid 5-chlorobenzo [b] thiophene-3-acetic acid 4-benzyloxy-3-methoxycinnamic acid 2-propylnonanoic acid indazole-3-carboxylic acid anthraquinone-2 boc-6-aminocaproic acid fmoc-nipecotinic acid 4 - ((2-hydroxy-5-methoxy-benzylidene) -amino) -benzoic acid hydroferulic acid pth-d / -cysteic acid (+/-) - cis s-1-amino-1-carboxycyclopentane-3-acetic acid 1-naphthol-3,6,8-trisulfonic acid 3- (4-chlorobenzoyl) -2- (4-fluorophenyl) propionic n-carbamyl-d-alanine t-hexahydro-n- (2-phenethyl) phthalic acid immobilized iminodiacetic acid trans-2- (4-fluorobenzoyl) -1-cyclohexanecarboxylic acid 2-pyridylacryloic acid 4-tert-butyl-3-nitrobenzoic acid 3- (4-methyl-3-nitrophenylureido) benzoic acid 2-benzhydrylidene-succinic acid 3-pentanoic acid 2- (1-indenylidene) glycolic acid 1 h, 1 h, 2h, 2h-Perfluorodecanoic acid 4- (3-chloro-1,4-dioxo-1-4-dihydro-naphthalen-2-ylamino) butyric acid φ

-67φφ φφφφ-67φφ φφφφ

Φ· φ φ · φφφ • t · · • φφφ φφ φφ φΦ φ · φ φ t t t t t

kyselina 3-(3-bróm-4-hydroxy-fenyl)-propiónová kyselina 2-chlór-6-metylfenoxyoctová kyselina alfa-beta-dibróm-4-nitrohydroškoricová kyselina alfa-(fenyltio)-o-toluylová kyselina heptakozánová kyselina 3,5-dibróm-2,4-dihydroxybenzoová kyselina 5-(9,10-dioxo-9,10-dihydro-antracén-2-yl)-penta-2,4-diénová kyselina 9-fluorenón-4-karboxylová kyselina alfa,alfa,alfa',alfa'-tetrametylheptándiová kyselina (+/-)-trans-2,3-piperidíndikarboxylová kyselina 4,5-dichlór-izotiazol-3-karboxylová kyselina 2-jódfenyloctová kyselina 4-jódfenoxyoctová kyselina 1 -amino-8-naftol-3,6-disulfónová kyselina 4-((4-chlór-benzylidén)-amino)-benzoová kyselina 2-kyano-3-metyl-but-2-énová kyselina 3-((adamantán-1 -karbonyl)-amino)-benzoová kyselina 5-(trifluórmetoxy)indol-2-karboxylová kyselina mezo-2,3-difenyljantárová kyselina cyklopentánkarboxylová kyselina 2-formylamino-2-fenyl-propiónová kyselina galová kyselina n-(2-butylsulfanyl-benzotiazol-6-yl)-sukcínamová kyselina 3-nitro-alfa-fenylškoricová kyselina 4-metoxyfenoxyoctová kyselina hex-4-ínová kyselina 5-(4-metoxybenzoyl)tiofén-2-octová kyselina 2-metyl-5-fenylfurán-3-karboxylová kyselina 3-((5-nitro-1,3-dioxo-1,3-dihydro-izoindol-2-ylmetyl)-amino)-benzoová kyselina n-etyl-d-asparágová kyselina d/-beta-hydroxycaprónová kyselina 3,5-dimetyl-2-jódbenzoová • · • · • · • ·3- (3-bromo-4-hydroxy-phenyl) -propionic acid 2-chloro-6-methylphenoxyacetic acid alpha-beta-dibromo-4-nitrohydrocinnamic acid alpha- (phenylthio) -o-toluic acid heptacosanoic acid 3,5 -dibromo-2,4-dihydroxybenzoic acid 5- (9,10-dioxo-9,10-dihydro-anthracen-2-yl) -penta-2,4-dienoic acid 9-fluorenone-4-carboxylic acid alpha, alpha [alpha], alpha ', alpha'-tetramethylheptanedioic acid (+/-) - trans-2,3-piperidinedicarboxylic acid 4,5-dichloro-isothiazole-3-carboxylic acid 2-iodophenylacetic acid 4-iodophenoxyacetic acid 1-amino-8-naphtholic acid -3,6-disulfonic acid 4 - ((4-chloro-benzylidene) -amino) -benzoic acid 2-cyano-3-methyl-but-2-enoic acid 3 - ((adamantane-1-carbonyl) -amino) -benzoic acid 5- (trifluoromethoxy) indole-2-carboxylic acid meso-2,3-diphenylsuccinic acid cyclopentanecarboxylic acid 2-formylamino-2-phenyl-propionic acid gallic acid n- (2-butylsulfanyl-benzothiazol-6-yl) - succinic acid 3-Nitro-alpha-phenyl cinnamic acid 4-methoxyphenoxyacetic acid hex-4-ynoic acid 5- (4-methoxybenzoyl) thiophene-2-acetic acid 2-methyl-5-phenylfuran-3-carboxylic acid 3 - ((5- nitro-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl) -amino) -benzoic acid n-ethyl-d-aspartic acid d-beta-hydroxycaproic acid 3,5-dimethyl-2-iodobenzoic acid • • • •

-68• » ·· · • ♦ · • · • e· ·· ···· • ·· • · · • Λ9 · ·· ·· ·· ··-68 »e e e e e9 e9 Λ9 Λ9 · Λ9

99

999 kyselina 2-etyl-2-metylhexánová kyselina diglykolová kyselina glutakónová kyselina 3-chlór-4-fluórbenzoová kyselina tricyklo(8.2.2.2(4,7))hexadeka-1 (13),4,6,10(14),11,15-hexaén-5-karboxylová kyselina 5-jódvanilová kyselina 3-metylškoricová kyselina 2-brómoktánová kyselina 2-bróm-6-metoxybenzoová kyselina boc-8-aminokaprylová kyselina 1,8-naftyridín-2-karboxylová kyselina 3-(4-sulfamoyl-fenyl)-akrylová kyselina 2-(3-(2,4-xylyl)ureido)benzoová kyselina 3-(3-tienyl)akrylová kyselina 2,2-dimetyl-3-hydroxypropiónová kyselina /?,n-bis((r)-(+)-1 -fenyletyl)ftalámová kyselina 1,3-fenyléndiakrylová kyselina 2-(2-(2-hydroxy-1 -naftoyl)vinyl)benzoová kyselina (+/-)-erytro-4-metylglutámová kyselina 7-(3-chlór-2-tienyl)-2,4-dimetylpyrol[1,2-a]pyrimidín-8-karboxylová kyselina 4-chlór-3-jódbenzoová kyselina 2-[2-chlór[(4-fluórfenyl)sulfonyl]anilino]octová kyselina glycyl-1-asparágová kyselina 5-[(4-chlórfenyl)sulfanyl]-1,2,3-tiadiazol-4-karboxylová kyselina 2-nitrobenzénsulfónová kyselina 3-(1,1,4,6,7-pentametyl-indán-5-yl)-akrylová kyselina 2,5-dimetylfenoxyoctová kyselina hypofosforná kyselina pyromelitová kyselina 2-metyl-2-fenyl-maslová kyselina 3-hydroxy-2,4,6-tribrómbenzoová999 2-ethyl-2-methylhexanoic acid diglycolic acid glutaconic acid 3-chloro-4-fluorobenzoic acid tricyclo (8.2.2.2 (4,7)) hexadeca-1 (13), 4,6,10 (14), 11 15-hexaene-5-carboxylic acid 5-iodoanilic acid 3-methylcinnamic acid 2-bromooctanoic acid 2-bromo-6-methoxybenzoic acid boc-8-aminocaprylic acid 1,8-naphthyridine-2-carboxylic acid 3- (4- sulfamoyl-phenyl) -acrylic acid 2- (3- (2,4-xylyl) ureido) benzoic acid 3- (3-thienyl) acrylic acid 2,2-dimethyl-3-hydroxypropionic acid p-n-bis (( r) - (+) - 1-phenylethyl) phthalic acid 1,3-phenylenediacrylic acid 2- (2- (2-hydroxy-1-naphthoyl) vinyl) benzoic acid (+/-) - erythro-4-methylglutamic acid 7 - (3-chloro-2-thienyl) -2,4-dimethylpyrrolo [1,2-a] pyrimidine-8-carboxylic acid 4-chloro-3-iodobenzoic acid 2- [2-chloro [(4-fluorophenyl) sulfonyl] anilino] acetic acid glycyl-1-aspartic acid 5 - [(4-chlorophenyl) sulfanyl] -1,2,3-thiadiazole-4-carboxylic acid 2-nitrobenzenesulfonic acid 3- (1,1,4,6,7-pentamethyl-indan-5-yl) -acrylic acid 2,5-dimethylphenoxyacetic acid hypophosphoric pyromellitic acid 2-methyl-2-phenylbutyric acid 3 hydroxy-2,4,6-tribromobenzoic

• · • ···· ·· • · ·· • · · · • · 9 ·· • · · ·· • ·· ·· kyselina 1 -(2-fluórfenyl)cyklohexánkarboxylová kyselina 3,4-dimetylhipurová kyselina 6,8-dichlór-2-hydroxy-4-chinolínkarboxylová kyselina n,n’-(1,3-fenylén)dimaleámová kyselina 1-butánsulfónová kyselina 2,3-difluórškoricová kyselina trifenylsilylkarboxylová kyselina etylfosfónová kyselina chlórgenínová kyselina (1 r,2s,3r)-1-hydroxy-3-hydroxymetyl-1,2,3,4-tetrahydronaftalén-2-karboxylová kyselina adamantán-2-yl-octová kyselina alfa-metyl-2-furánakrylová kyselina 4-oxatetradekánová kyselina 2,,5’-dimetyl-3l4,5,6-tetrachlórftalámová kyselina 4,4-difenyl-but-3-énová kyselina 4-anizidín-2,5-disulfónová kyselina 2-((3-alyl-2-hydroxy-benzylidén)-amino)-3-(1h-imidazol-4-yl)-propiónová kyselina benzylfosfónová kyselina metánsulfonyloctová kyselina 4,4-bis-(4-hydroxy-3-nitrofenyl)-valérová kyselina akrylová kyselina 1 -(4-chlórfenyl)etyliminoxyoctová kyselina 2-(2-chlór-1,1,2-trifluóretoxy)-benzoová kyselina c/s-2-(p-chlórbenzoyl)-1 -cyklohexán-karboxylová kyselina 3-acetamidobenzoová kyselina 2,4-bis(trifluórmetyl)benzoová kyselina 4-fluórškoricová n-acetyl-d,l-homotryptofán kyselina benzofurazán-5-karboxylová kyselina c/s-n-(5-chlór-2-metoxyfenyl)hexahydroftalámová kyselina 3-(3,4-dichlór-fenyl)-2-metyl-akrylová ·· ···· ··· • · · · · • · · · · ··· · ·· · · · · ·· φ· 99 99 ··1- (2-Fluorophenyl) cyclohexanecarboxylic acid 3,4-dimethylhipuric acid 6, 6, 9, 9, 9, 9, 9, 10, 11, 12, 13, 14 8-Dichloro-2-hydroxy-4-quinolinecarboxylic acid n, n '- (1,3-phenylene) dimaleamic acid 1-butanesulfonic acid 2,3-difluoro cinnamic acid triphenylsilylcarboxylic acid ethylphosphonic acid chlorgenenic acid (1 r, 2s, 3r) 1-hydroxy-3-hydroxymethyl-1,2,3,4-tetrahydronaphthalene-2-carboxylic acid adamantan-2-yl-acetic acid alpha-methyl-2-furánakrylová acid 4-oxatetradekánová acid 2 ', 5'-dimethyl -3 '4,5,6-tetrachlórftalámová 4,4-diphenyl-but-3-enoic acid 4-anisidine-2,5-disulfonic acid, 2 - ((3-allyl-2-hydroxy-benzylidene) -amino) -3- (1h-imidazol-4-yl) -propionic acid benzylphosphonic acid methanesulfonylacetic acid 4,4-bis- (4-hydroxy-3-nitrophenyl) -valeric acid 1- (4-chlorophenyl) ethyliminoxyacetate 2- (2-chloro-1,1,2-trifluoroethoxy) -benzoic acid cis-2- (p-chlorobenzoyl) -1-cyclohexanecarboxylic acid 3-acetamidobenzoic acid 2,4-bis (trifluoromethyl) benzoic acid 4-fluorocinnamic acid n-acetyl-1,1-homotryptophan benzofurazan-5-carboxylic acid cis- (5-chloro-2-methoxyphenyl) hexahydrophthalic acid 3- (3,4-dichlorophenyl) -2-methyl -acrylic ·················· 99 99 99

-70kyselina 4-chlór-2-jódbenzoová kyselina n-fenylantranilová kyselina (+/-)-ŕrans-2,5-piperidindikarboxylová kyselina 4-kyano-3,5-dimetyl-1 h-pyrol-2-karboxylová kyselina 3'-(trifluórmetyl)-1,2,3,6-tetrahydroftalámová kyselina 3-antracén-2-yl-propiónová kyselina n,n -(1,2-fenylén)dimaleámová kyselina (r)-(-)-4-metylglutárová-70 4-chloro-2-iodobenzoic acid n-phenylanthranilic acid (+/-) - trans -2,5-piperidinedicarboxylic acid 4-cyano-3,5-dimethyl-1H-pyrrole-2-carboxylic acid 3'- (trifluoromethyl) -1,2,3,6-tetrahydrophthalic acid 3-anthracen-2-yl-propionic acid n, n - (1,2-phenylene) dimaleamic acid (r) - (-) - 4-methylglutaric acid

-monometylester kyseliny 3-oxo-2-fenyl-1 -cyklopentánkarboxylovej kyselina 1-homocysteínsulfámová kyselina 2-(orto-tolyl)-heptánová kyselina 1 -(-)-treo-3-hydroxyasparágová kyselina 4-chlór-3-sulfamoyl-benzoová kyselina 3-(4-chlór-fenyl)-3-izobutyrylamino-propiónová kyselina dekánová kyselina 2-chlóretylfosfónová kyselina beta-d-aspartylaminometyl-fosfónová kyselina 3-n-propylglutárová kyselina alfa-acetamidoškoricová kyselina epsilon-/?-oxalyl-d-alfa,epsilon-diaminohexánová kyselina d-gáfrová kyselina 3-(1h-indol-3-yl)-2-(toluén-4-sulfonylamino)-propiónová kyselina alfa-metoxyškoricová kyselina „costic“ kyselina 4-oxo-4-(2-oxocyklohexyl)maslová kyselina n-(2-metoxyfenyl)maleámová kyselina 4-etoxykarboxy-3,5-dimetoxybenzoová kyselina 2-fluóren-9-ylidénmetyl-benzoová kyselina 4-dipropylamino-3,5-dinitro-benzoová kyselina 7,10,13,16,19-dokozapenténová kyselina 4-(3-chlór-5-trifluórmetyl-2-pyridyl)-4-fenylsulfonylbutánová kyselina 12-(n-metyl-n-[7-nitrobenz-2-oxa-1,3-diazol-4-yl])-aminododekánová3-oxo-2-phenyl-1-cyclopentanecarboxylic acid monomethyl ester 1-homocysteine sulfamic acid 2- (ortho-tolyl) -heptanoic acid 1- (-) - threo-3-hydroxyaspartic acid 4-chloro-3-sulfamoyl-benzoic acid 3- (4-chloro-phenyl) -3-isobutyrylamino-propionic acid decanoic acid 2-chloroethylphosphonic acid beta-d-aspartylaminomethylphosphonic acid 3-n-propylglutaric acid alpha-acetamido cinnamic acid epsilon - β-oxalyl-d- alpha, epsilon-diaminohexanoic acid d-camphoric acid 3- (1H-indol-3-yl) -2- (toluene-4-sulfonylamino) -propionic acid alpha-methoxycinnamic acid costic acid 4-oxo-4- (2 -oxocyclohexyl) butyric acid 4- (2-methoxyphenyl) maleic acid 4-ethoxycarboxy-3,5-dimethoxybenzoic acid 2-fluoren-9-ylidenemethylbenzoic acid 4-dipropylamino-3,5-dinitro-benzoic acid 7,10, 4- (3-chloro-5-trifluoromethyl-2-pyridyl) -4-phenylsulphonylbutanoic acid 13,16,19-docosapentenoic acid 12- (nm ethyl N- [7-nitrobenz-2-oxa-1,3-diazole-4-yl]) - aminododecanoic

-71 ·· ···· ·· kyselina 3,4,5-trietoxybenzoová kyselina 2-metoxypropiónová kyselina (r)-(+)-2-metylglutárová kyselina boc-10-aminodekánová kyselina c/s-akonitová kyselina n(alfa)-fmoc-n(beta)-alloc-1,2,3-diaminopropiónová kyselina 3-(4-butoxy-benzoylamino)-benzoová kyselina 4,6-dihydroxy-5-metánsulfonyl-1-ph-3a,6-metano-azulén-3-karboxylová kyselina 2-bróm-angeliková kyselina dodekándiová kyselina 2,3,4-trifluórfenyloctová kyselina (3-metoxystyryl)glyoxylová kyselina 4-[[(3-hydroxy-2-naftalenyl)karbonyl]amino]benzoová kyselina 2-benzyl-3-fenyl-propiónová kyselina 2-hydroxydodekánová kyselina 2,3-dibróm-2-metyl-propiónová kyselina 8-hydroxy-1 -naftylamín-4,6-disulfónová kyselina 3,4-dihydroxyfenyloctová kyselina 2,5-dimetyl-4-(etoxykarbonyl)-3-furoová kyselina 4-((5-bróm-1,3-dioxo-1,3-dihydro-izoindol-2-ylmetyl)-amino-benzoová n-karbobenzyloxy-2-metylalanín kyselina (3,4-dichlór-benzoylamino)-octová kyselina 5-ŕerc-butyl-2-furoová kyselina 2-hydroxy-3(s)-(n-ŕerc-boc-amino)hexánová kyselina cyklohexánpentánová kyselina 2’-nitroftalanilová kyselina 5-metoxy-3-metyl-ftalová kyselina ricínelaidová kyselina 2-oxo-6-pentyl-2h-pyrán-3-karboxylová kyselina 2-karboxyamino-3-(2-hydroxy-fenyl)akrylová kyselina 2-acetamido-5-nitrobenzoová kyselina 3-(n-fenylkarbamoyl)-5-norbornén-2-karboxylová-71 ·· ······ 3,4,5-Triethoxybenzoic acid 2-methoxypropionic acid (r) - (+) - 2-methylglutaric acid boc-10-aminodecanoic acid cis-aconitic acid n (alpha) ) -fmoc-n (beta) -alloc-1,2,3-diaminopropionic acid 3- (4-butoxy-benzoylamino) -benzoic acid 4,6-dihydroxy-5-methanesulfonyl-1-ph-3a, 6-metano -azulene-3-carboxylic acid 2-bromo-angelic acid dodecanedioic acid 2,3,4-trifluorophenylacetic acid (3-methoxystyryl) glyoxylic acid 4 - [[(3-hydroxy-2-naphthalenyl) carbonyl] amino] benzoic acid 2 -benzyl-3-phenyl-propionic acid 2-hydroxydodecanoic acid 2,3-dibromo-2-methyl-propionic acid 8-hydroxy-1-naphthylamine-4,6-disulfonic acid 3,4-dihydroxyphenylacetic acid 2,5-dimethyl 4- (ethoxycarbonyl) -3-furoic acid 4 - ((5-bromo-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl) -amino-benzoic acid n-carbobenzyloxy-2-methylalanine acid ( 3,4-Dichloro-benzoylamino) -acetic acid 5-tert-butyl-2-furoic acid and 2-hydroxy-3 (s) - (n-tert-boc-amino) hexanoic acid cyclohexanepentanoic acid 2'-nitropthalanilic acid 5-methoxy-3-methyl-phthalic acid ricinilaic acid 2-oxo-6-pentyl-2h- pyran-3-carboxylic acid 2-carboxyamino-3- (2-hydroxyphenyl) acrylic acid 2-acetamido-5-nitrobenzoic acid 3- (n-phenylcarbamoyl) -5-norbornene-2-carboxylic acid

·· ·· ··· · • · · · • · · kyselina d/-mandlová kyselina 3-fluóranten-1 -yl-akrylová kyselina 2-(4-brómfenyl)-3-(4-chlórbenzyl)propiónová kyselina 3-metyl-2-furoová kyselina (2-metylfenoxy)octová kyselina (4-metánsulfonyloxy-3-metoxy-fenyl)-octová kyselina 2-hydroxy-3-izopropyl-6-metylbenzoová kyselina 4-(5,6,7,8-tetrahydro-naftalén-2-yl)-maslová kyselina 3-benzoylakrylová kyselina 4-etoxybenzoová kyselina (4-hydroxy-3-metoxy-fenyl)-oxo-octová kyselina 2-((5-bróm-1,3-dioxo-1,3-dihydro-izoindol-2-ylmetyl)-amino)-benzoová kyselina 3-[[(1-acetyl-2,3-dihydro-(1h)-indol-7-yl)amino]karbonyl]propánová kyselina 5-metyl-4-oxohexánová kyselina (8-ho-3-meo-1,5,9,9-tetra-me-4,12-dioxo-benzocyklodecén-2-ylidén)octová kyselina 1 -(4-fluóranilíno)-6-metyl-4-oxo-1,4-dihydro-3-pyridínkarboxylová kyselina n-alfa-(9-fluórenylmetyloxykarbonyl)-[3s]-1,2,3,4-tetrahydroizochinolin-7hydroxy-3-karboxylová kyselina 2-[(adamantán-1-karbonyl)-amino]-3-(1h-indol-3-yl)-propiónová kyselina n-cbz-d/-asparágová kyselina karboxymetylmerkaptojantárová kyselina 3-bróm-4,5-dimetoxybenzoová kyselina 3,4-dichlóradipová kyselina 3’-brómftalanilová kyselina 6-metylpyrid-3-yloctová kyselina 3,5,6-trichlóroktafluórhexánová kyselina 3-(5-(4-chlór-fenyl)-furán-2-yl)-akrylová kyselina epsilon-maleimidokaprónová kyselina 6-(acetoxymetyl)-3-metyl-3-cyklohexén-1 -karboxylová kyselina fenylsulfonyloctová kyselina 2-metyl-2-fenyl-oktánová kyselina 2,5-dibrómadipová3-Fluoroanten-1-yl-acrylic acid 2- (4-bromophenyl) -3- (4-chlorobenzyl) propionic acid 3-fluoroanten-1-yl-acrylic acid methyl-2-furoic acid (2-methylphenoxy) acetic acid (4-methanesulfonyloxy-3-methoxyphenyl) -acetic acid 2-hydroxy-3-isopropyl-6-methylbenzoic acid 4- (5,6,7,8- tetrahydro-naphthalen-2-yl) butyric acid 3-benzoylacrylic acid 4-ethoxybenzoic acid (4-hydroxy-3-methoxyphenyl) -oxoacetic acid 2 - ((5-bromo-1,3-dioxo-1) 3-Dihydro-isoindol-2-ylmethyl) amino-benzoic acid 3 - [[(1-acetyl-2,3-dihydro- (1H) -indol-7-yl) amino] carbonyl] propanoic acid 5- methyl 4-oxohexanoic acid (8-ho-3-meo-1,5,9,9-tetra-me-4,12-dioxo-benzocyclodecen-2-ylidene) acetic acid 1- (4-fluoroanilino) -6 -methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid n-alpha- (9-fluorenylmethyloxycarbonyl) - [3s] -1,2,3,4-tetrahydroisoquinoline-7-hydroxy-3-carboxylic acid 2- [ (adamantan-1-carbonyl) -amino] -3- (1H-indol-3-yl l) -propionic acid n-cbz-d-aspartic acid carboxymethylmercaptosuccinic acid 3-bromo-4,5-dimethoxybenzoic acid 3,4-dichloro-adipic acid 3'-bromophthalanic acid 6-methylpyrid-3-ylacetic acid 3,5,6 trichloroctafluorohexanoic acid 3- (5- (4-chloro-phenyl) -furan-2-yl) -acrylic acid epsilon-maleimido-caproic acid 6- (acetoxymethyl) -3-methyl-3-cyclohexene-1-carboxylic acid phenylsulfonylacetic acid 2 -methyl-2-phenyl-octanoic acid 2,5-dibromadipic acid

-73··· kyselina 1,1-cyklohexándikarboxylová kyselina 2-metyl-bicyklo(2.2.1 )hept-5-én-2-karboxylová kyselina 2'-metyl-5’-nitromaleanilová kyselina 2-[benzyl-(toluén-4-sulfonyl)-amino]-benzoová kyselina (karboxy-fenyl-metylsulfanyl)-fenyl-octová kyselina indolizín-2-karboxylová kyselina alfa-metylhydroškoricová kyselina 10-metylundekánová kyselina alfa-kyano-beta-metyl-2-(metyltio)škoricová kyselina 3-hydroxypropánsulfónová kyselina 2-[[2-(2,4-dichlórfenyl)hydrazíno]karbonyl]benzoová kyselina 5-jód-orotová kyselina p-brómfenoxy-octová kyselina 2-hexínová kyselina 2,-chlór-5'-(trifluórmetyl)glutaranilová kyselina 5-metyl-2-fenylimidazo[1,2-a]pyridín-3-karboxylová kyselina 4-(3-chlórpropoxy)-benzoová kyselina 4-(4,4-dimetyl-2-oxocyklohexyl)maslová kyselina 2-metyl-5-nitro-3-furoová kyselina n-metyl-d-asparágová kyselina 4-hydroxyfenoxyoctová kyselina chlóroctová kyselina 4’-nitroglutaranilová kyselina (2s)-alfa-metylglutámová kyselina 9(s)-hydroxyoktadeka-10e,12z-diénová kyselina 2-sulfino-benzoová kyselina 3-(difluórmetoxy)fenyloctová kyselina 10-oxopalmitová kyselina 3-benzamidobenzoová kyselina hipurová fenyl-s-kyselina kyselina 2,7-d/-ŕerc-butyl-9,9-dimetyl-4,5-xanténdikarboxylová ·· ··· • · · • · • · ·· ···· •· •· •· •· · ·· ·· • ♦ · · ♦ 9· • · ·· • ·· •·· · kyselina 5-chlór-2-nitroškoricová kyselina delta-n-oxalyl-c/-alfa,delta-diaminopentánová kyselina 4’-pentyl-bifenyl-4-karboxylová kyselina n-(1-naftyl)glutarámová kyselina 3'-fluórftalanilová kyselina trikozánová kyselina 4-chlór-2,5-difluórbenzoová kyselina 16-fenyl-hexadekánová kyselina 3-[(r,s)-2-karboxypiperazín-4-yl]propyl-1 -fosfónová kyselina 2-naftalén-2-yl-1,3-dioxo-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina 2-pyrid í n-2-yl-chinol í η-4-karboxy lová kyselina 2-(4-metyl-benzoylamino)-3-(4-nitro-fenyl)-akrylová dihydroxychicago-kyselina kyselina 4-fluór-3-(trifluórrnetyl)fenyloctová kyselina 2-tolidín-3,3-disulfónová kyselina 2-((2-hydroxy-5-metoxy-benzylidén)-amino)-benzoová kyselina S’^’-dichlór-glutaranilová kyselina 4-(3-dodekanoyl-2-tioureido)benzoová kyselina 4-hydroxycyklohexánkarboxylová kyselina 3,5-dihydroxy-4-metoxybenzoová kyselina (s)-(+)-citrajablčná (ο-2-metyl-jablčná) kyselina 2-naftylamín-3,6,8-trisulfónová kyselina 3,5-dijód-4-hydroxyfenylpropiónová kyselina (s)-(-)-2-bróm 3-metylbutánová kyselina (r)-(-)-2-fenylmaslová kyselina fluorén-4-karboxylová kyselina n-2-karboxyfenyl)glycín-2-metoxy-3,6-dichlórbenzocvá kyselina 7-brómkynurénová kyselina 2-naftylamín-3,6,8-trisulfónová kyselina n-terc-butylsukcinamová (4-etyl-3,5-dimetyl-1h-pyrol-2-yl)octová kyselina cyklopropyloctová ·· ·· ····-73 ··· 1,1-cyclohexanedicarboxylic acid 2-methyl-bicyclo (2.2.1) hept-5-ene-2-carboxylic acid 2'-methyl-5'-nitromaleanilic acid 2- [benzyl- (toluene- 4-sulfonyl) amino] -benzoic acid (carboxy-phenyl-methylsulfanyl) -phenyl-acetic acid indolizine-2-carboxylic acid alpha-methylhydrocinnamic acid 10-methylundecanoic acid alpha-cyano-beta-methyl-2- (methylthio) cinnamic acid 3-hydroxypropanesulfonic acid 2 - [[2- (2,4-dichlorophenyl) hydrazino] carbonyl] benzoic acid 5-iodo-oroic acid p-bromophenoxy-acetic acid 2-hexanoic acid 2 , -chloro-5 '- (trifluoromethyl) ) Glutaranilic acid 5-methyl-2-phenylimidazo [1,2-a] pyridine-3-carboxylic acid 4- (3-chloropropoxy) -benzoic acid 4- (4,4-dimethyl-2-oxocyclohexyl) butyric acid 2- methyl-5-nitro-3-furoic acid n-methyl-d-aspartic acid 4-hydroxyphenoxyacetic acid chloroacetic acid 4'-nitroglutaranilic acid (2s) -alpha-methylglutamic acid 9 (s) -hydroxyoctadeca-10e, 12z-dienoic acid 2-sulfino-benzoic acid 3- (difluoromethoxy) phenylacetic acid 10-oxopalmitic acid 3-benzamidobenzoic acid hippuric acid phenyl-s-acid 2,7-d-tert-butyl-9, 9-Dimethyl-4,5-xanthene dicarboxylic acid 9-Dimethyl-4,5-xanthene dicarboxylic acid 9-Dimethyl-4,5-xanthene dicarboxylic acid 5-chloro-2-nitrocinnamic acid delta-n-oxalyl-cis-alpha, delta-diaminopentanoic acid 4'-pentyl-biphenyl-4-carboxylic acid n- (1-naphthyl) glutaramic acid 3'-fluorophthalanic acid tricosanoic acid 4-chloro-2,5-difluorobenzoic acid 16-phenyl-hexadecanoic acid 3 - [(r, s) -2-carboxypiperazin-4-yl] propyl-1-phosphonic acid 2- naphthalen-2-yl-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid 2-pyridin-2-yl-quinoline-4-carboxylic acid 2- (4 -methyl-benzoylamino) -3- (4-nitro-phenyl) -acrylic dihydroxychicago-4-fluoro-acid 2-tolidine-3,3-disulfonic acid 2-((2-hydroxy-5-methoxy-benzylidene) -amino) -benzoic acid 4-chloro-3- (trifluoromethyl) phenylacetic acid (3-dodecanoyl-2-thioureido) benzoic acid 4-hydroxycyclohexanecarboxylic acid 3,5-dihydroxy-4-methoxybenzoic acid (s) - (+) - citric acid (ο-2-methyl-malic acid) 2-naphthylamine-3, 6,8-Trisulfonic acid 3,5-diiodo-4-hydroxyphenylpropionic acid (s) - (-) - 2-bromo 3-methylbutanoic acid (R) - (-) - 2-phenylbutyric acid fluorene-4-carboxylic acid n -2-carboxyphenyl) glycine-2-methoxy-3,6-dichlorobenzoic acid 7-bromokynurenoic acid 2-naphthylamine-3,6,8-trisulfonic acid n-tert-butylsuccinamic acid (4-ethyl-3,5-dimethyl-1h) -pyrrol-2-yl) acetic acid cyclopropylacetic acid ·· ·· ····

-75kyselina 5-chlór-tetrazol-1 -octová kyselina ŕrans-2-hexénová kyselina 4-chlór-2-fluórškoricová kyselina tereftaloylbisoctová kyselina 5-(4-(4-karboxy-butyryl)-fenyl)-pentánová kyselina 3-bróm-4-metoxybenzoová kyselina ŕrans,ŕrans-9-kyano-2-dekalínkarboxylová kyselina n-(5-chlór-2-metylfenyl)ftalámová kyselina 1 -(s)-(+)-endo-bróm-gáfor-10-sulfónová kyselina 2-kyano-3-(4-metoxy-fenyl)-akrylová kyselina fmoc-1 -amino-1 -cyklohexán-karboxylová kyselina 3-(3,4-dimetoxy-pyridín-2-yl)-akrylová kyselina 3-metoxy-4-metylbenzoová kyselina 4-(2-fenyl-eténsulfonylamino)-maslová kyselina 4-hydroxy-6-(trifluórmetoxy)chinolín-3-karboxylová kyselina 3-hydroxymyristová kyselina 3-metyltio-4-oxo-4,5,6,7-tetrahydrobenzo[c]tiofén-1-karboxylová kyselina 2-oxo-4-fenyl-pyrolidín-3-karboxylová kyselina 3-chlórvalérová kyselina d-(-)-s-acetyl-beta-merkapto-izomaslová kyselina c/s-parinarová kyselina 2-(2,4-difenyltiazol-5-yl)octová kyselina 3-acetylamino-3-(4-metoxy-fenyl)-propiónová (2s, 1 ’r,2’s)-2-(karboxycyklopropyl)glycín kyselina 3-[fenyl-(toluén-4-sulfonyl)-amino]-maslová kyselina 4-chlór-alfa,beta-difenylakrylová kyselina 5-chlór-2,4-dinitrobenzoová kyselina kukurbová kyselina 2-decyldodekánová kyselina r-4-metyltiomandlová kyselina 2-(9h-fluorén-2-ylmetyl)-benzoová kyselina tricyklo( 12.2.2.2(6,9))eikoza-1 (17),6(20)7,9(19), 14(18), 15-hexaén-yl-octová-75 5-chloro-tetrazole-1-acetic acid trans-2-hexenoic acid 4-chloro-2-fluorocinnamic acid terephthaloylbisacetic acid 5- (4- (4-carboxy-butyryl) -phenyl) -pentanoic acid 3-bromo- 4-Methoxybenzoic acid trans, trans-9-cyano-2-decalinecarboxylic acid 1- (5-chloro-2-methylphenyl) phthalic acid 1- (s) - (+) - endo-bromo-camphor-10-sulfonic acid 2 cyano-3- (4-methoxy-phenyl) -acrylic acid fmoc-1-amino-1-cyclohexanecarboxylic acid 3- (3,4-dimethoxy-pyridin-2-yl) -acrylic acid 3-methoxy-4 4-hydroxy-6- (trifluoromethoxy) quinoline-3-carboxylic acid 4- (2-phenyl-etenesulfonylamino) -butyric acid 3-hydroxymyristic acid 3-methylthio-4-oxo-4,5,6,7- tetrahydrobenzo [c] thiophene-1-carboxylic acid 2-oxo-4-phenyl-pyrrolidine-3-carboxylic acid 3-chloro-valeric acid d - (-) - s-acetyl-beta-mercapto-isobutyric acid cis-parinaric acid 2- (2,4-Diphenylthiazol-5-yl) acetic acid 3-acetylamino-3- (4 -methoxy-phenyl) -propionic (2s, 1 ', 2's) -2- (carboxycyclopropyl) glycine 3- [phenyl- (toluene-4-sulfonyl) -amino] -butyric acid 4-chloro-alpha, beta- diphenylacrylic acid 5-chloro-2,4-dinitrobenzoic acid kucurbic acid 2-decyldodecanoic acid r-4-methylthiomandelic acid 2- (9h-fluoren-2-ylmethyl) -benzoic acid tricyclo (12.2.2.2 (6,9)) eicosis -1 (17), 6 (20) 7.9 (19), 14 (18), 15-hexaen-yl-acetic

-76·· ··· • · • · • ·· ·· ···· • · · • · · • · · · · • · · · ·· ··-76 ·····························

··· kyselina 4-(2-(metylsulfónamido)-etoxy)-meta-anízová kyselina fmoc-d-pipekolínová kyselina tiglinová kyselina fmoc-alfa,beta-dehydro-2-aminomaslová kyselina n,n-difenyl-oxalámová kyselina dehydrotio-p-toluidín-7-sulfónová kyselina 2-diazo-1 -naftol-4-sulfónová kyselina 2-chlór-6-fluórškoricová kyselina 2-etyldekánová kyselina terebinová kyselina 1 -benzoyl-piperazín-2,3-dikarboxylová kyselina 3,5-bis(trifluórmetyl)hydroškoricová kyselina 2,,4'-dimetoxymaleanilová kyselina 5-amino-m-toluylová kyselina 2-chlór-alfa-metylškoricová kyselina 1,4-cyklohexándikarboxylová kyselina gama-maleimidomaslová kyselina metyléndifosfónová kyselina n-(3-chlórfenyl)maleámová kyselina fmoc-2-aminobenzoová kyselina 2,,4’-dichlórftalanilová kyselina o-sulfobenzoová kyselina etyléndiamintetraoctová kyselina 1,4-benzodioxáne-5-karboxylová kyselina gama-oxo-1-pyrénmaslová kyselina n-fmoc-(2s,3s)-3-amino-2-hydroxy-4-fenylmaslová kyselina 2,4-dimetylbenzoová kyselina 3-oxo-1-fenyl-1-indánoctová kyselina 2-((2-(2,4-difluórfenyl)hydrazíno)karbonyl]benzoová kyselina (r)-(+)-3-metyljantárová··· 4- (2- (methylsulfonamido) -ethoxy) -methanesic acid fmoc-d-pipecolinic acid figoc-alpha, beta-dehydro-2-aminobutyric acid n, n-diphenyl-oxalamic acid dehydrothio- p-toluidine-7-sulfonic acid 2-diazo-1-naphthol-4-sulfonic acid 2-chloro-6-fluorocinnamic acid 2-ethyldecanoic acid terebinic acid 1-benzoyl-piperazine-2,3-dicarboxylic acid 3,5- bis (trifluoromethyl) hydrocinnamic acid 2 ', 4'-dimetoxymaleanilová 5-amino-m-toluic acid 2-chloro-methyl cinnamic acid, alpha-1,4-cyclohexanedicarboxylic acid gamma-methylene diphosphonic acid maleimidomaslová n- (3-chlorophenyl) maleamic acid, Fmoc-2-aminobenzoic acid, 2, 4 & apos dichlórftalanilová acid, o-sulfobenzoic acid ethylenediaminetetraacetic acid, 1,4-benzodioxane-5-carboxylic acid gamma-oxo-1-pyrénmaslová n-Fmoc- (2S, 3S) -3 amino-2-hydroxy-4-phenylbutyric acid 2,4-dimethylb enzoic acid 3-oxo-1-phenyl-1-indaneacetic acid 2 - ((2- (2,4-difluorophenyl) hydrazino) carbonyl] benzoic acid (r) - (+) - 3-methylsuccinic acid

1-monometylester kyseliny 2-chlórmetylsulfanyl-benzoovej kyselina d/-2-aminokorková ····2-chloromethylsulfanyl-benzoic acid 1-monomethyl ester d / -2-aminocork ····

-77kyselina 4-(6-butoxy-naftalén-2-yl)-maslová kyselina 3-(2',4’-difluórbenzoyl)propiónová kyselina 3'-nitromaleanilová kyselina 2-(4-kyanofenoxy)-2-metylpropiónová kyselina hexahydroftalová kyselina 5,6-difenyl-2,3-pyrazíndikarboxylová kyselina 5-(4-karboxy-benzoyl)-benzén-1,2,4-trikarboxylová kyselina (3r,4s)-(-)-n-boc-4-amino-3-hydroxy-6-metylheptánová kyselina 3,4-dimetoxy-alfa-merkaptoškoricová kyselina 1-adamantylmalónová kyselina 3-(trifluórmetyl)maslová kyselina 5-fluór-2-nitrobenzoová kyselina 2,3-dimetoxybenzoová kyselina 3,5-dijód-p-hydroxyfenylpyrohroznová kyselina 4-(4-acetylfenyl)maslová kyselina dicyklohexyloctová kyselina 9-fluór-1 -oxo-1 h,5h-pyrido[3,2,1 -ij]chinolín-2-karboxylová kyselina 3-metyl-3-fenylglutárová kyselina boc-d-2-aminoadipová kyselina 7-amino-4-metyl-kumarón-3-yl-octová kyselina homogentisínová kyselina kávová kyselina 2,2-dimetylglutárová kyselina 2-(4-chlórfenyl)-3-(3 -4-dichlórbenzoyl)propiónová kyselina 4-pentínová kyselina (r)-(-)-2-fenylpropiónová kyselina (2-propionyl-fenoxy)-octová kyselina n,n-dietyl-3,6-difluórftalámová kyselina 10,12-oktadekadiínová kyselina 2-hydroxyfenyloctová kyselina 2',3'-dichlórsukcinanilová sulfogama kyselina ···· , «· ·· ··· ·· ·· · · · · · • ··· · · · · ·· ·«· · ·· • · · · · · · · ··· ·· ·· ·· ·· ·-77- 4- (6-butoxy-naphthalen-2-yl) -butyric acid 3- (2 ', 4'-difluorobenzoyl) propionic acid 3'-nitromaleanilic acid 2- (4-cyanophenoxy) -2-methylpropionic acid hexahydrophthalic acid 5,6-Diphenyl-2,3-pyrazinedicarboxylic acid 5- (4-carboxy-benzoyl) -benzene-1,2,4-tricarboxylic acid (3r, 4s) - (-) - n-boc-4-amino- 3-hydroxy-6-methylheptanoic acid 3,4-dimethoxy-alpha-mercaptocinnamic acid 1-adamantylmalonic acid 3- (trifluoromethyl) butyric acid 5-fluoro-2-nitrobenzoic acid 2,3-dimethoxybenzoic acid 3,5-diiodo-p -hydroxyphenylpyruvic acid 4- (4-acetylphenyl) butyric dicyclohexylacetic acid 9-fluoro-1-oxo-1h, 5h-pyrido [3,2,1-i] quinoline-2-carboxylic acid 3-methyl-3-phenylglutaric acid boc-d-2-aminoadipic acid 7-amino-4-methyl-coumaron-3-yl-acetic acid homogentisic acid coffee 2,2-dimethylglutaric acid 2- (4-chlorophenyl) -3- (3 -4- dichlorobenzoyl) propionic acid 4-Pentinic acid (R) - (-) - 2-phenylpropionic acid (2-propionyl-phenoxy) -acetic acid n, n-Diethyl-3,6-difluorophthalic acid 10,12-octadecadiic acid 2-hydroxyphenylacetic acid 2 ', 3'-dichlorosuccinanilic sulfogama acid ···································· · · · ··· ·· ·· ·· ·· ·

-78kyselina 2-(2,4-dichlórfenoxy)propiónová kyselina (2-izopropylfenyl)fosfónová kyselina c/s-2'-etylhexahydroanilová kyselina 3-penténová kyselina 3-hydroxy-3-metyl-n-valérová kyselina 6-chlór-2-(metoxy-fenylamino)-3-nitro-benzoová kyselina 5,7-dichlór-4-hydroxychinolin-3-karboxylová kyselina 2-(2,5-dichlór-fenylkarbamoyl)cyklohexánkarboxylová kyselina atromliečna (2-hydroxy-2-fenylpropiónová) kyselina dibenzofurán-2-sulfónová kyselina 4-fluór-3-(trifluórmetyl)benzoová kyselina uracil-5-karboxylová kyselina 2,3,6-trifluórfenyloctová kyselina 1,3-dioxo-2-o-tolyl-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina 4-chlór-beta-metylhydroškoricová kyselina 1 -(meta-tolyl)-l -cyklopentánkarboxylová kyselina 3-chlórfenoxyoctová kyselina 2-chlór-5-metylbenzoová kyselina 3-(fenylsulfonyl)propiónová kyselina angeliková kyselina 2-hydroxypalmitová kyselina 4-metylkatechol-o,o-dioctová kyselina 4-(6-metoxy-naftalén-1-yl)-maslová kyselina 2,4-dihydroxypyridín-5-karboxylová kyselina 1-metionyl-1-glutámová kyselina 3-karboxymetyl-1-metyl-1 h-indol-2-karboxylová kyselina 4-(3,4,5-trimetoxybenzoyl)maslová kyselina 2-(p-anizyl)-3-fenyljantárová kyselina 2-metylsulfonylbenzoová kyselina 15-metylheptadekánová kyselina 2-cyklohexyl-propiónová kyselina 4-[fenyl-(toluén-4-sulfonyl)-amino]-maslová ·· ·· ····2- (2,4-dichlorophenoxy) propionic acid (2-isopropylphenyl) phosphonic acid cis-2'-ethylhexahydroanilic acid 3-pentenoic acid 3-hydroxy-3-methyl-n-valeric acid 6-chloro-2 - (Methoxy-phenylamino) -3-nitro-benzoic acid 5,7-dichloro-4-hydroxyquinoline-3-carboxylic acid 2- (2,5-dichloro-phenylcarbamoyl) -cyclohexanecarboxylic atromic acid (2-hydroxy-2-phenyl-propionic) dibenzofuran-2-sulfonic acid 4-fluoro-3- (trifluoromethyl) benzoic acid uracil-5-carboxylic acid 2,3,6-trifluorophenylacetic acid 1,3-dioxo-2-o-tolyl-2,3-dihydro- 1h-isoindole-5-carboxylic acid 4-chloro-beta-methylhydrocinnamic acid 1- (meta-tolyl) -1-cyclopentanecarboxylic acid 3-chlorophenoxyacetic acid 2-chloro-5-methylbenzoic acid 3- (phenylsulfonyl) propionic acid angelic acid 2-hydroxypalmitic acid 4-methylcatechol-o, o-diacetic acid 4- (6-methoxy-naphthalen-1-yl) butyric acid 2,4-dihydroxypy 1-Methionyl-1-glutamic acid 3-carboxymethyl-1-methyl-1H-indole-2-carboxylic acid 4- (3,4,5-trimethoxybenzoyl) butyric acid 2- (p-anisyl) ) -3-phenylsuccinic acid 2-methylsulfonylbenzoic acid 15-methylheptadecanoic acid 2-cyclohexyl-propionic acid 4- [phenyl- (toluene-4-sulfonyl) -amino] -butyric acid ·· ·· ····

·..··..· ·.·· ·ί·· .. ·· .. · · · · · · · ·

-79kyselina vinyloctová kyselina 1,3-cyklohexándikarboxylová kyselina 3-acetamino-6-brómbenzoová kyselina 2,3-dibenzylidén-jantárová kyselina 2,,4',6,-trimetylsukcínanilová kyselina n-fenylmaleámová kyselina (r)-(-)-3-hydroxytetradekánová kyselina boc-1 -glutámová kyselina n-furfurylglutarámová kyselina chromon-2-karboxylová kyselina 2,6-bis-( 1 -trimetylsilanyl-vinyl)-benzoová kyselina 5-ŕerc-butylizoftalová kyselina 3-(3,4-dimetoxyfenyl)-2-(2,4-dimetoxyfenyl)-akrylová kyselina n,n’-diglycyletyléndiamín-n,,,n”,n”’,n”’-tetraoctová kyselina 5-(3-nitrofenyl)-2-furoová kyselina 2-metyl-1,8-naftyridín-3-karboxylová kyselina 5-metylfurán-3-karboxylová kyselina 7-brómheptánová kyselina 1-adamantánoctová kyselina krokonová kyselina 2-hydroxy-trikozánová kyselina azelainová kyselina 3-metyl-naftalén-2-karboxylová kyselina 3-(hexadecyltio)benzoová kyselina 11,14-eikozadiénová kyselina (+/-)-írans-epoxyjantárová kyselina 4’-bróm-3’-metyl-1,2,3,6-tetrahydroftalanilová kyselina (1 s)-(-)-(1-amino-2-metylpropyl)fosfónová kyselina 4-(metyltio)benzoová kyselina n-(4-nitrofenyl)izonipekotinová kyselina o-anízová kyselina benzofenón-4,4'-dikarboxylová • ·· ·· ···· ·· ··· ·· · · · · • ··· · · · · ·-79kyselina, vinyl acid, 1,3-cyclohexanedicarboxylic acid, 3-acetylamino-6-bromobenzoic acid 2,3-dibenzylidene-succinic acid 2 ', 4', 6, N--trimetylsukcínanilová fenylmaleámová (R) - (-) - 3 -hydroxytetradecanoic acid boc-1-glutamic acid n-furfurylglutaramic acid chromone-2-carboxylic acid 2,6-bis- (1-trimethylsilanyl-vinyl) -benzoic acid 5-tert-butylisophthalic acid 3- (3,4-dimethoxyphenyl) -2- (2,4-dimethoxyphenyl) -acrylic acid n, n'-diglycylethylenediamine-n ' , n', n '', n '' - tetraacetic acid 5- (3-nitrophenyl) -2-furoic acid 2 -methyl-1,8-naphthyridine-3-carboxylic acid 5-methylfuran-3-carboxylic acid 7-bromoheptanoic acid 1-adamantanacetic acid croconic acid 2-hydroxy-tricosanoic acid azelaic acid 3-methyl-naphthalene-2-carboxylic acid 3 - (hexadecylthio) benzoic acid 11,14-eicosadienoic acid (+/-) - Trans-epoxysuccinic acid 4'-bromo-3'-meth yl-1,2,3,6-tetrahydrophthalanilic acid (1 s) - (-) - (1-amino-2-methylpropyl) phosphonic acid 4- (methylthio) benzoic acid n- (4-nitrophenyl) isonipecotinic acid o- benzophenone-4,4'-dicarboxylic anisic acid • anisic acid benzophenone-4,4'-dicarboxylic acid

-80mono-metylsukcinát kyselina 3-metoxy-9-oxo-8,9-dihydro-7h-benzocykloheptén-6-karboxylová kyselina 5-(terc-butyl)-4-hydroxy-m-toluylová kyselina 3-(5-fenyl-2,5-dihydro-furán-2-yl)-akrylová kyselina 16-bróm-hexadekánová kyselina c/s-1,2-cyklopropándikarboxylová kyselina 2-(1 -indolylkarbonyO-SAS.e-tetrachlórbenzoová kyselina (2-tioxo-benzotiazol-3-yl)-octová kyselina 4'-sulfamoylftalanilová kyselina oftalmová kyselina ftalová kyselina gama-linolénová kyselina 1-(4-chlórfenyl)-1-cyklopropánkarboxylová kyselina (rs)-alfa-metyl-4-karboxyfenylglycín-3-(2-nitrovinyl)benzoová kyselina 5-(3-chlórfenyl)-2,3-dihydro-1h-pyrolizín-6,7-dikarboxylová kyselina d/-gama-karboxyglutámová kyselina n-ŕerc-butyl-3,4,5,6-tetrachlórftalámová kyselina 2-fluór-4-metoxybenzoová kyselina 3,5-dichlórsalicylová kyselina bis(p-tolyl)octová kyselina 2-(4-hydroxyfenyl)izovalérová kyselina 3-(kyanometyltio)tiofén-2-karboxylová kyselina 3-metylindén-2-karboxylová kyselina 13-metyltetradekánová kyselina 2-propyloktánová kyselina hexahydro-n-(4-(metyltio)fenyl)ftalámová kyselina 8-hydroxy-2-metyl-chinolín-5-sulfónová kyselina 4-(2,4-bis-(2-2-dimetyl-propyl)-fenoxy)-maslová kyselina 4-chlórindoloctová kyselina 2,3-dihydrobenzo-furánoctová kyselina 5-oktadecyloxyizoftalová kyselina 4-(2-butylkarbamoyl-acetylamino)-benzoová-80-mono-methylsuccinate 3-methoxy-9-oxo-8,9-dihydro-7H-benzocycloheptene-6-carboxylic acid 5- (tert-butyl) -4-hydroxy-m-toluic acid 3- (5-phenyl- 2,5-dihydro-furan-2-yl) -acrylic acid 16-bromo-hexadecanoic acid cis-1,2-cyclopropanedicarboxylic acid 2- (1-indolylcarbonyl-O-SAS) .e-tetrachlorobenzoic acid (2-thioxobenzothiazole) -3-yl) -acetic acid 4'-sulfamoyl-phthalanic acid ophthalic acid phthalic acid gamma-linolenic acid 1- (4-chlorophenyl) -1-cyclopropanecarboxylic acid (rs) -α-methyl-4-carboxyphenylglycine-3- (2- nitrovinyl) benzoic acid 5- (3-chlorophenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid n-gamma-carboxyglutamic acid n-tert-butyl-3,4,5,6-tetrachlorophthalic acid 2-fluoro-4-methoxybenzoic acid 3,5-dichlorosalicylic acid bis (p-tolyl) acetic acid 2- (4-hydroxyphenyl) isovaleric acid 3- (cyanomethylthio) thiophene-2-carboxylic acid 3-methylindene-2-carboxylic acid Acid 1 3-methyltetradecanoic acid 2-propyloctanoic acid hexahydro-1- (4- (methylthio) phenyl) phthalic acid 8-hydroxy-2-methyl-quinoline-5-sulfonic acid 4- (2,4-bis- (2-2- dimethyl-propyl) -phenoxy) -butyric acid 4-chloroindole acetic acid 2,3-dihydrobenzo-furanacetic acid 5-octadecyloxyisophthalic acid 4- (2-butylcarbamoyl-acetylamino) -benzoic acid

• · · • · • ··· • · · • ··· • · • · • · • · • · • · ···· • • ···· • • 99 • · • · 99 • · • · • · • · • · · · • · · · ·· · · ·· · · • · • · • · • ·

kyselina 4-izopropyl-cyklohex-4-én-1,2-dikarboxylová kyselina fmoc-1-asparágová alfa-ŕerc-butylester kyseliny n-alfa-fmoc-n-gama-boc-1 -diaminomaslovej kyselina 9-metyl-9h-fluorén-3-karboxylová kyselina pentafluórbenzoová kyselina 3-butén-1,2,3-trikarboxylová kyselina 4-dibenzotiofénkarboxylová kyselina 2,2-dimetylmaslová kyselina m-toluylová kyselina 4-(4-hydroxy-benzénsulfonyl)-benzoová kyselina 2-dodecénová kyselina 4-[1 -(2-merkapto-4,5-dihydro)imidazolo]benzoová kyselina 5-chlórbicyklo[2.2.1 ]hept-2-en-5-endo-karboxylová kyselina c/s-4-(fosfonometyl)piperidín-2-karboxylová kyselina 2-jód-3-metylbenzoová kyselina 2-(4-etyl-fenyl)-1,3-dioxo-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina dimetylmalónová kyselina kuménsulfónová kyselina nl-ftaloyl-gly-alfa-aminoizomaslová tecloftalam kyselina 3-benzoylamino-n-hexylkarbamoylmetyl-sukcínamová kyselina 6,8-dibrómkumarín-3-karboxylová boc-d-homofenylalanín kyselina 2-fluórsukcínanilová kyselina 2-(4-nitrofenyl Jpropiónová kyselina 4-ŕrans-fenylcyklohexán-c/s-1,2-dikarboxylová o-sulfobenzaldehyd kyselina 4-brómškoricová kyselina 4-[2-(4-etoxy-benzoylamino)-3-fenyl-akryloylamino)rnaslová kyselina 5-sulfosalicylová kyselina 3'-fluórmaleanilová kyselina 4-(ŕerc-butoxy)benzoová • ·· ·· ···· ·· ··· ·· ···· • ··· · · · · ·4-isopropyl-cyclohex-4-ene-1,2-dicarboxylic acid fmoc-1-aspartic n-alpha-fmoc-n-gamma-boc-1-diaminobutyric acid alpha-tert-butyl ester 9-methyl-9h- fluorene-3-carboxylic acid pentafluorobenzoic acid 3-butene-1,2,3-tricarboxylic acid 4-dibenzothiophenecarboxylic acid 2,2-dimethylbutyric acid m-toluic acid 4- (4-hydroxy-benzenesulfonyl) -benzoic acid 2-dodecenoic acid 4- [1- (2-mercapto-4,5-dihydro) imidazolo] benzoic acid 5-chlorobicyclo [2.2.1] hept-2-ene-5-endo-carboxylic acid cis-4- (phosphonomethyl) piperidine -2-carboxylic acid 2-iodo-3-methylbenzoic acid 2- (4-ethylphenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid dimethyl malonic acid cumenesulfonic acid nl- phthaloyl-gly-alpha-aminoisobutyric acid tecloftalam 3-benzoylamino-n-hexylcarbamoylmethyl-succinamic acid 6,8-dibromocoumarin-3-carboxylic acid boc-d-homophenylalanine 2-fluorosuccinanilic acid 2 - (4-nitrophenyl) propionic acid 4-trans-phenylcyclohexane-cis-1,2-dicarboxylic o-sulfobenzaldehyde 4-bromocinnamic acid 4- [2- (4-ethoxy-benzoylamino) -3-phenyl-acryloylamino) -sonic acid 5-Sulfosalicylic acid 3'-fluoro-maleanoic acid 4- (tert-butoxy) benzoic acid • ·····················

-82kyselina 2-(4-(4-kyano-fenoxy)-ph)-1,3-clioxo-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina c/s-n-(4-acetylfenyl)hexahydroftalámová kyselina (s)-2-metyloktánová kyselina 9-hydroxyfluorén-9-karboxylová kyselina 2-metyl-1-naftyloctová kyselina 2,4-dihydroxy-3,6-dinnetylbenzoová kyselina 2,2,5,7-tetrametylindán-1 -όη-4-karboxylová kyselina 5-(dimetyôaminosulfonyl)2,3-dihydro-gama-oxo-1 -(1 h)-indolbutánová kyselina 4-chlórfenylsulfonyloctová kyselina 4-[2-(propán-2-sulfonyl)-acetylamino]-benzoová kyselina 2-(2-{2-metoxyetoxy)etoxy)octová kyselina 3,4,5-trichlór-2-tiofénkarboxylová-82- 2- (4- (4-cyano-phenoxy) -ph) -1,3-clioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid cis- (4-acetylphenyl) hexahydrophthalic acid (s) -2-methyloctanoic acid 9-hydroxyfluorene-9-carboxylic acid 2-methyl-1-naphthylacetic acid 2,4-dihydroxy-3,6-dinomethylbenzoic acid 2,2,5,7-tetramethylindan-1-one- 4- (2- (Propane-2-sulfonyl) -acetylamino) -benzoic acid 4-carboxylic acid 5- (dimethylamino-sulfonyl) -2,3-dihydro-gamma-oxo-1- (1 h) -indole-butanoic acid 4-Chloro-phenylsulfonylacetic acid 2- (2- (2-methoxyethoxy) ethoxy) acetic acid 3,4,5-trichloro-2-thiophenecarboxylic acid

4-karboxybenzaldehyd kyselina n-etyl-n-(p-toluénsulfonyl)antranilová kyselina (s)-(+)-2-hydroxy-2-fenylpropiónová kyselina 2-karboxymetyl-4,6-dimetoxy-benzoová kyselina n-alfa-z-glycyl-1 -glutámová kyselina 4-(2-karbamoylfenylamino)-2,3-dichlór-2-buténová kyselina 4-metyl-2-hepténová kyselina 2-karboxy-alfa-oxobenzénoctová kyselina (+/-)-1-aminocyklopentán-c/s-1,3-dikarboxylová kyselina (-)-1,2,3-trimetyl-2-cyklopenténakrylová kyselina 2,,4,-difluórglutaranilová kyselina 3-fenyl-1,3,5-pentántrikarboxylová ftalylsulfacetamid kyselina 4-(etoxykarbonylmetoxy)-1 -hydroxy-2-naftoová kyselina 2-(2-kyanofenyltio)benzoová kyselina 3-chlór-5-jódbenzoová kyselina 2-(3-(2,2,2-trichlór-1-izobutylylamino-etyl)-tioureido)-benzoová kyselina 10,12-nonakozadiínová kyselina 2-hydroxytetrakozánová kyselina 2-ftalimidobenzoová • ·· ·· ···· · ·4-carboxybenzaldehyde n-ethyl-N- (p-toluenesulfonyl) anthranilic acid (s) - (+) - 2-hydroxy-2-phenylpropionic acid 2-carboxymethyl-4,6-dimethoxybenzoic acid n-alpha-z Glycyl-1-glutamic acid 4- (2-carbamoylphenylamino) -2,3-dichloro-2-butenoic acid 4-methyl-2-heptenoic acid 2-carboxy-alpha-oxobenzeneacetic acid (+/-) - 1-aminocyclopentane c / s-1,3-dicarboxylic acid (-) - 1,2,3-trimethyl-2-cyklopenténakrylová acid, 2, 4, -difluórglutaranilová acid, 3-phenyl-1,3,5-pentanetricarboxylic ftalylsulfacetamid 4- (ethoxycarbonylmethoxy) -1-hydroxy-2-naphthoic acid 2- (2-cyanophenylthio) benzoic acid 3-chloro-5-iodobenzoic acid 2- (3- (2,2,2-trichloro-1-isobutylylaminoethyl) - thioureido) -benzoic acid 10,12-nonacosadiic acid 2-hydroxytetracosanoic acid 2-phthalimidobenzoic acid · ·· ····· · ·

BBB B · · ···BBB B · · ···

B BBB BBB B BBBB BBB

-83kyselina 4'-etoxyftalanilová kyselina 4-jódacetamidosalicylová kyselina n-(terc-butoxykarbonyl)-1 -asparágová-83 4'-ethoxyphtalanilic acid 4-iodoacetamidosalicylic acid n- (tert-butoxycarbonyl) -1-aspartic acid

4-benzylester kyseliny 4-benzoylbenzoovej kyselina 4'-bróm-1,2,3,6-tetrahydroftalanilová kyselina 1-naftylmetylfosfónová kyselina 3-jód-4-metylbenzoová kyselina (s)-3-hydroxy-3-fenylpropánová kyselina (s)-2-etyloktánová kyselina n-(2-metyl-4-nitro-fenyl)jantárová kyselina 3-aminopropylfosfónová kyselina (+)-4'-chlórtartranilová kyselina boc-(3s,4s)-4-amino-3-hydroxy-6-metylheptánová kyselina c//-beta-hydroxylaurová kyselina (+/-)-2-hydroxypentadekánová kyselina n-metylmaleámová kyselina 3-metylhipurová kyselina 3-nitroškoricová kyselina mesakonová kyselina 3-hydroxybenzoová kyselina 2-bróm-4,5-dimetoxyhydroškoricová kyselina 1-alanyl-4-asparágová kyselina 4-benzoyloxybenzoová kyselina n-fmoc-1-1,2,3,4-tetrahydroizochinolín-3-karboxylová kyselina 3,4-diacetoxybenzoová kyselina 1,2-dihydroxycyklobutánkarboxylová kyselina 2,,3’-dimetylmaleanilová kyselina 1 -metyl-1 h-indazol-3-karboxylová kyselina 22-trikozénová kyselina n-ŕerc-boc-7-aminoheptánová kyselina 5-nitro-2-(fenyltio)benzénsulinic kyselina 1-(3,4-dimetoxy-ph)-hydroxy-5,6,7-trimetoxynaftalén-2-karboxylová ·· ·· ···· ·· • · · · · · ♦ ··· · · · · ·4-benzyl 4-benzoylbenzoic acid 4'-bromo-1,2,3,6-tetrahydrophthalanilic acid 1-naphthylmethylphosphonic acid 3-iodo-4-methylbenzoic acid (s) -3-hydroxy-3-phenylpropanoic acid (s) 2-ethyloctanoic acid n- (2-methyl-4-nitrophenyl) succinic acid 3-aminopropylphosphonic acid (+) - 4'-chlorotartranilic acid boc- (3s, 4s) -4-amino-3-hydroxy-6 - methylheptanoic acid cis - beta-hydroxylauric acid (+/-) - 2-hydroxypentadecanoic acid n-methylmaleamic acid 3-methylhipuric acid 3-nitrocinnamic acid mesaconic acid 3-hydroxybenzoic acid 2-bromo-4,5-dimethoxyhydrocinnamic acid 1 alanyl-4-aspartic acid 4-benzoyloxybenzoová n-fmoc-1-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid 3,4-diacetoxybenzoová acid 1,2-dihydroxycyklobutánkarboxylová acid, 2, 3 ' dimetylmaleanilová 1-methyl-1H-indazole-3-carboxylic acid 22-tricosenoic acid n-tert-boc-7-aminohep 5-nitro-2- (phenylthio) benzenesulfonic acid 1- (3,4-dimethoxy-ph) -hydroxy-5,6,7-trimethoxynaphthalene-2-carboxylic acid ·· ·· ···· ·· · · · · · ♦ ··· · · · · ·

-84• ·· ·· ·· kyselina 3-(3,4-dimetoxy-fenyl)-3-(3,4,5-trimetoxyfenyl)-propiónová kyselina di(cyklohexyl)-ditiofosforečná kyselina 4-metylfenoxyoctová kyselina 3-(trifluórmetyl)škoricová kyselina trimetylpyrohroznová kyselina n-(benzyl)-3,4,5,6-tetrachlórftalámová kyselina 2-etyl-3-(4-nitro-fenyl)-akrylová kyselina 5-(3-chlór-5-trifluórmetyl-2-pyridylmetyl)tiofén-2-sulfónová kyselina boc-5-aminovalérová kyselina 3-p-tolyloxymetyl-benzoová kyselina 2-amino-1,5-naftaléndisulfónová kyselina d/-alfa-metoxyfenyloctová kyselina 1 -cyklopenténkarboxylová kyselina 2-metyl-1 -naftalénkarboxylová kyselina 2-fluór-3-metylbenzoová kyselina (r)-3-chlórmliečna kyselina 2-fenoxybenzoová kyselina (-)-3-pinánkarboxylová kyselina 5-metyl-2-furoová kyselina 213-dibróm-2’-metoxy-3'-nitrosukcínanilová beta-cyklohexyl-ester kyseliny n-boc-4-asparágovej kyselina (1 -metyl-heptyl)-fenyl-fosfínová kyselina 3-jód-4-metoxybenzoová (+)-dimetyl-2,3-o-benzylidén-d-vínan kyselina d/-o-metoxymandlová kyselina 2-chlór-para-anízová kyselina (2-karboxyfenylimino)dioctová kyselina mekonová kyselina 3-metyl-1-oxo-1,2-dihydro-izochinolín-4-karboxylová kyselina 3-(4-metylsulfanyl-fenyl)-3-oxo-propiónová kyselina 4-(diacetoxymetyl)benzoová kyselina 3-fn-(2,5-xylyl)karbamoyl)-5-norbornén-2-karboxylová • ·· ·· φφφφ ·· ·· · ·· φφφφ • φφφ φ · φ · φ kyselina 3-(4-chlór-fenylamino)-maslová kyselina 3-acenaftén-5-yl-akrylová kyselina 2,4-dimetylfenoxyoctová kyselina 5,7-dodekadiíndiová kyselina 3,5-difenylbenzoová kyselina (2s,4r)-4-metylglutámová kyselina nitrotereftalová kyselina c/s-n-cyklohexylhexahydroftalámová kyselina 5-nitroindol-2-karboxylová kyselina d(-)-2-amino-6-fosfonohexánová kyselina (etyltio)octová kyselina 4'-brómmaleanilová kyselina 2-(p-tolyltio)octová kyselina tiooctová kyselina (6-terc-butyl-l,1-dimetyl-indán-4-yl)-octová kyselina 3-metyl-1,1-cyklopentándioctová kyselina 2-(karboxy-4-hydroxyfenyl)chinolín-4-karboxylová kyselina dnp-1-asparágová kyselina 2-(4-etoxybenzoyl)akrylová kyselina 1-(2,5-dichlór-4-sulfofenyl)-5-pyrazolón-3-karboxylová kyselina 2-[3-(n’-nonanoyl-hydrazíno)-3-oxo-propionylamino]benzoová kyselina 3-chlór-2-(toluén-4-sulfonylamino)-benzoová kyselina 2-tridecénová kyselina 4,5,6,7-tetrafluór-2I3-dihydro-gama-oxo-1 -(1 h)-indolibutánová kyselina 3'-brómglutaranilová kyselina 3-(4-fluórbenzoyl)propiónová kyselina 3-(ac-(5-bróm-1,3-dioxo-1,3-dihydroizoindol-2-ylmetyl)amono)-benzoová kyselina 5-(chlóracetyl)tiofén-2-octová kyselina 3-(fenyltio)akrylová kyselina o-hydroxyhipurová kyselina 4-izopropoxybenzoová kyselina (r)-(-)-2-chlór 3-fenylpropiónová-84 • ····· 3- (3,4-Dimethoxyphenyl) -3- (3,4,5-trimethoxyphenyl) -propionic acid di (cyclohexyl) -dithiophosphoric acid 4-methylphenoxyacetic acid 3- ( trifluoromethyl) cinnamic acid trimethylpyruvic acid n- (benzyl) -3,4,5,6-tetrachlorophthalic acid 2-ethyl-3- (4-nitro-phenyl) -acrylic acid 5- (3-chloro-5-trifluoromethyl-2) -pyridylmethyl) thiophene-2-sulfonic acid boc-5-aminovaleric acid 3-p-tolyloxymethyl-benzoic acid 2-amino-1,5-naphthalenedisulfonic acid d-alpha-methoxyphenylacetic acid 1-cyclopentenecarboxylic acid 2-methyl-1- naphthalenecarboxylic acid 2-fluoro-3-methylbenzoic acid (R) -3-chloro-lactic acid 2-phenoxybenzoic acid (-) - 3-pinanecarboxylic acid 5-methyl-2-furoic acid 2 1 3-dibromo-2'-methoxy-3 n-boc-4-aspartic acid (1-methyl-heptyl) -phenyl-phosphinic acid 3-iodo-4-methoxy-benzoic acid (+) - dimethyl-2,3-o-benzylide 1'-nitrosucciniline beta-cyclohexyl ester n-tartrate d -o-methoxy-butyric acid 2-chloro-para-anisic acid (2-carboxyphenylimino) diacetic acid meconic acid 3-methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxylic acid 3- (4-Methylsulfanyl-phenyl) -3-oxo-propionic acid 4- (diacetoxymethyl) -benzoic acid 3-N- (2,5-xylyl) -carbamoyl) -5-norbornene-2-carboxylic acid · ·· ·· φφφφ ·· 3- (4-chloro-phenylamino) -butyric acid 3-acenaphthen-5-yl-acrylic acid 2,4-dimethylphenoxyacetic acid 5,7-dodecadienedioic acid 3, 5-diphenylbenzoic acid (2s, 4r) -4-methylglutamic acid nitroterephthalic acid cis -cyclohexylhexahydrophthalic acid 5-nitroindole-2-carboxylic acid d (-) - 2-amino-6-phosphonohexanoic acid (ethylthio) acetic acid 4 ' 2- (p-tolylthio) acetic acid thioacetic acid (6-tert-butyl-1,1-dimethyl-indan-4-yl) -acetic acid 3-methyl-1,1-cyclopentanediacetic acid 2- (carboxy-4-hydroxyphenyl) quinoline-4-carboxylic acid dnp-1-aspartic acid 2- (4-ethoxybenzoyl) acrylic acid 1- (2,5-dichloro-4-sulfophenyl) -5-pyrazolone-3 -carboxylic acid 2- [3- (n'-nonanoyl-hydrazino) -3-oxo-propionylamino] benzoic acid 3-chloro-2- (toluene-4-sulfonylamino) -benzoic acid 2-tridecenoic acid 4,5,6 , 7-tetrafluoro-2 L 3-dihydro-gamma-oxo-1 - (1 h) -indolibutánová 3'-brómglutaranilová 3- (4-fluorobenzoyl) propionic acid 3- (ac- (5-bromo-1, 3-dioxo-1,3-dihydro-isoindol-2-ylmethyl) -amono) -benzoic acid 5- (chloroacetyl) -thiophene-2-acetic acid 3- (phenylthio) acrylic acid o-hydroxyhipuric acid 4-isopropoxybenzoic acid (r) - ( -) - 2-Chloro-3-phenylpropionic

-86• ·· ·· · • ··· ··· ·· kyselina 11-eikozénová kyselina ((3-chlór-fenyl)-(toluén-4-sulfonyl)-amino)-octová kyselina 4-izotiokyanátobenzénsulfónová kyselina 4-chlór-5-nitro-o-toluénsulfónová kyselina 2-chlórstearová kyselina 3-(3,4-dimetoxy-fenyl)-propínová kyselina 3-(n-(3-nitrofenyl)karbamoyl)bicyklo(2.2.1 )hept-5-én-2-karboxylová kyselina cyklohexyloctová kyselina 5-norbornén-2-karboxylová kyselina brómmaleínová kyselina 4-oktyloxybenzoová kyselina tymoxyoctová kyselina 4-(4-chlór-benzénsulfonyl)-ftalová kyselina 2,2-difluórjantárová /7-ŕerc-boc-5-cyklohexylstatín kyselina (+/-)-3-exo-aminotricyklo[2.2.1.0(2,6)]heptán-3-endo-7-anti-dikarboxylová kyselina (r)-(+)-2-chlórhexánová kyselina 2-(3,4-dimetoxy-alfa-metylbenzyl)-6-metoxy-benzoová kyselina tridekafluór-2-nonénová kyselina 3-metyl-2-(orto-tolyl)-hexánová kyselina 2-metyl-7-oxononánová kyselina /?-alfa-formyl-1 -glutámová kyselina (l-aminobutyl)fosfónová kyselina exo-3,6-epoxy-1,2,3,6-tetrahydroftalová kyselina n-(2,5-xylyl)glutarámová kyselina 3-amino-2,6-naftalén-disulfónová kyselina 12(r)-hydroxyeikoza-5z,8z, 14z-triénová kyselina 3-metyl-2-fenylhexánová kyselina 3-chlór-2,4,6-trimetyl-benzoová kyselina 6-(4-ŕerc-butylfenyl)-4-oxo-5-hexénová kyselina n-etyl-d-glutámová kyselina d/-tropová • ·· ·· ···· ·· ··· ·· · · · · • ··· · · · Λ ·-86 11-Eicosenoic acid ((3-chloro-phenyl) - (toluene-4-sulfonyl) -amino) -acetic acid 4-isothiocyanate-benzenesulfonic acid 4- chloro-5-nitro-o-toluenesulfonic acid 2-chloro-stearic acid 3- (3,4-dimethoxyphenyl) -propionic acid 3- (n- (3-nitrophenyl) carbamoyl) bicyclo (2.2.1) hept-5- en-2-carboxylic acid cyclohexylacetic acid 5-norbornene-2-carboxylic acid bromaleanoic acid 4-octyloxybenzoic acid thyloxyacetic acid 4- (4-chloro-benzenesulfonyl) -phthalic acid 2,2-difluoro succinic acid / 7-tert-boc-5- cyclohexylstatin (+/-) - 3-exo-aminotricyclo [2.2.1.0 (2,6)] heptane-3-endo-7-anti-dicarboxylic acid (r) - (+) - 2-chlorohexanoic acid 2- ( 3,4-dimethoxy-alpha-methylbenzyl) -6-methoxy-benzoic acid tridecafluoro-2-nonenoic acid 3-methyl-2- (ortho-tolyl) -hexanoic acid 2-methyl-7-oxononanoic acid p-alpha- formyl-1-glutamic acid (1-aminobutyl) phosphonic acid Exo-3,6-epoxy-1,2,3,6-tetrahydrophthalic acid n- (2,5-xylyl) glutaramic acid 3-Amino-2,6-naphthalene disulfonic acid 12 (r) -Hydroxyicose-5z 8z, 14z-Trienoic acid 3-methyl-2-phenylhexanoic acid 3-chloro-2,4,6-trimethyl-benzoic acid 6- (4-tert-butylphenyl) -4-oxo-5-hexenoic acid n-ethyl -d-glutamic acid d / -tropic acid d trop trop trop d d d d d d d d d

-87kyselina 8-metylnon-6-énová kyselina alfa-chlórfenyloctová kyselina n-oktadecylmaleámová kyselina 3-(3,4,5-trimetoxyfenyl)propiónová kyselina 1,3-dioxo-2-m-tolyl-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina ŕrans-2-decénová kyselina 3-(4-metylfenyl)propiónová kyselina 6-metoxy-1-naftoová kyselina 2-(4-acetoxy-3-ŕerc-butylfenoxy)-tetradekánová kyselina 2-(2-cl-4-(2-metyl-akryloylamino)-fenylkarbamoyl)-3,3-dimetyl-maslová kyselina 2-[[(2,4-dichlórfenyl)sulfonyl]-3-(trifluórmetyl)anilino]octová kyselina 3-cyklohexénkarboxylová kyselina 3-bróm-5-nitrobenzoová bis(2-etylhexyl)-hydrogenfosfát kyselina 3-sukcínimidopropiónová kyselina 2-(hydroxy-fenyl-fosfinoyl)-benzoová kyselina 3-(4-chlórbenzoyl)-2-(4-metylfenyl)propiónová kyselina 4-bróm-2-chlórbenzoová kyselina 2,4-dinitrobenzoová kyselina 2,4,6-trimetyl-benzénstulfínová kyselina cyklopentenyloctová kyselina n-alfa-acetyl-/?-gama-boc-1 -diaminomaslová kyselina 3-(4-chlór-fenyl)-3-fenylacetylamino-propiónová kyselina 2,3,4,5-tetrafluórbenzoová kyselina 3-[4-(4-fluórbenzyloxy)fenyl]akrylová kyselina 1-cyklopentén-1,2-dikarboxylová kyselina 3-ŕerc-butyl-5-metylsalicylová kyselina pmp(p-mbzl)-87-8-methylnon-6-enoic acid alpha-chlorophenylacetic acid n-octadecylmaleamic acid 3- (3,4,5-trimethoxyphenyl) propionic acid 1,3-dioxo-2-m-tolyl-2,3-dihydro-1 h-Isoindole-5-carboxylic acid trans-2-decenoic acid 3- (4-methylphenyl) propionic acid 6-methoxy-1-naphthoic acid 2- (4-acetoxy-3-tert-butylphenoxy) -tetradecanoic acid 2- ( 2-cl-4- (2-methyl-acryloylamino) -phenylcarbamoyl) -3,3-dimethyl-butyric acid 2 - [[(2,4-dichlorophenyl) sulfonyl] -3- (trifluoromethyl) anilino] acetic acid 3- 3-Bromo-5-nitrobenzoic acid, cyclohexenecarboxylic acid bis (2-ethylhexyl) -hydrogenphosphate 3-Succinimidopropionic acid 2- (hydroxyphenylphosphinoyl) -benzoic acid 3- (4-chlorobenzoyl) -2- (4-methylphenyl) propionic acid 4-bromo-2-chlorobenzoic acid 2,4-dinitrobenzoic acid 2,4,6-trimethyl-benzenesulfonic acid cyclopentenylacetic acid n-alpha-acetyl-R-gamma-boc-1-diaminobutyric acid 3- (4-chloro) phenyl) -3-phenylacetamido 2,3,4,5-tetrafluorobenzoic acid ylamino-propionic acid 3- [4- (4-fluorobenzyloxy) phenyl] acrylic acid 1-cyclopentene-1,2-dicarboxylic acid 3-tert-butyl-5-methylsalicylic acid pmp ( p-MBzl)

3-(4-hydroxy-2-metyl-cyklohex-2-enyl)-propiónová kyselina 1,3-dikyano-2,2-dimetyl-cyklobután-1,3-dikarboxylová kyselina 4,5-bis-(4-amino-fenoxy)-ftalová kyselina 9-brómnonánová3- (4-hydroxy-2-methyl-cyclohex-2-enyl) -propionic acid 1,3-dicyano-2,2-dimethyl-cyclobutane-1,3-dicarboxylic acid 4,5-bis- (4-amino) -phenoxy) -phthalic acid 9-bromonanoic acid

• ·· • · • ··· • ·· • · • ··· ·· • · • · · · • · • · ···· • • ···· • • ·· · • · · · • · · ·· · • · · • · · · • · · · ·· · · ·· · · ·· ·· ·· ··

kyselina 7,7-dimetyl-(5z,8z)-eikoza-diénová kyselina 2,4,6-tri-ŕerc-butyl-benzoová kyselina 2-akrylamido-2-metylpropánsulfónová kyselina n-metyl-d/-glutámová kyselina 1 -hydroxy-4-(metoxykarbonylmetoxy)-2-naftoová kyselina 4-etylbenzoová kyselina 3-[2-(4-etoxy-benzoylamino)-3-fenyl-akryloylamino]-propiónová kyselina 4-(brómmetyl)benzoová kyselina 2-chlór-5-fluórbenzoová kyselina 3-(4-chlórfenyl)glutárová kyselina bis(4-metoxyfenyl)fosfinová kyselina 18-fenyloktadekánová kyselina (s)-(-)-alfa-metoxy-alfa-(trifluórmetyl)fenyloctová kyselina (r)-(+)-citronelová kyselina 4-(hydroxymetyl)fenoxyoctová kyselina 4,5-dichlór-4,5,5-trifluórpentánová kyselina 4,4-bis-etoxykarbonyl-heptándiová kyselina (s)-(-)-2-brómpentánová kyselina 1 h-imidazo(4,5-c)pyridín-2-sulfónová kyselina 3-(2-hydroxy-5-metylbenzoyl)propiónová kyselina neononánová kyselina 4-ho-6,7-dimetoxy-1-(3,4,5-trimetoxyfenyl)-aftalén-2-karboxylová kyselina 1 -2-(benzyloxykarbonylamino)-4-sulfamoylmaslová kyselina c/s-1 -amino-3-(2-fosfono-1 -hydroxyetyl)-cyklobután-1 -karboxylová kyselina 10-brómdekánová kyselina 3-nitrosalicylová kyselina z-3-(2-benzimidazolyltio)propénová kyselina 4'-(etoxykarbonyl)-maleanilová kyselina 4'-fluór-1,2,3,6-tetrahyroftalanilová kyselina 6-hydroxykaprónová kyselina (r)-(-)-alfa-metoxyfenyloctová kyselina dibróm-maleínová • ·· ······ ·· ·· · ·· ···· • ··· BBB B B7,7-Dimethyl- (5z, 8z) -eicoza-dienoic acid 2,4,6-tert-butyl-benzoic acid 2-acrylamido-2-methylpropanesulfonic acid n-methyl-d-glutamic acid 1- hydroxy-4- (methoxycarbonylmethoxy) -2-naphthoic acid 4-ethylbenzoic acid 3- [2- (4-ethoxy-benzoylamino) -3-phenyl-acryloylamino] -propionic acid 4- (bromomethyl) benzoic acid 2-chloro-5 -fluorobenzoic acid 3- (4-chlorophenyl) glutaric acid bis (4-methoxyphenyl) phosphinic acid 18-phenyloctadecanoic acid (s) - (-) - alpha-methoxy-alpha- (trifluoromethyl) phenylacetic acid (r) - (+) -citronelic acid 4- (hydroxymethyl) phenoxyacetic acid 4,5-dichloro-4,5,5-trifluoropentanoic acid 4,4-bis-ethoxycarbonyl-heptanedioic acid (s) - (-) - 2-bromopentanoic acid 1 h-imidazo (4,5-c) pyridine-2-sulfonic acid 3- (2-hydroxy-5-methylbenzoyl) propionic acid neononanoic acid 4-ho-6,7-dimethoxy-1- (3,4,5-trimethoxyphenyl) - Aphthalene-2-carboxylic acid 1 - 2- (benzyloxycarbonylamino) -4 -sulfamoylbutyric acid cis-1-amino-3- (2-phosphono-1-hydroxyethyl) -cyclobutane-1-carboxylic acid 10-bromodecanoic acid 3-nitrosalicylic acid z-3- (2-benzimidazolylthio) propenoic acid 4 ' - (ethoxycarbonyl) -maleeanilic acid 4'-fluoro-1,2,3,6-tetrahyropthalanilic acid 6-hydroxycaproic acid (r) - (-) - alpha-methoxyphenylacetic acid dibromo-maleic acid • ·· ······ ···················· BBB BB

-89kyselina 13-oxooktadekánová kyselina 1 -formyl-3-cyklohexén-1 -propiónová kyselina 2-(3,4-dichlórfenylkarbamoyl)cyklohexánkarboxylová kyselina 2-metyl-3,3,3-trifenyl-propiónová kyselina (8r,15s)-dihydroxy-(5z,9e,11z,13e)-eikozatetraénová kyselina 3-(4-metylsulfonylbenzoyl)propiónová kyselina c/-glukurónová kyselina 4’,6-dinitro-2,-metoxyftalanilová kyselina 5,8-dioxo-1,4,4a,5,8,8a-hexahydro-1 -naftalénkarboxylová kyselina hemimelitová kyselina 4-metyl-4-fenyl-hexánová kyselina n-(4-brómfenyl)glutaranilová kyselina monofluórfosforečná kyselina 2-etylmaslová kyselina boc-(3-aminometyl)-benzoová kyselina n-(2-pentylsulfanyl-benzotiazol-6-yl)-sukcínamová kyselina 6-metoxysalicylová kyselina alfa-merkapto-2-metoxy-beta-metylškoricová kyselina c/s-hexahydro-n-(2,4-dichlórfenyl)ftalámová kyselina 2-(3-(1-butyrylamino-2,2I2-trichlór-etyl)-tioureido)-benzoová kyselina 2-[3-(n-heptanoyl-hydrazíno)-3-oxo-propionylamino]-benzoová kyselina (-)-c/s-izoketopinová kyselina 2-chlór-4,5-dimetoxybenzoová kyselina 2-etoxyškoricová kyselina 5-(2-tienoyl)maslová kyselina 3-(2,5-dimetylbenzoyl)propiónová kyselina pentachlór-c/s-2,4-pentadiénová kyselina 4'-(2-hydroxyetyl)glutaranilová kyselina n-(4-fenoxyfenyl)malonámová kyselina (4-ŕerc-butyl-fenylsulfanyl)-octová kyselina 4-(ŕerc-butyl)škoricová n-(p-toluoyl)-glycín ·· ·· ···· ·· • · · · · ··· · · · · · ····· · · · ·-89-13-oxooctadecanoic acid 1-formyl-3-cyclohexene-1-propionic acid 2- (3,4-dichlorophenylcarbamoyl) cyclohexanecarboxylic acid 2-methyl-3,3,3-triphenyl-propionic acid (8r, 15s) -dihydroxy - (5z, 9e, 11z, 13e) -eicosatetraenoic acid 3- (4-methylsulfonylbenzoyl) propionic acid cis -glucuronic acid 4 ', 6-dinitro-2 , -methoxyphthalanic acid 5,8-dioxo-1,4,4a 5,8,8a-hexahydro-1-naphthalenecarboxylic acid hemimelitic acid 4-methyl-4-phenyl-hexanoic acid n- (4-bromophenyl) glutaranilic acid monofluorophosphoric acid 2-ethylbutyric acid boc- (3-aminomethyl) -benzoic acid n- (2-Pentylsulfanyl-benzothiazol-6-yl) -succinamic acid 6-Methoxy-salicylic acid alpha-mercapto-2-methoxy-beta-methylcinnamic acid cis-hexahydro-n- (2,4-dichlorophenyl) phthalic acid 2 - (3- (1-butyrylamino-2-I, 2,2-trichloro-ethyl) -thioureido) -benzoic acid 2- [3- (n-heptanoyl-hydrazino) -3-oxo-propionylamino] -benzoic acid, (-) c / s-isopropyl ketopinic acid 2-chloro-4,5-dimethoxybenzoic acid 2-ethoxycinnamic acid 5- (2-thienoyl) butyric acid 3- (2,5-dimethylbenzoyl) propionic acid pentachloro-cis-2,4-pentadienoic acid 4 ' - (2-hydroxyethyl) glutaranilic acid n- (4-phenoxyphenyl) malonamic acid (4-tert-butyl-phenylsulfanyl) -acetic acid 4- (tert-butyl) cinnamic n- (p-toluoyl) -glycine ·· ··· ·····················

-90kyselina antrachinón-disulfónová kyselina 4'-bróm-2'-metylglutaranilová kyselina 2,2'-ditiodibenzoová kyselina 2,4-difluórfenyloctová kyselina trifluórmetánsulfónová kyselina 4-etenyl-3-metyl-5-(metyltio)tiofén-2-karboxylová kyselina 2-brómhexánová kyselina 5-(2-karboxyfenylaminosulfo)-2-chlórbenzoová p-nitrofenyl-beta-d-galakturonid kyselina 2-nitrotoluén-4-sulfónová kyselina 3-(4-brómbenzoyl)-2-(4-chlórfenyl)propiónová kyselina 4-hydroxy-6-metoxy-1-(4-metoxy-fenyl)-naftalén-2-karboxylová kyselina (2-aminotiazol-4-yl)glyoxylová kyselina (+/-)-1 -amino-ŕrans-3-fosfonocyklohexánkarboxylová kyselina n,n’-etylénbis(sukcínamová) kyselina 2,2-difenylmaslová kyselina (s)-4,9-dihydro-1-metyl-3h-pyrido[3,4-b]indol-3-karboxylová kyselina 3,4,5,6-tetrachlór-2',4',5'-trimetylftalanilová kyselina 5-bróm-2-metyl-pyrimidín-4-karboxylová kyselina (4-ho-4-ph-1,3,4,5-4h-2-tia-4a,10-diaza-indeno(2,1-a)inden-3-yl)-octová kyselina (+/-)-1-aminocyklohexán-c/s-1,2-dikarboxylová kyselina 2,3,4,5,6-pentafluórškoricová kyselina 2-(3-chlór-benzoylamino)-3-hydroxy-propiónová kyselina boc-2-aminoizomaslová kyselina n-(2-tiazolyl)glutarámová kyselina 4-(ac-(5-bróm-1,3-dioxo-1,3-dihydro-izoindol-2-ylmetyl)-amino)-benzoová kyselina 2-kyano-3-(2-hydroxyfenyl)propiónová kyselina alfa-(orto-tolyl)-cyklohexánoctová kyselina [etylénbis(oxyetylénnitrilo)]tetraoctová kyselina 4-antracén-2-yl-4-oxo-maslová kyselina 1-(-)-3-fenylmliečna n-chlóracetyl-dehydroalanin • ·· ·· ···· ·*-90 anthraquinone disulfonic acid 4'-bromo-2'-methylglutaranilic acid 2,2'-dithiodibenzoic acid 2,4-difluorophenylacetic acid trifluoromethanesulfonic acid 4-ethenyl-3-methyl-5- (methylthio) thiophene-2-carboxylic acid 2-Bromohexanoic acid 5- (2-Carboxyphenylaminosulfo) -2-chlorobenzoic acid p-Nitrophenyl-beta-d-galacturonide 2-Nitrotoluene-4-sulfonic acid 3- (4-Bromobenzoyl) -2- (4-chlorophenyl) propionic acid 4-Hydroxy-6-methoxy-1- (4-methoxy-phenyl) -naphthalene-2-carboxylic acid (2-aminothiazol-4-yl) glyoxylic acid (+/-) - 1-amino-trans-3-phosphonocyclohexanecarboxylic acid n, n'-ethylenebis (succinamic acid) 2,2-diphenylbutyric acid (s) -4,9-dihydro-1-methyl-3h-pyrido [3,4-b] indole-3-carboxylic acid 3,4 5,6-tetrachloro-2 ', 4', 5'-trimethylphthalanilic acid 5-bromo-2-methyl-pyrimidine-4-carboxylic acid (4-ho-4-ph-1,3,4,5-4h) -2-thia-4α, 10-diaza-indeno (2,1-a) inden-3-yl) -acetic acid (+/-) -1-aminocyclohexane-cis s-1,2-dicarboxylic acid 2,3,4,5,6-pentafluorocinnamic acid 2- (3-chloro-benzoylamino) -3-hydroxy-propionic acid boc-2-aminoisobutyric acid n- (2-thiazolyl) glutaramic acid 4- (ac- (5-Bromo-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl) -amino) -benzoic acid 2-Cyano-3- (2-hydroxyphenyl) propionic acid alpha- (ortho-tolyl) -cyclohexaneacetic acid [ethylenebis (oxyethylenenitrilo)] tetraacetic acid 4-anthracen-2-yl-4-oxo-butyric acid 1 - (-) - 3-phenyl-lactic n-chloroacetyl-dehydroalanine • ·· ·· · ··· · *

9 9 9 9 9 9 99 9 9 9 9

999 999 99..

-91 kyselina 3-(4-fluórfenyl)propiónová kyselina boc-1 -alfa-amino-gama-(4-metylbenzylmerkapto)maslová kyselina 5-sulfo-2,4-chinolíndikarboxylová kyselina c/s-2-(2-tiofénkarbonyl)-1 -cyklohexánkarboxylová kyselina 5-(4-(3-metoxykarbonyl-propyl)-fenyl)-5-oxo-pentánová kyselina c/s-hexahydro-n-(2-metylfenyl)ftalámová kyselina 4-decyloxy-2-fluórbenzoová kyselina fmoc-ŕra/?s-4-(aminometyl)cyklohexánkarboxylová kyselina 4-(4-chlór-benzénsulfonyloxy)-benzoová kyselina 2,3-dibróm-4l-fluórsukcínanilová kyselina stearolová kyselina boc-(3s,4s)-4-amino-3-hydroxy-5-(3-indolyl)-pentánová kyselina dokozahexaénová kyselina 3,5-dibróm-7-metyl-1 -adamantánoctová kyselina 3-(3-(2l2I2-trichlór-1-izobutyrylamino-etyl)-tioureido)-benzoová kyselina 2-heptínová kyselina dnp-d/-alfa-aminokaprylová kyselina (r)-2-(4-hydroxyfenoxy)propánová kyselina 3-(3-(2,2,2-trichlór-1-[(furán-2-karbonyl)-amino]-et)-tioureido)-benzoová kyselina 1 -fenyl-1 -cyklopentánkarboxylová kyselina d/-6,8-ditiooktánová-91 3- (4-Fluorophenyl) propionic acid boc-1-alpha-amino-gamma- (4-methylbenzylmercapto) butyric acid 5-sulfo-2,4-quinolinedicarboxylic acid cis-2- (2-thiophenecarbonyl) 1-Cyclohexanecarboxylic acid 5- (4- (3-methoxycarbonyl-propyl) -phenyl) -5-oxo-pentanoic acid cis-hexahydro-1- (2-methylphenyl) phthalic acid 4-decyloxy-2-fluorobenzoic acid fmoc-trans-4- (aminomethyl) cyclohexanecarboxylic acid 4- (4-chloro-benzenesulfonyloxy) -benzoic acid 2,3-dibromo-4- fluoro- succinilic acid stearic acid boc- (3s, 4s) -4-amino -3-hydroxy-5- (3-indolyl) -pentanoic acid docosahexaenoic acid 3,5-dibromo-7-methyl-1-adamantaneacetic acid 3- (3- ( 2L 2 L 2-trichloro-1-isobutyrylamino-ethyl) 1-Thioureido) -benzoic acid 2-heptinoic acid n 3 -D-.alpha.-aminocaprylic acid (R) -2- (4-hydroxyphenoxy) propanoic acid 3- (3- (2,2,2-trichloro-1- [ (Furan-2-carbonyl) -amino] -ethyl) -thioureido) -benzoic acid 1-Phenyl-1-cyclopentanecarboxy d) -6,8-dithioctanoic acid

3-sulfofenylgama kyselina kyselina 3-chlór-5-trifluórmetyl-2-pyridyltiooctová kyselina 2,3-dimetyl-2-fenyljantárová kyselina d(-)-2-amino-4-fosfonomaslová kyselina 5-ŕerc-butyl-2-metylfurán-3-karboxylová kyselina 1-metionyl-1-asparágová kyselina boc-d-tiazolidín-4-karboxylová, boc-d-tioprolín kyselina s-4-metylmandlová kyselina 4-(trifluórmetyl)cyklohexánkarboxylová kyselina 2,4-dichlór-5-sulfamoyl-benzoová kyselina 5(s),6(r), 15(s)-trihydroxyeikoza-7e,9e, 11 z, 13e-tetraénová3-Sulfophenylgama 3-chloro-5-trifluoromethyl-2-pyridylthioacetic acid 2,3-dimethyl-2-phenylsuccinic acid d (-) - 2-amino-4-phosphonomasic acid 5-tert-butyl-2-methylfuran- 3-carboxylic acid 1-methionyl-1-aspartic acid boc-d-thiazolidine-4-carboxylic acid, boc-d-thioproline s-4-methylmandelic acid 4- (trifluoromethyl) cyclohexanecarboxylic acid 2,4-dichloro-5-sulfamoyl -benzoic acid 5 (s), 6 (r), 15 (s) -trihydroxyeicose-7e, 9e, 11 z, 13e-tetraenoic acid

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · • · · · • • • · · · • ·· • · • · ·· • · • · • · · · • · · · ·· · · • · • · ·· · ·

kyselina 3-(5-oxo-4,5,6>7-tetrahydro-1h-pyrolo(2,3-c)pyridín-3-yl)-propiónová kyselina (4-oktyl-fenoxy)-octová kyselina 4-n-hexylbenzoová kyselina 2-(4,5,6-trihydroxy-3-oxo-3h-xantén-9-yl)-benzoová kyselina ty m í n-1-octová kyselina 4-chlór-3-nitrobenzénsulfónová kyselina n-alfa-boc-n-beta-dnp-1 -diaminopropiónová kyselina 3-hydroxy-4-nitrobenzoová kyselina 3-(3-trifluórmetylbenzyltio)tiofén-2-karboxylová kyselina (r)-(-)-5-oxo-2-tetrahydrofuránkarboxylová kyselina 2-(2-(4-chlórfenyl)-4-fenyltiazol-5-yl)octová kyselina 3-(4-ŕerc-butylbenzyloxy)tiofén-2-karboxylová kyselina rezorcinol-(4-azo-1 )-2-naftol-4-sulfónová kyselina 2-fenoxyfenyloctová kyselina 4-(3-fenylureido)benzoová kyselina 2-(3-fluór-fenyl)-1,3-dioxo-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina 3-(p-hydroxyfenyl)-2-fenylpropiónová kyselina 2-(dimetyltiokarbamoyltio)octová kyselina 5-(p-toluénsulfonyl)merkaptooctová kyselina 2,3-bis-(3,4-dimetoxy-benzylidén)-jantárová kyselina (s)-2-amino-2-metyl-4-fosfonobutánová kyselina 2,3-dihydro-5-(metylsulfinyl)-gama-oxo-(1h)-indolbutánová kyselina 5-brómtiofén-2-karboxylová kyselina 4-amino-3-bróm-naftalén-1-sulfónová kyselina 2-(metoxymetyl)jantárová kyselina 1-leucyl-1-asparágová kyselina 4-aminoazobenzén-3,4,-disulfónová kyselina 2-chlór-6-fluórfenyloctová kyselina 2-cyklohexylidénmaslová kyselina 2-metyl-oktánová kyselina n-oktylfosfónová kyselina 3-dimetylaminobenzoová • ·· ·· ···· ·· ··· · · · · · · • ··· · · · · ·3- (5-oxo-4,5,6> 7-tetrahydro-1 H-pyrrolo (2,3-c) pyridin-3-yl) -propionic acid (4-octyl-phenoxy) -acetic acid 4-n -hexylbenzoic acid 2- (4,5,6-trihydroxy-3-oxo-3h-xanthen-9-yl) -benzoic acid thin-1-acetic acid 4-chloro-3-nitrobenzenesulfonic acid n-alpha- boc-n-beta-dnp-1-diaminopropionic acid 3-hydroxy-4-nitrobenzoic acid 3- (3-trifluoromethylbenzylthio) thiophene-2-carboxylic acid (r) - (-) - 5-oxo-2-tetrahydrofuranecarboxylic acid 2 - (2- (4-chlorophenyl) -4-phenylthiazol-5-yl) acetic acid 3- (4-tert-butylbenzyloxy) thiophene-2-carboxylic acid resorcinol- (4-azo-1) -2-naphthol-4 sulfonic acid 2-phenoxyphenylacetic acid 4- (3-phenylureido) benzoic acid 2- (3-fluorophenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid 3- ( p-hydroxyphenyl) -2-phenylpropionic acid 2- (dimethylthiocarbamoylthio) acetic acid 5- (p-toluenesulfonyl) mercaptoacetic acid 2,3-bis- (3,4-dimethoxybenzylidene) succinic acid (s) -2-amino-2-methyl-4-phosphonobutanoic acid 2,3-dihydro-5- (methylsulfinyl) -gamato-oxo- (1h) -indolbutanoic acid 5-bromothiophene-2-carboxylic acid 4-amino- 3-bromo-naphthalene-1-sulfonic acid 2- (methoxymethyl) succinic acid 1-leucyl-1-aspartic acid 4-aminoazobenzene-3,4 , -disulfonic acid 2-chloro-6-fluorophenylacetic acid 2-cyclohexylideneabutyric acid 2- methyl-octanoic acid n-octylphosphonic acid 3-dimethylaminobenzoic acid 3-dimethylaminobenzoic acid

-93kyselina 3,4-tioféndikarboxylová kyselina 1 -hydroxy-4-(1 -fenyl-1 h-tetrazol-5-yl-tio)-2-naftoová kyselina n-acetylneuramínová kyselina (-)-dibenzoyl-l-vínna kyselina 2-(2-metyl-1 -fenylpropyl)benzoová kyselina 8-metyl-naftalén-1 -karboxylová kyselina 4-(4-bróm-2,5-dimetoxyfenyl)maslová kyselina 2-chlór-4-hydroxybenzoová kyselina 2-chlór-3-metylbenzoová kyselina (4,4-dimetyl-3,7-dioxo-2,3,4,5,6,7-hexahydro-1 h-indén-1 -yl)-octová kyselina 2,3-dihydro-4-etoxyftalová kyselina 2-(trifluórmetyl)-1,6-naftyridín-3-karboxylová kyselina 1-pyrénhexánová kyselina 2-metoxy-4-(metyltio)benzoová kyselina n-acetyl-1-glutamín kyselina 2,4-pentadekadiínová kyselina 2-(2-hydroxyimino-propionylamino)-jantárová kyselina 5-antracén-9-yl-pentánová kyselina n-(2,3-dimetylfenyl)- 12,3,6-tetrahydroftalámová kyselina 2-hydroxy-3(s)-(n-terc-boc-amino)-4-fenylbutánová kyselina 3,3-dichlór-2-fluór-propiónová kyselina 5-bróm-2-metoxyfenyloctová kyselina 2-aminoetylfosfónová kyselina 4'-n-decyloxybifenyl-4-karboxylová kyselina c/s-5-eikozénová kyselina 2-hydroxyamino-4-metyl-pentánová kyselina 4-chlór-3,5-dinitrofenyloctová kyselina 8-(3-oxo-4,5,6-trihydroxy-3h-xantén-9-yl)-1 -naftoová kyselina n-acetyl-1-glutámová kyselina 10,12-pentakozadiínová kyselina tricyklo( 11.2.2.2(5,8))nonadeka-hexaén-7-karboxylová kyselina 4-fluórfenoxyoctová-93-3,4-thiophenedicarboxylic acid 1-hydroxy-4- (1-phenyl-1H-tetrazol-5-yl-thio) -2-naphthoic acid n-acetylneuraminic acid (-) - dibenzoyl-1-tartaric acid 2 - (2-methyl-1-phenylpropyl) benzoic acid 8-methyl-naphthalene-1-carboxylic acid 4- (4-bromo-2,5-dimethoxyphenyl) butyric acid 2-chloro-4-hydroxybenzoic acid 2-chloro-3 -methyl-benzoic acid (4,4-dimethyl-3,7-dioxo-2,3,4,5,6,7-hexahydro-1H-inden-1-yl) -acetic acid 2,3-dihydro-4- 2- (trifluoromethyl) -1,6-naphthyridine-3-carboxylic acid ethoxyphthalic acid 1-pyrene-hexanoic acid 2-methoxy-4- (methylthio) benzoic acid n-acetyl-1-glutamine 2,4-pentadecadiic acid 2- ( 2-hydroxyimino-propionylamino) -succinic acid 5-anthracen-9-yl-pentanoic acid n- (2,3-dimethylphenyl) -12,3,6-tetrahydrophthalic acid 2-hydroxy-3 (s) - (n-tert-butyl) -boc-amino) -4-phenylbutanoic acid 3,3-dichloro-2-fluoro-propionic acid 5-bromo-2-methoxyphenylacetic acid 2-aminoethylphos phonic acid 4'-n-decyloxybiphenyl-4-carboxylic acid cis-5-eicosenoic acid 2-hydroxyamino-4-methylpentanoic acid 4-chloro-3,5-dinitrophenylacetic acid 8- (3-oxo-4, 5,6-trihydroxy-3h-xanthen-9-yl) -1-naphthoic acid n-acetyl-1-glutamic acid 10,12-pentacosadioic acid tricyclo (11.2.2.2 (5,8)) nonadeca-hexaen-7- 4-fluorophenoxyacetic acid carboxylic acid

• ·· • ·· 99 99 ···· ···· ·· · · • · • · 9 9 9 9 9 9 • ··· • ··· 9 9 • · · • · · 9 9 • · • · 9 9 ·· ·· ·· ·· 99 99 ·· · · 99 99

kyselina 2,3-difenylakrylová kyselina n-(2,4-difluórfenyl)malónová kyselina 5h-perfluórpentánová kyselina behenová kyselina 4-(2-nitro-fenylsulfanylamino)-benzoová kyselina 2-hexyldekánová kyselina n-íerc-boc-1 -alfa-aminoadipová kyselina beta-brómangeliková kyselina 4,5-dihydroxy-2-metylbenzoová kyselina (-)-kamfanová kyselina evernová kyselina 5,6,7-trimetoxy-3,4-dihydro-naftalén-2-karboxylová kyselina 2,4-nonadekadiínová kyselina 2-[3-oxo-3-(n’-pentanoyl-hydrazíno)-propionylamino]-benzoová kyselina 4-(3-(2-chlór-6-metylfenyl)ureido)salicylová kyselina 3-o-tolyl-but-2-énová kyselina alfa-(ŕerc-butyl)hydroškoricová kyselina 3,5-dimetyl-4-hydroxybenzoová kyselina 3,4-dimetoxyfenyloctová kyselina 3-hydroxypropiónová kyselina n-decylmaleámová kyselina 2-(2-metoxyfenyl)-1 -metyl-6-oxo-3-piperidínkarboxylová kyselina 5-aminoazelainová kyselina 5-formyl-2-furánkarboxylová kyselina 4-alyl-2,3,5,6-tetrafluórbenzoová kyselina 2’,5'-dichlórftalanilová kyselina 3'-hydroxyhexahydroftalanilová kyselina 2-butoxy-3-nitrosalicylová kyselina 4'-butyl-bifenyl-4-karboxylová kyselina 3-benzo[1,3]dioxol-5-yl-2-benzoylamino-propiónová kyselina 3,4-dimetoxy-ftalová kyselina 2-ketopimelová2,3-diphenylacrylic acid n- (2,4-difluorophenyl) malonic acid 5h-perfluoropentanoic acid behenic acid 4- (2-nitro-phenylsulfanylamino) -benzoic acid 2-hexyldecanoic acid n-tert-boc-1-alpha- amino-adipic acid beta-bromoanonic acid 4,5-dihydroxy-2-methylbenzoic acid (-) - camphoric acid evernic acid 5,6,7-trimethoxy-3,4-dihydro-naphthalene-2-carboxylic acid 2,4-nonadecadioic acid 2- [3-oxo-3- (n'-pentanoyl-hydrazino) -propionylamino] -benzoic acid 4- (3- (2-chloro-6-methylphenyl) ureido) salicylic acid 3-o-tolyl-but-2 -enic acid alpha- (tert-butyl) cinnamic acid 3,5-dimethyl-4-hydroxybenzoic acid 3,4-dimethoxyphenylacetic acid 3-hydroxypropionic acid n-decylmaleamic acid 2- (2-methoxyphenyl) -1-methyl-6- oxo-3-piperidinecarboxylic acid 5-aminoazelaic acid 5-formyl-2-furancarboxylic acid 4-allyl-2,3,5,6-tetrafluorobenzoic acid 2 ', 5'-dichlorophthalate ilic acid 3'-hydroxyhexahydrophthalanic acid 2-butoxy-3-nitrosalicylic acid 4'-butyl-biphenyl-4-carboxylic acid 3-benzo [1,3] dioxol-5-yl-2-benzoylamino-propionic acid 3,4- dimethoxyphthalic acid 2-ketopimelic acid

·· · · • e • e ···· ···· • e • e • « • « ··· · · · • · • · • · • · • ·· • ·· • e • e ·· · · ·· · · « «

kyselina n2-fmoc-n4-boc-1 -2,4-diaminomaslová kyselina pyrogalol-4-karboxylová kyselina 4-(1-brómetyl)benzoová kyselina 5-hexínová kyselina ŕrans-vakcénová kyselina 3-hydroxy-2-naftoová kyselina 3,6-dichlór-2-hydroxy-benzoová kyselina 3-(4-fenoxybenzoyl)propiónová kyselina lekanorová kyselina 5-(4-fltiórfenyl)valérová kyselina 2-(4-(4-benzyloxy)fenylsulfonyl)fenoxy)maslová kyselina 3-(4-hydroxymetylfenoxy)propiónová pyridoxal-5-fosfát kyselina 2-(2-metoxykarbonyl-etylamino)-benzoová kyselina 3,4,5-trifluórbenzoová kyselina 2,3-pyridíndikarboxylová kyselina 2,6-dimetyl-tereftalámová kyselina 4-(4-(3-metyl-3h-benzotiazol-2-ylidén)-but-2-énylidénamino)-benzoová kyselina 2-fluór-4-izo-propoxybenzoová kyselina o-propionylbenzoová kyselina tricyklo(16.2.2.2(8,11 ))tetrakoza-hexaén-9-karboxylová kyselina fmoc-ŕrans-3-fenylazetidín-2-karboxylová kyselina (+/-)-1-aminocyklopentán-ŕrans-1,3-dikarboxylová kyselina (r)-(+)-2-(fenylkarbamoyloxy)propiónová kyselina benzoylsulfanyl-octová kyselina fmoc-aV-alfa-aminomaslová kyselina 1 -aminocyklobután-frans-13-dikarboxylová kyselina 2,4-difenylpyrimidín-5-karboxylová kyselina 3-(3-hydroxyfenyl)propiónová kyselina 7-hydroxy-13-naftaléndisulfónová kyselina /?-alfa-z-4-amino-maslová kyselina 2,3,5-trifluórškoricová • ·· ·· ···· ·· ·· · · · · · · · • ··· · · · · tn2-fmoc-n4-boc-1 -2,4-diaminobutyric acid pyrogalol-4-carboxylic acid 4- (1-bromomethyl) benzoic acid 5-hexanoic acid trans-vaccenoic acid 3-hydroxy-2-naphthoic acid 3, 6-Dichloro-2-hydroxy-benzoic acid 3- (4-phenoxybenzoyl) propionic acid Lecanic acid 5- (4-fluorophenyl) valeric acid 2- (4- (4-benzyloxy) phenylsulfonyl) phenoxy) butyric acid 3- (4 -hydroxymethylphenoxy) propionic pyridoxal-5-phosphate 2- (2-methoxycarbonyl-ethylamino) -benzoic acid 3,4,5-trifluorobenzoic acid 2,3-pyridinedicarboxylic acid 2,6-dimethyl-terephthalic acid 4- (4- ( 3-Methyl-3h-benzothiazol-2-ylidene) -but-2-phenyleneamino) -benzoic acid 2-fluoro-4-iso-propoxybenzoic acid o-propionylbenzoic acid tricyclo (16.2.2.2 (8,11)) tetracos-hexaene -9-carboxylic acid fmoc-trans-3-phenylazetidine-2-carboxylic acid (+/-) -1-aminocyclopentane-trans-1,3-dicarboxylic acid (r) - (+) - 2- (phenylcarbamoyloxy) propiones Benzoylsulfanyl-acetic acid fmoc-N-alpha-aminobutyric acid 1-Aminocyclobutane-trans-13-dicarboxylic acid 2,4-diphenylpyrimidine-5-carboxylic acid 3- (3-hydroxyphenyl) propionic acid 7-hydroxy-13-naphthalenedisulfonic acid β-alpha-z-4-amino-butyric acid 2,3,5-trifluorocinnamic acid · t · · · t · t · t · t · t

-96kyselina beta-hydroxypyrohroznová kyselina ftalidénoctová kyselina 2-metylimidazol-4-karboxylová kyselina 9,10-dihydro-9,10-etanoantracén-11,12-dikarboxylová kyselina 3I3-dichlór-2-(4-chlór-benzoylamino)-akrylová kyselina 3-bróm-[3-(4-chlórbenzoyl)propiónová kyselina 2-(4-(3-(5-chlór-2,4-dimetoxyfenyl)ureido)fenyltio)octová kyselina 3-metyl-1-oxo-1 h-izochromén-4-karboxylová kyselina 2-[(4-metoxykarbonyl)fenoxymetyl]benzoová kyselina 4-bróm-2I3,5,6-tetrafluórbenzoová kyselina 2-metyl-3-buténová kyselina ((2-hydroxy-benzylidén)-amino)-fenyl-octová kyselina 2,5-dimetyltereftalová kyselina bis-(hydroxymetyl)-fosfínová kyselina 5-jódsalicylová kyselina (2,4-dimetoxy-fenyl)-octová kyselina 3-(4-chlórbenzoyl)-2-(4-chlórfenyl)propiónová kyselina 4-(6-hexyloxy-naftalén-2-yl)-maslová kyselina pth-asparágová kyselina 2-amino-6-fluórbenzoová kyselina 2l2',2,, I2,-(1,2-etán-diylidén-tetrakis[tio])-tetrakis-octová kyselina n-acetyl-1-asparágová kyselina 3-(hexadecyloxy)benzoová kyselina fmoc-d-beta-aminomaslová kyselina 1 -diazo-2-hydroxy-5-nitronaftalén-4-sulfónová kyselina n-alfa-chlóracetyl-1 -glutámová kyselina 1 -fenyl-1 -cyklopropánkarboxylová kyselina 3,4-difluórhydroškoricová kyselina (3-ho-3-ph-2,3,5,6,7,8-6h-benzo(4,5)imidazo(2,1-b)tiazol-2-yl)-octová (r)-cbz-oxaprolín kyselina (1 s,3s)-1 -aminocyklopentán-1,3-dikarboxylová kyselina boe- ŕrans-4-(aminometyl)cyklohexánkarboxylová • ·· ·· ···· ·· ··· · · ···· • ··· · · · · ·-96kyselina beta-hydroxypyruvic acid ftalidénoctová acid 2-methylimidazole-4-carboxylic acid, 9,10-dihydro-9,10-ethanoanthracene-11,12-dicarboxylic acid 3 I, 3-dichloro-2- (4-chloro-benzoylamino) - Acrylic acid 3-bromo- [3- (4-chlorobenzoyl) propionic acid 2- (4- (3- (5-chloro-2,4-dimethoxyphenyl) ureido) phenylthio) acetic acid 3-methyl-1-oxo-1 h-isochromene-4-carboxylic acid 2 - [(4-methoxycarbonyl) phenoxymethyl] benzoic acid 4-bromo-2 L 3,5,6-tetrafluorobenzoic acid 2-methyl-3-butenoic acid ((2-hydroxy-benzylidene) -amino) -phenyl-acetic acid 2,5-dimethylterephthalic acid bis- (hydroxymethyl) -phosphinic acid 5-iodosalicylic acid (2,4-dimethoxyphenyl) -acetic acid 3- (4-chlorobenzoyl) -2- (4 chlorophenyl) propionic acid 4- (6-hexyloxy-naphthalen-2-yl) -butyric acid pth-aspartic acid 2-amino-6-fluorobenzoic acid, 2 l 2 ', 2 ,, I 2 - (1,2- ethane-diylidene-tetrakis [thio]) - tetrakis-acetic acid n-acetyl-1-aspartate 3- (hexadecyloxy) benzoic acid fmoc-d-beta-aminobutyric acid 1-diazo-2-hydroxy-5-nitronaphthalene-4-sulfonic acid n-alpha-chloroacetyl-1-glutamic acid 1-phenyl-1-cyclopropanecarboxylic acid 3,4-difluorocinnamic acid (3-ho-3-ph-2,3,5,6,7,8-6h-benzo (4,5) imidazo (2,1-b) thiazol-2-yl) -acetic (r) -cbz-oxaproline (1s, 3s) -1-aminocyclopentane-1,3-dicarboxylic acid bo-trans-4- (aminomethyl) cyclohexanecarboxylic acid • ·· ·· ········ · · · ··· · ··· · · · · ·

-97kyselina 2,2-dichlórcyklopropán-karboxylová kyselina (4-chlórfenyl)fosfónová kyselina 2,5-dichlór-3-nitrobenzoová kyselina 2-acetamidoakrylová kyselina 1-glutámová kyselina 3-(4-brómbenzoyl)-akrylová kyselina 3,5-dibróm-4-metylbenzoová kyselina 5-amino-n-(2,3-dihydroxy-1 -propyl)izoftalámová kyselina 3-benzoyl-2-tiofénkarboxylová kyselina d-homocysteínová kyselina 3,4-furándikarboxylová kyselina 2-(3,4-dimetoxyfenyl)-1-metyl-5-oxopyrolidín-3-karboxylová kyselina me-tricyklo(8.2.2.2(4,7))hexadeka-1 (13),4,6,10(14),11,15-hexaén-karboxylová kyselina 1 -fenylalanyl-1 -glutámová kyselina 6,6,7,7-tetrafluór-bicyklo(3.2.0)heptán-2,4-dikarboxylová kyselina n-glykolylneuramínová kyselina 6,15-dioxo-1,20-eikozándikarboxylová kyselina 1-benzyl-5-oxo-3-pyrolidínkarboxylová kyselina 2'-kyanoglutaranilová kyselina (z)-3-[(aminoiminometyl)tio]prop-2-énová kyselina dicyklopentadién-dikarboxylová kyselina 4-heptylbenzoová kyselina o-etylbenzoová kyselina (1s,3r)-1-aminocyklopentán-1,3-dikarboxylová kyselina 5-fenyl-2,3-dihydro-1 h-pyrolizín-6,7-dikarboxylová kyselina 3-(2-naftyltio)propiónová kyselina 4-((2-hydroxy-benzylidén)-amino)-benzoová kyselina 2-(hexadecyloxy)škoricová kyselina d/-alfa-hydroxykaprónová kyselina trikarbalylová kyselina 3-metyl-4-oxo-2-penténová-97 2,2-dichlorocyclopropanecarboxylic acid (4-chlorophenyl) phosphonic acid 2,5-dichloro-3-nitrobenzoic acid 2-acetamidoacrylic acid 1-glutamic acid 3- (4-bromobenzoyl) -acrylic acid 3,5-dibromo 4-methylbenzoic acid 5-amino-N- (2,3-dihydroxy-1-propyl) isophthalic acid 3-benzoyl-2-thiophenecarboxylic acid d-homocysteic acid 3,4-furanedicarboxylic acid 2- (3,4-dimethoxyphenyl) ) -1-methyl-5-oxopyrrolidine-3-carboxylic acid methicyclo (8.2.2.2 (4,7)) hexadeca-1 (13), 4,6,10 (14), 11,15-hexaenecarboxylic acid 1-phenylalanyl-1-glutamic acid 6,6,7,7-tetrafluorobicyclo (3.2.0) heptane-2,4-dicarboxylic acid n-glycolylneuraminic acid 6,15-dioxo-1,20-eicosandicarboxylic acid 1 -benzyl-5-oxo-3-pyrrolidinecarboxylic acid 2'-cyanoglutaranilic acid (z) -3 - [(aminoiminomethyl) thio] prop-2-enoic acid dicyclopentadiene-dicarboxylic acid 4-heptylbenzoic acid o-ethylbenzoic acid (1s, 3r) -1-Aminocyclopentane-1,3-dicarboxylic acid 5-phenyl-2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid 3- (2-naphthylthio) propionic acid 4 - (( 2-hydroxy-benzylidene) -amino) -benzoic acid 2- (hexadecyloxy) cinnamic acid d-alpha-hydroxycaproic acid tricarbalyl 3-methyl-4-oxo-2-pentenoic acid

-98• ·· ·· ·» ·· · kyselina (1,4-dioxa-spiro(4,5)dec-6-yl)-octová kyselina fenylmalónová kyselina n-(4-etoxyfenyl)maleámová kyselina tiazolidín-2,4-dikarboxylová kyselina 4-(3-bróm-propoxy)-benzoová kyselina n-(3-acetylfenyl)glutarámová kyselina 3-bróm-4-chlórbenzoová kyselina 4-chlór-alfa-metylškoricová kyselina 2-benzamido-3-metoxy-3-fenylpropiónová kyselina 2-etyl-3-(3-hydroxy-fenyl)-akrylová kyselina c/s-4,7,10,13,16,19-dokozahexaénová kyselina (r)-(+)-2-bróm 3-metylbutánová kyselina 2,6-dichlór-3-nitrobenzoová kyselina (s)-(-)-n-(1 -fenyletyl)ftalámová kyselina 2-fluór-5-(trifluórmetyl)fenyloctová kyselina 2,2-difenylheptánová kyselina 4-amino-4'-metoxydifenylamín-2-sulfónová kyselina 6,6-dimetyl-3-oxo-bicyklo(2.2.2)oktán-2-karboxylová kyselina 2,-(trifluórmetyl)ftalanilová kyselina 2-(4-ferc-butyl-benzoylamino)-benzoová kyselina beta-metyl-3-nitrohydroškoricová kyselina 7a-metánsulfonylacetyl-3,6-dioxooktahydro-indén-1-karboxylová kyselina alfa-chlór-2-norbornánoctová kyselina 4-(3,4-dihydro-4-oxo-1,2,3-benzotriazín-3-yl)fenyloctová kyselina fmoc-9-aminononánová kyselina dietylfosfonopropánová kyselina metyliminodioctová kyselina 3-endo-aminobicyklo[2.2.1 ]hept-5-én-2-endo-karboxylová kyselina 3-jód-4-hydroxybenzoová kyselina 1 h-dibenz(a,kl)-7-antracenón-13-karboxylová kyselina 4,4,4-trifluór-3-(4-metoxy-naftalén-1 -yl)-but-2-énová kyselina 3-(4-metoxy-febyl)-3-(4-metyl-benzoylamono)-propiónová(1,4-dioxa-spiro (4,5) dec-6-yl) -acetic acid phenyl malonic acid n- (4-ethoxyphenyl) maleic acid thiazolidin-2 -98; 4-Dicarboxylic acid 4- (3-bromo-propoxy) -benzoic acid n- (3-acetylphenyl) glutaramic acid 3-bromo-4-chlorobenzoic acid 4-chloro-alpha-methylcinnamic acid 2-benzamido-3-methoxy-3 -phenylpropionic acid 2-ethyl-3- (3-hydroxy-phenyl) -acrylic acid cis-4,7,10,13,16,19-docosahexaenoic acid (r) - (+) - 2-bromo 3- methylbutanoic acid 2,6-dichloro-3-nitrobenzoic acid (s) - (-) - n- (1-phenylethyl) phthalic acid 2-fluoro-5- (trifluoromethyl) phenylacetic acid 2,2-diphenylheptanoic acid 4-amino- 4'-metoxydifenylamín-2-sulfonic acid 6,6-dimethyl-3-oxo-bicyclo (2.2.2) octane-2-carboxylic acid 2, - (trifluoromethyl) ftalanilová 2- (4-tert-butyl-benzoylamino) -benzoic acid beta-methyl-3-nitrohydrocinnamic acid 7α-methanesulfonylacetyl-3,6-dioxooctahydro-inden-1-ka 4- (3,4-dihydro-4-oxo-1,2,3-benzotriazin-3-yl) phenylacetic acid fmoc-9-aminononanoic acid diethylphosphonopropanoic acid methyliminodioacetic acid alpha-chloro-2-norboronic acetic acid -aminobicyclo [2.2.1] hept-5-ene-2-endo-carboxylic acid 3-iodo-4-hydroxybenzoic acid 1 h-dibenz (a, kl) -7-anthracenone-13-carboxylic acid 4,4,4 -trifluoro-3- (4-methoxy-naphthalen-1-yl) -but-2-enoic acid 3- (4-methoxy-phenyl) -3- (4-methyl-benzoylamono) -propionic acid

• · · • 8 • ··· 8 • ··· 88 8888 9 · · 8 8 8 88 8888 9 · · 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 88 88 88 88 • 8 88 8 88 88 88 88 88

kyselina 2-fluór-4-(trifluórmetyl)benzoová kyselina 3-metyladipová kyselina 4-(2-metoxy-fenyl)-maslová kyselina 4-metylsalicylová kyselina 2-metoxy-2-fenyl-propiónová kyselina 4-(2-chlór-1,1,2-trifluóretoxy)-benzoová kyselina 2-oxo-1 -fenylpyrolidin-4-karboxylová kyselina beta-karboxyasparágová kyselina 2-(1 -fenyl-2,2,2-trifliióretoxy)octová kyselina 1 -((1,1 -dimetyletoxy)karbonyl)-4-piperidínoctová kyselina 11 (s), 12(s)-epoxy-13(s)-hydroxy-9z-oktadecénová kyselina 3-nitropropiónová kyselina 2-(2-hydroxy-fenyl)-tiazolidín-4-karboxylová kyselina 3-karboxy-1,2,2-trimetylcyklopentánakrylová kyselina 4-{2-hydroxy-fenyl)-maslová kyselina fenyloctová kyselina 9,10-dihydroxystearová kyselina 7-dimetylaminokiimarín-4-octová kyselina (4-hydroxy-3-sulfo-fenylamino)-octová kyselina r-ftalimido-alfa-hydroxy-n-maslová kyselina n-(4-fluórfenyl)maleámová kyselina 4-[[4-[(4,6-dimetylpyrimidín-2-yl)pxy]fenyl]amino]-2-metyl-4-oxo-(2z)-buténová kyselina (2-metoxyfenyl)fosfónová kyselina 3'-nitroftalanilová kyselina indol-3-jantárová kyselina d/-2-amino-7-fosfonoheptánová kyselina 5-sulfoantronilová kyselina 3-(2-oxocyklododecyl)propiónová kyselina 19-metyleikozánová kyselina 3-(3-metylfenyl)propiónová kyselina 7-etyl-3-oxo-2-aza-bicyklo(2.2.2)oktán-6-karboxylová2-fluoro-4- (trifluoromethyl) benzoic acid 3-methyladipic acid 4- (2-methoxyphenyl) butyric acid 4-methylsalicylic acid 2-methoxy-2-phenylpropionic acid 4- (2-chloro-1) 1,2-trifluoroethoxy) -benzoic acid 2-oxo-1-phenylpyrrolidine-4-carboxylic acid beta-carboxyaspartic acid 2- (1-phenyl-2,2,2-trifluoroethoxy) acetic acid 1 - ((1,1 (dimethylethoxy) carbonyl) -4-piperidineacetic acid 11 (s), 12 (s) -epoxy-13 (s) -hydroxy-9z-octadecenic acid 3-nitropropionic acid 2- (2-hydroxy-phenyl) -thiazolidin-4 -carboxylic acid 3-carboxy-1,2,2-trimethylcyclopentanacrylic acid 4- (2-hydroxy-phenyl) -butyric acid 9,10-dihydroxystearic acid 7-dimethylaminociimarin-4-acetic acid (4-hydroxy-3- sulfo-phenylamino) -acetic acid r-phthalimido-alpha-hydroxy-n-butyric acid 4- (4-fluorophenyl) maleic acid 4 - [[4 - [(4,6-dimethylpyrimidin-2-yl) pxy] phenyl] amino] -2-methyl-4-oxo- (2z) -butyric acid (2-methoxy) phenyl) phosphonic acid 3'-nitropthalanic acid indole-3-succinic acid d / -2-amino-7-phosphonoheptanoic acid 5-sulfoantronic acid 3- (2-oxocyclododecyl) propionic acid 19-methylicosanoic acid 3- (3-methylphenyl) Propionic acid 7-ethyl-3-oxo-2-aza-bicyclo (2.2.2) octane-6-carboxylic acid

-100--100-

• ·· • · • III • ·· • · • III • · • B B B B B B • BBB • A • BBB • A BB • · • · BB • · • · ·· · · ·· ·· ·· ·· • B • B • · • · BB BB • B • B

kyselina n-(1 -cyklopropyl-etyl)-n-fenyl-sukcínamová kyselina (r)-1 -amino-(3-metylbután)fosfónová kyselina 3-naftalén-2-yl-propínová kyselina propiónová kyselina 1 -(4-metoxyfenyl)-1 -cyklohexánkarboxylová kyselina malónová kyselina izodehydroctová kyselina /7-alfa-(benzyloxykarbonyl)-d-glutámová kyselina n-(3,4-xylyl)ftalámová kyselina 8-amino-5-(4-hydroxy-fenylamino)-naftalén-2-sulfónová kyselina pentametylbenzoová kyselina n-acetyl-8-hydroxy-1 -naftylamín-3,6-disulfónová kyselina 2-(2-chlóracetamido)-4-tiazoloctová kyselina (4-etyl-fenoxy)-octová kyselina 3-(4-chlórbenzoyl)propiónová kyselina p-chlórfenyl-izovalérová kyselina 3,3-dichlór-cyklopropán-1,2-dikarboxylová kyselina n-(2-bróm-4-nitro-fenyl)-ftalámová kyselina 1 (+)-2-amino-4-fosfonomaslová kyselina bicyklo(2.2.2)okt-5-én-2,3-dikarboxylová kyselina 2-chlór-5-nitroškoricová kyselina 3-(3-benzyloxy-4,5-dimetoxy-fenyl)-akrylová kyselina 5-bróm-2-metoxyškoricová kyselina 3-(4-karboxyfenyl)propiónová kyselina metylfosfónová kyselina 2-metyl-3-fenyljantárová kyselina boc-(3s,4s)-4amino-3-hydroxy-5-(4-benzyloxyfenyl)-pentánová kyselina n-alfa-(benzyloxykarbonyl)-alfa-(benzylester)-1-glutámová kyselina (s)-(+)-2-(4-bifenylyl)propiónová kyselina 4-hexadecyloxy-3-metoxyškoricová kyselina 6-benzoylhexánová kyselina 3-nitro-4-trifluórmetyl-benzoován- (1-cyclopropyl-ethyl) -n-phenyl-succinamic acid (r) -1-amino- (3-methylbutane) phosphonic acid 3-naphthalen-2-yl-propionic acid propionic acid 1- (4-methoxyphenyl) -1-Cyclohexanecarboxylic acid Malonic acid Isodehydroacetic acid / 7-alpha- (Benzyloxycarbonyl) -d-glutamic acid N- (3,4-xylyl) phthalic acid 8-amino-5- (4-hydroxy-phenylamino) -naphthalene- 2-sulfonic acid pentamethylbenzoic acid n-acetyl-8-hydroxy-1-naphthylamine-3,6-disulfonic acid 2- (2-chloroacetamido) -4-thiazoleacetic acid (4-ethyl-phenoxy) -acetic acid 3- (4 -chlorobenzoyl) propionic acid p-chlorophenyl-isovaleric acid 3,3-dichloro-cyclopropane-1,2-dicarboxylic acid 1- (2-bromo-4-nitro-phenyl) -phthalic acid 1 (+) - 2-amino- 4-Phosphonomyric acid bicyclo (2.2.2) oct-5-ene-2,3-dicarboxylic acid 2-chloro-5-nitrocinnamic acid 3- (3-benzyloxy-4,5-dimethoxyphenyl) -acrylic acid 5- Bromo-2-methoxycinnamic acid 3- (4- carboxyphenyl) propionic acid methylphosphonic acid 2-methyl-3-phenylsuccinic acid boc- (3s, 4s) -4amino-3-hydroxy-5- (4-benzyloxyphenyl) -pentanoic acid n-alpha- (benzyloxycarbonyl) -alpha- (benzyl ester) ) -1-glutamic acid (s) - (+) - 2- (4-biphenylyl) propionic acid 4-hexadecyloxy-3-methoxycinnamic acid 6-benzoylhexanoic acid 3-nitro-4-trifluoromethyl-benzoic acid

• · · 8 * • ··· • · · 8 * • ··· ·· ···· • · · • 8 8 ·· ···· · · · • 8 8 88 « • 8 88 • 8 · 88 «• • 8 · • · ·· • · ·· ·· 88 ·· 88 88 88 88 88

- 101 kyselina 3-vinylbenzoová kyselina izopropylmalónová kyselina 2,2-bis(trifluórmetyl)-2-hydroxyoctová kyselina r(+)-2-(4-chlór-2-metyl fenoxy) propiónová kyselina 5-(3-metoxy-fenyl)-hexánová kyselina 4-trifluórmetyl-2-aminobenzoová kyselina 4-(4-metoxyfenyl)maslová kyselina tetrafluór-izoftalová kyselina 2-antracén-1 -yl-propiónová kyselina 2,2-difluórbenzodioxol-5-karboxylová kyselina 2-(3,5-dinitro-tiofén-2-ylamino)-4-metyl-pentánová kyselina [2-(4-chlórbenzénsulfonyl)etyltio]octová kyselina 3-metoxypropiónová kyselina 9,10-epitio-oktadekánová kyselina 4-(2-(3,4-dimetyl-fenoxy)-acetylamino)-benzoová kyselina 3-benzoylbenzoová kyselina 4,4,5,5,6,6,7,7,8,8,9,9,9-tridekafluórnonánová kyselina 3-metylpentánová kyselina 6-metoxy-2-naftalénškoricová kyselina 14-br-tricyklo(8.2.2.2(4,7))hexadeka-hexaén-5-karboxylová kyselina 3-(4-metoxy-2,3-dimetyl-fenyl)-propiónová kyselina 3-(2,2-dimetylpropiónamido)benzoová kyselina 3-(2,4I6-trimetyl-fenyl)-akrylová kyselina (2,4,6-trimetylfenyl)fosfónová kyselina (+/-)5-hydroxyeikoza-6e,8z,11z,14z-tetraénová kyselina 5-[2-chlór-4-(trifluórmetyl)-fenoxy]-2-nitrobenzoová kyselina 5-fluór-6-hydroxy-2-metyl-pyrimidin-4-karboxylová kyselina n-(2-hydroxyetyl)iminodioctová kyselina 2-(benzoyloxymetyl)benzoová kyselina 4-(3,4-(metyléndioxy)benzylidénamino)salicylová kyselina 5-(2-brómbenzoyl)pentánová kyselina 1,4,4a,5,8,8a-hexahydro-5-hydroxy-8-oxo-1 -naftalénkarboxylová101 101 3-vinylbenzoic acid isopropylmalonic acid 2,2-bis (trifluoromethyl) -2-hydroxyacetic acid r (+) - 2- (4-chloro-2-methylphenoxy) propionic acid 5- (3-methoxyphenyl) -hexanoic acid 4-trifluoromethyl-2-aminobenzoic acid 4- (4-methoxyphenyl) butyric acid tetrafluoro-isophthalic acid 2-anthracen-1-yl-propionic acid 2,2-difluorobenzodioxole-5-carboxylic acid 2- (3,5 -Dinitro-thiophen-2-ylamino) -4-methyl-pentanoic acid [2- (4-chlorobenzenesulfonyl) -ethylthio] -acetic acid 3-methoxy-propionic acid 9,10-epithio-octadecanoic acid 4- (2- (3,4- dimethyl-phenoxy) -acetylamino) -benzoic acid 3-benzoylbenzoic acid 4,4,5,5,6,6,7,7,8,8,9,9,9-tridecafluorononic acid 3-methylpentanoic acid 6-methoxy- 2-Naphthalenic cinnamic acid 14-br-tricyclo (8.2.2.2 (4,7)) hexadeca-hexaene-5-carboxylic acid 3- (4-methoxy-2,3-dimethyl-phenyl) -propionic acid 3- (2, 2-dimethylpropionamido) benzoic acid 3- (2,4 L 6-trimethyl-phe) nyl) -acrylic acid (2,4,6-trimethylphenyl) phosphonic acid (+/-) 5-hydroxyeicoza-6e, 8z, 11z, 14z-tetraenoic acid 5- [2-chloro-4- (trifluoromethyl) phenoxy] 2-nitrobenzoic acid 5-fluoro-6-hydroxy-2-methyl-pyrimidine-4-carboxylic acid n- (2-hydroxyethyl) iminodiacetic acid 2- (benzoyloxymethyl) benzoic acid 4- (3,4- (methylenedioxy) benzylideneamino Salicylic acid 5- (2-bromobenzoyl) pentanoic acid 1,4,4a, 5,8,8a-hexahydro-5-hydroxy-8-oxo-1-naphthalenecarboxylic acid

-102 --102 -

9 99 9 99 99 9999 99 9999 ·· · · 9 9 9 9 • · • · 9 * 9 * 99 99 9 999 9 999 • 9 • 9 4 9 4 9 99 9 9 99 9 9 • 4 • 4 • 4 • 4 99 99 99 99

kyselina n-( 1 -naftyl)-6-nitroftalámová kyselina 3-(2,4,6-trimetylbenzoyl)-2-bifenylkarboxylová kyselina (+/-)-erytro-3-metylglutámová kyselina 5-metoxybenzofurán-2-karboxylová kyselina 2-imino-4-oxytiazol-5-octová kyselina 2-(trifluórmetyl)-2-hydroxypropiónová kyselina brómpivalová kyselina cyklopropánkarboxylová kyselina cyklopropán-1,2,3-trikarboxylová kyselina 7-oxo-8-nonénová kyselina nonakozánová kyselina 4-(4-brómbenzoyl)pentánová kyselina 2',4',6,-trimetylftalanilová kyselina 1-metyl-2-oxo-1,2-dihydrochinoxalín-3-propiónová kyselina tribrómoctová kyselina (3-acetyl-2-metyl-5-oxo-2-pyrolín-4-yl)-octová kyselina 4-ŕerc-butylbenzoová kyselina c/s-n-(2-fluórfenyl)hexahydroftalámová kyselina fmoc-4-aminobenzoová kyselina 2-(2-chlóracetamido)benzoová acetyl-asp-glu-oh kyselina laktobiónová kyselina 1 -brómcyklohexánkarboxylová kyselina 2-metyl-2-naftalén-1 -ylmetyl-malónová kyselina 2-(4-izopropyl-benzylidén)-pent-4-énová kyselina 2,-metoxy-3,4,5,5',6-pentachlórftalanilová kyselina 2-(cinamylidén)-2-fenyloctová kyselina glycyl-1-glutámová kyselina 3-fosfonopropiónová kyselina 2-(4-chlórfenoxy)-2-metylpropiónová kyselina 2,3-dichlórbenzoová kyselina (r)-2-metylhexánová3- (2,4,6-trimethylbenzoyl) -2-biphenylcarboxylic acid (+/-) - erythro-3-methylglutamic acid 5-methoxybenzofuran-2-carboxylic acid 2- (1-naphthyl) -6-nitrophthalic acid 2 -imino-4-oxytiazole-5-acetic acid 2- (trifluoromethyl) -2-hydroxypropionic acid bromopivalic acid cyclopropanecarboxylic acid cyclopropane-1,2,3-tricarboxylic acid 7-oxo-8-nonenoic acid nonacosanoic acid 4- (4- bromobenzoyl) pentanoic acid 2 ', 4', 6 , -trimethylphthalanic acid 1-methyl-2-oxo-1,2-dihydroquinoxaline-3-propionic acid tribromoacetic acid (3-acetyl-2-methyl-5-oxo-2- pyrrolidin-4-yl) -acetic acid 4- tert -butylbenzoic acid cis- (2-fluorophenyl) hexahydrophthalic acid fmoc-4-aminobenzoic acid 2- (2-chloroacetamido) benzoic acetyl-asp-glu-oh lactobionic acid 1-Bromocyclohexanecarboxylic acid 2-methyl-2-naphthalen-1-ylmethyl-malonic acid 2- (4-isopropyl-benzylidene) -pent-4-enoic acid 2 , -methoxy-3,4,5,5 ', 6-pentachlorophthalanic acid 2- (cinamylidene) -2-phenylacetic acid glycyl-1-glutamic acid 3-phosphonopropionic acid 2- (4-chlorophenoxy) -2-methylpropionic acid (R) -2-methylhexanoic acid 2,3-dichlorobenzoic acid

-103-103-

• ·· • ·· • · • · ···· ···· ·· · · • · • · • · • · B B 9 9 9 9 9 9 • ··· • ··· • · · • · · 9 9 9 9 • e ·· • e ·· ·· · · ·· · · 9 9 9 9 9 9 9 9

kyselina 4'-fluórglutaranilová kyselina 2-tetradecénová kyselina 2-metyl-5-nitrobenzoová kyselina 4-hexadecyloxy-meta-anízová kyselina 1 (+)-2-amino-7-fosfonoheptánová kyselina spiro(5.5)undekán-2,2-dioctová kyselina 1 -acetylpiperidín-4-karboxylová kyselina 3-naftalén-1 -yl-propiónová kyselina p-propoxybenzoová kyselina (1 r)-(+)-(1-amino-2-metylpropyl)fosfónová kyselina 3-(4-brómbenzoyl)propiónová kyselina alfa-1 -glutamyl-1 -tyrozín-1 -glutámová kyselina 3,3-difenylpropiónová kyselina 2-dibenzofuránsulfínová kyselina 2-(difluórmetoxy)fenyloctová kyselina n-alfa-boc-n-beta-(z)-1 -diaminopropiónová kyselina d/-2-amino-7-sulfoheptánová kyselina 3-(4-nitrofenoxy)-2-tiofénkarboxylová kyselina d/-2-metylglutámová kyselina r-2-chlórmandlová kyselina n-boc-d/-alfa-aminoadipová kyselina 7-(4-(2-karboxy-etyl)-fenyl)-heptánová kyselina 1-sulfoantrachinón4'-fluoroglutaranilic acid 2-tetradecenoic acid 2-methyl-5-nitrobenzoic acid 4-hexadecyloxy-meta-ananoic acid 1 (+) - 2-amino-7-phosphonoheptanoic acid spiro (5.5) undecane-2,2-diacetic acid 1-acetylpiperidine-4-carboxylic acid 3-naphthalen-1-yl-propionic acid p-propoxybenzoic acid (1R) - (+) - (1-amino-2-methylpropyl) phosphonic acid 3- (4-bromobenzoyl) propionic acid alpha-1-glutamyl-1-tyrosine-1-glutamic acid 3,3-diphenylpropionic acid 2-dibenzofuran sulphonic acid 2- (difluoromethoxy) phenylacetic acid n-alpha-boc-n-beta- (z) -1-diaminopropionic acid d) -2-amino-7-sulfoheptanoic acid 3- (4-nitrophenoxy) -2-thiophenecarboxylic acid d] -2-methylglutamic acid r-2-chloro-mandelic acid n-boc-d-alpha-aminoadipic acid 7- (4- (2-Carboxy-ethyl) -phenyl) -heptanoic acid 1-Sulfoanthraquinone

4-(4-(hexadecyloxy)fenyl)maslová kyselina 4-pentylbicyklo(2.2.2)oktán-1 -karboxylová kyselina (bifenyl-4-yloxy)-octová kyselina 6,12-dioxo-1,17-heptadekándikarboxylová kyselina 5-benzoylamino-2-bróm-pentánová kyselina 3-cyklopentyloxy-4-metoxybenzoová kyselina (2,2-dimetyl-5-oxo-(1,3)dioxolán-4-yl)-octová kyselina (s)-(+)-2-amino-6-0ód-acetamido)hexánová kyselina 6-(2-nitro-fenylsulfanylamino)-hexánová4- (4- (hexadecyloxy) phenyl) butyric acid 4-Pentylbicyclo (2.2.2) octane-1-carboxylic acid (biphenyl-4-yloxy) acetic acid 6,12-dioxo-1,17-heptadecanedicarboxylic acid 5- benzoylamino-2-bromo-pentanoic acid 3-cyclopentyloxy-4-methoxybenzoic acid (2,2-dimethyl-5-oxo- (1,3) dioxolan-4-yl) -acetic acid (s) - (+) - 2 6- (2-nitro-phenylsulfanylamino) -hexanoic acid-amino-6-oxo-acetamido) hexanoic acid

• ·· • · • ··· • ·· • · • ··· ·· • a • · · · • a • · ···· e • ···· e • ·· • · 9 9 ·· • · 9 9 • · • · • · a a • · a a • a • a ·· · · • · • · 9 9 9 9

-104 kyselina c/s-2,5-piperidíndikarboxylová kyselina 3-(2,3-dimetoxy-fenyl)-2-metyl-akrylová kyselina tricyklo(10.2.2.2(4,7))oktadeka-heptaén-9-karboxylová kyselina 4,6-heptadekadiínová kyselina arteannuová kyselina 5-(4-chlórfenyl)-2,3-dihydro-1h-pyrolizín-6,7-dikarboxylová kyselina 6,7,8,8a,9,10-hexahydro-2-metoxyfenantrén-7,8-dikarboxylová kyselina 2-benzylidén-malónová kyselina benzo[b]tiofén-3-octová kyselina 2-acetylamino-3-(1 h-imidazol-4-yl)-akrylová kyselina (9h-xantén-9-ylsulfanyl)-octová kyselina 3,3'-tiodipropiónová kyselina tetrafluórftalová kyselina 6-butylamino-pyrimidín-4-karboxylová kyselina n-dodecylfosfónová kyselina m-tolyloctová kyselina mykofenolová kyselina 3-acetoxybenzoová kyselina 1 -(3,4-dichlórfenyl)-2-oxopyrolidín-4-karboxylová kyselina (2s,5r)-fmoc-5-fenyl-pyrolidín-2-karboxylová kyselina fluorovodíková kyselina 3-chlór-4-(izopropylsulfonyl)tiofén-2-karboxylová kyselina 4-chlórsalicylová kyselina beta-metyl-4-nitrohydroškoricová kyselina trichlór-pyrohroznová kyselina 3,5-d/-terc-butylbenzoová kyselina 3-(trifluórmetoxy)fenyloctová kyselina bicyklo(2.2.2)oktán-2-karboxylová kyselina 2-fenylindol-3-octová kyselina 2,2-bifenyldioctová kyselina 2-mezitylénsulfónová kyselina gama-oxo-5-acenafténmaslová-104 cis -2,5-piperidinedicarboxylic acid 3- (2,3-dimethoxyphenyl) -2-methyl-acrylic acid tricyclo (10.2.2.2 (4,7)) octadeca-heptaene-9-carboxylic acid 4,6-heptadecadioic acid arteannuic acid 5- (4-chlorophenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid 6,7,8,8a, 9,10-hexahydro-2-methoxyphenanthrene- 7,8-Dicarboxylic acid 2-benzylidene-malonic acid benzo [b] thiophene-3-acetic acid 2-acetylamino-3- (1H-imidazol-4-yl) -acrylic acid (9h-xanthen-9-ylsulfanyl) -acetic acid 3,3'-thiodipropionic acid tetrafluorophthalic acid 6-butylamino-pyrimidine-4-carboxylic acid n-dodecylphosphonic acid m-tolylacetic acid mycophenolic acid 3-acetoxybenzoic acid 1- (3,4-dichlorophenyl) -2-oxopyrrolidine- (2s, 5r) -fmoc-5-phenyl-pyrrolidine-2-carboxylic acid 4-carboxylic acid 3-chloro-4- (isopropylsulfonyl) -thiophene-2-carboxylic acid 4-chlorosalicylic acid beta-methyl-4-ni Trichloro-pyruvic acid 3,5-di-tert-butylbenzoic acid 3- (trifluoromethoxy) phenylacetic acid Bicyclo (2.2.2) octane-2-carboxylic acid 2-Phenylindole-3-acetic acid 2,2-Biphenyldiacetic acid 2-mesitylene sulfonic acid gamma-oxo-5-acenaphthenebutyric acid

-105--105-

• ·· • · • ··· • ·· • · • ··· ·· «··· • · · • · · ··· · · · · ·· • · • · ·· • · • · • · • · ·· · · ·· · · • 9 ·· • 9 ·· • · • · β · β ·

kyselina 3-trifluórmetylfenoxydifluóroctová kyselina s-2-chlórmandlová kyselina 2-nonínová kyselina 2,6-dichlór-3-metylbenzoová kyselina n,n -(1,4-cyklohexyléndimetylén)-dimaleámová kyselina 7-nitro-9-oxo-1 -fluorénkarboxylová kyselina eikozándiová kyselina 12-metánsulfonyloxy-dodekánová kyselina tiosalicylová kyselina 3-acetyl-2-naftoová kyselina poly(akrylová) kyselina 3-fenylmaslová kyselina 1 -(3,5-dimetylfenyl)-6-metyl-4-oxo-1,4-dihydro-3-pyridínkarboxylová kyselina 2-bróm-4-chlórbenzoová kyselina n-(4-etoxyfenyl)-1,2,3,6-tetrahydroftalámová kyselina fenylundekánová n-acetyl-s-(4-nitrofenyl)-1-cysteín kyselina 3-acetylbenzoová kyselina terc-butylfosfónová kyselina c/s-epoxyjantárová kyselina 4-brómbenzoová kyselina for-1-2-aminohexánová kyselina 4-(4’-nitro-bifenyl-4-sulfonyl)-benzoová kyselina krotónová kyselina 15(r)-hydroxyeikoza-5z,8z, 11 z, 13e-tetraénová kyselina 3-[4-oxo-5-(5-ph-furán-2-ylmetylén)-2-tioxo-tiazolidín-3-yl]-propiónová kyselina palmitová kyselina 5-metoxy-2-(2,2,2-trifluóretoxy)benzoová kyselina alfa-chlór-3,5,7-trimetyl-1 -adamantánoctová kyselina (5,6,7,8-tetrahydro-chinazolín-4-ylsulfanyl)-octová kyselina ŕrans-(+)-chryzantémová kyselina 1,4-dihydro-1 -(2-fluóretyl)-4-oxo-6,7,8-trifluór-3-chinolínkarboxylová ·· ·· ···· ·· • · · · · · · • ·Φ · · *) · ·3-Trifluoromethylphenoxydifluoroacetic acid s-2-Chloromandelic acid 2-Nonanoic acid 2,6-dichloro-3-methylbenzoic acid n, N- (1,4-Cyclohexylenedimethylene) -dimaleamic acid 7-nitro-9-oxo-1-fluorocarboxylic acid eicosanedioic acid 12-methanesulfonyloxy-dodecanoic acid thiosalicylic acid 3-acetyl-2-naphthoic acid poly (acrylic) 3-phenylbutyric acid 1- (3,5-dimethylphenyl) -6-methyl-4-oxo-1,4- dihydro-3-pyridinecarboxylic acid 2-bromo-4-chlorobenzoic acid n- (4-ethoxyphenyl) -1,2,3,6-tetrahydrophthalamic acid phenylundecanoic acid n-acetyl-s- (4-nitrophenyl) -1-cysteine acid 3 -acetylbenzoic acid tert-butylphosphonic acid cis-epoxysuccinic acid 4-bromobenzoic acid for-1-2-aminohexanoic acid 4- (4'-nitro-biphenyl-4-sulfonyl) -benzoic acid crotonic acid 15 (r) -hydroxyeicosis -5z, 8z, 11z, 13e-tetraenoic acid 3- [4-oxo-5- (5-ph-furan-2-ylmethylene) -2-thioxothiazolidin-3-yl] -propionic acid palmitic acid 5-methoxy-2- (2,2,2-trifluoroethoxy) benzoic acid alpha-chloro-3,5,7-trimethyl-1-adamantaneacetic acid (5,6,7,8-tetrahydroquinazoline) -4-Ylsulfanyl) -acetic acid trans - (+) - Chrysanthemic acid 1,4-dihydro-1- (2-fluoroethyl) -4-oxo-6,7,8-trifluoro-3-quinolinecarboxylic acid ·· ·· · ··· ·· · · · · · · Φ · *) · ·

-106kyselina 3-(fenyltio)propiónová kyselina 2-(2-benzoyloxyfenoxy)octová kyselina 3-(4-(6-(4-(2-metoxykarbonyl-etyl)-fenyl)-hexyl)-fenyl)-propiónová kyselina 4-hydroxyftalová kyselina n-boc-aminovalérová kyselina 2'-chlórftalanilová kyselina 3-(2-nonylsulfanyl-benzotiazol-6-ylkarbamoyl)-akrylová kyselina 2-(trifluórmetyl)propénová kyselina 2-karboxy-3-indolmaslová kyselina 13c, 16c-dokozadiénová kyselina 11-p-tolylsulfanyl-undekánová kyselina propargylová kyselina p-metylbenzyl-3-tio-propiónová kyselina 13-eikozínová kyselina 2-(2,3-dichlórfenyltio)octová kyselina (+/-)-12,13-epoxyoktadec-9z-énová kyselina 3,5-dichlór-o-anízová kyselina 3,5-dibrómsalicylová kyselina 3,4-(metyléndioxy)-6-nitroškoricová kyselina c/s-vakcénová kyselina 4-nitrofenyljantárová kyselina p-chlórbenzoylakrylová kyselina 3-(4-ŕerc-butyl-fenyl)-propiónová kyselina 2,,6,-dimetyl-3,4,5,6-tetrachlórftalanilová kyselina 11,14,17-eikozatriénová kyselina 3-(2,4-dichlórbenzyltio)tiofén-2-karboxylová kyselina 2-(2,6-dichlórfenyltio)octová kyselina 4,5-dimetoxylodobenzoová kyselina 3,5,6-trichlórsalicylová kyselina 6-bróm-1,3-dioxo-1 h-benz[de]-izochinolín-2(3h)-octová kyselina 3-bróm-4-fluórbenzoová kyselina trichlóroctová-106 3- (Phenylthio) propionic acid 2- (2-benzoyloxyphenoxy) acetic acid 3- (4- (6- (4- (2-methoxycarbonyl-ethyl) -phenyl) -hexyl) -phenyl) -propionic acid 4- hydroxyphthalic acid n-boc-aminovaleric acid 2'-chlorophthalanilic acid 3- (2-nonylsulfanyl-benzothiazol-6-ylcarbamoyl) -acrylic acid 2- (trifluoromethyl) propenoic acid 2-carboxy-3-indolebutyric acid 13c, 16c-docosadienoic acid 11-p-tolylsulfanyl-undecanoic acid propargylic acid p-methylbenzyl-3-thio-propionic acid 13-eicosic acid 2- (2,3-dichlorophenylthio) acetic acid (+/-) - 12,13-epoxyoctadec-9z-enoic acid 3,5-dichloro-o-anisic acid 3,5-dibromosalicylic acid 3,4- (methylenedioxy) -6-nitrocinnamic acid cis-vaccenoic acid 4-nitrophenylsuccinic acid p-chlorobenzoylacrylic acid 3- (4-tert- butyl-phenyl) -propionic acid 2, 6-dimethyl-3,4,5,6-tetrachlórftalanilová 11,14,17-eicosatrienoic acid, 3- (2,4-dich lorobenzylthio) thiophene-2-carboxylic acid 2- (2,6-dichlorophenylthio) acetic acid 4,5-dimethoxyylbenzoic acid 3,5,6-trichlorosalicylic acid 6-bromo-1,3-dioxo-1 h-benz [de] -isoquinoline-2 (3h) -acetic acid 3-bromo-4-fluorobenzoic acid trichloroacetic acid

-107 kyselina (+/-)-1 -amino-ŕrans-3-fosfonocyklopentán-karboxylová kyselina 2-(2-(2-amino-acetylamino)-4-karbamoyl-1-butyrilamino)-3-(4-ho-ph)-propiónová kyselina 2-kyano-2-hexénová kyselina 3,3-dimetylakrylová kyselina 2-brómtereftalová kyselina 8-fenyloktánová kyselina 3-(benzyltio)-propiónová kyselina 2-(dodecyloxy)benzoová kyselina 4,5-dibrómtiofén-2-karboxylová kyselina (n,n-dietyltiokarbamoyltio)-octová kyselina 2 (4-metoxykarbonyl-ph)-1,3-dioxo-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina 2,3-dimetoxyškoricová kyselina n-acetyl-d/-metionín-9-fluorénkarboxylová kyselina (+/-)-treo-3-metylglutámová kyselina 7c, 10c, 13c, 16c-dokozatetraénová kyselina 3-(4-n-propyloxybenzoyl)propiónová kyselina perfluór(4-metylpent-2-énová) kyselina 4-(2-hydroxy-1 -naftylmetylénamino)benzoová kyselina etyléndiamín-n.n-dioctan-n.n-dipropiónová kyselina c/s-n-furfurylhexahydroftalámová kyselina /?-[3-(6-chlór)pyridazinyl]izonipekotínová kyselina n-(1-metyl-5-metyltio-1,2,4-triazol-3-yl)malonámová kyselina (r)-(-)-3-chlórmandlová kyselina (r)-(-)-o-acetylmandlová kyselina beta-metyl-1 -pyrénpropiónová kyselina 4-(difluórmetoxy)fenyloctová fenyl-beta-d-glukuronid kyselina 2-bróm-5-metylbenzoová kyselina n-(4-jódfenyl)glutarámová kyselina m-etylbenzoová kyselina 2,2-bis-(4-benzyloxy-butyl)-malónová-107 (+/-) - 1-amino-trans-3-phosphonocyclopentanecarboxylic acid 2- (2- (2-amino-acetylamino) -4-carbamoyl-1-butyrilamino) -3- (4-ho- ph) -propionic acid 2-cyano-2-hexenoic acid 3,3-dimethylacrylic acid 2-bromo-terephthalic acid 8-phenyloctanoic acid 3- (benzylthio) -propionic acid 2- (dodecyloxy) benzoic acid 4,5-dibromothiophene-2- (n, n-Diethylthiocarbamoylthio) -acetic acid 2- (4-methoxycarbonyl-ph) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid 2,3-dimethoxycinnamic acid n- (+/-) - Threo-3-methylglutamic acid acetyl-d-methionine-9-fluorenecarboxylic acid 7c, 10c, 13c, 16c-docosatetraenoic acid 3- (4-n-propyloxybenzoyl) propionic acid perfluoro (4-methylpent- 2-enoic acid 4- (2-hydroxy-1-naphthylmethyleneamino) benzoic acid ethylenediamine-n-dioctane-n-dipropionic acid cis -furfurylhexahydrophthalic acid p - [3- (6-chloro) pyridazinyl] isonipecotinic acid n - (1-m ethyl-5-methylthio-1,2,4-triazol-3-yl) malonamic acid (R) - (-) - 3-chloro-butyric acid (R) - (-) - o-acetyl-butyric acid beta-methyl-1- pyrene-propionic acid 4- (difluoromethoxy) phenylacetic phenyl-beta-d-glucuronide 2-bromo-5-methylbenzoic acid n- (4-iodophenyl) glutaramic acid m-ethylbenzoic acid 2,2-bis- (4-benzyloxy-butyl) -malonic

-108 --108 -

« ·· • · • ··· «·· • · • ··· ·· • · • e · · • · • e ···· • • ···· • • ·· • · B · ·· • · B · 9 9 9 9 • · · · • · · · • · • · ·· · · • · • · 9 9 9 9

kyselina 5-bróm-2-fluórškoricová kyselina 3,4-dihydro-2,2-dimetyl-4-oxo-2h-pyrán-6-karboxylová kyselina 7-nitrofluorén-1 -karboxylová kyselina boc-2-aminobenzoová kyselina S'-metylmaleanilová kyselina 15-(3,4-dichlórfenyl)-pentadekánová kyselina 4-vinylbenzoová kyselina 2,3,6-trifluórbenzoová kyselina tetratiafulvaléntetrakarbónová kyselina 4-((pyridín-3-karbonyl)-amino)-maslová kyselina 6-metoxy-2-naftyloctová kyselina z-1-2-aminohexándiová kyselina (+/-)-13-hydroxyoktadeka-9z, 11e-diénová kyselina 1-hexánsulfónová kyselina tnp-1-asparágová kyselina 3-(2,4-dichlórbenzyloxy)tiofén-2-karboxylová kyselina karbobenzyloxy-d-2-aminomaslová kyselina 11-dodecylsulfanyl-iindekánová kyselina 8-(3-(5-f-2-ho-fenyl)-3-oxo-propenyl)-4h-benzo(1,3)dioxín-6-karboxylová kyselina 4-(1,3-dioxo-1 h,3h-benzo(de)izochinolín-2-yl)-benzoová kyselina 2-(2-chlór-acetylamino)-3-(4-hydroxy-fenyl)-propiónová kyselina 3-(chlórmetyl)benzoová kyselina 7-etoxybenzofurán-2-karboxylová kyselina acetylsalicylová kyselina 4-(3-(3-fluórfenyl)ureido)benzoová kyselina 3-hydroxy-2-metyl-eikozánová kyselina 2-naftalén-2-yl-benzoová kyselina 1-valyl-1-asparágová kyselina 3,3-dimetylglutárová kyselina 3,5-bis(trifluórmetyl)benzoová kysel ina (-)-2-(4-metoxyfenyl )maslová kyselina (s)-3-(4-fluórfenyl)butánová5-Bromo-2-fluorocinnamic acid 3,4-dihydro-2,2-dimethyl-4-oxo-2h-pyran-6-carboxylic acid 7-nitrofluorene-1-carboxylic acid boc-2-aminobenzoic acid S'- methylmaleanilic acid 15- (3,4-dichlorophenyl) -pentadecanoic acid 4-vinylbenzoic acid 2,3,6-trifluorobenzoic acid tetrathifulvalenetretracarboxylic acid 4 - ((pyridine-3-carbonyl) amino) butyric acid 6-methoxy-2- naphthylacetic acid z-1-2-aminohexanedioic acid (+/-) - 13-hydroxyoctadeca-9z, 11e-dienoic acid 1-hexanesulfonic acid tnp-1-aspartic acid 3- (2,4-dichlorobenzyloxy) thiophene-2-carboxylic acid carbobenzyloxy-d-2-aminobutyric acid 11-dodecylsulfanylindecanoic acid 8- (3- (5-f-2-ho-phenyl) -3-oxo-propenyl) -4h-benzo (1,3) dioxin-6 -carboxylic acid 4- (1,3-dioxo-1h, 3h-benzo (de) isoquinolin-2-yl) -benzoic acid 2- (2-chloro-acetylamino) -3- (4-hydroxy-phenyl) - propionic acid 3- (chloromethyl) benzoic acid 7-ethoxybenzofuran-2 carboxylic acid acetylsalicylic acid 4- (3- (3-fluorophenyl) ureido) benzoic acid 3-hydroxy-2-methyl-eicosanoic acid 2-naphthalen-2-yl-benzoic acid 1-valyl-1-aspartic acid 3,3 -dimethylglutaric acid 3,5-bis (trifluoromethyl) benzoic acid (-) - 2- (4-methoxyphenyl) butyric acid (s) -3- (4-fluorophenyl) butanoic acid

-109--109-

• ·· • · • ··· • ·· • · • ··· • · • · • · • · • · • · ···· • • ···· • • ·· · • · · · • · · ·· · • · · ·· ·· ·· ·· ·· · · • · • · ·· ·· ·· ··

kyselina 2-(2-metyl-3-fenyl-propionyl)-benzoová kyselina 4-(4-/7-propylfenyl)benzoová kyselina 5 alebo 6 alebo 7 alebo 8-nitro-2-antrachinónkarboxylová kyselina 1,2-dihydro-3-metyl-2-oxo-4-chinolínkarboxylová kyselina 1,8-naftalaldehydová kyselina 1 -(4-ch lórfeny I)-1 -cyklopentánkarboxylová kyselina 2,5-dimetyl-2,4-hexadiéndiová kyselina 3-(4-fluórbenzyloxy)tiofén-2-karboxylová kyselina (+/-)-ŕrans-azetidín-2,4-dikarboxylová kyselina 2-(4-nitrofenyltio)octová kyselina (3,5-xylyl)fosfónová kyselina 3,4-dimetylfenoxyoctová kyselina 2-etylhexánová kyselina (+/-)-2-hydroxynonánová kyselina adipová kyselina 2-(4-izopropyl-benzoyl)-benzoová kyselina 2-(6-bróm-2-naftyloxy)-propiónová kyselina 3,5-dibróm-2-(2-etoxykarbonyl-acetylamino)benzoová kyselina n-(2,4,6-trimetylfenyl)maleámová kyselina 4-morfol ín-4-yl-4-oxo-but-2-énová kyselina n-(2-alylsulfanyl-benzotiazol-6-yl)-sukcínamová kyselina 4-metylsulfonyl-3-nitrobenzoová kyselina 3,4-difluórmandlová kyselina 3-(4-chlórfenyl)-glutarámová kyselina 3,5-dibrómbenzoová kyselina 1 h-indén-2-karboxylová kyselina s-(-)-2-[(fenylamino)karbonyloxy]propiónová kyselina alizarín-5-sulfónová kyselina 4-acetoxyfenyloctová kyselina 2,4-dichlórbenzoová kyselina n-(2-tiazolyl)ftalámová kyselina dibenzo(a,d)cyklohepten-5-ylidén-octová2- (2-Methyl-3-phenyl-propionyl) -benzoic acid 4- (4- / 7-propyl-phenyl) -benzoic acid 5 or 6 or 7 or 8-nitro-2-anthraquinone carboxylic acid 1,2-dihydro-3 methyl-2-oxo-4-quinolinecarboxylic acid 1- (4-chlorophenyl) -1-cyclopentanecarboxylic acid 1,8-naphthaldehyde 2,5-dimethyl-2,4-hexadienedioic acid 3- (4-fluorobenzyloxy) thiophene-2-carboxylic acid (+/-) - trans -azetidine-2,4-dicarboxylic acid 2- (4-nitrophenylthio) acetic acid (3,5-xylyl) phosphonic acid 3,4-dimethylphenoxyacetic acid 2-ethylhexanoic acid (+/-) - 2-hydroxynonanoic acid adipic acid 2- (4-isopropyl-benzoyl) -benzoic acid 2- (6-bromo-2-naphthyloxy) -propionic acid 3,5-dibromo-2- (2-ethoxycarbonyl) -acetylamino) benzoic acid 4- (2,4,6-trimethylphenyl) maleic acid 4-morpholin-4-yl-4-oxo-but-2-enoic acid n- (2-allylsulfanyl-benzothiazol-6-yl) -Succinamic acid 4-methylsulfonyl-3-nitrobenzoic acid 3,4-difluoromethyl 3- (4-chlorophenyl) -glutaramic acid 3,5-dibromobenzoic acid 1H-indene-2-carboxylic acid with - (-) - 2 - [(phenylamino) carbonyloxy] propionic acid alizarin-5-sulfonic acid 4 -acetoxyphenylacetic acid 2,4-dichlorobenzoic acid n- (2-thiazolyl) phthalic acid dibenzo (a, d) cyclohepten-5-ylidene-acetic acid

-110·· ·· ···· ·· • · · · · · · • 99 9 9 9 · · kyselina tiofén-3-octová kyselina 3,3-dimetyl-(1,1,3',1)terfenyl-2'-karboxylová kyselina 5-(4-metoxy-fenyl)-pentánová kyselina 3-oxo-1 -indánkarboxylová kyselina 6-brómhexánová kyselina (4-(2-acetyl-3-oxo-cyklopent-1-enylamino)-benzoylamino)-octová kyselina 4-(4-(2-karboxybenzoyl)fenyl)maslová kyselina 2-dicyklohexylkarbamoyl-cyklohexánkarboxylová kyselina 13-oxopentadekánová kyselina 2,3,4,4a,4b,5,8,8a,9,10-dekahydro-8a-metyl-2-oxo-1-fenantrénpropiónová kyselina 3-(7-metoxy-2,2-difenyl-benzo(1,3)dioxol-5-yl)-propiónová kyselina fenylpyrohroznová kyselina 4-(3-(2-fenoxypropionyl)-2-tioureido)benzoová kyselina 3-(4-etylbenzoyl)propiónová kyselina 4-hydroxyazobenzén-4'-sulfónová kyselina 2-acetylamino-3-(1 h-indol-3-yl)-propiónová kyselina 2,3,4,6-tetrametyl-benzoová kyselina linolová kyselina 4-(2,6-dimetyl-4-hydroxyfenylazo)benzénsulfónová kyselina 3-(3-bróm-4-metoxy-fenyl)-propiónová kyselina 3-[(4-metoxyfenyl)-(toluén-4-sulfonyl)-amino]propiónová kyselina 5-(3-amino-4-chlór-fenylsulfamoyl)-izoftalová kyselina 3-bróm-2,6-dimetoxy-5-nitrobenzoová kyselina (+/-)-c/s-2,3-piperidín-dikarboxylová kyselina n-acetyl-n-n-butylantranilová kyselina 3,5-dimetylfenoxyoctová kyselina 2-kyanobenzoová kyselina n-alfa-boc-n-gama-aloc-1 -diaminomaslová kyselina 3,4-metyléndioxyfenylpyrohroznová kyselina 6-hydroxy-2,5,7,5-tetrametylchroman-2-karboxylová kyselina 1-benzylorotová kyselina boc-1 -7-hydroxy-1,2,3,4-tetrahydroizochinolín-3-karboxylová-110 99 9 9 9 thiophene-3-acetic acid 3,3-dimethyl- (1,1,3 ', 1) terphenyl 2'-carboxylic acid 5- (4-methoxy-phenyl) -pentanoic acid 3-oxo-1-indanecarboxylic acid 6-bromohexanoic acid (4- (2-acetyl-3-oxo-cyclopent-1-enylamino) -benzoylamino) ) -acetic acid 4- (4- (2-carboxybenzoyl) phenyl) butyric acid 2-dicyclohexylcarbamoyl-cyclohexanecarboxylic acid 13-oxopentadecanoic acid 2,3,4,4a, 4b, 5,8,8a, 9,10-decahydro- 8α-Methyl-2-oxo-1-phenanthrenepropionic acid 3- (7-methoxy-2,2-diphenyl-benzo (1,3) dioxol-5-yl) -propionic acid phenylpyruvic acid 4- (3- (2- phenoxypropionyl) -2-thioureido) benzoic acid 3- (4-ethylbenzoyl) propionic acid 4-hydroxyazobenzene-4'-sulfonic acid 2-acetylamino-3- (1H-indol-3-yl) -propionic acid 2,3, 4,6-tetramethyl-benzoic acid linoleic acid 4- (2,6-dimethyl-4-hydroxyphenylazo) benzenesulfonic acid 3- (3-bromo-4-methoxyphenyl) -propion 3 - [(4-Methoxyphenyl) - (toluene-4-sulfonyl) amino] propionic acid 5- (3-amino-4-chloro-phenylsulfamoyl) -isophthalic acid 3-bromo-2,6-dimethoxy-5 -nitrobenzoic acid (+/-) - cis-2,3-piperidine-dicarboxylic acid n-acetyl-n-butylantranilic acid 3,5-dimethylphenoxyacetic acid 2-cyanobenzoic acid n-alpha-boc-n-gamma-aloc -1-diaminobutyric acid 3,4-methylenedioxyphenylpyruvic acid 6-hydroxy-2,5,7,5-tetramethylchroman-2-carboxylic acid 1-benzylorotic acid boc-1-7-hydroxy-1,2,3,4-tetrahydroisoquinoline 3-carboxylic acid

-111 --111 -

• ·· • · • ··· • ·· • · • ··· ·· ···· • · · • · · ·· ···· · · · · · · ·· · • · ·· • · · ·· · • · ·· • · · ·· ·· ·· ·· ·· ·· ·· ·· ·· ·· ·· ··

kyselina (3-metoxyfenyl)fenylfosfínová kyselina 3-(3,6-dimetoxy-2-naftoyl)propiónová kyselina 4-(3-(2,5-xylyl)ureido)benzoová kyselina d-alfa-hydroxyizovalérová kyselina 5,5,6,6,7,7,7-heptafluór-4,4-bis(trifluórmetyl)heptánová kyselina 2-chlór-4-fluórškoricová kyselina acetyléndikarboxylová kyselina n-acetyl-d/-2-amino-/?-maslová kyselina 2-hydroxyvalérová kyselina 2,5-difluórmandlová kyselina n-boc-1 -1,2,3,4-tetrahydro-beta-karbolín-3-karboxylová kyselina 5-(1-metyletoxy)-1,3-benzéndikarboxylová kyselina 2,,4'-dichlórglutaranilová kyselina tiopivalová kyselina 5’-chlór-2’,4'-dimetoxymaleanilová kyselina (4-(3-(4-meo-fenyl)-tioureido)-6-metyl-pyrimidín-2-ylsulfanyl)octová kyselina 2,2-dichlórpropiónová kyselina 3-chlór-4-hydroxybenzoová kyselina 4-etoxy-2-hydroxybenzoová kyselina 1,2,3,4-tetrahydro-2-naftoová kyselina 2-(1-(3-chlórbenzyl)-1 h-3-indolyl]octová kyselina ŕrans-beta-hydromukonová kyselina 2-(3-chlór-1,4-dioxo-1,4-dihydro-naftalén-2-ylamino)-jantárová kyselina 4-fluór-3-hydroxybenzoová kyselina 2-fenoxynikotínová kyselina 6-(2-benzoylamino-3-fenyl-akryloylamino)-hexánová kyselina 2-metoxy-5-sulfamoyl-benzoová kyselina 5-oxotricyklo(2.2.1.0(2,6))heptán-2,3-dikarboxylová(3-Methoxyphenyl) phenylphosphinic acid 3- (3,6-dimethoxy-2-naphthoyl) propionic acid 4- (3- (2,5-xylyl) ureido) benzoic acid d-alpha-hydroxyisovaleric acid 5,5,6 , 6,7,7,7-heptafluoro-4,4-bis (trifluoromethyl) heptanoic acid 2-chloro-4-fluorocinnamic acid acetylenedicarboxylic acid n-acetyl-d-2-amino-β-butyric acid 2-hydroxyvaleric acid acid, 2,5-difluoromandelic acid, n-boc-1 -1,2,3,4-tetrahydro-.beta.-carboline-3-carboxylic acid 5- (1-methylethoxy) -1,3-benzenedicarboxylic acid, 2, 4 ' Dichloroglutaranilic acid Thiopivalic acid 5'-chloro-2 ', 4'-dimethoxymaleanilic acid (4- (3- (4-Meophenyl) thioureido) -6-methyl-pyrimidin-2-ylsulfanyl) acetic acid 2,2 -dichloropropionic acid 3-chloro-4-hydroxybenzoic acid 4-ethoxy-2-hydroxybenzoic acid 1,2,3,4-tetrahydro-2-naphthoic acid 2- (1- (3-chlorobenzyl) -1H-3-indolyl) acetic acid trans-beta-hydromuconic acid 2- (3-chloro-1,4-dioxo-1,4-dihydro-naphtha) alen-2-ylamino) succinic acid 4-fluoro-3-hydroxybenzoic acid 2-phenoxynicotinic acid 6- (2-benzoylamino-3-phenyl-acryloylamino) -hexanoic acid 2-methoxy-5-sulfamoyl-benzoic acid 5-oxotricyclo (2.2.1.0 (2,6)) heptane-2,3-dicarboxylic acid

2,2-bis(4-karboxyfenyl)hexafluórpropán kyselina 3-(trimetylsilyl)propínová kyselina (2s,3s)-2-chlór-3-metyl-n-valérová kyselina 6-nitro-3-(fenylacetamido)benzoová2,2-Bis (4-carboxyphenyl) hexafluoropropane 3- (trimethylsilyl) propionic acid (2s, 3s) -2-chloro-3-methyl-n-valeric acid 6-nitro-3- (phenylacetamido) benzoic acid

-112 --112 -

• ·· • · • ··· • ·· • · • ··· ·· ···· • · · • · · ·· ···· · · · · · · ·· • · • · · · • · • · ·· · · ·· ·· ·· ·· ·· ·· ·· ·· ·· · · • · • ·

kyselina 6-(2,3-dioxo-3-fenyl-propyl)-2,3-dimetoxy-benzoová kyselina 5-(n-benzoylamino)-n-valérová kyselina d/-3-hydroxyglutámová kyselina 13(s)-hydroperoxyoktadeka-9z,11e-diénová kyselina (2,4-d/-ferc-pentylfenoxy)octová kyselina 2-metylundekánová kyselina 2-hydroxy-2-metylmaslová kyselina 4'-metoxysukcínanilová kyselina 2-anilinonaftalén-6-sulfónová kyselina (4l-karboxymetánsulfonyl-bifenyl-4-sulfonyl)-octová kyselina beta-acetylmerkaptoizomaslová kyselina 3,5-dijódbenzoová kyselina 4-((fenyl-(toluén-4-sulfonylimino)-metyl)-amino)-benzoová kyselina 3-(4-metylbenzoyl)propiónová kyselina 2,2-dichlórtetradekánová kyselina 2-(2’-nitro-4,-trifluórmetylfenyltio)benzoová kyselina 2,8,14,20-dokozatetraín-1,22-diová kyselina (2-bróm-4-metylfenoxy)octová kyselina 2-fluór-4-nitrobenzoová kyselina izostearová kyselina (+/-)-3-endo-aminotricyklo[2.2.1.0(2,6)]heptán-3-endo-7-anti-dikarboxylová kyselina 4-brómizoftalová kyselina 6-bróm-alfa-kyano-1,3-benzodioxol-5-akrylová kyselina 1 -karboetoxyamino-7-naftol-3-sulfónová kyselina 6-(2-benzoylamino-3-(4-metoxy-fenyl)-akryloylamino)hexánová6- (2,3-dioxo-3-phenyl-propyl) -2,3-dimethoxy-benzoic acid 5- (n-benzoylamino) -n-valeric acid 1,3-hydroxyglutamic acid 13 (s) -hydroperoxyoctadeca -9z, 11e-dienoic acid (2,4-D / N-tert-pentylphenoxy) acetic acid, 2-methylundecane 2-hydroxy-2-methylbutyric acid 4'-metoxysukcínanilová acid 2-anilinonaftalén-6-sulfonic acid (4 l - carboxymethanesulfonyl-biphenyl-4-sulfonyl) -acetic acid beta-acetylmercaptoisobutyric acid 3,5-diiodo-benzoic acid 4 - ((phenyl- (toluene-4-sulfonylimino) -methyl) -amino) -benzoic acid 3- (4-methylbenzoyl) propionic acid, 2,2-dichlorotetradecanoic 2- (2'-nitro-4, -trifluórmetylfenyltio) benzoic acid, 2,8,14,20-dokozatetraín-1,22-dioic acid, (2-bromo-4-methyl-phenoxy) -acetic acid 2-fluoro-4-nitrobenzoic acid isostearic acid (+/-) - 3-endo-aminotricyclo [2.2.1.0 (2,6)] heptane-3-endo-7-anti-dicarboxylic acid 4-bromoisophthalic acid 6-bromo alpha-cyano-1,3-be nzodioxole-5-acrylic acid 1-Carboethoxyamino-7-naphthol-3-sulfonic acid 6- (2-benzoylamino-3- (4-methoxyphenyl) acryloylamino) hexanoic acid

2'-karboxy-2,5-dimetylbenzofenón kyselina 2-metylmaslová kyselina 3,3-bis(trifluórmetyl)-3-hydroxypropiónová kyselina alfa-fenyl-o-toluylová kyselina 6-oxotrikozánová kyselina 3,6-dihydroxyftalová kyselina 4-(3,4,5-trihydroxy-6-hydroxymetyl-tetrahydropyrán-2-ylamino)-benzoová2'-carboxy-2,5-dimethylbenzophenone 2-methylbutyric acid 3,3-bis (trifluoromethyl) -3-hydroxypropionic acid alpha-phenyl-o-toluic acid 6-oxotricosanoic acid 3,6-dihydroxyphthalic acid 4- (3 , 4,5-trihydroxy-6-hydroxymethyl-tetrahydropyran-2-ylamino) -benzoic acid

-113 --113 -

• ·· • · • ··· • ·· • · • ··· * * • · • · * * • · • · ···· • • ···· • • ·· • · • · ·· • · • · • · • · ·· ·· ·· ·· ·· · · ·· · · • · • · • · • ·

kyselina 2-brómhexadekánová kyselina 6-acetoxy-2-naftoová kyselina oktakozánová kyselina 3-karbamoyl-2,4-difenyl-cyklobutánkarboxylová kyselina 4'-bróm-2,,6,-dimetylftalanilová kyselina 3-acetyl-3-metylpentán-1,5-dikarboxylová kyselina tiobenzoová kyselina 2-[3-oxo-3-(n-propionyl-hydrazíno)-propionylamino]-benzoová kyselina c/s-1,4-cyklohexándikarboxylová kyselina tricyklo( 11.2.2.2(5,8))nonadekán-7-karboxylová kyselina guanidínojantárová kyselina 2-(karboxymetyltio)benzoová kyselina 1 (-)-2-amino-3-fosfonopropiónová kyselina 4-(4-brómbenzoyl)maslová kyselina 3,5-dibróm-4-metoxybenzoová kyselina 3-jódbenzoová kyselina 4-bróm-4-metyl-pentánová kyselina 18,18,18-trifluóroktadekánová kyselina 4-(hexadecylsulfonyl)benzoová kyselina 1 -(2-chlór-6-fluórfenyl)cyklohexánkarboxylová kyselina 2,3-dinitrobenzoová kyselina (1 r,3r)-1-amino-1-karboxycyklopentán-3-octová kyselina 1,3-fenyléndioctová kyselina 2’-(morfolín-4-karbonyl)-bifenyl-2-karboxylová kyselina n-(2,6-xylyl)ftalámová kyselina agarová kyselina n-hexadecylmaleámová kyselina (s)-4-karboxyfenylglycin-4'-fluór-3'-nitroftalanilová kyselina 3,3,3-trifluórpropiónová kyselina 4,5-dimetoxy-2-nitrobenzoová kyselina (1 r,3s)-1 -amino-1-karboxycyklopentán-3-octová kyselina n-(2,6-dietylfenylkarbamoylmetyl)iminodioctová • ·· ·· ···· ·· ··· ·· ···· ··« · · · · ·acid 2-brómhexadekánová 6-acetoxy-2-naphthoic acid oktakozánová acid, 3-carbamoyl-2,4-diphenyl-cyclobutanecarboxylic acid 4'-bromo-2, 6, -dimetylftalanilová acid, 3-acetyl-3-methylpentane-1, 5-Dicarboxylic acid thiobenzoic acid 2- [3-oxo-3- (n-propionyl-hydrazino) -propionylamino] -benzoic acid cis-1,4-cyclohexanedicarboxylic acid tricyclo (11.2.2.2 (5,8)) nonadecane 2- (carboxymethylthio) benzoic acid 1 (-) - 2-amino-3-phosphonopropionic acid 4- (4-bromobenzoyl) butyric acid 3,5-dibromo-4-methoxybenzoic acid 3-iodobenzoic acid 4-bromo-4-methylpentanoic acid 18,18,18-trifluorooctadecanoic acid 4- (hexadecylsulfonyl) benzoic acid 1- (2-chloro-6-fluorophenyl) cyclohexanecarboxylic acid 2,3-dinitrobenzoic acid (1 r, 3r) -1-amino-1-carboxycyclopentane-3-acetic acid 1,3-phenylenediacetic acid 2 '- (morpholine-4-carbonyl) -biphenyl-2-carbo xylic acid n- (2,6-xylyl) phthalic acid agaric acid n-hexadecylmaleamic acid (s) -4-carboxyphenylglycine-4'-fluoro-3'-nitropthalanic acid 3,3,3-trifluoropropionic acid 4,5-dimethoxy -2-nitrobenzoic acid (1 r, 3s) -1-amino-1-carboxycyclopentane-3-acetic acid n- (2,6-diethylphenylcarbamoylmethyl) iminodiacetic acid • ·· ·· ··········· ······ · · · · · ·

- 114kyselina jódoctová kyselina 2-(trifluórmetyltio)fenyloctová kyselina 4-(3-(2,2,2-trichlór-1-[(furán-2-karbonyl)-amino]-et)-tioureido)-benzoová kyselina cyklopentylidénoctová kyselina 2-fluór-3-(trifluórmetyl)benzoová kyselina 2,6-dioxo-5-etyl-1 -(3-metoxyfenyl)-1,2,3,6-tetra-h-4-pyrimidínkarboxylová kyselina fmoc-d-2-aminohexánová kyselina 2,6-dihydroxy-3-(3-(trifluórmetyl)fenylazo)benzoová kyselina 5-oxoundekánová kyselina 5-acetylamino-izoftalová kyselina 3-(trifluórmetoxy)benzoová kyselina 2-(toluén-4-sulfonylamino)-propiónová kyselina 2-(3,4-dimetyl-benzoyl)-benzoová kyselina tetrahydro-3-furoová kyselina 1-erytro-4-fluórglutámová kyselina 6-(karbobenzyloxyamino)kaprónová kyselina 3',4'-dimetylsukcínanilová kyselina 2-(2-nitro-4-trifluórmetyl-fenylamino)-propiónová kyselina 4-(4-hydroxy-fenylazo)-benzoová kyselina 9h-hexadekafluórnonánová kyselina 2-fluórškoricová kyselina 3-chlór-6-fluór-benzo(b)tiofén-2-karboxylová kyselina 2-furamido-4-nitrobenzoová kyselina 2-(2,-(3’-chlór-5,-trifluórmetyl)pyridyltio)nikotínová kyselina 3,3'-metylénbis[6-chlórbenzoová] kyselina 3-(4-n-hexylbenzoyl)propiónová kyselina 2-benzyloxyfenyloctová kyselina 4-(3,4-etyléndioxyfenyl)maslová kyselina 3,6,9-trioxaundekándiová kyselina 2-metyl-6-nitrobenzoová kyselina 6-(4-brómbenzoyl)hexánová kyselina 4-oktylbenzoová- 114 Iodoacetic acid 2- (trifluoromethylthio) phenylacetic acid 4- (3- (2,2,2-trichloro-1 - [(furan-2-carbonyl) -amino] -ethyl) thioureido) -benzoic acid Cyclopentylideneacetic acid 2 -fluoro-3- (trifluoromethyl) benzoic acid 2,6-dioxo-5-ethyl-1- (3-methoxyphenyl) -1,2,3,6-tetra-h-4-pyrimidinecarboxylic acid fmoc-d-2- aminohexanoic acid 2,6-dihydroxy-3- (3- (trifluoromethyl) phenylazo) benzoic acid 5-oxoundecanoic acid 5-acetylamino-isophthalic acid 3- (trifluoromethoxy) benzoic acid 2- (toluene-4-sulfonylamino) -propionic acid 2 - (3,4-Dimethyl-benzoyl) -benzoic acid tetrahydro-3-furoic acid 1-erythro-4-fluoroglutamic acid 6- (carbobenzyloxyamino) caproic acid 3 ', 4'-dimethylsuccinic acid 2- (2-nitro-4) -trifluoromethyl-phenylamino) -propionic acid 4- (4-hydroxy-phenylazo) -benzoic acid 9h-hexadecafluoronanoic acid 2-fluorocinnamic acid 3-chloro-6-fluoro-benzo (b) thiophene-2-carboxylic acid 2- furamide-4-nitrobenzoic acid 2- (2 '- (3'-chloro-5-trifluoromethyl) pyridylthio) nicotinic acid 3,3'-methylenebis [6-chlorobenzoic acid] 3- (4-n-hexylbenzoyl) propionic acid 2-Benzyloxyphenylacetic acid 4- (3,4-ethylenedioxyphenyl) butyric acid 3,6,9-trioxaundecanedioic acid 2-methyl-6-nitrobenzoic acid 6- (4-bromobenzoyl) hexanoic acid 4-octylbenzoic acid

-115--115-

• ·· • · • ··· • ·· • · • ··· • · • · • · • · ···· • • ···· • • ·· · • · · · • · · ·· · • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 2-(trifluórmetoxy)tereftalová kyselina 10-undecínová kyselina trans-13-oktadecénová kyselina 2-fenyl-2-propyljantárová kyselina 5,7-oktadekadiínová kyselina cysteamín-s-fosforečná n-acetyl-d/-alanín n-alfa-boc-1 -norvalín kyselina benzyloxyoctová kyselina 3,5-dimetoxybenzoová kyselina d/-alfa-brómizokaprónová kyselina meta-fosforečná kyselina 4'-fluórftalanilová kyselina 4’-bróm-2'-chlór-1,2,3,6-tetrahydroftalanilová kyselina fenyloin-n-maslová kyselina hydroxyimino-fenyl-octová kyselina (+/-)-1-aminocyklohexán-ŕrans-1,3-dikarboxylová kyselina d/-2-amino-5-fosfonovalérová kyselina 2-kyano-3-(5-naftalén-1 -yl-furán-2-yl)-akrylová kyselina ŕrans-parinarová kyselina 3-(2-benzotiazolyltio)propiónová kyselina 2-[1-(4-fluórbenzyl)-1 h-3-indolyl)octová kyselina 4-(4-metoxy-fenyl)-2-oxo-pyrolidín-3-karboxylová kyselina komanová kyselina 4-chlór-2-nitrobenzoová kyselina beta-metyl-levulová kyselina 1 -[2-(3-chlór-5-trifluórmetyl)pyridyl]indol-3-octová kyselina 4-dibenzotiofén-2-yl-4-oxo-maslová kyselina 3,5-difluórbenzoová n-alfa-benzoylasparagín kyselina c/s-n-(3-chlór-2-metylfenyl)hexahydroftalámová kyselina 4-butoxy-2-fluórbenzoová2- (trifluoromethoxy) terephthalic acid 10-undecinic acid trans-13-octadecenic acid 2-phenyl-2-propylsuccinic acid 5,7-octadecadiic acid cysteamine-s-phosphoric n-acetyl-d-alanine n-alpha-boc -1 -norvaline benzyloxyacetic acid 3,5-dimethoxybenzoic acid d-alpha-bromoisocaproic acid meta-phosphoric acid 4'-fluorophthalanic acid 4'-bromo-2'-chloro-1,2,3,6-tetrahydrophthalanic acid phenyloin -n-butyric acid hydroxyimino-phenyl-acetic acid (+/-) -1-aminocyclohexane-trans-1,3-dicarboxylic acid d-2-amino-5-phosphonovaleric acid 2-cyano-3- (5-naphthalene) -1-yl-furan-2-yl) -acrylic acid trans-parinic acid 3- (2-benzothiazolylthio) propionic acid 2- [1- (4-fluorobenzyl) -1H-3-indolyl] acetic acid 4- ( 4-methoxy-phenyl) -2-oxo-pyrrolidine-3-carboxylic acid comanoic acid 4-chloro-2-nitrobenzoic acid beta-methyl-levulinic acid 1- [2- (3-chloro-5-trifluoromethyl) pyri dyl] indole-3-acetic acid 4-dibenzothiophen-2-yl-4-oxo-butyric acid 3,5-difluorobenzoic acid n-alpha-benzoylasparagine cis- (3-chloro-2-methylphenyl) hexahydrophthalic acid 4- butoxy-2-fluorobenzoic acid

-116 --116 -

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kyselina (+/-)-ŕrans-2,4-piperidíndikarboxylová kyselina kantaridínová kyselina d/-alfa-hydroxyhexakozánová kyselina 4-(4-cyklopentyl-naftalén-1 -yl)-4-oxo-maslová kyselina 1 -(p-toly I)-1 -cyklohexánkarboxylová kyselina 1 -karboxy-3-cyklohexén-1 -octová kyselina olejová kyselina n-(difenylmetyl)ftalámová(+/-) - trans-2,4-piperidinedicarboxylic acid cantaridinic acid N-alpha-hydroxyhexacosanoic acid 4- (4-cyclopentyl-naphthalen-1-yl) -4-oxo-butyric acid 1- (p-tols) I) -1-cyclohexanecarboxylic acid 1-carboxy-3-cyclohexene-1-acetic acid oleic acid n- (diphenylmethyl) phthalic acid

2-karboxybenzaldehyd kyselina tetrafluórjantárová kyselina izo-oktánová kyselina 3-kyanoškoricová kyselina 2,3,5-trifluórfenyloctová kalceínová modrá kyselina 4-etoxy-3-metoxyfenyloctová kyselina 1 -amino-4-bróm-9,10-dioxo-9,10-dihydro-antracén-2-karboxylová kyselina karboxymetoxymetyl-pentaoxa-bicyklo(15.3.1)heneikoza-trién-21-karboxylová kyselina 3-((r)-2-karboxypiperazín-4-yl)-propyl-1 -fosfónová kyselina tetraoxa-23-aza-tricyklo( 17.3.1.1 (8,12))tetrakoza-hexaén-24-karboxylová kyselina [4-oxo-5-(5-fenyl-furán-2-ylmetylén)-2-tioxo-tioxo-tiazolidín-3-yl]octová kyselina 2-(4-(3,5-dichlór-pyridín-2-yloxy)-fenoxy)-propiónová kyselina 2,6-dimetoxy-3-nitrobenzoová kyselina 4-sulfoftalová kyselina 15-(4-jódfenyl)-pentadekánová kyselina 13-fenylsulfanyl-tridekánová kyselina 2-oktyldodekánová kyselina c/s-1O-heptadecénová kyselina n-etyl-1-glutámová kyselina 2’-chlór-5’-(trifluórmetyl)sukcínanilová kyselina 2,6-dichlórbenzoová kyselina brasidová2-carboxybenzaldehyde tetrafluorosuccinic acid iso-octanoic acid 3-cyanocinnamic acid 2,3,5-trifluorophenylacetic acid calceinic blue 4-ethoxy-3-methoxyphenylacetic acid 1-amino-4-bromo-9,10-dioxo-9,10- dihydro-anthracene-2-carboxylic acid carboxymethoxymethyl-pentaoxa-bicyclo (15.3.1) heneicoza-triene-21-carboxylic acid 3 - ((r) -2-carboxypiperazin-4-yl) -propyl-1-phosphonic acid tetraoxa- 23-aza-tricyclo (17.3.1.1 (8,12)) tetracoza-hexaene-24-carboxylic acid [4-oxo-5- (5-phenyl-furan-2-ylmethylene) -2-thioxo-thioxo-thiazolidine- 3-yl] acetic acid 2- (4- (3,5-dichloro-pyridin-2-yloxy) -phenoxy) -propionic acid 2,6-dimethoxy-3-nitrobenzoic acid 4-sulfophthalic acid 15- (4-iodophenyl) ) -pentadecanoic acid 13-phenylsulfanyl-tridecanoic acid 2-octyldodecanoic acid cis-10-heptadecenoic acid n-ethyl-1-glutamic acid 2'-chloro-5 '- (trifluoromethyl) succinilic acid 2,6-dichlorobenzoic acid br asidová

-117 --117 -

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kyselina naftazín-8,8'-disulfónovánaphthasin-8,8'-disulfonic acid

5-karboxy-3-metylflavón kyselina 1,6-dibróm-2-hydroxynaftalén-3-karboxylová kyselina alfa-brómheptánová kyselina (4-metyl-5-(2,2,2-trichlór-etyl)-tiazol.2-ylsulfanyl)octová kyselina d-(+)-treo-3-hydroxyasparágová kyselina 5-(metyltio)-salicylová kyselina 4-hydroxybenzoová kyselina 2-[[2-(4-fluórfenyl)hydrazíno]karbonyl]benzoová kyselina 3-(4-n-oktyloxybenzoyl)propiónová kyselina 3-fenyl-naftalén-2-karboxylová kyselina 4-metyloktánová kyselina fenantrén-4-karboxylová kyselina benzénpentakarboxylová kyselina 9-decénová kyselina 4,5-dihydro-3-metyl-5-oxo-1-fenyl-pyrazol-4-ditiokarboxylová kyselina 3-(3-(3,4,5-trimetoxy-fenyl)-akryloylamino)-benzoová kyselina 4,5,5,5-tetrafluór-4-trifluórmetyl-2-penténová kyselina fenyl-(toluén-4-sulfonyl)-octová kyselina 11-kyanoundekánová kyselina 2,5-dibrómtereftalová kyselina 2-chlór-5-(trichlórmetyltio)benzoová kyselina (rs)-1-amino-3-(fosfonometylén)cyklobután-karboxylová kyselina (r)-1 -amino(1-fenyl)metán-fosfónová kyselina (+)-4'-nitrotartranilová kyselina 5-metoxy-1,3-benzéndikarboxylová kyselina (s)-2-chlór-3-metylmaslová kyselina 5-etyl-2-metyl-1 -oxy-izonikotínová kyselina 1,3,5-trimetyl-1,3,5-cyklohexántrikarboxylová kyselina 5-hydroxy-2-metyl-4-nitrobenzoová kyselina 2,6-dimetyl-4-hexadecyloxybenzénsulfónová kyselina p-(trimetylsilyl)fenyl-octová5-carboxy-3-methylflavone 1,6-dibromo-2-hydroxynaphthalene-3-carboxylic acid alpha-bromoheptanoic acid (4-methyl-5- (2,2,2-trichloroethyl) thiazol-2-ylsulfanyl) ) acetic acid d - (+) - Threo-3-hydroxyaspartic acid 5- (methylthio) -salicylic acid 4-hydroxybenzoic acid 2 - [[2- (4-fluorophenyl) hydrazino] carbonyl] benzoic acid 3- (4-n) -octyloxybenzoyl) propionic acid 3-phenyl-naphthalene-2-carboxylic acid 4-methyloctanoic acid phenanthrene-4-carboxylic acid benzenepentacarboxylic acid 9-decenic acid 4,5-dihydro-3-methyl-5-oxo-1-phenyl-pyrazole -4-dithiocarboxylic acid 3- (3- (3,4,5-trimethoxy-phenyl) -acryloylamino) -benzoic acid 4,5,5,5-tetrafluoro-4-trifluoromethyl-2-pentenoic acid phenyl- (toluene- 4-sulfonyl) -acetic acid 11-cyanoundecanoic acid 2,5-dibromo-terephthalic acid 2-chloro-5- (trichloromethylthio) benzoic acid (rs) -1-amino-3- (phosphonomethylene) cyclobutanecarboxylic acid (r) -1 amino (1-phenyl) methyl ан-phosphonic acid (+) - 4'-nitrotartranilic acid 5-methoxy-1,3-benzenedicarboxylic acid (s) -2-chloro-3-methylbutyric acid 5-ethyl-2-methyl-1-oxy-isonicotinic acid 1 3,5-trimethyl-1,3,5-cyclohexanetricarboxylic acid 5-hydroxy-2-methyl-4-nitrobenzoic acid 2,6-dimethyl-4-hexadecyloxybenzenesulfonic acid p- (trimethylsilyl) phenyl acetic acid

-118--118-

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kyselina boc-1-asparágová kyselina izoindolin-1 -ón-2-(3-metyl-2-maslová) kyselina 3-(/?’-fenylacetyl-hydrazínokarbonyl)-propiónová kyselina glutárová kyselina 2-(1,3-dioxo-1,3-dihydro-izoindol-2-yl)-3-metyl-maslová kyselina 3-(p-chlórfenoxy)propiónová kyselina n-n-propyl-1-asparágová kyselina 3-fosfono-benzoová kyselina (z)-5-fluór-2-metyl-1 -[[4-(metyl-sulfinyl)fenyl]metylén]-1 -h-indén-3-octová kyselina difenylmetán-4-karboxylová kyselina (+/-)-1,1'-bi nafty l-2,2'-d i karboxylová kyselina (m-tolyl)-fosfónová kyselina chlórmetylfosfónová kyselina 2-(dibenzotiofén-2-ylkarbonyl)benzoová kyselina d-(-)-a-(4-etyl-2,3-dioxo piperzinyl)-karbocamid-4-hydroxyfenyl-octová kyselina 2,-terc-butyl-bifenyl-3-karboxylová kyselina linolénlaidová kyselina sulfojantárová kyselina 5-metyl-2-(orto-tolyl)-hexánová kyselina 3-terc-butyl-4-hydroxybenzoová kyselina n-butylfosfónová kyselina 4-amino-2,7-naftaléndisulfónová kyselina 3-(4-(6-(4-(2-karboxy-etyl)-6-oxo-hexanoyl)-fenyl)-propiónová kyselina 1 -(2-kyano-etyl)-5-oxo-pyrolidín-2-karboxylová kyselina 3-(2-oxo-benzotiazol-3-yl)-propiónová kyselina 2-metylvalérová kyselina beta-azido-o-benzoyl-mliečna kyselina 4-(2-hydroxyetoxy)salicylová kyselina 2,4-dihydroxytiazol-5-octová kyselina n-alfa-fmoc-n-gama-aloc-1 -diaminomaslová kyselina nitrometántrispropiónová kyselina ŕrans-chryzantémum monokarboxylováboc-1-aspartic acid isoindolin-1-one-2- (3-methyl-2-butyric) 3- (R-phenylacetyl-hydrazinocarbonyl) -propionic acid glutaric acid 2- (1,3-dioxo- 1,3-dihydro-isoindol-2-yl) -3-methylbutyric acid 3- (p-chlorophenoxy) propionic acid n-propyl-1-aspartic acid 3-phosphonobenzoic acid (z) -5-fluoro- 2-Methyl-1 - [[4- (methylsulfinyl) phenyl] methylene] -1-h-indene-3-acetic acid Diphenylmethane-4-carboxylic acid (+/-) - 1,1'-Bi naphthyl -2,2'-di-carboxylic acid (m-tolyl) -phosphonic acid chloromethylphosphonic acid 2- (dibenzothiophen-2-ylcarbonyl) benzoic acid d - (-) - α- (4-ethyl-2,3-dioxo piperzinyl) -carbocamide-4-hydroxyphenyl-acetic acid 2 , -tert-butyl-biphenyl-3-carboxylic acid linolenlaidic acid sulfosuccinic acid 5-methyl-2- (ortho-tolyl) -hexanoic acid 3-tert-butyl-4-hydroxybenzoic acid n-butylphosphonic acid 4-amino-2,7-naphthalenedisulfonic acid 3- (4- (6- (4- (2-carboxyethyl) -6-o) xo-hexanoyl) -phenyl) -propionic acid 1- (2-cyano-ethyl) -5-oxo-pyrrolidine-2-carboxylic acid 3- (2-oxo-benzothiazol-3-yl) -propionic acid 2-methylvaleric acid beta-azido-o-benzoyl-lactic acid 4- (2-hydroxyethoxy) salicylic acid 2,4-dihydroxytiazole-5-acetic acid n-alpha-fmoc-n-gamma-aloc-1-diaminobutyric acid nitromethane trispropionic acid trans-chrysanthemum monocarboxylic

-119--119-

• · · • · • 888 • · · • · • 888 e e 8 8 • · e e 8 8 • · 8888 * 8 8888 * 8 8 8 8 8 8 88 8 8 8 8 8 8 8 8 88 8 8 8 • 8 ·· • 8 ·· • 8 • 8 88 88 8 8 88 8 8 88

kyselina n-(2-metyl-4-nitrofenyl)ftalámová kyselina 2-etylundekánová kyselina 2',6'-dichlórmaleanilová kyselina dodecylsulfanyl-octová kyselina 1,2,3,4-cyklobutántetrakarboxylová kyselina trans-9,10-epoxystearová kyselina 5-acetoxy-izokaprónová kyselina tricyklo(9.2.2.1 (4,8))hexadeka-1 (14),4(16),5,7,11(15),12-hexaén-karboxylová kyselina 2-hydroxy-2-trifluórmetyl-dokoz-4-énová kyselina 4-ŕerc-butylfenyloctová kyselina 5-chlór-2-prop-2-inyloxy-benzoová kyselina 3-(3,4-dimetoxyfenyl)propiónová kyselina 2-acetylamino-3-(3-nitro-fenyl)-akrylová kyselina 2-(3-(2-fenylcyklopropyl)ureido)octová kyselina 4-metoxysalicylová kyselina 2-hexadecénová kyselina o-yodozobenzoová kyselina n-(3-acetylfenyl)-maleanilová kyselina acetylneuramínová kyselina 4-hydroxy-1 -fenyl-naftalén-2-karboxylová kyselina 4-bifenyloctová kyselina 5-bróm-4-chlór-2-fluórbenzoová kyselina 2'-metoxy-5'-metylsukcínanilová kyselina 2-karbamoyl-2-fenyl-maslová kyselina (4-amino-5-(4-chlór-fenyl)-pyrimidín-2-ylsulfanyl)-octová kyselina 2-bróm-5-nitrobenzoová kyselina dichrostachinová kyselina (s)-3-(4-ŕerc-butoxyfenyl)butánová kyselina 9-fluorénoctová kyselina n-butylmaleámová kyselina 4-bróm-1-naftoová • ·· ·· ···· ·· ·· · ·· 4 4 4 4 • ··· · 4 4 · · · ··· f 444 4n- (2-methyl-4-nitrophenyl) phthalic acid 2-ethylenedecanoic acid 2 ', 6'-dichloromaleanilic acid dodecylsulfanyl acetic acid 1,2,3,4-cyclobutanetetracarboxylic acid trans-9,10-epoxystearic acid 5- acetoxy-isocaproic acid tricyclo (9.2.2.1 (4,8)) hexadeca-1 (14), 4 (16), 5,7,11 (15), 12-hexaenecarboxylic acid 2-hydroxy-2-trifluoromethyl- docos-4-enoic acid 4-tert-butylphenylacetic acid 5-chloro-2-prop-2-ynyloxybenzoic acid 3- (3,4-dimethoxyphenyl) propionic acid 2-acetylamino-3- (3-nitrophenyl) -acrylic acid 2- (3- (2-phenylcyclopropyl) ureido) acetic acid 4-methoxysalicylic acid 2-hexadecenoic acid o-yodozobenzoic acid n- (3-acetylphenyl) -maleanil acetylneuraminic acid 4-hydroxy-1-phenyl-naphthalene 2-carboxylic acid 4-biphenylacetic acid 5-bromo-4-chloro-2-fluorobenzoic acid 2'-methoxy-5'-methylsuccinilic acid 2-carbamoyl-2-phenylbutyric acid (4-amino-5- (4 -c 2-Bromo-5-nitrobenzoic acid Dichrostachinic acid (s) -3- (4-tert-butoxyphenyl) butanoic acid 9-Fluoro-acetic acid n-butylmaleamic acid 4-bromo-phenyl) -pyrimidin-2-ylsulfanyl) -acetic acid -1-naphtha 4 4 4 4 4 4 4 4 44

-120kyselina 3-fenylglutárová kyselina 4-bróm-2-metylbenzoová kyselina arachová kyselina 2-(p-ŕerc-butylbenzoyl)akrylová kyselina nitrilotris(metylén)trifosfónová kyselina ketomalónová kyselina 5-chlórsalicylová kyselina 2,4,6-trichlórfenoxyoctová kyselina (4-acetylamino-fenyl)-octová kyselina 4-(2-(1-metyl-1 h-chinolín-4-ylidén)-etylidénamino)-benzoová kyselina n-(4-chlórfenyl)malonámová kyselina 2-(4-cyklohexylbenzoyl)akrylová kyselina c/s-hexahydro-n-(2-(trifluórmetyl)fenyl)ftalámová fmoc-d-homofenylalanín kyselina 1 -fenyl-1 -cyklohexánkarboxylová kyselina dibenzyl-fosfínová kyselina (2-hydroxyfenoxy)octová kyselina (2-brómfenyl)fosfónová kyselina 3,4-dimetoxy-2,5-furándikarboxylová kyselina n-acetylmuramová kyselina pentakozánová kyselina 5-fluór-2-metoxyfenyloctová kyselina n-(2,6-dimetylfenyl)maleámová kyselina 3-(pentametylbenzoyl)akrylová kyselina 1,2-acetamidomaslová kyselina ŕrans-2-(p-chlórbenzoyl)-1 -cyklohexán-karboxylová kyselina 1,1-cyklohexándioctová kyselina 2-(1 -oktadecenyl)jantárová kyselina n-(4-chlórfenyl)glutarámová kyselina c/s-11,14,17-eikozatriénová kyselina antracén-9,10-dikarboxylová kyselina 2,3,4-trifenylmaslová • · * ·· ···· · · ·· · · · · · · · • ··· · · · β ·-120 acid 3-phenylglutaric acid 4-bromo-2-methylbenzoic acid arachic acid 2- (p-tert-butylbenzoyl) acrylic acid nitrilotris (methylene) triphosphonic acid ketomalonic acid 5-chlorosalicylic acid 2,4,6-trichlorophenoxyacetic acid (4- Acetylamino-phenyl) -acetic acid 4- (2- (1-methyl-1H-quinolin-4-ylidene) -ethylidenamino) -benzoic acid 2- (4-Cyclohexyl-benzoyl) -acrylic acid cis-Hexahydro-1- (2- (trifluoromethyl) phenyl) phthalic fmoc-d-homophenylalanine 1-Phenyl-1-cyclohexanecarboxylic acid dibenzylphosphinic acid (2-hydroxyphenoxy) acetic acid (2-bromophenyl) phosphonic acid 3 4-dimethoxy-2,5-furanedicarboxylic acid n-acetylmuramic acid pentacosanoic acid 5-fluoro-2-methoxyphenylacetic acid n- (2,6-dimethylphenyl) maleic acid 3- (pentamethylbenzoyl) acrylic acid 1,2-acetamidobutyric acid trans -2- (p-chlorobenzoyl) -1-cyclohexanecarboxylic acid 1,1-cyclohexanediacetic acid 2- (1-octadecenyl) succinic acid n- (4-chlorophenyl) glutaramic acid cis-11,14,17-eicosatrienoic acid anthracene-9,10-dicarboxylic acid 2,3,4 -triphenylbuttered • β · tr tr · β tr tr tr

-121 kyselina 4'-(etoxykarbonyl)glutaranilová kyselina 1 -(n-cbz-amino)cyklo-propánkarboxylová kyselina n-(chlóracetyl)-1 -asparágová kyselina 4-etoxy-3-metoxyškoricová kyselina dipivaloyl-1 -vínna kyselina 2,6-bis-fenoxymetyl-benzoová kyselina 4-acetamido-3-nitrobenzoová kyselina omega-ketoheptánová kyselina 3,5-d/-ŕerc-butyl-4-hydroxyfenylpropiónová kyselina 8(r)-hydroxy-(5z,9e,11z,14z)-eikozatetraénová kyselina 3-antracén-9-yl-propínová kyselina 3-[4-(4-chlórfenyltio)-3-nitrofenyl]akrylová kyselina d/-treo-4-fluórglutámová kyselina n-p-toluénsulfonylimino-S.S'-dipropiónová kyselina 2,,5,-dichlórmaleanilová kyselina o-tolyloctová kyselina oktafluóradipová kyselina 3-[2,2,3,3A4,5l5-oktafluór-1-(tnfluórmetyl)cyklopentyl)propánová kyselina 7-epi-jasmonová kyselina n-karbamyl-d/-asparágová kyselina 3-kyano-5-metoxy-2-metyl-benzoová kyselina tetradekándiová kyselina 5,5-dimetyl-4-hydroxy-4-(4-fenoxyfenyl)-2-hexínová kyselina d-ftalimidobenzoová kyselina 4-fluórsulfonyl-1 -hydroxy-2-naftoová kyselina 4-(2-chlór-5-(trifluórmetyl)fenylazo)-3-hydroxy-2-naftoová kyselina oxalurová kyselina c/s-2-benzoyl-1 -cyklohexánkarboxylová kyselina 4-oxo-4-fenantren-2-yl-maslová kyselina 15-fenylpentadekánová kyselina benzylizovanilová kyselina 21-brómhenikozánová *· ······ ·· ··· ·· · ··· • ··· · · · · · • · * · · · · · · ·-121 4 '- (ethoxycarbonyl) glutaranilic acid 1- (n-cbz-amino) cyclopropanecarboxylic acid n- (chloroacetyl) -1-aspartic acid 4-ethoxy-3-methoxycinnamic acid dipivaloyl-1-tartaric acid 2, 6-bis-phenoxymethyl-benzoic acid 4-acetamido-3-nitrobenzoic acid omega-ketoheptanoic acid 3,5-di-tert-butyl-4-hydroxyphenylpropionic acid 8 (r) -hydroxy- (5z, 9e, 11z, 14z 3-Anthracen-9-yl-propionic acid 3- [4- (4-chlorophenylthio) -3-nitrophenyl] acrylic acid 1-threo-4-fluoroglutamic acid n-toluenesulfonylimino-5'-dipropionic acid acid 2, 5, -dichlórmaleanilová acid, tolyl acid, oktafluóradipová-3- [l 2,2,3,3A4,5 5-octafluoro-1- (trifluoromethyl) cyclopentyl) propanoic acid, 7-epi jasmonic acid, n-carbamyl 3-cyano-5-methoxy-2-methylbenzoic acid tetradecanedioic acid 5,5-dimethyl-4-hydroxy-4- (4-phenoxyphenyl) -2-hexanoic acid d-phthalimidobe 4-Fluorosulfonyl-1-hydroxy-2-naphthoic acid 4- (2-chloro-5- (trifluoromethyl) phenylazo) -3-hydroxy-2-naphthoic acid oxaluric acid cis-2-benzoyl-1-cyclohexanecarboxylic acid 4-oxo-4-phenanthren-2-yl-butyric acid 15-phenylpentadecanoic acid benzylizovanilic acid 21-bromoenicosanoic acid * · ················ · · · · · · · · · · · · ·

-122kyselina 6-hydroxypyrazíne-2-karboxylová kyselina n-(2,4-dimetylfenyl)-1,2,3,6-tetrahydroftalámová kyselina 2-(2-nitrobenzyltio)octová kyselina neodekánová kyselina 4-(2-fenoxyetoxy)benzoová kyselina 2-(6-metoxy-3-nitropyrid-2-yltio)propiónová kyselina 12-hydroxystearová kyselina 3-jód-2-metylbenzoová kyselina difenolová kyselina 3-(trifluórmetyltio)fenyloctová kyselina 4-metyl-2-[4-trifluórmetyl)fenyl]tiazol-5-karboxylová kyselina 3-etoxytiofén-2-karboxylová kyselina (-)-4'-chlórtartranilová kyselina 2,5-difenyl-furán-3,4-dikarboxylová kyselina metylmalónová kyselina p-pentyloxyškoricová kyselina 6-oxo-1,14-tetradekándikarboxylová kyselina 2-(metylaminometyl)tartronová kyselina (3-kyano-2-metoxykarbonylmetylén-6-(meo-ph)-3-me-cyklohexyl)-octová kyselina 2-fenylpropiónová kyselina 1-cyklohexenyloctová kyselina 3-(4-hydroxy-fenyl)-2-((naftalén-2-ylmetylén)-amino)-propiónová kyselina (5-karboxymetylsulfanyl-2-tioxo-[1,3]ditiol-4-ylsulfanyl)-octová kyselina alfa-kyano-4-hydroxy-3-metoxyškoricová kyselina 6-trifluórmetyltieno[3,2-b]pyridín-2-karboxylová kyselina boc-1-alfa terc-butylglycín kyselina (5-etyl-4-hydroxy-5-metyl-pyrimidín-2-ylsulfanyl)-octová kyselina 4-metoxytiofén-3-karboxylová kyselina 4'-bróm-3'-metylhexahydroftalanilová kyselina 3-[2-(4-chlórfenyltio)-5-nitrofenyl]akrylová kyselina c/s-n-(4-(etoxykarbonyl)fenyl)hexahydroftalámová kyselina 8-oxo-bicyklo(3.2.1 )okt-6-én-3-karboxylová-122 6-hydroxypyrazine-2-carboxylic acid n- (2,4-dimethylphenyl) -1,2,3,6-tetrahydrophthalic acid 2- (2-nitrobenzylthio) acetic acid neodecanoic acid 4- (2-phenoxyethoxy) benzoic acid 2- (6-methoxy-3-nitropyrid-2-ylthio) propionic acid 12-hydroxystearic acid 3-iodo-2-methylbenzoic acid diphenolic acid 3- (trifluoromethylthio) phenylacetic acid 4-methyl-2- [4-trifluoromethyl) phenyl ] thiazole-5-carboxylic acid 3-ethoxythiophene-2-carboxylic acid (-) - 4'-chlorotartranilic acid 2,5-diphenyl-furan-3,4-dicarboxylic acid methyl malonic acid p-pentyloxycinnamic acid 6-oxo-1, 14-Tetradecanedicarboxylic acid 2- (methylaminomethyl) tartronic acid (3-cyano-2-methoxycarbonylmethylene-6- (meo-ph) -3-methoxycyclohexyl) -acetic acid 2-phenylpropionic acid 1-cyclohexenylacetic acid 3- (4- hydroxy-phenyl) -2 - ((naphthalen-2-ylmethylene) -amino) -propionic acid (5-carboxymethylsulfanyl-2-thioxo- [1,3] dithiol-4-ylsulfanyl) -acetic acid 6-Trifluoromethylthieno [3,2-b] pyridine-2-carboxylic acid alpha-cyano-4-hydroxy-3-methoxy cinnamic acid boc-1-alpha tert-butylglycine (5-ethyl-4-hydroxy-5- methyl-pyrimidin-2-ylsulfanyl) -acetic acid 4-Methoxythiophene-3-carboxylic acid 4'-bromo-3'-methylhexahydrophthalanic acid 3- [2- (4-chlorophenylthio) -5-nitrophenyl] acrylic acid cis / n- (4- (ethoxycarbonyl) phenyl) hexahydrophthalic acid 8-oxo-bicyclo (3.2.1) oct-6-ene-3-carboxylic acid

ΦΦ Μ ···· ΦΦ • φ · φ «. φ · φφφ φφφ φ ·Φ · ···· ΦΦ • φ · φ «. φ · φφφ φφφ φ ·

-123kyselina 2-(trifluórmetoxy)fenyloctová kyselina n-boc-d.1-2-aminotetralín-2-karboxylová kyselina 2-(3-chlór-5-trifluórmetyl-2-pyridyltio)-1-metylimidazol-5-karboxylová kyselina 4-(2-(4,4-dimetyl-chroman-6-yl)-propenyl)-benzoová kyselina 2-formyl-4-nitrofenoxyoctová kyselina 2-chlór-5-(metylsulfamoyl)-benzoová kyselina 4-chlór-2-(2-kyano-etylamino)-benzoová kyselina pentafluórpropiónová kyselina ŕrans-6-oktadecénová kyselina n-alfa-z-glycyl-1 -asparágová kyselina n-acetylglycín kyselina (+)-lich-esterová kyselina 3-hydroxyoktadekánová kyselina 4'-etylsukcínanilová kyselina 3,4,5-trifluórfenyloctová kyselina c/s-hexahydro-n-(4-nitrofenyl)ftalámová kyselina fmoc-(4-karboxymetyl)-piperidín-(2-acetyl-4,5-dimetoxy-fenyl)-octová kyselina 2-(4-metoxy-1 -naftyl)-1 -metyl-5-oxo-3-pyrolidínkarboxylová kyselina 3-(4-etoxybenzoyl)akrylová kyselina acetopyrohroznová kyselina aceaftén-5-karboxylová kyselina 3-hydroxy-6-metoxy-indán-1-karboxylová kyselina 4-(2-cyklohexenyloxy)benzoová kyselina 2-hydroxy-6-izopropyl-3-metylbenzoová kyselina 3,5-dichlór-4-metoxybenzoová kyselina nonánová kyselina 2-nitrofenyloctová kyselina 4-[(3-nitro-2-pyridyl)amino]butánová kyselina 3’-chlór-4’-metylmaleanilová kyselina 3-(2-brómbenzoyl)propiónová kyselina 3-fluór-adamantán-1 -karboxylová kyselina 2-(trifluórmetyl)benzoová-123 2- (trifluoromethoxy) phenylacetic acid n-boc-d -1-2-aminotetraline-2-carboxylic acid 2- (3-chloro-5-trifluoromethyl-2-pyridylthio) -1-methylimidazole-5-carboxylic acid 4 - (2- (4,4-Dimethyl-chroman-6-yl) -propenyl) -benzoic acid 2-formyl-4-nitrophenoxyacetic acid 2-chloro-5- (methylsulfamoyl) -benzoic acid 4-chloro-2- ( 2-cyano-ethylamino) -benzoic acid pentafluoropropionic acid trans-6-octadecenoic acid n-alpha-z-glycyl-1-aspartic acid n-acetylglycine (+) - odd-ester acid 3-hydroxyoctadecanoic acid 4'-ethylsuccinilic acid 3,4,5-Trifluorophenylacetic acid cis-hexahydro-1- (4-nitrophenyl) phthalic acid fmoc- (4-carboxymethyl) -piperidine- (2-acetyl-4,5-dimethoxy-phenyl) -acetic acid 2 - (4-Methoxy-1-naphthyl) -1-methyl-5-oxo-3-pyrrolidinecarboxylic acid 3- (4-ethoxybenzoyl) acrylic acetopyruvic acid Aceaphthene-5-carboxylic acid 3-hydroxy-6-methoxy-indan- 1-carboxylic acid 4 - (2-cyclohexenyloxy) benzoic acid 2-hydroxy-6-isopropyl-3-methylbenzoic acid 3,5-dichloro-4-methoxybenzoic acid nonanoic acid 2-nitrophenylacetic acid 4 - [(3-nitro-2-pyridyl) amino] butanoic acid 3'-chloro-4'-methylmaleanilic acid 3- (2-bromobenzoyl) propionic acid 3-fluoro-adamantane-1-carboxylic acid 2- (trifluoromethyl) benzoic acid

Φ φ φ φ · ·· · ·· • φ · · · · · ··· φ φ φ φ ·Φ · · · · • · • · • · • · · ·

-124kyselina 17-oktadecínová kyselina 1 -(4-metoxyfenyl)-6-metyl-4-oxo-1,4-dihydro-3-pyridínkarboxylová kyselina 3-fluór-2,4,6-trimetyl-benzoová kyselina 4,4'-azobis-(4-kyanovaleriánová) kyselina 5-aminoizoftalová kyselina 6-metyl-2-fenyl-5,7b-diaza-cyklopenta(cd)indén-3-karboxylová kyselina alfa-ketoglutárová kyselina 2-chlór-4-nitrobenzoová kyselina 4-hydroxy-10-oxo-9-oxa-tricyklo(6.2.1.0(1,5))undekáin-2-karboxylová kyselina n-(2-tienylmetylén)antranilová kyselina /7-(3-metoxyfenyl)maleámová kyselina 10-doxyl-stearová kyselina 1-hydroxy-2-naftoová kyselina 3'-οΙίΙ0γ-3,4,5,6-tetrachlórftalanilová kyselina pentán-1-fosfónová kyselina 1-cysteinsulfínová kyselina 3-fenyl-3-propylglutárová kyselina 6-ŕerc-butyl-1,1-dimetyl-indán-4-karboxylová kyselina 3,5-diacetoxybenzoová kyselina 3-(4-chlór-fenyl)-3-(2,2-dimetyl-propionylamino)-propiónová kyselina 8a-metyl-oktahydro-naftalén-4a-karboxylová kyselina rezorcinol-o,o-dioctová kyselina 5-bróm-4-chlór-4,5,5-trifluór-2-penténová kyselina (1 .ľ^'.ľ'Jterfenyl-S'.S'-dikarboxylová kyselina maleámová kyselina 2-amino-4-metoxy-benzoová gama-cyklohexylester kyseliny n-boc-1-glutámovej kyselina 4-(difluórmetoxy)benzoová kyselina 3,4,5,6-tetrachlór-34trifluórmetyl)ftalanilová kyselina 3,7,11,15-tetrametylhexadekánová kyselina 4-nitro-2-fosfono-benzoová kyselina 3-[2-(4-metylfenyltio)-5-nitrofenyl]akrylová-124 17-octadecinic acid 1- (4-methoxyphenyl) -6-methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid 3-fluoro-2,4,6-trimethylbenzoic acid 4,4 ' -azobis- (4-cyanovalerioic acid) 5-aminoisophthalic acid 6-methyl-2-phenyl-5,7b-diaza-cyclopenta (cd) indene-3-carboxylic acid alpha-ketoglutaric acid 2-chloro-4-nitrobenzoic acid 4 -hydroxy-10-oxo-9-oxa-tricyclo (6.2.1.0 (1,5)) undecain-2-carboxylic acid n- (2-thienylmethylene) anthranilic acid / 7- (3-methoxyphenyl) maleic acid 10-doxyl -stearic acid 1-hydroxy-2-naphthoic acid 3'-ωΙΙΙΙγ-3,4,5,6-tetrachlorophthalanilic acid pentane-1-phosphonic acid 1-cysteine sulphonic acid 3-phenyl-3-propylglutaric acid 6-tert-butyl- 1,1-Dimethyl-indane-4-carboxylic acid 3,5-diacetoxybenzoic acid 3- (4-chloro-phenyl) -3- (2,2-dimethyl-propionylamino) -propionic acid 8a-Methyl-octahydro-naphthalene- 4α-carboxylic acid resorcinol-o, o-diacetic acid 5-bromo-4 - Chloro-4,5,5-trifluoro-2-pentenoic acid (1,1'''''-Phenyl-5'''''-dicarboxylic acid maleic acid 2-Amino-4-methoxy-benzoic acid gamma-cyclohexyl ester n -boc-1-glutamic acid 4- (difluoromethoxy) benzoic acid 3,4,5,6-tetrachloro-34-trifluoromethyl) phthalic acid 3,7,11,15-tetramethylhexadecanoic acid 4-nitro-2-phosphonobenzoic acid 3- [2- (4-methylphenylthio) -5-nitrophenyl] acrylic acid

-125 --125 -

• BB • B • BBB • BB • B • BBB BB BB BBBB • • BBBB • • • I B B B BB • B B • I B B B BB • B B • t • t • • • • • · B · • · B · BB BB BB BB • B BB • B BB

kyselina imidazol-2-karboxylová kyselina 4-jódbenzoová kyselina 2-(4-fluórfenyl )-acetooctová kyselina 2,2-dimetyl-but-3-énová kyselina 4'-acetoxy-bifenyl-4-karboxylová kyselina 2-bróm-5-fluórbenzoová kyselina n-(3,5-dimetylfenyl)-1,2,3,6-tetrahydroftalámová kyselina 2,3-dihydro-1-(1 h)-indolpropánová kyselina 5-benzyloxykarbonylamino-pentánová kyselina alfa-izopropylidénaminooxypropiónová kyselina alfa-bróm-1 -adamantánoctová kyselina 5-bróm-4-chlór-4,5,5-trifluórpentánová kyselina 4-(2,4-dimetylfenyl)maslová kyselina 5-(4-(4-(4-karboxy-butyl)-benzyl)-fenyl)-pentánová kyselina 1,4-dihydro-2-metylbenzoová kyselina difenyloctová kyselina 2,7-naftaléndikarboxylová fenyl-beta-d-tioglukuronid kyselina exo-2-chlór-5,5-etyléndioxy-bicyklo[2.2.1 ]heptán-syn-7-karboxylová kyselina 4-(3-butenyloxy)benzoová kyselina 3-(2-(4-nitro-fenyl)-acetylamino)-propiónová kyselina 3-chlór-6-metylbenzoová kyselina 3-fluórbenzoová kyselina hydroxy(3-)2,4,5-trifluórbenzoová kyselina 10-bróm-9-antracénkarboxylová kyselina difenová kyselina p-anízová kyselina (r)-(+)-2-brómhexánová kyselina 3-bróm-6-(karboxymetyl-amino)-2-chlór-benzoová kyselina n-metyl-d/-asparágová kyselina homoftalová kyselina cinamylidén-octováimidazole-2-carboxylic acid 4-iodobenzoic acid 2- (4-fluorophenyl) -acetoacetic acid 2,2-dimethyl-but-3-enoic acid 4'-acetoxy-biphenyl-4-carboxylic acid 2-bromo-5- fluorobenzoic acid n- (3,5-dimethylphenyl) -1,2,3,6-tetrahydrophthalic acid 2,3-dihydro-1- (1h) -indolpropanoic acid 5-benzyloxycarbonylamino-pentanoic acid alpha-isopropylideneamininooxypropionic acid alpha-bromo 5-Bromo-4-chloro-4,5,5-trifluoropentanoic acid 5-bromo-4-chloro-4- (2,4-dimethylphenyl) butyric acid 5- (4- (4- (4-carboxy-butyl) -benzyl)) -phenyl) -pentanoic acid 1,4-dihydro-2-methylbenzoic acid diphenylacetic acid 2,7-naphthalenedicarboxylic acid phenyl-beta-d-thioglucuronide exo-2-chloro-5,5-ethylenedioxy-bicyclo [2.2.1] heptane -syn-7-carboxylic acid 4- (3-butenyloxy) benzoic acid 3- (2- (4-nitro-phenyl) -acetylamino) -propionic acid 3-chloro-6-methylbenzoic acid 3-fluorobenzoic acid hydroxy (3- ) of 2,4,5-trifluoro- rbenzoic acid 10-bromo-9-anthracenecarboxylic acid diphenoic acid p-anisic acid (r) - (+) - 2-bromohexanoic acid 3-bromo-6- (carboxymethylamino) -2-chloro-benzoic acid n-methyl- d) aspartic acid, homophthalic acid, cinamylidene acetic acid

-126--126-

• ·· • · • ··· « · · • ·· • · • ··· «· · • · • • • · • · • • • · • · · · • « • · • · · • · · · • « • · • · · • · • · • · • · • · • · • · • · « · «· ·· «· ·· «· ·· · · • * • * • · • · • · • ·

kyselina 2,4,5-trifluórbenzoová kyselina oxo-(1 -oxo-1 -2,3,4-tetrahydro-fenantrén-2-yl)-octová kyselina 12-nitrododekánová kyselina dichlórdianilínotereftalová kyselina 3-p-tolyl-adamantán-1 -karboxylová kyselina 3-metoxy-9-oxo-5,7,8,9-tetrahydro-benzocykloheptén-6,6-dikarboxylová kyselina 4-chlór-3-nitro-benzénsulfínová kyselina 4-(2-metylkarbamoyl-acetylamino)-benzoová kyselina asym-hydrazíndioctová kyselina (4-(4-karboxymetánsulfonyl-fenylsulfanyl)-benzénsulfonyl)-octová kyselina 2-chlór-3-nitrobenzoová kyselina 2-etoxybenzoová kyselina 2-[(3-karboxy-propyl)-(toluén-4-sulfonyl)-amino]-benzoová kyselina 4'-brómhexahydroftalanilová kyselina (2-metoxykarbonylmetyl-cyklopropyl)-octová kyselina 2-(4-metylbenzylkarbamoyl)benzoová kyselina 2-hydroxyimino-3-fenyl-propiónová kyselina aminomalónová kyselina 2,5-bis(trifluórnietyl)hydroškoricová kyselina 2,6-difluórbenzoová kyselina 3,3'-ditiodipropiónová kyselina 9-oxo-1,2,4,5-tetrahydro-3h-10-oxo-2a-aza-aceantrylén-8-karboxylová kyselina 2-hydroxy-1 -naftalénoctová kyselina anilín-2,5-disulfónová kyselina 2-acetylbenzoová kyselina 2-tiofénglyoxylová kyselina 4'-metylglutaranilová kyselina 3-chlór-4-metylbenzoová kyselina 4-hydroxy-7-jód-10-oxo-9-oxa-tricyklo(6.2.1.0(1,5))undekán-2-karboxylová kyselina (3,5-dioxo-2,3,4,5-tetrahydro-(1,2,4)triazín-6-ylsulfanyl)-octová kyselina 2,5-bis(trifluórmetyl)benzoová kyselina 4-etyl-3-metyl-2-pyrolkarboxylová2,4,5-trifluorobenzoic acid oxo- (1-oxo-1 -2,3,4-tetrahydro-phenanthren-2-yl) -acetic acid 12-nitrododecanoic acid dichlorodianiline-terephthalic acid 3-p-tolyl-adamantane-1 3-Methoxy-9-oxo-5,7,8,9-tetrahydro-benzocycloheptene-6,6-dicarboxylic acid 4-chloro-3-nitro-benzenesulfonic acid 4- (2-methylcarbamoyl-acetylamino) -benzoic acid (4-carboxymethanesulfonyl-phenylsulfanyl) -benzenesulfonyl) -acetic acid 2-chloro-3-nitrobenzoic acid 2-ethoxybenzoic acid 2 - [(3-carboxypropyl) - (toluene-4-sulfonyl) (amino) -benzoic acid 4'-Bromo-hexahydrophthalanilic acid (2-methoxycarbonylmethyl-cyclopropyl) -acetic acid 2- (4-methylbenzylcarbamoyl) benzoic acid 2-hydroxyimino-3-phenylpropionic acid aminomalonic acid 2,5-bis (trifluoromethyl) ) cinnamic acid 2,6-difluorobenzoic acid 3,3'-dithiodipropionic acid 9-oxo-1,2,4,5-tetrahydro-3h-10-oxo-2 α-aza-aceantrylene-8-carboxylic acid 2-hydroxy-1-naphthaleneacetic acid aniline-2,5-disulfonic acid 2-acetylbenzoic acid 2-thiophene-glyoxylic acid 4'-methylglutaranilic acid 3-chloro-4-methylbenzoic acid 4-hydroxy -7-iodo-10-oxo-9-oxa-tricyclo (6.2.1.0 (1,5)) undecane-2-carboxylic acid (3,5-dioxo-2,3,4,5-tetrahydro- 2,4-triazin-6-ylsulfanyl) -acetic acid 2,5-bis (trifluoromethyl) benzoic acid 4-ethyl-3-methyl-2-pyrrolecarboxylic acid

-127--127-

• ·· • ·· ·· ···· ·· ···· ·· · ·· · • · • · • · · • · · • · ·· • · ·· • ··· • ··· • · · • · · • · · • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 1,2-fenyléndioxydioctová kyselina 5-fluór-2-(trifluórmetyl)fenyloctová kyselina 4-((2,4-dihydroxy-benzylidén)-amino)-benzoová kyselina 2-metyl-1 h-benzimidazol-5-karboxylová kyselina 4-( 1 ’, 1 '-dimetyl-1 '-hydroxypropyl)fenoxy-octová kyselina 11-(2-oxo-tetrahydro-furán-3-yl)-undekánová kyselina n-(4-fenoxyfenyl)glutarámová kyselina linolénová kyselina 2-(fenyltio)propiónová kyselina 2-(trifluórmety I)-1,8-naftyridín-3-karboxylová kyselina 7-oxooktánová kyselina 2-chlór-3-metoxytiofén-4-karboxylová kyselina benzilová kyselina anti-3-oxotricyklo(2.2.1.02,6)heptán-7-karboxylová kyselina íerc-butyloctová kyselina (3-benzyloxy-4-metoxy-fenyl)-hydroxy-octová kyselina jodovodíková kyselina 4-hydroxyfenyloctová kyselina 15-fenyl-3,3-dimetyl-pentadekánová kyselina r-4-metylmandlová kyselina 2-(4-fluórfenyl)-3-(3-metoxybenzoyl)propiónová kyselina 5-(4-karboxy-2-nitrofenoxy)izoftalová kyselina 5-nitro-1,10-fenantrolín-2,9-dikarboxylová kyselina 3-bróm-5-jódbenzoová kyselina tricyklo(8.2.2.2(4,7))hexadeka-hexaén-5,12-dikarboxylová kyselina 7-metoxykumarín-3-karboxylová kyselina (+)-4’-fluórtartranilová kyselina 2-[4-(4-chlórbenzoyl)-fenoxy]-2'-metylpropánová kyselina 5-fluór-izoftalová kyselina 3-(5-(2-karboxy-etánsulfonyl)-naftalén-1-sulfonyl)-propiónová kyselina salicylová kyselina (s)-2-(4-fluórfenyl)-3-metylmaslová * ·· ···· ·· ··· ·· · · · « • ··· · · · · ·1,2-phenylenedioxydiacetic acid 5-fluoro-2- (trifluoromethyl) phenylacetic acid 4 - ((2,4-dihydroxy-benzylidene) -amino) -benzoic acid 2-methyl-1H-benzimidazole-5-carboxylic acid 4 - (1 ', 1'-Dimethyl-1'-hydroxypropyl) phenoxyacetic acid 11- (2-oxo-tetrahydro-furan-3-yl) -undecanoic acid n- (4-phenoxyphenyl) glutaramic acid linolenic acid 2- (phenylthio) propionic acid 2- (trifluoromethyl) -1,8-naphthyridine-3-carboxylic acid 7-oxooctanoic acid 2-chloro-3-methoxythiophene-4-carboxylic acid benzilic acid anti-3-oxotricyclo (2.2.1.02, 6) heptane-7-carboxylic acid tert-butylacetic acid (3-benzyloxy-4-methoxy-phenyl) -hydroxy-acetic acid hydroiodic acid 4-hydroxyphenylacetic acid 15-phenyl-3,3-dimethyl-pentadecanoic acid r-4- 2- (4-fluorophenyl) -3- (3-methoxybenzoyl) propionic acid 5- (4-carboxy-2-nitrophenoxy) isophthalic acid 5-nitro-1,10-phenanthroline-2,9-dicarboxylic acid 3-Bromo-5-iodobenzoic acid tricyclo (8.2.2.2 (4,7)) hexadeca-hexaene-5,12-dicarboxylic acid 7-methoxycoumarin-3-carboxylic acid (+) - 4'-fluorotartranilic acid 2- [ 4- (4-chlorobenzoyl) -phenoxy] -2'-methylpropanoic acid 5-fluoro-isophthalic acid 3- (5- (2-carboxyethanesulfonyl) -naphthalene-1-sulfonyl) -propionic acid salicylic acid (s) - 2- (4-fluorophenyl) -3-methylbutyric acid

-128kyselina 4-acetamidobenzoová kyselina alfa.alfa-dimetylfenyloctová kyselina cyklopropyl-fenylglykolová kyselina 2-keto-d-galaktónová kyselina 2-[[(4-metoxyfenyl)sulfonyl](2-pyridyl)amino]octová kyselina 5-(4-chlór-2-nitrofenyl)-2-furoová kyselina etyléndiamín-n,n -bis(izopropylfosfónová), hydrát kyselina z-1-2-aminohexánová kyselina 1 -4-hydroxyprolín-o-fosforečná kyselina 2-(2-karboxy-fenylsulfanyl)-malónová kyselina melitová kyselina 1 -hydroxy-1 -cyklopropánkarboxylová kyselina (1 r)-(-)-(1-aminohexyl)fosfónová gama-benzylester kyseliny n-boc-d-glutámovej kyselina 4-(3-metoxy-benzoylamino)-benzoová kyselina 4-hydrazobenzoová kyselina 4-fluór-1-naftoová kyselina benzoyl-mliečna kyselina 3-buty 1-5-(2.6.6-trimetyl-1 -cyklohexén-1 -yl)-2,4-pentadiénová kyselina fmoc-1 -beta-aminomaslová kyselina (s)-3-hydroxymaslová kyselina n-(3,5-xylyl)glutarámová kyselina 4,5-dichlórftalová kyselina (s)-1-amino(1-fenyl)metán fosfónová kyselina 6-amino-2,3-dimetoxy-benzoová kyselina 4-(trifluórmetyl)škoricová kyselina /i-alfa-n-gama-d/-z-1 -diaminomaslová kyselina 2,3-dibrómmaslová kyselina ô^'-karbonylbis-Orimelitová) kyselina 4-(2-brómbenzoyl)maslová kyselina 6-hydroxypikolínová kyselina 4-(3-hydroxy-propylamino)-3-nitro-benzoová ·· ·· ···· ·· • · · · · · · ··« · · · 9 ·-128 4-acetamidobenzoic acid alpha.alpha.-dimethylphenylacetic acid cyclopropylphenylglycolic acid 2-keto-d-galactonic acid 2 - [[(4-methoxyphenyl) sulfonyl] (2-pyridyl) amino] acetic acid 5- (4-chloro) -2-nitrophenyl) -2-furoic acid ethylenediamine-n, n -bis (isopropylphosphonic acid) z-1-2-aminohexanoic acid hydrate 1-4-hydroxyproline-o-phosphoric acid 2- (2-carboxyphenylsulfanyl) 1-hydroxy-1-cyclopropanecarboxylic acid (1R) - (-) - (1-aminohexyl) phosphonic acid n-boc-d-glutamic acid 4- (3-methoxybenzoylamino) - benzoic acid 4-hydrazobenzoic acid 4-fluoro-1-naphthoic acid benzoyl-lactic acid 3-butyl 1-5- (2,6,6-trimethyl-1-cyclohexen-1-yl) -2,4-pentadienoic acid fmoc-1 -beta-aminobutyric acid (s) -3-hydroxybutyric acid n- (3,5-xylyl) glutaramic acid 4,5-dichlorophthalic acid (s) -1-amino (1-phenyl) methane phosphonic acid 6-amino-2 3-dimethoxy-benzoic acid 4- (trifluoromethyl) cinnamic acid (1-alpha-n-gamma-d) -z-1-diaminobutyric acid 2,3-dibromobutyric acid 6 '- carbonylbis-Orimelitic acid 4- ( 2-bromobenzoyl) butyric acid 6-hydroxypicolinic acid 4- (3-hydroxy-propylamino) -3-nitro-benzoic acid · 9 · 9 · 9

-129kyselina 4-toludín-2,5-disulfónová kyselina 4-izopropylfenoxyoctová kyselina 2-fluór-6-metoxybenzoová kyselina 13-fenyl-10.12-tridekadiínová kyselina 4-chlórškoricová kyselina 2-acetyl-3,5-dibrómsalicylová kyselina mezityloctová kyselina 4-(4-(3,4-dimetyl-benzénsulfonyl)-fenoxy)-benzoová kyselina 4-karboxyškoricová kyselina 2-bróm-5-sulfobenzoová kyselina c/s-2-(4-brómbenzoyl)-1 -cyklohexán-karboxylová kyselina 4-(3,4-dimetoxy-fenyl)-4-oxo-maslová kyselina 3-(2-tenoyl)-propiónová kyselina cykloheptánkarboxylová kyselina n-chlóracetyl-1,2-amino-n-maslová kyselina 1-tryptofyl-1-asparágová kyselina 3-(n-(4-chlór-3-nitrofenyl)karbamoyl)-5-norbornén-2-karboxylová kyselina hipuryl-d/-fenylmliečna kyselina 3-bróm-adamantán-1 -karboxylová kyselina (s)-(-)-citronelová kyselina 1-(3,4-dimetoxy-fenyl)-4-hydroxy-6,7-dometoxy-naftalén-2-karboxylová kyselina (s)-2-metylhexánová kyselina 4-(2,2,2-trichlóracetamido)salicylová kyselina 1,2,3,4-tetrahydro-gama-oxo-2-pyrido[4.3-b]naftyrilidénbutánová kyselina 1,3-dioxo-2-(4-p-tolylkarbamoyl-ph)-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina 3,4,5,6-tetrachlórftalanilová kyselina n-benzoyl-1-glutámová kyselina (s)-(-)-4-oxo-2-azetidínkarboxylová kyselina dibrómoctová kyselina 5,5,5-trifluór-4,4-bis(trifluórmetyl)pentánová kyselina 3-(2-(2-karboxy-et)-1,1,3,3-tetraoxo-5-ph-,-(1,3)ditian-2-yl)-propiónová kyselina 3-oxoadipová • ·· ·· «··· ·· ·· · ·· ···· • ··· · · · · ·-129 4-toludine-2,5-disulfonic acid 4-isopropylphenoxyacetic acid 2-fluoro-6-methoxybenzoic acid 13-phenyl-10,12-tridecadioic acid 4-chlorocinnamic acid 2-acetyl-3,5-dibromosalicylic acid mesitylacetic acid 4- (4- (3,4-Dimethyl-benzenesulfonyl) -phenoxy) -benzoic acid 4-Carboxylic cinnamic acid 2-bromo-5-sulfobenzoic acid cis-2- (4-bromobenzoyl) -1-cyclohexanecarboxylic acid 4- (3,4-dimethoxy-phenyl) -4-oxo-butyric acid 3- (2-tenoyl) -propionic acid cycloheptanecarboxylic acid n-chloroacetyl-1,2-amino-n-butyric acid 1-tryptophyll-1-aspartic acid 3- (n- (4-Chloro-3-nitrophenyl) carbamoyl) -5-norbornene-2-carboxylic acid hipuryl-1-phenyl-lactic acid 3-bromo-adamantane-1-carboxylic acid (s) - (-) - 1- (3,4-dimethoxyphenyl) -4-hydroxy-6,7-domethoxy-naphthalene-2-carboxylic acid (s) -2-methylhexanoic acid 4- (2,2,2-trichloroacetamido) salicylic acid 1,2,3,4-tetrahydric acid o-gamma-oxo-2-pyrido [4,3-b] naphthyridenebutanoic acid 1,3-dioxo-2- (4-p-tolylcarbamoyl-ph) -2,3-dihydro-1H-isoindole-5-carboxylic acid 3 4,5,6-tetrachlorophthalanic acid n-benzoyl-1-glutamic acid (s) - (-) - 4-oxo-2-azetidinecarboxylic acid dibromoacetic acid 5,5,5-trifluoro-4,4-bis (trifluoromethyl) ) pentanoic acid 3- (2- (2-carboxy-et) -1,1,3,3-tetraoxo-5-ph -, - (1,3) dithian-2-yl) -propionic acid 3-oxoadipic acid • ·················

-130kyselina n-(o-tolyl)sukcínamová kyselina (z)-(3)-brómakrylová kyselina 2,5-dimetyladipová kyselina fmoc-4-fenyl-piperidín-4-karboxylová kyselina 3,4-dichlór-alfa-metoxyfenyloctová kyselina 2,2'-bitiofén-5-karboxylová kyselina 2’-chlór-3,4,5,6-tetrachlórftalámová kyselina 5-chlór-3-metylbenzo[b]tiofén-2-octová kyselina n-(2,4-dinitrofenyl)-1,2-aminomaslová kyselina 2-nitrofenol-4-sulfónová kyselina 3-imidazolakrylová kyselina 2,3-dihydroxybenzoová kyselina 4-((4-dimetylamino-benzylidén)-amino)-benzoová kyselina 4-(2,5-dimetyl-fenyl)-pentánová kyselina 2-[(2-chlór-alyl)-(toluén-4-sulfonyl)-amino]-benzoová kyselina bis-(2-metyl-5-nitro-fenyl)-fosfínová kyselina c/s,c/s-1,3,5-tripropyl-1,3,5-cyklohexántrikarboxylová kyselina 3-chlór-2-nitrobenzoová kyselina 2-[(4I6-dimetoxypyrimidín-2-yl)oxy]-3-metylbutánová kyselina 3,5-d/-ŕerc-butyl-4-hydroxyfenyloctová kyselina tetrachlórtereftalová kyselina furyloctová kyselina 3-(3-(2-metoxy-5-nitrofenyl)ureido)benzoová kyselina 1,2-diaminocyklohexán-n,n,/?',n’-tetraoctová fosphatidovaný glycerol kyselina ŕrans-2-(4-brómbenzoyl)-1 -cyklohexán-karboxylová kyselina 2-(2-bróm-benzoylamino)-3-fenyl-propiónová kyselina 3-(4-ŕerc-butyl-benzoyl)akrylová kyselina n-boc-d-glutámová kyselina c/s-hexahydro-n-(4-jódfenyl)ftalámová kyselina 1,4-fenyléndioctová kyselina 7-metyldekánová ·· ·· ···· ·· • · · · · · · ··· · · · · ·-130 n- (o-Tolyl) succinamic acid (z) - (3) -bromoacrylic acid 2,5-dimethyladipic acid fmoc-4-phenyl-piperidine-4-carboxylic acid 3,4-dichloro-alpha-methoxyphenylacetic acid 2 , 2'-bitiophene-5-carboxylic acid 2'-chloro-3,4,5,6-tetrachlorophthalic acid 5-chloro-3-methylbenzo [b] thiophene-2-acetic acid n- (2,4-dinitrophenyl) -1,2-aminobutyric acid 2-nitrophenol-4-sulfonic acid 3-imidazolacrylic acid 2,3-dihydroxybenzoic acid 4 - ((4-dimethylamino-benzylidene) -amino) -benzoic acid 4- (2,5-dimethyl- phenyl) -pentanoic acid 2 - [(2-chloro-allyl) - (toluene-4-sulfonyl) -amino] -benzoic acid bis- (2-methyl-5-nitro-phenyl) -phosphinic acid cis / c s-1,3,5-tripropyl-1,3,5-cyclohexanetricarboxylic acid 3-chloro-2-nitrobenzoic acid 2 - [( 4L 6-dimethoxypyrimidin-2-yl) oxy] -3-methylbutanoic acid 3, 5-tert-butyl-4-hydroxyphenylacetic acid tetrachloro-terephthalic acid furylacetic acid 3- (3- (2-methoxy-5-nitrophen) yl) ureido) benzoic acid 1,2-diaminocyclohexane-n, n ', N', n'-tetraacetic acid Phosphatidated glycerol trans-2- (4-bromobenzoyl) -1-cyclohexanecarboxylic acid 2- (2-bromo- benzoylamino) -3-phenyl-propionic acid 3- (4-tert-butyl-benzoyl) acrylic acid n-boc-d-glutamic acid cis-hexahydro-1- (4-iodophenyl) phthalic acid 1,4-phenylenediacetic acid 7-methyldecanoic acid ··· ··············

-131 kyselina 4-nitroftalová kyselina p-toluylová kyselina 2-[(4,6-dimetoxypyrimidín-2-yl)oxy]-3-metylpentánová kyselina 4-acetylglutárová kyselina 3-hydroxy-7-metoxy-2-naftoová kyselina 2-(4-(3,4-dimetyl-fenoxy)-ph)-1,3-dioxo-2,3-2h-1 h-izoindol-5-karboxylová kyselina 2,5-dimetoxy-3-nitrobenzoová kyselina 1-metoxy-2-naftoová kyselina (2,4,6-trimetyl-fenoxy)-octová kyselina n,n-dietyl-4-sulfamoylbenzoová kyselina 4-benzyloxy-3-metoxy-benzoová kyselina 3-chlór-antrachinón-2-karboxylová kyselina 3-(imidazol-4-yl)propiónová kyselina (+/-)-pinolová kyselina 2,5-dihydroxy-1,4-benzéndioctová kyselina d/-alfa-metylasparágová kyselina n-(2,6-xylyl)glutarámová kyselina 3-(2-(1,3,3-trimetyl-1,3-dihydro-indol-2-ylidén)-etylidénamino)benzoová kyselina 4-antracén-9-yl-4-oxo-maslová kyselina perfluór(2-etoxyetán)sulfónová kyselina 3,5-diizotiokyanatobenzoová kyselina 4-metoxy-1,7-dimetyl-indán-5-karboxylová kyselina n,n-dietylmaleámová kyselina 2-undecénová kyselina 2-metyl-3-o-tolyl-akrylová kyselina 4,4’-azobis(4-kyanovalérová) kyselina 4-(4-chlór-benzoyl)-ftalová kyselina d/-alfa-aminoadipová kyselina 4-(metyltio)fenyloctová kyselina glycyl-d/-asparágová kyselina sulfo-octová kyselina (+l-)-trans-1 -amino-1 -karboxycyklopentán-3-octová-131 4-nitrophthalic acid p-toluic acid 2 - [(4,6-dimethoxypyrimidin-2-yl) oxy] -3-methylpentanoic acid 4-acetylglutaric acid 3-hydroxy-7-methoxy-2-naphthoic acid 2- (4- (3,4-Dimethyl-phenoxy) -ph) -1,3-dioxo-2,3-2h-1H-isoindole-5-carboxylic acid 2,5-dimethoxy-3-nitrobenzoic acid 1-methoxy -2-naphthoic acid (2,4,6-trimethyl-phenoxy) -acetic acid n, n-diethyl-4-sulfamoylbenzoic acid 4-benzyloxy-3-methoxy-benzoic acid 3-chloro-anthraquinone-2-carboxylic acid 3 - (imidazol-4-yl) propionic acid (+/-) - pinoleic acid 2,5-dihydroxy-1,4-benzenediacetic acid d-alpha-methylaseparic acid n- (2,6-xylyl) glutaramic acid 3- (2- (1,3,3-trimethyl-1,3-dihydro-indol-2-ylidene) -ethylidenamino) benzoic acid 4-anthracen-9-yl-4-oxo-butyric acid perfluoro (2-ethoxyethane) sulfonic acid 3,5-diisothiocyanatobenzoic acid 4-methoxy-1,7-dimethyl-indane-5-carboxylic acid n, n-diethylmaleamic acid 2-undecenoic acid 2-Methyl-3-o-tolyl-acrylic acid 4,4'-azobis (4-cyanovaleric) 4- (4-chloro-benzoyl) -phthalic acid d-alpha-aminoadipic acid 4- (methylthio) phenylacetic acid glycyl-d-aspartic acid sulfoacetic acid (+ 1 -) - trans-1-amino-1-carboxycyclopentane-3-acetic acid

-132·· ·· ···· ·· • · · · e · · ··· · · · e · kyselina 3-hydroxy-2-metyl-3-(3-nitro-fenyl)-propiónová kyselina 4-(n-metyl(metylsulfónamido))benzoová kyselina 1,2,3-tiadiazol-4-karboxylová kyselina 2-metylhexadekánová kyselina 3’-nitro-3,4,5,6-tetrachlórftalanilová kyselina psoromová kyselina 4-nonyloxybenzoová kyselina d-erytro-4-fluórglutámová kyselina 2-[[2-(4-chlórfenyl)hydrazíno]karbonyl]benzoová kyselina eb.ľ.ľa-trimetyl-ľ.ya-dihydro-ebh-cyklopropaíajacenaftylén-ľ-karboxylová kyselina 3-(trifluórmetoxy)škoricová kyselina 2,6-dietoxybenzoová kyselina 1-(ŕerc-butoxykarbonyl)-4-hydroxy-2-pyrolidínkarboxylová kyselina 4-fluór-alfa-metylfenyloctová kyselina 3,3'-ditiobishydroškoricová kyselina 2-metyl-2-sulfooktadekánová kyselina 2-chlór-4-metyltiobutánová kyselina 2-hydroxy-3-(2-hydroxybenzoyl)-6-trifluórmetylpyridín-5-karboxylová kyselina 2-terc-butoxykarbonylamino-3-(4-hydroxy-fenyl)-propiónová kyselina 3-(4-chlórbenzoyl)-2-(4-etylfenyl)propiónová kyselina (r)-(+)-alfa-metoxy-alfa-(trifluórmetyl)fenyloctová kyselina 2-kyano-2-(2,3-dimetoxybenzylidén)octová kyselina 2-(4-karbamoylfenoxy)-2-metylpropiónová kyselina 2'-chlórmaleanilová kyselina 2-(3,4-dikyano-fenyl)-1,3-dioxo-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina 1,4-naftaléndikarboxylová kyselina 3-(2-metoxy-fenyl)-3-metyl-maslová kyselina d/-2-amino-4-fosfonomaslová kyselina 4-izopropylškoricová kyselina 5-(4-metyl-2-nitrofenyl)-2-furoová kyselina trans-1,2-cyklohexándikarboxylová kyselina 3-(4-metoxy-3-metylfenyl)propiónová-132 3-hydroxy-2-methyl-3- (3-nitro-phenyl) -propionic acid 4- (n-methyl (methylsulfonamido)) benzoic acid 1,2,3-thiadiazole-4-carboxylic acid 2-methylhexadecanoic acid 3'-nitro-3,4,5,6-tetrachlorophthalanilic acid psoromic acid 4-nonyloxybenzoic acid d-erythro 4-fluoroglutamic acid 2 - [[2- (4-chlorophenyl) hydrazino] carbonyl] benzoic acid eb.l.1'-trimethyl-1'-dihydro-eb-cyclopropayl-naphthylene-1'-carboxylic acid 3- (trifluoromethoxy) cinnamic acid 2,6-diethoxybenzoic acid 1- (tert-butoxycarbonyl) -4-hydroxy-2-pyrrolidinecarboxylic acid 4-fluoro-alpha-methylphenylacetic acid 3,3'-dithiobishydicinnamic acid 2-methyl-2-sulfooctadecanoic acid 2-chloro- 4-methylthiobutanoic acid 2-hydroxy-3- (2-hydroxybenzoyl) -6-trifluoromethylpyridine-5-carboxylic acid 2-tert-butoxycarbonylamino-3- (4-hydroxyphenyl) -propionic acid 3- (4-chloro) (benzoyl) -2- (4-ethylphenyl) propionic acid (R) - (+) - alpha-methoxy-alpha- (trifluoromethyl) phenylacetic acid 2-cyano-2- (2,3-dimethoxybenzylidene) acetic acid 2- (4 -carbamoylphenoxy) -2-methylpropionic acid 2'-chloromaleanilic acid 2- (3,4-dicyanophenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid 1,4- naphthalenedicarboxylic acid 3- (2-methoxyphenyl) -3-methylbutyric acid d-2-amino-4-phosphonomasic acid 4-isopropylcinnamic acid 5- (4-methyl-2-nitrophenyl) -2-furoic acid trans -1,2-Cyclohexanedicarboxylic acid 3- (4-methoxy-3-methylphenyl) propionic acid

-133·· ··· • · • · ·· ·· ···· ·· • · · · ·· • · · · · • · · · · ·· • · · · ·· ·· ·· ·· · ·· ···· kyselina 2-(4-bróm-fenylamino)-malónová kyselina 2-dibenzotiofénmaslová kyselina polystyrénsulfónová kyselina (8-hydroxy-5,7-dinitro-2-naftalénsulfónová) kyselina p-metyl-alfa-fenylhydroškoricová kyselina 1-naftol-3,6-disulfónová kyselina 5,6-dihydro-(1,4)dioxín-2-karboxylová kyselina 6-(3-brómbenzoyl)hexánová kyselina 2,6,2I6-tetrametyl-(1,1 ‘,3', 1 )-terfenyl-2'-karboxylová kyselina 3-chlór-3-fenylkarbamoyl-akrylová kyselina 4-amino-1,7-naftaléndisulfónová kyselina 4-bróm-2-fluórškoricová-133 ·· ··· ······························ 2- (4-bromo-phenylamino) -malonic acid 2-dibenzothiophenebutyric acid polystyrenesulfonic acid (8-hydroxy-5,7-dinitro-2-naphthalenesulfonic acid) p-methyl-alpha-phenylhydrocinnamic acid 1-Naphthol-3,6-disulfonic acid 5,6-dihydro- (1,4) dioxine-2-carboxylic acid 6- (3-bromobenzoyl) hexanoic acid 2,6,2 L 6-tetramethyl- (1, 3-bromobenzoyl) hexanoic acid 1 ', 3', 1) -phenyl-2'-carboxylic acid 3-chloro-3-phenylcarbamoyl-acrylic acid 4-amino-1,7-naphthalenedisulfonic acid 4-bromo-2-fluorocinnamic acid

4,4'-dikarboxydifenyl-éter kyselina 2-(4-chlórbenzoyl)benzoová kyselina linoelaidová kyselina 2-etyl-5-metoxy-izoftalová kyselina 1,5-naftalén-disulfónová kyselina 4-(2,4-dichlórfenoxy)maslová kyselina fmoc-12-aminododekánová kyselina pivalová kyselina benzofuroxán-5-karboxylová kyselina 4-amino-3-(trifluórmetoxy)benzoová kyselina 3-(3-metylindol 1-yl)propiónová kyselina 2,5-dimetylškoricová kyselina 6,7,8-trifluór-4-oxo-1-propa-12-diényl-1,4-dihydro-chinolín-3-karboxylová kyselina 2-chlór-5-maleimidobenzoová kyselina 3-fenoxyfenyloctová kyselina indazolón-4-karboxylová kyselina 3-(n-(4-fluórfenyl)karbamoyl)-5-norbomén-2-karboxylová kyselina 4-(4-benzyloxybenzylidénamino)benzoová kyselina 3'-acetyl-1,2,3,6-tetrahydroftalanilová kyselina 4-oxo-4,5,6,7-tetrahydrobenzo[b]furán-3-karboxylová • ·· ·· ···· ·· ·· · ·· ···· • ··· · · · · ·4,4'-dicarboxydiphenyl ether 2- (4-chlorobenzoyl) benzoic acid linoelaidic acid 2-ethyl-5-methoxy-isophthalic acid 1,5-naphthalene disulfonic acid 4- (2,4-dichlorophenoxy) butyric acid fmoc -12-aminododecanoic acid pivalic acid benzofuroxane-5-carboxylic acid 4-amino-3- (trifluoromethoxy) benzoic acid 3- (3-methylindol 1-yl) propionic acid 2,5-dimethyl cinnamic acid 6,7,8-trifluoro- 4-oxo-1-propa-12-dienyl-1,4-dihydroquinoline-3-carboxylic acid 2-chloro-5-maleimidobenzoic acid 3-phenoxyphenylacetic acid indazolone-4-carboxylic acid 3- (n- (4- fluorophenyl) carbamoyl) -5-norbomene-2-carboxylic acid 4- (4-benzyloxybenzylidenamino) benzoic acid 3'-acetyl-1,2,3,6-tetrahydrophthalanilic acid 4-oxo-4,5,6,7-tetrahydrobenzo [b] furan-3-carboxylic acid • furan-3-carboxylic acid

-134kyselina 3-bróm-3-(3-nitrofenyl)propiónová kyselina 3-metyl-2-(2-nitro-4-trifluórmetyl-fenylamino)-maslová kyselina c/s-8-eikozénová kyselina 2,2'-iminodibenzoová kyselina 4,4'-bifenyldisulfónová kyselina 3,3,3-trifenylpropiónová kyselina 3-(dodekán-1 -sulfonyl)-propiónová kyselina hydroxyvalerénová kyselina 3-chinolín-2-yl-akrylová kyselina c/s-hexahydro-n-(3-metylfenyl)ftalámová kyselina 1-benzyl-3-hydroxy-1,2,3,3a,4,7-hexahydro-indén-1,7a-dikarboxylová kyselina 4-metoxy-3-metylfenyloctová kyselina n-formylantranilová kyselina 4-(3-fenyl-propyl)-benzoová kyselina cyklopentylmalónová kyselina alfa-hydroxyfarnesylfosfónová kyselina 3,5-dinitro-4-hydroxybenzoová kyselina 4-fenoxymaslová kyselina 3-izobutyrylamino-benzoová kyselina c/s-2',6'-dimetylhexahydroftalanilová kyselina 4-(4-(4-(2-karboxy-etyl)-benzyl)-fenyl)-maslová kyselina 4-[2-(4-metyl-4h-[1,2,4]triazol-3-ylsulfanyl)-acetylamiino]-benzoová kyselina /?-(1,2-dimetyl-propyl)-ftalámová kyselina eikoza-5,8,11-triénová kyselina 2,3-dibróm-3-(4-sulfamoyl-fenyl)-propiónová kyselina tridekándiová kyselina 3,5-dihydroxybenzoová kyselina chinizarin-2-sulfónová kyselina 4-(2,2-dimetylpropyl)benzénsulfínová kyselina 4’-jód-1,2,3,6-tetrahydroftalanilová kyselina 2,,4'-dimetylglutaranilová kyselina 4-metyl-3-fenyl-pentánová • · · φ ·-134-3-bromo-3- (3-nitrophenyl) propionic acid 3-methyl-2- (2-nitro-4-trifluoromethyl-phenylamino) -butyric acid cis-8-eicosenoic acid 2,2'-iminodibenzoic acid 4,4'-biphenyldisulfonic acid 3,3,3-triphenylpropionic acid 3- (dodecane-1-sulfonyl) -propionic acid hydroxyvalerenic acid 3-quinolin-2-yl-acrylic acid cis-hexahydro-n- (3- methylphenyl) phthalic acid 1-benzyl-3-hydroxy-1,2,3,3a, 4,7-hexahydro-indene-1,7a-dicarboxylic acid 4-methoxy-3-methylphenylacetic acid n-formylantranilic acid 4- (3 -phenyl-propyl) -benzoic acid cyclopentylmalonic acid alpha-hydroxypharnesylphosphonic acid 3,5-dinitro-4-hydroxybenzoic acid 4-phenoxybutyric acid 3-isobutyrylaminobenzoic acid cis-2 ', 6'-dimethylhexahydrophthalanic acid 4- (4 - (4- (2-Carboxy-ethyl) -benzyl) -phenyl) -butyric acid 4- [2- (4-methyl-4h- [1,2,4] triazol-3-ylsulfanyl) -acetylamino] -benzoic acid N - (1,2-dimethyl-propyl) -phthalic acid eicoza-5,8,11-trienoic acid 2,3-dibromo-3- (4-sulfamoyl-phenyl) -propionic acid tridecanedioic acid 3,5-dihydroxybenzoic acid quinizarin-2-sulfonic acid 4- (2,2- dimethylpropyl) benzenesulfinic acid, 4'-iodo-1,2,3,6-tetrahydroftalanilová acid, 2, 4 & apos dimetylglutaranilová acid 4-methyl-3-phenyl-pentanoic • φ · · ·

ΦΦ· · • · · ·ΦΦ · · · · · ·

135 ·· ·· ·· ···· • · · • · * ·· φ · ·· ·· ·· · kyselina 2-(3-hydroxy-4-metoxyfenyl)glyoxylová135 2- (3-Hydroxy-4-methoxyphenyl) glyoxylic acid 135 ··· ·······

3-karboxy-7-hydroxykumarín kyselina opianová kyselina 4-metyl-3-(2-nitroetyl)-2,5-pyroldikarboxylová kyselina 3-(2-hydroxy-1 -naftylmetylénamino)benzoová kyselina 2-fluór-6-metoxyfenyloctová kyselina c/s-6-oktadecénová kyselina 2-[(5-oxotetrahydro-1 h-2-pyrolyl)sulfanyl]benzoová kyselina (s)-2-chlór-4-metyl-n-valérová kyselina 3-metyl-2-tiofénkarboxylová kyselina 2,5-dimetylimidazo[1,2-a]pyridin-3-karboxylová kyselina 3-(p-nitrofenoxy)propiónová kyselina 2-(orto-tolyl)-valérová kyselina brómjantárová kyselina 4,4,-ditiodimaslová kyselina 2-[3-(n-dekanoyl-hydrazíno)-3-oxo-propionylamino]-benzoová kyselina hexahydro-4-metylftalová kyselina 1,5-naftaléndisulfónová kyselina 2-[(4,6-dimetoxypyrimidín-2-yl)oxy]benzoová kyselina 3-(2-alylsulfanyl-benzotiazol-6-ylkarbamoyl)-akrylová kyselina 5-fenylsalicylová kyselina 3-(2-furyl)akrylová kyselina 4-metoxy-2-(3-metoxy-benzoyl)-benzoová kyselina 3-acetyl-2,2-dimetyltiazolidín-4-karboxylová kyselina 6-bróm-1,3-benzodioxol-5-karboxylová kyselina 1-cyklohexénkarboxylová kyselina 3,4,5-trichlór-6-hydroxy-pyridín-2-karboxylová kyselina 3-(4-metoxybenzoyl)propiónová kyselina 5-oxo-4-oxa-tricyklo(4,2,1,0(3,7))nonán-9-karboxylová kyselina 2-oxo-4-fenyl-but-3-énová kyselina (4-( 1 -(4-karboxymetoxy-3-me-ph)-1 -metyl-etyl)-2-melyl-fenoxy)-octová kyselina 2-benzoylamino-3-fenyl-akrylová3-carboxy-7-hydroxycoumarin opianic acid 4-methyl-3- (2-nitroethyl) -2,5-pyrroleicarboxylic acid 3- (2-hydroxy-1-naphthylmethyleneamino) benzoic acid 2-fluoro-6-methoxyphenylacetic acid c s-6-octadecenic acid 2 - [(5-oxotetrahydro-1H-2-pyrrolyl) sulfanyl] benzoic acid (s) -2-chloro-4-methyl-n-valeric acid 3-methyl-2-thiophenecarboxylic acid 2,5-dimethylimidazo [1,2-a] pyridine-3-carboxylic acid 3- (p-nitrophenoxy) propionic acid 2- (ortho-tolyl) -valeric bromosuccinic acid 4,4 , -dithiodimasic acid 2- [3 - (n-decanoyl-hydrazino) -3-oxo-propionylamino] -benzoic acid hexahydro-4-methylphthalic acid 1,5-naphthalenedisulfonic acid 2 - [(4,6-dimethoxypyrimidin-2-yl) oxy] benzoic acid 3- (2-Allylsulfanyl-benzothiazol-6-ylcarbamoyl) -acrylic acid 5-Phenylsalicylic acid 3- (2-furyl) acrylic acid 4-methoxy-2- (3-methoxy-benzoyl) -benzoic acid 3-acetyl-2,2 6-bromo-dimethylthiazolidine-4-carboxylic acid -1,3-benzodioxole-5-carboxylic acid 1-cyclohexenecarboxylic acid 3,4,5-trichloro-6-hydroxy-pyridine-2-carboxylic acid 3- (4-methoxybenzoyl) propionic acid 5-oxo-4-oxa- tricyclo (4,2,1,0 (3,7)) nonane-9-carboxylic acid 2-oxo-4-phenyl-but-3-enoic acid (4- (1- (4-carboxymethoxy-3-methoxy)) ph) -1-methyl-ethyl) -2-melyl-phenoxy) -acetic acid 2-benzoylamino-3-phenyl-acrylic acid

-136--136-

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · ···· • • ···· • • ·· · • · ·· • · · ·· · • · ·· • · · ·· ·· ·· ·· • e • e • · • · ·· ·· ·· ··

kyselina beta-5-dimetyl-2-(metyltio)škoricová kyselina 4-(4-oktadecyl)-4-oxobenzénbuténová kyselina 4-(2-etoxykarbonyl-acetylamino)-benzoová kyselina 4-(3-metoxy-5-metyl-fenyl)-4-oxo-maslová kyselina 3-hydroxypentadekánová kyselina z-styrénsulfonyloctová kyselina 3-(4-metoxyfenoxy)propiónová kyselina 3’-(trifluórmetyl)ftalanilová kyselina 3,6-dioxaoktándiová kyselina 3'-chlór-4'-metylftalanilová kyselina 2-[2-chlór[(2,5-dichlórfenyl)sulfonyl]anilíno]octová kyselina 3-hydroxy-3-(2-oxo-1,2-dihydro-indol-3-ylidén)-propiónová kyselina 6-fenylhexánová kyselina 3-(metylsulfonyloxy)-4-nitrobenzoová kyselina (2-jódfenyl)fosfónová kyselina 4-fenoxyfenyloctová kyselina (1 -aminopropyl)fosfónová kyselina p-chlórbenzénsulfónová kyselina 4,5-dibróm-cyklohexán-1,2-dikarboxylová kyselina (-)-2-oxo-4-tiazolidín-karboxylová kyselina 4,6-dichlórindol-2-karboxylová kyselina 2-chlór-6-nitrobenzoová kyselina indol-3-acetyl-1-asparágová kyselina kuminová kyselina 9,12-oktadekadiínová kyselina 2,2,-dimetoxy-5,5,-dimetyl-bifenyl-3,3,dikarboxylová kyselina 6-(benzoylamino)-2-brómhexánová kyselina 3-fenoxybenzoová kyselina 3,4-dimetylškoricová kyselina (oxo-d/-pr-tioxo-imidazolín-ylidén-etylidén)benzoxazol-yl-propiónová kyselina 7-formyl-naftalén-2-karboxylová kyselina n-lauroyl-1-asparágovábeta-5-dimethyl-2- (methylthio) cinnamic acid 4- (4-octadecyl) -4-oxobenzenebutenic acid 4- (2-ethoxycarbonyl-acetylamino) -benzoic acid 4- (3-methoxy-5-methyl-phenyl) ) -4-oxo-butyric acid 3-hydroxypentadecanoic acid z-styrene sulfonylacetic acid 3- (4-methoxyphenoxy) propionic acid 3 '- (trifluoromethyl) phthalanilic acid 3,6-dioxaoctanedioic acid 3'-chloro-4'-methylphthalanilic acid 2 - [2-chloro [(2,5-dichlorophenyl) sulfonyl] anilino] acetic acid 3-hydroxy-3- (2-oxo-1,2-dihydro-indol-3-ylidene) -propionic acid 6-phenylhexanoic acid 3 - (methylsulfonyloxy) -4-nitrobenzoic acid (2-iodophenyl) phosphonic acid 4-phenoxyphenylacetic acid (1-aminopropyl) phosphonic acid p-chlorobenzenesulfonic acid 4,5-dibromocyclohexane-1,2-dicarboxylic acid (-) - 2 -oxo-4-thiazolidine-carboxylic acid 4,6-dichloroindole-2-carboxylic acid 2-chloro-6-nitrobenzoic acid indole-3-acetyl-1-aspartic acid 9,12-octadecadiic acid 2,2 , -dimethoxy-5,5 , -dimethyl-biphenyl-3,3 , dicarboxylic acid 6- (benzoylamino) -2-bromohexanoic acid 3-phenoxybenzoic acid 3,4-dimethyl cinnamic acid ( oxo-d-pr-thioxo-imidazolin-ylidene-ethylidene) benzoxazol-yl-propionic acid 7-formyl-naphthalene-2-carboxylic acid n-lauroyl-1-aspartic acid

-137--137-

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · ···· • • ···· • • ·· • · • · · · • · • · ·· · · ·· ·· ·· ·· ·· · · ·· · · ·· · · ·· · ·

kyselina n-(4-chlórfenyl)maleámová kyselina 6-karboxymetyl-2,3-dihydroxy-benzoová kyselina 2-chlór-5-(metyltio)benzoová kyselina 4-p-tolyl-1,10-fenantrolín-2,9-dikarboxylová kyselina homochinolínová kyselina 5-sulfoizoftalová kyselina 5-(4-trifluórmetylfenyl)-2h-tetrazol-2-octová kyselina 4'-oktyl-4-bifenylkarboxylová kyselina 1,3-dioxo-ih-benz[de]izochinolín-2(3h)-octová kyselina 3-oxo-tetrametyl-perhydrofenantro(2,3-d)(1,3)dioxol-propiónová kyselina 4-(5-bróm-1,3-dioxo-1,3-dihydro-izoindol-2-yl)-benzoová kyselina formimino-1-asparágová kyselina 2-(4-etylbenzoyl)-benzoová kyselina metyltiohydantoín-d/-glutámová kyselina 2-(4-aminofenyl)propiónová kyselina 2’-metyl-3,-nitro-3,4,5,6-tetrachlórftalanilová kyselina 4-n-oktadecyloxyškoricován- (4-chlorophenyl) maleic acid 6-carboxymethyl-2,3-dihydroxybenzoic acid 2-chloro-5- (methylthio) benzoic acid 4-p-tolyl-1,10-phenanthroline-2,9-dicarboxylic acid 5-sulfoisophthalic acid 5- (4-trifluoromethylphenyl) -2h-tetrazole-2-acetic acid 4'-octyl-4-biphenylcarboxylic acid 1,3-dioxo-1 H -benzo [de] isoquinolin-2 (3h) -acetic acid 3-oxo-tetramethyl-perhydrophenantro (2,3-d) (1,3) dioxol-propionic acid 4- (5-bromo-1,3-dioxo-1,3-dihydro-isoindol-2-yl) ) -benzoic acid formimino-1-aspartic acid 2- (4-ethylbenzoyl) -benzoic acid methylthiohydantoin-d-glutamic acid 2- (4-aminophenyl) propionic acid 2'-methyl-3 , -nitro-3,4, 5,6-Tetrachlorophthalic acid 4-n-octadecyloxycinnamic acid

-aspartyl-1 -fenylalanín-diketopiperazín kyselina /7-(2,6-dietyl-fenyl)-3-nitro-ftalámová /?-ftaloyl-d/-fenylalanín kyselina metánsulfónová kyselina 1 -(3-chlórbenzoyl)piperazín-2,3-dikarboxylová kyselina 3,4-benzo-9-oxofluorén-1 -karboxylová kyselina 1-pyrénsulfónová kyselina dehydrooctová kyselina 2-(p-chlórfenyl)-3-metylmaslová kyselina 5-metyl-1,1-dioxo-tetrahydro-tiofén-2-karboxylová kyselina 3-fluór-5-(trifliiórmetyl)škoricová alfa-benzylester kyseliny n-boc-1-glutámovej kyselina n-hexylfosfónová kyselina 2-acetamido-2-alylmalónová kyselina difenylmetán-4,4'-dikarboxylová ·· ·· ···· ·· • · · · · · ··· · · · · · • · · · · ··· ·- [1- (3-chlorobenzoyl) piperazin-2] -aspartyl-1-phenylalanine-diketopiperazine [7- (2,6-diethylphenyl) -3-nitro-phthalic acid] -phthaloyl-d] phenylalanine methanesulfonic acid 3-dicarboxylic acid 3,4-benzo-9-oxofluorene-1-carboxylic acid 1-pyrenesulfonic acid dehydroacetic acid 2- (p-chlorophenyl) -3-methylbutyric acid 5-methyl-1,1-dioxo-tetrahydro-thiophene- 2-carboxylic acid 3-fluoro-5- (trifluoromethyl) cinnamic alpha-benzyl n-boc-1-glutamic acid n-hexylphosphonic acid 2-acetamido-2-allylmalonic acid diphenylmethane-4,4'-dicarboxylic acid ·· ·· ··························

-138kyselina z-(-)-alfa-amino-4-fenylmaslová kyselina 3,5-oktadekadiínová kyselina 4-chlór-2,6-dinitrobenzénsulfónová kyselina n,n-bis((s)-(-)-1-fenyletyl)ftalámová kyselina 4-(3-brómbenzoyl)maslová kyselina 8,10-henikozadiínová kyselina 4,4'-ditiobisbenzoová kyselina n-(4-karboxyfenyl)sukcínimid-3,4-dihydroxybenzoová kyselina 5-[[(4-chlórfenyl)sulfonyl]amino]-5-oxopentánová kyselina 3,5-dichlór-4-hydroxybenzénsulfónová kyselina n-(2-hydroxybenzoyl)glutámová kyselina 2-benzénsulfonyl-2-metyl-oktánová kyselina 2,3-difenylpropiónová kyselina 3,4-dimetyltieno(2,3-b)tiofén-2,5-dikarboxylová kyselina 4-(3-(3-(trifluórmetyl)fenyl)ureido)benzoová kyselina 2-metyl-3-nitrobenzoová kyselina 2-izopropyljablčná kyselina 4-(2-fenyl-eténsulfonylamino)-benzoová kyselina 4-fluórfenyloctová kyselina exo-2-chlór-5-oxo-bicyklo[2.2.1]heptán-syn-7-karboxylová kyselina 2,5-dimetylfenyloctová kyselina S'^'-dichlórftalanilová kyselina tricyklo(12.2.2.2(6,9))eikoza-1(16),6(20)7,9(19),14l17-hexaén-dikarboxylová kyselina (3,4,5,6-tetrahydroxy-tetrahydro-pyran-2-yl)-octová kyselina 3'-chlór-2'-metylftalanilová kyselina S-^-ÍS^-dichlórbenzyloxyJfenyljakrylová kyselina 3-brómmaslová kyselina n-(4-jódfenyl)maleámová kyselina (+)-s-2-amino-6-jódacetamidohexánová kyselina 2,4-dimetoxybenzoová kyselina 3-(4-(hexadecyloxy)-benzoyl)-propiónová • ·· ······ ·· ·· · · · ···· • ··· · · · · ·-138 acid from - (-) - alpha-amino-4-phenylbutyric acid 3,5-octadecadiic acid 4-chloro-2,6-dinitrobenzenesulfonic acid n, n-bis ((s) - (-) - 1-phenylethyl) 4- (3-Bromobenzoyl) butyric acid 8,10-hensosadioic acid 4,4'-dithiobisbenzoic acid 4- (4-carboxyphenyl) succinimide-3,4-dihydroxybenzoic acid 5 - [[(4-chlorophenyl) sulfonyl] amino] -5-oxopentanoic acid 3,5-dichloro-4-hydroxybenzenesulfonic acid n- (2-hydroxybenzoyl) glutamic acid 2-benzenesulfonyl-2-methyl-octanoic acid 2,3-diphenylpropionic acid 3,4-dimethylthieno (2, 3-b) Thiophene-2,5-dicarboxylic acid 4- (3- (3- (trifluoromethyl) phenyl) ureido) benzoic acid 2-methyl-3-nitrobenzoic acid 2-isopropyl malic acid 4- (2-phenyl-etenesulfonylamino) -benzoic acid 4-fluorophenylacetic acid exo-2-chloro-5-oxo-bicyclo [2.2.1] heptane-syn-7-carboxylic acid 2,5-dimethylphenylacetic acid S '-4' - dichlorophthalanic acid tricyclo (12.2.2.2 ( 6.9)) eicos a-1 (16), 6 (20) 7.9 (19), 14 L 17-hexaen-dicarboxylic acid (3,4,5,6-tetrahydroxy-tetrahydro-pyran-2-yl) -acetic acid 3 ' 3-bromobutyric acid 3- (4-iodophenyl) maleic acid (+) - s-2-amino-6-iodoacetamidohexanoic acid 2,4-dimethoxybenzoic acid 3-bromobutyric acid 3-bromobutyric acid 3- (4- (Hexadecyloxy) -benzoyl) -propionic • (hex op op pr · · · · · · ·

-139kyselina (r)-(-)-2-bróm-3-fenylpropiónová kyselina (r)-(-)-gáfor-10-sulfónová kyselina antipyrínová kyselina 2-indanyloctová kyselina n-(3,4-dimetylfenyl)maleámová kyselina 4-palmitamidobenzoová kyselina 2-[1,6-naftyridín-2-yl]benzoová kyselina 2-(n-dodecylkarbamoylmetyl)-2-hydroxyjantárová kyselina 4-(2-hydroxy-5-fenylanilíno)-1 -butánsulfónová kyselina 14c-trikozénová kyselina 3-{toluén-4-sulfonyl)-propiónová kyselina pentafluórfenyloctová kyselina (+/-)-1-aminocyklohexán-c/s-1,3-dikarboxylová kyselina 4-amino-4,-chlórdifenylamín-2-sulfónová kyselina pimelová kyselina 2-[(fenylsulfonyl)-3 -(trifluórmetyl)anilínojoctová kyselina (s)-(-)-2-brómpropiónová kyselina 4-(2-ftalimidofenyl)maslová kyselina 6-metylsulfanyl-pyrimidín-4-karboxylová kyselina 3-metyl-2-nitrobenzoová kyselina 3,4-dichlórbenzoová kyselina 5-metylhexánová kyselina 4-(trifluóracetyl)benzoová kyselina 3-(3-(2,2,2-trichlór-1-(2-fluór-acetylamino)-etyl)-tioureido)benzoová kyselina 4-(2-metoxy-fenyl)-pent-3-énová kyselina 2-(4-fluór-fenyl)-1,3-dioxo-2,3-dihydro-1 h-izoindol-5-karboxylová kyselina bicyklo(3.3.1 )nonán-1-karboxylová kyselina 3,7-dimetyl-1-adamantánoctová kyselina 4-kyanobenzoová kyselina 7-izopropylidén-bicyklo(2.2.1)hept-5-én-2,3-dikarboxylová kyselina 2-(hexadecyltio)benzoová kyselina n-(3-karboxy-propyl)-ftalámová ·· ·· BBBB ·· • · B BBBB •*· · · B · ·-139 (r) - (-) - 2-bromo-3-phenylpropionic acid (r) - (-) - camphor-10-sulfonic acid antipyric acid 2-indanylacetic acid n- (3,4-dimethylphenyl) maleic acid 4 2- [1,6-naphthyridin-2-yl] benzoic acid 2- (n-dodecylcarbamoylmethyl) -2-hydroxysuccinic acid 4- (2-hydroxy-5-phenylanilino) -1-butanesulfonic acid 14c-tricosenoic acid 3- (toluene-4-sulfonyl) -propionic acid pentafluorophenylacetic acid (+/-) - 1-aminocyclohexane-cis-1,3-dicarboxylic acid 4-amino-4 , -chlorodiphenylamine-2-sulfonic acid pimelic acid 2 - [(phenylsulfonyl) -3- (trifluoromethyl) anilinoacetic acid (s) - (-) - 2-bromopropionic acid 4- (2-phthalimidophenyl) butyric acid 6-methylsulfanyl-pyrimidine-4-carboxylic acid 3-methyl-2- nitrobenzoic acid 3,4-dichlorobenzoic acid 5-methylhexanoic acid 4- (trifluoroacetyl) benzoic acid 3- (3- (2,2,2-trichloro-1- (2-fluoro-acetylamino) ethyl) thioureido) benzoic acid 4- (2-methoxy-phenyl) -pent-3-enoic acid 2- (4-fluoro-phenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid bicyclo (3.3.1) nonane-1-carboxylic acid 3,7-dimethyl-1-adamantaneacetic acid 4-cyanobenzoic acid 7-isopropylidene-bicyclo (2.2.1) hept-5-ene-2,3-dicarboxylic acid 2- ( hexadecylthio) benzoic acid n- (3-carboxy-propyl) -phthalic acid ··· BBBB · B BBBB

-140kyselina alfa-(2,6-dimetoxybenzylidén)hipurová kyselina írans-7-oktadecénová kyselina 4-penténová kyselina 5-(4-metylfenyl)-2,3-dihydro-1h-pyrolizín-6,7-dikarboxylová kyselina 4'-brómsukcínanilová kyselina 4-acetyl-1 -metylpyridol-2-karboxylová kyselina 2-(1 -naftyl)-2-fenyloctová kyselina 2'-hydroxy-5,-metylmaleanilová kyselina c/s-n-(4-fluórfenyl)hexahydroftalámová kyselina 4-(3-(piperidín-1 -sulfonyl)-benzoylamino)-benzoová kyselina 4,-bróm-2,-chlórftalanilová kyselina 3,3'-(karbonyldiimino)bis-benzoová kyselina (7-metoxy-5,8-dioxo-1,4,5,8-tetrahydro-naftalén-1 -yl)-octová kyselina 2-fenylmaslová kyselina n-íerc-boc-(2s,3r)-3-amino-2-hydroxy-4-fenylmaslová kyselina 2-(4-fluórfenyl)-1 -izochinolón-4-karboxylová kyselina 11c,14c-eikozadiénová kyselina (4(s)-trans)-4,5-dihydroxy-3-oxo-1 -cyklohexén-1 -karboxylová kyselina 2-(n-(2,4l6-trimetylfenyl)karbamoyl)cyklohexánkarboxylová kyselina beta-hydroxyizovalérová kyselina n-benzoyl-n-fenylantranilová kyselina 3-(brómmetyl)krotónová kopolymér etylén/kyselina akrylová kyselina n-benzyl-d/-asparágová kyselina beta-(naftylmerkapto)octová kyselina pentadekándiová kyselina 3,4-dimetyl-2,5-pyroldikarboxylová kyselina 2,3-bis-(3-metoxy-benzylidén)-jantárová kyselina 2-(2-hexylkarbamoyl-acetylamino)-benzoová kyselina n-oktadecylfosfónová kyselina 1-(2,-(3,-chlór-5,-trifluórmetyl)pyridyl)piperid-4-ón-metylén-karboxylová kyselina 1,1,2-etántrikarboxylová e ·> ·· ···· ·· ··· · · · ··· • bbb · · · e B-140-alpha- (2,6-dimethoxybenzylidene) hippuric acid trans-7-octadecenic acid 4-pentenoic acid 5- (4-methylphenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid 4'- brómsukcínanilová acid 4-acetyl-1-methylpyrid-2-carboxylic acid 2- (1-naphthyl) -2-phenylacetic acid, 2 ' -hydroxy-5, -metylmaleanilová cis / SN- (4-fluorophenyl) hexahydroftalámová 4- ( 3- (piperidine-1-sulfonyl) -benzoylamino) -benzoic acid 4-bromo-2, -chlórftalanilová 3,3 '- (carbonyldiimino) bis-benzoic acid (7-methoxy-5,8-dioxo-1, 4,5,8-tetrahydro-naphthalen-1-yl) -acetic acid 2-phenylbutyric acid n-tert -boc- (2s, 3r) -3-amino-2-hydroxy-4-phenylbutyric acid 2- (4- Fluorophenyl) -1-isoquinolone-4-carboxylic acid 11c, 14c-eicosadienoic acid (4 (s) -trans) -4,5-dihydroxy-3-oxo-1-cyclohexene-1-carboxylic acid 2- (n- ( 2,4 1 6-trimethylphenyl) carbamoyl) cyclohexanecarboxylic acid beta-hydroxyisovaleric acid n-benzoyl-n-phen ylanthranilic acid 3- (bromomethyl) crotonic copolymer ethylene / acrylic acid n-benzyl-d / -aspartic acid beta- (naphthylmercapto) acetic acid pentadecanedioic acid 3,4-dimethyl-2,5-pyrrole dicarboxylic acid 2,3-bis- (3-methoxy-benzylidene) -succinic acid, 2- (2-hexylcarbamoyl-acetylamino) -benzoic acid n-octadecylphosphonic acid 1- (2 - (3-chloro-5-trifluoromethyl) pyridyl) piperidin-4-one -methylene-carboxylic acid 1,1,2-ethanetricarboxylic acid e ·> · B · bbb · e · B

-141 kyselina d(-)-2-amino-3-fosfonopropiónová kyselina 5-bróm-n-(karboxymetyl)antranilová kyselina 16,17-dichlórheptadekánová kyselina 8-hydroxy-7-chinolínkarboxylová kyselina 4-(4-fluórbenzoyl)maslová kyselina 4,4,4-trifluór-3-(trifluórmetyl)maslová kyselina 2,4,6,8-dekatetraénová kyselina 6-(3,4-dimetoxy-fenyl)-hexánová kyselina 2-(n-(2,5-dimetylbenzyl)karbamoyl)cyklohexánkarboxylová kyselina 2-(1 -metyl-2,2-difenyl-etoxy)-benzoová-141 d (-) - 2-amino-3-phosphonopropionic acid 5-bromo-n- (carboxymethyl) anthranilic acid 16,17-dichloroheptadecanoic acid 8-hydroxy-7-quinolinecarboxylic acid 4- (4-fluorobenzoyl) butyric acid 4,4,4-trifluoro-3- (trifluoromethyl) butyric acid 2,4,6,8-decatetraenoic acid 6- (3,4-dimethoxyphenyl) -hexanoic acid 2- (n- (2,5-dimethylbenzyl) (carbamoyl) cyclohexanecarboxylic acid 2- (1-methyl-2,2-diphenyl-ethoxy) -benzoic acid

4,5-dikarboxy-gama-pentadekanolaktón kyselina 6-hepténová kyselina pentadec-14-énová kyselina d-(-)-chinová kyselina 4,7-dioxo-7-fenylheptánová kyselina 3-hydroxy-pyridín-4-karboxylová kyselina acetylsalicylsalicylová kyselina 4-(brómirietyl)-3-nitrobenzoová kyselina 2-metyl-4,4,4-trifluórmaslová kyselina n-ferc-boc-(2r,3r)-3-amino-2-hydroxy-4-fenylmaslová kyselina alfa-hydroxyhipurová kyselina 3-(karboxymetylaminometyl)-4-hydroxybenzoová kyselina 3-(4-etoxyfenylkarbamoyl)propiónová kyselina 2-jód-4,6-dibenzofurandikarboxylová kyselina 5-ŕerc-butylsalicylová kyselina 3,3-(5-chlór-2,4-dimetoxyfenyl)ureido)benzoová kyselina 4,5-dimetoxy-3-oxo-1,3-dihydro-izobenzofurán-1 -karboxylová kyselina 4,4,4-trifluór-3-metyl-2-buténová kyselina 2-metoxyškoricová kyselina (1s,3r)-(-)-gáfrová kyselina 3',4'-dimetyl-1,2,3,6-tetrahydroftalanilová kyselina (r)-n-(1-(1-naftyl)etyl)sukcínamová4,5-dicarboxy-gamma-pentadecanolactone 6-heptenoic acid pentadec-14-enoic acid d - (-) - quinic acid 4,7-dioxo-7-phenylheptanoic acid 3-hydroxy-pyridine-4-carboxylic acid acetylsalicylsalicylic acid 4- (Bromoethyl) -3-nitrobenzoic acid 2-methyl-4,4,4-trifluorobutyric acid n-tert-boc- (2r, 3r) -3-amino-2-hydroxy-4-phenylbutyric acid alpha-hydroxyhipuric acid 3- (carboxmethylaminomethyl) -4-hydroxybenzoic acid 3- (4-ethoxyphenylcarbamoyl) propionic acid 2-iodo-4,6-dibenzofuranedioic acid 5-tert-butylsalicylic acid 3,3- (5-chloro-2,4-dimethoxyphenyl) ureido) benzoic acid 4,5-dimethoxy-3-oxo-1,3-dihydro-isobenzofuran-1-carboxylic acid 4,4,4-trifluoro-3-methyl-2-butenoic acid 2-methoxycinnamic acid (1s, 3r - (-) - Camphoric acid 3 ', 4'-dimethyl-1,2,3,6-tetrahydrophthalanilic acid (R) -N- (1- (1-naphthyl) ethyl) succinamic acid

-142Φ ΦΦ ······ · · · ·· · φ φ φ φ φ ΦΦ • ΦΦΦ · · φ ·· · φ J · φφφφ ·· · •ΦΦ ·· φφφφ ΦΦ ··· kyselina 4-nitrobenzénsulfónová kyselina 3-(5,6,7,8-tetrahydro-naftalén-l -yl)-propiónová kyselina pseudokumén-5-sulfónová kyselina fenol-disulfónová kyselina 3-(2,4-dichlórbenzylidénamino)benzoová kyselina 5-benzoylpentánová kyselina 4-(4-chlórbenzylidénamino)salicylová kyselina 2-((1 h-indol-3-karbonyl)-amino)-benzoová kyselina 5-metyl-sulfónamido-indol-2-karboxylová kyselina 2,3-dichlórfenoxyoctová kyselina 5-chlór-2-furoová kyselina 2-benzyloxybenzoová kyselina p-chlórfenylpropargylová kyselina 1 -alfa-hydroxyizokaprónová kyselina 4’-chlór-2’-metoxyftalanilová kyselina gama-oxo-1 -pyrolidínmaslová kyselina trans-2,5-bis(trifluórmetyl)škoricová kyselina 2-[(4,6-dimetoxypyrimidín-2-yl)oxy]-6-fluórbenzoová kyselina d-(+)-10-gáforsulfónová kyselina 2,5-dichlórbenzénsulfónová kyselina 2-[3-(n-hexanoyl-hydrazíno)-3-oxo-propionylamino]-benzoová kyselina 3-metoxyškoricová n-(o-toluoyl)glycín kyselina 2-naftylamín-4,6,8-trisulfónová kyselina 2-chlór-5-nitrobenzoová kyselina 6-oxo-1,2-dihydro-6h-pyrol[3.2.1-ij]chinolín-5-karboxylová kyselina 2-bróm-5-chlórbenzoová kyselina 3-(2,6-dichlórfenyl)-5-metylizoxazol-4-karboxylová kyselina 1-bróm-2-naftoová kyselina d/-beta-hydroxykaprylová kyselina 1 -(2-chlór-6-fluórfenyl)cyklopentánkarboxylová kyselina 2-chlór-5-nitrobenzénsulfónová-142Φ · ······ · · · · · · · · · φ · φ · J · J · J · · · φ · · · · · φ · φ · · · φ · · · ··φ 4-nitrobenzenesulfonic acid 3- (5,6,7,8-tetrahydro-naphthalen-1-yl) -propionic acid pseudocuman-5-sulfonic acid phenol disulfonic acid 3- (2,4-dichlorobenzylidenamino) benzoic acid 5-benzoylpentanoic acid 4- ( 4-chlorobenzylidenamino) salicylic acid 2 - ((1H-indole-3-carbonyl) -amino) -benzoic acid 5-methylsulfonamido-indole-2-carboxylic acid 2,3-dichlorophenoxyacetic acid 5-chloro-2-furoic acid 2-benzyloxybenzoic acid p-chlorophenylpropargylic acid 1-alpha-hydroxyisocaproic acid 4'-chloro-2'-methoxyphthalanilic acid gamma-oxo-1-pyrrolidinebutyric acid trans-2,5-bis (trifluoromethyl) cinnamic acid 2 - [(4 6-dimethoxypyrimidin-2-yl) oxy] -6-fluorobenzoic acid d - (+) - 10-camphorsulfonic acid 2,5-dichlorobenzenesulfonic acid 2- [3 - (n-hexanoyl-hydrazino) -3-oxo-propionylamino] -benzoic acid 3-methoxycinnamic acid n- (o-toluoyl) glycine 2-naphthylamine-4,6,8-trisulfonic acid 2-chloro-5-nitrobenzoic acid 6-oxo-1,2-dihydro-6h-pyrrolo [3.2.1-ij] quinoline-5-carboxylic acid 2-bromo-5-chlorobenzoic acid 3- (2,6-dichlorophenyl) -5-methylisoxazole-4- 1-Bromo-2-naphthoic acid d-beta-hydroxycaprylic acid 1- (2-chloro-6-fluorophenyl) cyclopentanecarboxylic acid 2-chloro-5-nitrobenzenesulfonic acid

-143--143-

* «8 • 8 8 III * «8 • 8 8 III 88 88 8888 8 0 8888 8 0 88 88 O 8 O 8 8 0 8 0 8 8 8 8 8 0 8 0 O 8 ABOUT 8 0 8 8 0 8 8 0 0 8 8 8 8 8 8 8 8 8 8 88 88 88 88 8 e 8 e 8 8 8 8 8 8 8 8 «8 «8

kyselina 4-(4-hydroxy-1 -naftylazo)benzénsulfónová kyselina 2,-metoxy-5,-metylftalanilová kyselina 4-benzyloxyfenoxyoctová kyselina beta-butylhydroškoricová kyselina n-(4-nitrobenzoyl)antranilová kyselina 2-fenylmetánsulfinyl-benzoová kyselina 2-(trifluórmetyl)škoricová kyselina 5-hydroxyindol-3-b-propiónová kyselina (2r,3r)-2-benzyl-3-hydroxymaslová kyselina 5-(3,4-dimetoxy-fenyl)-penta-2,4-diénová kyselina 4-nitro-2-ftalimidobenzoová kyselina o-chlórfenoxyoctová kyselina beta-brómhydroškoricová kyselina 2-(2-cyklohexen-1 -yl)-2-metylmalónová kyselina 2,5-dimetoxybenzoová kyselina hydrokávová kyselina n-(2-etylfenyl)ftalámová kyselina (1r)-(+)-kamfanová kyselina 4-chlór-6-(2I4-dihydroxyfenyl-azo)-1-hydroxybenzén-2-sulfónová kyselina 1-cykloundecén-1-karboxylová kyselina sulfosalicylová kyselina 5,5'-dinitro-2,2'-bifenyldikarboxylová kyselina 2-furán-propiónová kyselina 3-(4-ho-3-meo-6-oxo-dekahydro-4ah-benzo(c)chromén-1-yl)-propiónová kyselina 3-[(2-metoxy-fenyl)-(toluén-4-sulfonyl)-amino]-propiónová kyselina izoindolín-1 -ón-2-(3-fenyl-2-propiónová) kyselina 4-bróm-4,4-difluór-2-buténová kyselina p-nitrofenylpyrohroznová kyselina 3-metyl-2-fenylvalérová kyselina (s)-(-)-2-brómhexánová kyselina 3,5-dibróm-2-anízová kyselina 3-cyklopentylpropiónová • · ·· ···· ·· • · · · <4- (4-hydroxy-1-naphthylazo) benzenesulfonic acid 2 , -methoxy-5 , -methylphthalanilic acid 4-benzyloxyphenoxyacetic acid beta-butylhydrocinnamic acid n- (4-nitrobenzoyl) anthranilic acid 2-phenylmethanesulfinyl-benzoic acid 2- ( 5-hydroxyindole-3-b-propionic acid (2r, 3r) -2-benzyl-3-hydroxybutyric acid 5- (3,4-dimethoxyphenyl) -penta-2,4-dienoic acid nitro-2-phthalimidobenzoic acid o-chlorophenoxyacetic acid beta-bromocinnamic acid 2- (2-cyclohexen-1-yl) -2-methylmalonic acid 2,5-dimethoxybenzoic acid hydrocavic acid n- (2-ethylphenyl) phthalic acid (1r) - (+) - camphanic acid, 4-chloro-6- (2 L 4-dihydroxyphenyl-azo) -1-hydroxybenzene-2-sulfonic acid 1-cycloundecene-1-carboxylic acid, sulfosalicylic acid, 5,5-dinitro-2, 2'-Biphenyldicarboxylic acid 2-furan-propionic acid 3- (4-ho-3-meo-6-oxo-decahydro-4H-benzo (c) chromen-1-yl) -propiones 3 - [(2-Methoxy-phenyl) - (toluene-4-sulfonyl) -amino] -propionic acid Isoindolin-1-one-2- (3-phenyl-2-propionic acid) 4-bromo-4,4 -difluoro-2-butenoic acid p-nitrophenylpyruvic acid 3-methyl-2-phenylvaleric acid (s) - (-) - 2-bromohexanoic acid 3,5-dibromo-2-anisic acid 3-cyclopentylpropionic acid · · ·· ·· ·· ·· • · · · <

999 · 9 · «999 · 8 · «

-144kyselina 2,3,6-trichlórbenzoová kyselina 2,6-difluórfenyloctová kyselina c/s-9,10-epoxystearová kyselina 6-oxo-1,4,5,6-tetrahydropyridazín-3-karboxylová kyselina 3,5,7-trimetyl-adamantán-l -karboxylová kyselina 3-hexín-1,1,6,6-tetrakarboxylová kyselina 3-hydroxy-4-metoxyškoricová kyselina 4-ŕerc-butyl-2,6-dimetylbenzoová kyselina 3-metylbenzofurán-2-karboxylová kyselina 2-hydroxyimino-3-(4-metoxy-fenyl)-propiónová kyselina 2,3,4-trimetyl-cyklopentánkarboxylová kyselina 4-bróm-2-(fenoxy)benzoová kyselina 4-(etyltio)benzoová kyselina (4-etoxy-2-oxo-3-pyrolín-1 -yl)octová kyselina 2-naftoxyoctová kyselina (4,6-dihydroxy-5-fenyl-pyrimidín-2-ylsulfanyl)-octová kyselina 11-(4-acetylfenoxy)-undekánová kyselina kyanooctová kyselina 3-metylglutárová kyselina 4,5-dimetoxy-2-metylbenzoová kyselina 2-etyl-2-metyljantárová kyselina 2-ŕerc-butyl-5-pyridínsulfónová kyselina 4-(trimetylsilyl)benzoová kyselina boc-1 -tiazolidín-4-karboxylová kyselina (1 s,3r)-1 -amino-1 -karboxycyklopentán-3-octová kyselina 2-(3-fenyl-tioureido)-benzoová kyselina 2-(3-nitropyrid-2-yltio)propiónová kyselina 4'-chlór-3'-nitroftalanilová kyselina 3,4,5-triacetoxybenzoová kyselina pyrazín-2,3-dikarboxylová, monoamid kyselina 3-etoxykarbonyl-4,4-difenyl-but-3-énová kyselina n-(3-metoxyfenyl)glutarámová • ·· ·· ···· ··-144 2,3,6-trichlorobenzoic acid 2,6-difluorophenylacetic acid cis-9,10-epoxystearic acid 6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxylic acid 3,5,7- trimethyl-adamantane-1-carboxylic acid 3-hexine-1,1,6,6-tetracarboxylic acid 3-hydroxy-4-methoxycinnamic acid 4-tert-butyl-2,6-dimethylbenzoic acid 3-methylbenzofuran-2-carboxylic acid 2-hydroxyimino-3- (4-methoxyphenyl) -propionic acid 2,3,4-trimethyl-cyclopentanecarboxylic acid 4-bromo-2- (phenoxy) benzoic acid 4- (ethylthio) benzoic acid (4-ethoxy-2) -oxo-3-pyrrolin-1-yl) acetic acid 2-naphthoxyacetic acid (4,6-dihydroxy-5-phenyl-pyrimidin-2-ylsulfanyl) -acetic acid 11- (4-acetylphenoxy) -undecanoic acid cyanoacetic acid 3 methyl-glutaric acid 4,5-dimethoxy-2-methylbenzoic acid 2-ethyl-2-methylsuccinic acid 2- tert -butyl-5-pyridinesulfonic acid 4- (trimethylsilyl) benzoic acid boc-1-thiazolidine-4-carboxylic acid (1) with 3r) -1-amino-1-carboxycyclopentane-3-acetic acid 2- (3-phenylthioureido) -benzoic acid 2- (3-nitropyrid-2-ylthio) propionic acid 4'-chloro-3'-nitropthalanilic acid 3,4,5-triacetoxybenzoic acid pyrazine-2,3-dicarboxylic acid, 3-ethoxycarbonyl-4,4-diphenyl-but-3-enoic acid, monoamide n- (3-methoxyphenyl) glutaramic acid • ·· ·· ·· ·· ··

B · · ·· · · · · • ··* · · · 99B · 99 · 99

-145kyselina oktenyl-dijantárová kyselina 3-amino-2-chlórbenzoová kyselina n-n-propyl-d-asparágová kyselina 4-benzyloxy-3,5-dimetbylbenzoová kyselina (+/-)-9-hydroxyoktadeka-1 Oe, 12z-diénová kyselina (r)-(+)-indolín-2-karboxylová kyselina 4-chlórbenzoová kyselina 2-(2,2-dichlór-etyl)-5-metoxy-benzoová kyselina 1,2-dihydro-6-metoxy-1 -metyl-2-oxo-4-chinolínkarboxylová kyselina 2,2-diizopropylmalonámová kyselina 3-fluór-4-metylbenzoová kyselina 3-nitrobenzénsulfónová kyselina n-p-nitrobenzoyl-1 -glutámová kyselina 5-(2-fluórbenzoyl)tiofén-2-octová kyselina 2-hydroxy-4-metoxybenzofenón-5-sulfónová kyselina chromotropová kyselina 2-(trifluórmetyltio)benzoová kyselina d/-4-hydroxyfenylmliečna kyselina (3-metyl-4-oxo-4,9-dihydro-pyrazolo(3,4-b)chinolín-1-yl)-octová kyselina 3-(4-oktyloxy-fenyl)-akrylová kyselina n-alfa-terc-boc-5,5-dimetyl-d-tiazolidín-4-karboxylová kyselina 2-metoxyizoftalová kyselina n-alfa-z-1 -alanyl-1 -glutámová kyselina z-gama-amino-beta-hydroxy-maslová kyselina 4-(1,2,3,4-tetrahydro-naftalén-1-yl)-maslová kyselina n-(4-nitrobenzoyl)-6-aminokaprónová kyselina 2-karboxymetyl-oktahydro-indén-2-karboxylová kyselina o-krezol-4-sulfónová kyselina 2,3,3,4,4-pentachlór-maslová kyselina trichlórmetylfosfónová kyselina 3-formyl-4-hydroxybenzoová kyselina n-lauroyliminodioctová-145 octenyl-disuccinic acid 3-amino-2-chlorobenzoic acid n-propyl-d-aspartic acid 4-benzyloxy-3,5-dimethylbenzoic acid (+/-) - 9-hydroxyoctadeca-10e, 12z-dienoic acid ( r) - (+) - Indoline-2-carboxylic acid 4-chlorobenzoic acid 2- (2,2-dichloroethyl) -5-methoxybenzoic acid 1,2-dihydro-6-methoxy-1-methyl-2 -oxo-4-quinolinecarboxylic acid 2,2-diisopropylmalonamic acid 3-fluoro-4-methylbenzoic acid 3-nitrobenzenesulfonic acid np-nitrobenzoyl-1-glutamic acid 5- (2-fluorobenzoyl) thiophene-2-acetic acid 2-hydroxy- 4-Methoxybenzophenone-5-sulfonic acid chromotropic acid 2- (trifluoromethylthio) benzoic acid d] -4-hydroxyphenyl-lactic acid (3-methyl-4-oxo-4,9-dihydro-pyrazolo (3,4-b) quinolin-1) -yl) -acetic acid 3- (4-octyloxy-phenyl) -acrylic acid n-alpha-tert-boc-5,5-dimethyl-d-thiazolidine-4-carboxylic acid 2-methoxyisophthalic acid n-alpha-z- 1 -alanyl-1-glutamic acid z-ga 4- (1,2,3,4-Tetrahydro-naphthalen-1-yl) -butyric acid n- (4-nitrobenzoyl) -6-aminocaproic acid 2-carboxymethyl-octahydro- indene-2-carboxylic acid o-cresol-4-sulfonic acid 2,3,3,4,4-pentachloro-butyric acid trichloromethylphosphonic acid 3-formyl-4-hydroxybenzoic acid n-lauroyliminodioacetic acid

-146--146-

• ·· B B • II· • B B • II · B B B · e b B B B · e b BBBB B B BBBB B B BB B B B B BB B B B B B B B B ·· BB ·· BB BB BB e b e b B B B B B B B B

kyselina 2,3,5,6-tetrafluórbenzoová kyselina 3-formylsalicylová kyselina 4-bróm-2-chlór-5-fluórbenzoová kyselina 3-(3-brómbenzoyl)propiónová kyselina 2-hydroxy-2-trifluórmetyl-eikoz-4-énová kyselina 2',3,4-benzofenóntrikarboxylová kyselina 2-hydroxyimino-maslová kyselina nafto(2,3-d)-1,3-dioxolén-2-karboxylová kyselina 2-(8-chlór-1 -naftyltio)octová kyselina dihydronaftalén-1,4-dikarboxylová kyselina cyklobután-1,2,3,4-tetrakarboxylová kyselina alfa-metyl-2,4,5-trimetoxyškoricová kyselina p-tolyl-fosfónová kyselina c/s-3A4,4-tetrachlórkrotónová kyselina alfa-ketooktánová kyselina 1,8-naftaléndikarboxylová kyselina 2,2-dimetylvalérová kyselina 3-fluór-2-metyl-benzoová kyselina (s)-(+)-2-chlór-3-fenylpropiónová kyselina 3-chlórtetrafluórpropiónová kyselina 2,4-dibrómbenzoová kyselina 4-(5-(amino-karboxy-metyl)-tiofén-2-yl)-maslová kyselina p-krezidín-6-sulfónová beta ŕerc-butylester kyseliny fmoc-d-asparágovej kyselina 3,4-diacetamidobenzoová kyselina 2-( 1 -trimetylsilanyl-vinyl)-benzoová formylglycín kyselina 2,6-dimetoxybenzoová kyselina 4-bróm-3-hydroxy-naftalén-2-karboxylová kyselina cyklohexándiamíntetraoctová kyselina 4-pentylbenzoová kyselina 2-amino-4,5-dibróm-3,6-dimetyl-benzoová ·· ·· ···· ·· • · · · · ··· · · · ·2,3,5,6-tetrafluorobenzoic acid 3-formylsalicylic acid 4-bromo-2-chloro-5-fluorobenzoic acid 3- (3-bromobenzoyl) propionic acid 2-hydroxy-2-trifluoromethyl-eicos-4-enoic acid 2 ', 3,4-benzophenone tricarboxylic acid 2-hydroxyimino-butyric acid naphtho (2,3-d) -1,3-dioxolene-2-carboxylic acid 2- (8-chloro-1-naphthylthio) acetic acid dihydronaphthalene-1 4-dicarboxylic acid cyclobutane-1,2,3,4-tetracarboxylic acid alpha-methyl-2,4,5-trimethoxycinnamic acid p-tolylphosphonic acid cis-3A4,4-tetrachlorocrotonic acid alpha-ketoctanoic acid 1 8-naphthalenedicarboxylic acid 2,2-dimethylvaleric acid 3-fluoro-2-methylbenzoic acid (s) - (+) - 2-chloro-3-phenylpropionic acid 3-chlorotetrafluoropropionic acid 2,4-dibromobenzoic acid 4- ( 5- (Amino-carboxymethyl) -thiophen-2-yl) -butyric acid p-cresidine-6-sulfonic acid fmoc-d-aspartic acid tert-butyl ester 3,4-diacetamide obenzoic acid 2- (1-trimethylsilanyl-vinyl) -benzoic formylglycine 2,6-dimethoxybenzoic acid 4-bromo-3-hydroxy-naphthalene-2-carboxylic acid cyclohexanediaminetetraacetic acid 4-pentylbenzoic acid 2-amino-4,5-dibromo -3,6-Dimethyl-benzoic acid

-147kyselina 2-(4-fluórfenyl)-2-adamantán-octová kyselina 2-cyklohexylglykolová kyselina 4,5,515-tetrafluór-4-trifluórmetoxy-2-penténová kyselina beta-hydroxyasparágová kyselina 4-(2-benzoylamino-3-(4-metoxy-fenyl)-akryloylamino)-maslová kyselina c/s-7-oktadecénová kyselina 1-bróm-4,4-dichlór-1,3-butadién-1-karboxylová kyselina 4'-etylmaleanilová kyselina 2-hydroxy-3-nitroacetanilid-5-sulfónová kyselina (-)-diacetyl-l-vínna kyselina 4,4'-( 1,4-fenylén)bis(2-oxo-3-buténová) kyselina 5-nitroizoftalová kyselina 4-chlór-o-anízová kyselina 2-amino-3-(4-karboxyfenyl)propiónová kyselina s-trifenylmetyl-3-merkaptopropiónová kyselina 5-bróm-3,4-dihydroxybenzoová kyselina 3-(n-propylkarbamoyl)-5-norbornén-2-karboxylová kyselina (5s, 12s)-dihydroxy-(6e,8e, 10e, 14z)-eikozatetraénová kyselina heptánová kyselina adamantán-1 -yl-benzoylamino-octová kyselina 3-(1h-imidazol-2-yl)-2-(4-metoxy-benzoylamino)-propiónová kyselina n-(2-(3-chlór-5-trifluórmetyl)pyridylaminoetyl)maleámová kyselina 6-chlór-2-(1,3-dioxo-indán-2-yl)-chinolín-8-sulfónová kyselina 3-fenylmetánsulfonyl-propiónová kyselina (5,6,7,8-tetrahydro-naftalén-2-yl)-octová kyselina (4-(3-fenyl-propyl)-fenyl)-octová kyselina 2l3-dibróm-4’-(etoxykarbonyl)sukcínanilová kyselina 3,4-dietoxybenzoová kyselina fmoc-1 -tiazolidín-4-karboxylová kyselina 4-(6-(3-karboxy-propylamino)-5-nitro-pyridín-2-ylamino)-maslová kyselina 2-(trifluórmetoxy)benzoová kyselina (3-kyano-6-(4-metoxy-fenyl)-2-oxo-cyklohexyl)-octová-147 2- (4-fluorophenyl) -2-adamantan-acetic acid 2-cyclohexylglycolic acid 4,5,5 1 5-Tetrafluoro-4-trifluoromethoxy-2-pentenoic acid beta-hydroxyaspartic acid 4- (2-benzoylamino-3) - (4-Methoxy-phenyl) -acryloylamino) -butyric acid cis-7-octadecenic acid 1-bromo-4,4-dichloro-1,3-butadiene-1-carboxylic acid 4'-ethylmaleanilic acid 2-hydroxy 3-nitroacetanilide-5-sulfonic acid (-) - diacetyl-1-tartaric acid 4,4 '- (1,4-phenylene) bis (2-oxo-3-butenoic) 5-nitroisophthalic acid 4-chloro- o-anisic acid 2-amino-3- (4-carboxyphenyl) propionic acid s-triphenylmethyl-3-mercaptopropionic acid 5-bromo-3,4-dihydroxybenzoic acid 3- (n-propylcarbamoyl) -5-norbornene-2-carboxylic acid (5s, 12s) -dihydroxy- (6e, 8e, 10e, 14z) -eicosatetraenoic acid heptanoic acid adamantan-1-yl-benzoylamino-acetic acid 3- (1H-imidazol-2-yl) -2- (4- methoxy-benzoylamino) propionic acid n- (2- (3-chloro-5-trifluoromethyl) 6-chloro-2- (1,3-dioxo-indan-2-yl) -quinoline-8-sulfonic acid 3-phenylmethanesulfonyl-propionic acid (5,6,7,8-tetrahydro-naphthalene-) 2-yl) -acetic acid (4- (3-phenyl-propyl) -phenyl) -acetic acid 2 l 3-dibromo-4 '- (ethoxycarbonyl) sukcínanilová 3,4-diethoxy-benzoic acid, fmoc-1-thiazolidine-4 4- (6- (3-carboxy-propylamino) -5-nitro-pyridin-2-ylamino) -butyric acid 2- (trifluoromethoxy) benzoic acid (3-cyano-6- (4-methoxy-phenyl)) 2-oxo-cyclohexyl) -acetic acid

-148--148-

• ·· • ·· 99 99 9999 9999 99 9 99 9 • · • · 9 9 9 9 9 9 9 9 99 9 9 999 9 999 9 9 9 9 9 9 9 9 9 9 9 9 99 9 99 99 99 99 99 9 9 99 9 9

kyselina 4-acetamido-4,-aminostilbén-2,2'-disulfónová kyselina 2-bibenzylkarboxylová kyselina tricyklo(12.2.2.2(6I9))eikoza-1(17)I6,8,14(18),15,19-hexaén-7-karboxylová kyselina 4l-bróm-3,-metylglutáranilová kyselina 4-(3-(3-nitrobenzoyl)-2-tioureido)benzoová kyselina 5-(ŕerc-butyl)-2-hydroxycyklohexánkarboxylová kyselina cyklododekánkarboxylová kyselina 5-hydroxymetyl-2,6-dimetyl-nikotínová kyselina 3,-chlór-2'-metylsukcínanilová boc-d-norleucín kyselina tetraoxa-bicyklo(12.3.1 )oktadeka-1 (17), 14(18), 15-trién-18-karboxylová kyselina 2-metylimidazo[1,2-a]pyridín-3-karboxylová kyselina 6-chlór-2h-1 -benzopyrán-3-karboxylová kyselina 4-(2-(3,3-dimetyl-2,3-dihydro-benzo(b)tiofén-5-yl)-propenyl)benzoová kyselina 3-(2-acetylamino-3-(4-metoxy-fenyl)-akryloylamino)-propiónová kyselina stearidónová kyselina (+/-)-1 -amino-c/s-3-fosfonocyklohexánkarboxylová kyselina 6-metylchromón-2-karboxylová kyselina 4-acetoxyhydroškoricová kyselina 3,4,5-tribróm-2-furoová kyselina 1 -(p-tolyl )-1 -cyklopentánkarboxylová kyselina 5,7-bis(trifluórmetyl)-4-hydroxychinolín-3-karboxylová kyselina n-(2-hydroxyetyl)etyléndiamíntrioctová kyselina alfa-brómškoricová kyselina 2,3,4-trichlórglutakónová kyselina 4-acetyl-ftalová kyselina 3-(4-oktadecyl)-benzoylakrylová kyselina n-alfa-z-/?-beta-boc-1 -diaminopropiónová kyselina n-(2-hydroxybenzoyl)-1-asparágová metyl-4-karboxy-2-nitrobenzoát kyselina 4-amino-2-chlórpyridín-5-karboxylová kyselina 3,5-dihydroxy-2-naftoová • 99 99 ···· 9· ·· · 9 9 9 4 9·acid, 4-acetamido-4, -aminostilbén-2,2'-disulfonic acid, 2-bibenzylcarboxylic acid tricyclo (12.2.2.2 (6 I 9)) eicosa-1 (17) I, 6,8,14 (18), 15, 19-Hexaen-7-carboxylic acid 4 1 -Bromo-3 , -methylglutananilic acid 4- (3- (3-nitrobenzoyl) -2-thioureido) benzoic acid 5- (tert-butyl) -2-hydroxycyclohexanecarboxylic acid cyclododecanecarboxylic acid 5 -hydroxymethyl-2,6-dimethyl-nicotinic acid 3 , -chloro-2'-methylsucciniline boc-d-norleucine tetraoxa-bicyclo (12.3.1) octadeca-1 (17), 14 (18), 15-triene- 18-carboxylic acid 2-methylimidazo [1,2-a] pyridine-3-carboxylic acid 6-chloro-2h-1-benzopyran-3-carboxylic acid 4- (2- (3,3-dimethyl-2,3- dihydro-benzo (b) thiophen-5-yl) -propenyl) benzoic acid 3- (2-acetylamino-3- (4-methoxy-phenyl) -acryloylamino) -propionic acid stearidonic acid (+/-) - 1-amino cis-3-phosphonocyclohexanecarboxylic acid 6-methylchromone-2-carboxylic acid 4-acetoxyhydrocinnamic acid 3,4,5 -tribromo-2-furoic acid 1- (p-tolyl) -1-cyclopentanecarboxylic acid 5,7-bis (trifluoromethyl) -4-hydroxyquinoline-3-carboxylic acid n- (2-hydroxyethyl) ethylenediaminetriacetic acid 3,4-trichloroglutaconic acid 4-acetyl-phthalic acid 3- (4-octadecyl) -benzoylacrylic acid n-alpha-2-R-beta-boc-1-diaminopropionic acid n- (2-hydroxybenzoyl) -1- aspartic methyl 4-carboxy-2-nitrobenzoate 4-amino-2-chloropyridine-5-carboxylic acid 3,5-dihydroxy-2-naphthoic acid • 99 99 ··· 9 · ·· · 9 9 9 4 9 ·

999 999 99..

-149kyselina p-kumarová kyselina 9-hydroxydekánová kyselina 2-(3-chlór-1,4-dioxo-1,4-dihydronaftalén-2-ylamino)-hexánová kyselina 3-(2,4-dimetoxy-fenyl)-propiónová kyselina 4,4,4-trifluórmaslová kyselina ŕrans-2-fenyl-1 -cyklopropánkarboxylová kyselina 4-jódfenyloctová kyselina [fenetyl-(toluén-4-sulfonyl)-amino]-octová kyselina 2,3-dihydro-3-oxo-(1h)izoindol-1-ylidénoctová kyselina boc-12-aminododekánová kyselina 2-acetyl-3,4,5,6-tetrachlórbenzoová kyselina 1 -benzoylpiperidín-4-karboxylová kyselina (s)-2-metyldekánová kyselina 1 -hydroxyamino-cyklohexánkarboxylová kyselina 8-chlórmetyl-7-metoxy-4-oxo-4h-chromén-2-karboxylová kyselina 2-bróm-3-nitrobenzoová kyselina 3-(trifluórmetyl)fenyloctová kyselina 3-(2-benzoylamino-3-fenyl-akryloylamino)-propiónová kyselina n-(3,4-dimetoxyfenetyl)-maleámová kyselina 4,6-dioxoheptánová kyselina 4-chlór-alfa-metylfenyloctová kyselina 4,-metyl-2-bifenylkarboxylová kyselina alfa-guanidínoglutárová kyselina n-(2,3-xylyl)ftalámová kyselina 5-nitro-2-(4-(1,1,3,3-tetrametylbutyl)fenoxy)benzénsulfónová kyselina 4-propyloxybifenyl-4,-karboxylová kyselina 1 -(4-chlóranilíno)-6-metyl-4-oxo-1,4-dihydro-3-pyridínkarboxylová kyselina 2-amino-4-metyl-tiazol-5-sulfónová-149 p-coumaric acid 9-hydroxydecanoic acid 2- (3-chloro-1,4-dioxo-1,4-dihydronaphthalen-2-ylamino) -hexanoic acid 3- (2,4-dimethoxyphenyl) -propionic acid Trans-2-phenyl-1-cyclopropanecarboxylic acid 4,4,4-trifluorobutyric acid 4-iodophenylacetic acid [phenethyl- (toluene-4-sulfonyl) -amino] -acetic acid 2,3-dihydro-3-oxo- (1h ) isoindol-1-ylideneacetic acid boc-12-aminododecanoic acid 2-acetyl-3,4,5,6-tetrachlorobenzoic acid 1-benzoylpiperidine-4-carboxylic acid (s) -2-methyldecanoic acid 1 -hydroxyamino-cyclohexanecarboxylic acid 8 -chloromethyl-7-methoxy-4-oxo-4h-chromene-2-carboxylic acid 2-bromo-3-nitrobenzoic acid 3- (trifluoromethyl) phenylacetic acid 3- (2-benzoylamino-3-phenyl-acryloylamino) -propionic acid n- (3,4-dimethoxyphenethyl) -maleamic acid 4,6-dioxoheptanoic acid 4-chloro-alpha-methylphenylacetic acid 4 , -methyl-2-biphenylcarboxylic acid alpha-guanidinoglutaric acid k yselina of N- (2,3-xylyl) phthalamic acid 5-nitro-2- (4- (1,1,3,3-tetramethylbutyl) phenoxy) benzenesulfonic acid 4-propyloxybifenyl-4-carboxylic acid 1 - (4- chloroanilino) -6-methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid 2-amino-4-methyl-thiazole-5-sulfonic acid

3-chlór-4-(metylsulfonyl)tiofén-2-karbonyl-chloride kyselina 2-(2-o-tolyloxy-acetylamino)-benzoová kyselina 3'-metylglutaranilová kyselina 3-oktylsulfanyl-propiónová • ·· ·· ···· ·· ·· · · · · « • ··· · · 9 93-chloro-4- (methylsulfonyl) thiophene-2-carbonyl chloride 2- (2-o-tolyloxy-acetylamino) -benzoic acid 3'-methylglutaranilic acid 3-octylsulfanyl-propionic acid • ·· ·· ···· 9 9

-150·· kyselina 2,3-dihydroxy-4-metoxybenzoová kyselina 2-furánglyoxylová kyselina chlórdifluór-octová kyselina 1,3,3al6,7,7a-hexahydro-1-oxo-4,5,6-trimetyl-7-izobenzofuránkarboxylová kyselina (+)-benzylmetylfenylsilyloctová kyselina 4,4'-stilbéndikarboxylová kyselina 4-(2-benzotiazolyltio)-maslová kyselina 2-(1 -acetyl-2-naftyloxy)-propiónová kyselina 2-hydroxy-6-fenyl-3,5-pyridíndikarboxylová kyselina o-benzamidoglykolová kyselina 2-hydroxy-3-butínová-150 ·· 2,3-dihydroxy-4-methoxybenzoic acid 2-furanglyoxylic acid chlorodifluoroacetic acid 1,3,3a 1 6,7,7a-hexahydro-1-oxo-4,5,6-trimethyl-7 -isobenzofuranecarboxylic acid (+) - benzylmethylphenylsilylacetic acid 4,4'-stilbenedicarboxylic acid 4- (2-benzothiazolylthio) butyric acid 2- (1-acetyl-2-naphthyloxy) -propionic acid 2-hydroxy-6-phenyl-3, 5-pyridinedicarboxylic acid o-benzamidoglycolic acid 2-hydroxy-3-butanoic acid

2-karboxy-4-(trifluórmetyl)difenyl-sulfid boc-1 -homofenylalanín kyselina n-alfa-fmoc-fn-beta-boc)-diaminopropiónová kyselina (e)-10-hydroxy-2-decénová kyselina 2-benzoylamino-3-(1 h-imidazol-4-yl)-akrylová kyselina 9-tetradecínová kyselina 3-(2-karboxy-etyl)-tiazol-2-yl-amino)-propiónová kyselina 5-(4-(4-metoxykarbonyl-butyl)-fenyl)-5-oxo-pentánová kyselina 2,3,4-trimetoxyškoricová kyselina 4-dodekanoylamino-benzoová kyselina 3-metylpikolínová kyselina 2-chlór-n-maslová kyselina fmoc-2-aminoindán-2-karboxylová kyselina oktadekadiénová, konjugovaná kyselina 3-(4-n-butoxybenzoyl)propiónová kyselina (2-metoxy-4-nitro-fenyl)-fosfónová kyselina 2,4,6-oktatriénová kyselina 5-chlór-2-nitrobenzoová kyselina 3-(4-metoxy-fenyl)-propínová kyselina 2-chlórfenyloctová kyselina 5-(4-morfolíno)-2h-tetrazol-2-octová2-Carboxy-4- (trifluoromethyl) diphenyl sulfide boc-1-homophenylalanine n-alpha-fmoc-fn-beta-boc) -diaminopropionic acid (e) -10-hydroxy-2-decenoic acid 2-benzoylamino-3 - (1 H -imidazol-4-yl) -acrylic acid 9-Tetradecinic acid 3- (2-carboxy-ethyl) -thiazol-2-yl-amino) -propionic acid 5- (4- (4-methoxycarbonyl-butyl) (phenyl) -5-oxo-pentanoic acid 2,3,4-trimethoxycinnamic acid 4-dodecanoylamino-benzoic acid 3-methyl-picolinic acid 2-chloro-n-butyric acid fmoc-2-aminoindane-2-carboxylic acid octadecadienoic acid, conjugated 3- (4-n-butoxybenzoyl) propionic acid (2-methoxy-4-nitro-phenyl) -phosphonic acid 2,4,6-octatrienoic acid 5-chloro-2-nitrobenzoic acid 3- (4-methoxy-phenyl) 2-Chlorophenylacetic acid 5- (4-morpholino) -2h-tetrazole-2-acetic acid

-151 --151 -

• ·· • · • ··· • ·· • · • ··· ·· • · • · · · • · • · ···· • • ···· • • ·· 9 • · · · • · 9 ·· 9 9 • · · · • · · · • · • · • · • · 99 99 99 99

kyselina 6-metyl-4-oxo-1-(4-toluidíno)-1,4-dihydro-3-pyridínkarboxylová kyselina cbz-1-alfa-aminokorková kyselina 3-adamantán-1 -yl-propiónová kyselina 4-(6-butoxy-naftalén-2-yl)-4-oxo-maslová kyselina 4-[(5,6,718-tetrahydro-5,5,8,8-tetrametyl-2-naftalényl)karboxamido]benzoová kyselina 3,4-difluórbenzoová kyselina 2-oxo-1 -cyklohexánpropiónová kyselina 2',4'-dichlór-1,2,3,6-tetrahydroftalanilová kyselina 3-brómmetyl-benzoová kyselina c/s-hexahydro-/7-(4-chlórfenyl)ftalámová kyselina m-xylén-4-sulfónová kyselina 2-(2-chlór-1,1,2-trifluóretoxy)-p-anízová kyselina 2-(1,2,3,4-tetrahydro-6-naftylmetyl)benzoová kyselina 3-(4-dimetylamino-fenyl)-2-metyl-akrylová kyselina boc-d/-alfa-aminomaslová kyselina 3-[(4,6-dimetoxypyrinnidín-2-yl)oxy]benzoová kyselina 2,5-dinitrobenzoová kyselina trans-12-oktadecénová kyselina 2-chlór-adamantán-2-karboxylová kyselina 3-fluór-4-metoxyfenyloctová kyselina 2,4,6-tribrómbenzoová kyselina 2-[[2-(4-metylfenyl)hydrazíno]-karbonyl]-benzoová kyselina 1 -(3-fluórfenyl)cyklohexánkarboxylová kyselina mezitylénsulfónová kyselina 2,5-difluórškoricová kyselina 3-(4-metoxyfenyl)propiónová kyselina metakrylová kyselina d/-s-acetyl-2-benzyl-3-merkaptopropiónová kyselina 2,5-difluórbenzoová kyselina 2-nitroizoftalová kyselina 2,3-difluór-4-(trifluórmetyl)benzoová • ·· ·· ···· ·· ·· · · · · · · · • ··· · · · · ·6-methyl-4-oxo-1- (4-toluidino) -1,4-dihydro-3-pyridinecarboxylic acid cbz-1-alpha-aminocorkic acid 3-adamantan-1-yl-propionic acid 4- (6- butoxy-naphthalen-2-yl) -4-oxo-butyric acid 4 - [(5,6,7 1 8-5,5,8,8-tetramethyl-2-naphthalenyl) carboxamido] benzoic acid 3,4- 2-oxo-1-cyclohexanepropionic acid 2 ', 4'-dichloro-1,2,3,6-tetrahydrophthalanilic acid 3-bromomethylbenzoic acid cis-hexahydro- [7- (4-chlorophenyl) phthalic acid] -difluorobenzoic acid m-xylene-4-sulfonic acid 2- (2-chloro-1,1,2-trifluoroethoxy) -p-anisic acid 2- (1,2,3,4-tetrahydro-6-naphthylmethyl) benzoic acid 3- (4-dimethylamino-phenyl) -2-methyl-acrylic acid boc-d-alpha-aminobutyric acid 3 - [(4,6-dimethoxypyrinnidin-2-yl) oxy] benzoic acid 2,5-dinitrobenzoic acid trans-12 2-chloro-adamantane-2-carboxylic acid 3-fluoro-4-methoxyphenylacetic acid 2,4,6-tribromobenzoic acid 2 - [[2- (4-methylphenyl) hyd] Razino] carbonyl] -benzoic acid 1- (3-fluorophenyl) cyclohexanecarboxylic acid mesitylenesulfonic acid 2,5-difluorocinnamic acid 3- (4-methoxyphenyl) propionic acid methacrylic acid d -s-acetyl-2-benzyl-3-mercaptopropionic acid 2,5-Difluorobenzoic acid 2-Nitroisophthalic acid 2,3-Difluoro-4- (trifluoromethyl) benzoic acid · ··· ················ · ·

- 152kyselina 6-(2-hydroxybenzylidénamino)hexánová kyselina (1r-(1alfa,2beta,3alfa))-(+)-3-metyl-2-(nitrometyl)-5-oxocyklopentánoctová kyselina 4-(4'-metoxybenzylidén)aminoškoricová kyselina 4-bróm-3-nitrobenzoová kyselina 9-benzoylnonánová kyselina 4'-acetamidosukcínanilová kyselina n-toluénsulfonyl-1 -glutámová kyselina 2,4,6-triizopropylbenzoová kyselina 5-azido-2-nitrobenzoová kyselina 4-hexadecyloxybenzoová kyselina 1,2-dihydroxyantrachinón-3-sulfónová kyselina 1,3-adamantándioctová kyselina 4-[2-(benzotiazol-2-ylsulfanyl)-acetylamino]-benzoová kyselina fosfoglykolová kyselina n-alfa-boc-n-beta-aloc-1 -diaminopropiónová kyselina 2-chlór-6-fluórbenzoová kyselina 1 -(4-metoxyfenyl)etyliminoxy-octová kyselina 4-(3-(1-butyrylamino-2,2,2-trichlór-etyl)-tioureido)-benzoová kyselina (+/-)-5-jód-3-izopropylpentánová kyselina 4-fluórmandlová kyselina alfa-kyano-3-hydroxyškoricová kyselina 5-metoxy-2-nitrobenzoová kyselina 4-fluór-2-(trifluórmetyl)fenyloctová kyselina oktán-2-sulfónová kyselina krezolsírová kyselina aleuritová- 152 (6- (2-hydroxybenzylideneamino) hexanoic acid) (1R- (1alpha, 2beta, 3alpha)) - (+) - 3-methyl-2- (nitromethyl) -5-oxocyclopentaneacetic acid 4- (4'-methoxybenzylidene) amino cinnamic acid 4-bromo-3-nitrobenzoic acid 9-benzoylnonanoic acid 4'-acetamidosuccinilic acid n-toluenesulfonyl-1-glutamic acid 2,4,6-triisopropylbenzoic acid 5-azido-2-nitrobenzoic acid 4-hexadecyloxybenzoic acid 1,2- dihydroxyantraquinone-3-sulfonic acid 1,3-adamantanediacetic acid 4- [2- (benzothiazol-2-ylsulfanyl) -acetylamino] -benzoic acid phosphoglycolic acid n-alpha-boc-n-beta-aloc-1-diaminopropionic acid 2- chloro-6-fluorobenzoic acid 1- (4-methoxyphenyl) ethyliminoxy-acetic acid 4- (3- (1-butyrylamino-2,2,2-trichloroethyl) thioureido) -benzoic acid (+/-) - 5 -iodo-3-isopropylpentanoic acid 4-fluoro-butyric acid alpha-cyano-3-hydroxycinnamic acid 5-methoxy-2-nitrobenzoic acid 4-fluoro-2- (trifluoromethyl) (l) phenylacetic acid octane-2-sulfonic acid cresolsulfuric acid aleuritic acid

1-(2-chlór-5-sulfofenyl)-3-metyl-5-pyrazolón kyselina pentadekafluóroktánová kyselina n-(5-nitro-2-tiazolyl)ftalámová kyselina 2-(2-chlórfenoxy)propiónová kyselina 1-gama-karboxyglutámová kyselina (r)-(-)-fenyljantárová • ·· ·· ···· ·· ··· ·· · ··· • ··· 999 991- (2-chloro-5-sulfophenyl) -3-methyl-5-pyrazolone pentadecafluorooctanoic acid n- (5-nitro-2-thiazolyl) phthalic acid 2- (2-chlorophenoxy) propionic acid 1-gamma-carboxyglutamic acid (r) - (-) - phenylsuccinate 999 99

-153kyselina 1,18-oktadekándiová kyselina 3-amino-5-bróm-benzoová kyselina 5-chlór-tricyklo(2.2.1.0(2,6))heptán-3-karboxylová kyselina 2-hydroxydokozánová kyselina 4-metoxyfenyloctová kyselina palmito-olejová kyselina 3-benzo[1 .SJdioxol-S-yl^-metyl-akrylová kyselina 2’-(piperid í n-1 -karbonyl)-bifenyl-2-karboxylová kyselina 3-benzoylamino-3-(4-chlór-fenyl)-propiónová kyselina 2-metylbenzylfosfónová kyselina mukobromičná kyselina 2,3,6-trimetoxybenzoová kyselina 2-metylheptánová kyselina 3-metyl-1 -cyklohexánkarboxylová kyselina fenyl-(2,4,6-trimetylfenyl)-octová kyselina 2-tiofénkarboxylová kyselina 3-(n-(4-etoxyfenyl)karbamoyl)bicyklo(2.2.1)hept-5-én-2-karboxylová kyselina 2-metyl-4-fenyl-maslová kyselina 2-(3-metoxy-fenyl)-jantárová kyselina (s)-n-(1-(1-naftyl)etyl)sukcínamová kyselina 2,-metoxy-5,-metyl-3,4I5,6-tetrachlórftalanilová kyselina 5-ŕerc-butylsulfanyl-tiofén-2-karboxylová kyselina 4-(oktadekánamido)benzoová kyselina d(-)-2-amino-7-fosfonoheptánová kyselina 4-metyl-1 -cyklohexánkarboxylová kyselina 3-(2,4-dichlór-fenyl)-2-metyl-akrylová boc-d-norvalín kyselina 4-[5-(2,4-dichlórfenyl)-2-furyl]tiazol-2-octová kyselina 3-hydroxy-3-metylglutárová kyselina 3-hydroxy-4-metoxyfenyloctová kyselina (s)-(-)-2-(6-metoxy-2-naftyl)propiónová kyselina 6-brómkumarín-3-karboxylová-153 1,18-octadecanedioic acid 3-amino-5-bromo-benzoic acid 5-chloro-tricyclo (2.2.1.0 (2,6)) heptane-3-carboxylic acid 2-hydroxydocosanoic acid 4-methoxyphenylacetic acid palmito-oleic acid 3-Benzo [1,1'-dioxol-S-yl-4-methyl-acrylic acid 2 '- (piperidin-1-carbonyl) -biphenyl-2-carboxylic acid 3-benzoylamino-3- (4-chloro-phenyl) -propionic acid 2-methylbenzylphosphonic acid mucobromic acid 2,3,6-trimethoxybenzoic acid 2-methylheptanoic acid 3-methyl-1-cyclohexanecarboxylic acid phenyl- (2,4,6-trimethylphenyl) -acetic acid 2-thiophenecarboxylic acid 3- ( n- (4-ethoxyphenyl) carbamoyl) bicyclo (2.2.1) hept-5-ene-2-carboxylic acid 2-methyl-4-phenylbutyric acid 2- (3-methoxyphenyl) succinic acid (s) N- (1- (1-naphthyl) ethyl) succinamic acid 2'-methoxy-5-methyl-3,4 5,6, tetrachlórftalanilová acid 5-tert-butylsulfanyl-thiophene-2-carboxylic acid 4- ( octadecanamido) benzoic acid d (-) - 2-Amino-7-phosphonoheptanoic acid 4-methyl-1-cyclohexanecarboxylic acid 3- (2,4-dichlorophenyl) -2-methyl-acrylic boc-d-norvaline 4- [5- (2,4-dichlorophenyl) -2-furyl] thiazole-2-acetic acid 3-hydroxy-3-methylglutaric acid 3-hydroxy-4-methoxyphenylacetic acid (s) - (-) - 2- (6-methoxy-2-naphthyl) propionic acid 6 -brómkumarín-3-carboxylic acid

-154--154-

• ·· • · • ··· • ·· • · • ··· • · • · • · • · • · • · ···· • • ···· • • ·· · • · ·· • e · ·· · • · ·· • e · ·· ·· ·· ·· ·· · · • · • · • e ·· • e ··

kyselina 3-(2-butylsulfanyl-benzotiazol-6-ylkarbamoyl)-akrylová kyselina 2-naftylamín-1,5,7-trisulfónová kyselina s-3-chlórmandlová kyselina orselová kyselina 2-(2-oxo-2-(4-(3-trifluórmetyl-fenyl)-piperazín-1-yl)-etyl)-malónová kyselina 1,1-cykloheptándioctová kyselina 3-etoxybenzoová kyselina 2-metyl-1 -cyklohexánkarboxylová kyselina 5-metoxy-2-metyl-izoftalámová kyselina n-(p-toluénsulfonyl)antranilová kyselina 4-nitro-naftalén-1 -karboxylová kyselina 2-norbornánoctová benzyloxykarbonyl-4-norval i n kyselina 3-fenylcinolín-4-karboxylová kyselina 3-fluór-4-(trifluórmetyl)fenyloctová kyselina 4-(3-karboxypropiónamido)-benzoová kyselina 2-(karbamoylmetyltio)benzoová kyselina 2,4-dimetyl-5-oxohexánová kyselina n-(2,5-dichlórfenyl)-1,2,3,6-tetrahydroftalámová kyselina d/-cyklohexylmandlová kyselina n-cyklohexylftatámová kyselina 4-fosfonomaslová kyselina 5-fluór-2-metoxybenzoová kyselina 1,3-acetóndikarboxylová kyselina 4-(trifluórmetyl)hydroškoricová kyselina (2-tienyl)maslová kyselina s-4-metyltiomandlová kyselina 3-hydroxy-2-nitrobenzoová kyselina 3-hydroxyškoricová kyselina ferulová kyselina 3-bróm-4-oxo-4-tiofén-2-yl-maslová kyselina 2,4,5-trimetylškoricová3- (2-Butylsulphanyl-benzothiazol-6-ylcarbamoyl) -acrylic acid 3-Trifluoromethyl-phenyl) -piperazin-1-yl) -ethyl) -malonic acid 1,1-cycloheptanedioic acid 3-ethoxybenzoic acid 2-methyl-1-cyclohexanecarboxylic acid 5-methoxy-2-methyl-isophthalic acid n- ( p-toluenesulfonyl) anthranilic acid 4-nitro-naphthalene-1-carboxylic acid 2-norboranacetic acid benzyloxycarbonyl-4-norvaline 3-phenylcinoline-4-carboxylic acid 3-fluoro-4- (trifluoromethyl) phenylacetic acid 4- (3- carboxypropionamido) benzoic acid 2- (carbamoylmethylthio) benzoic acid 2,4-dimethyl-5-oxohexanoic acid n- (2,5-dichlorophenyl) -1,2,3,6-tetrahydrophthalic acid d -cyclohexylmandelic acid n-cyclohexylphthamic acid 5-fluoro-2-methoxybenzoic acid 1,3-acetone dicarboxylic acid 4- (trifluoromethyl) hydro (2-thienyl) butyric acid s-4-methylthiomandelic acid 3-hydroxy-2-nitrobenzoic acid 3-hydroxycinnamic acid ferulic acid 3-bromo-4-oxo-4-thiophen-2-yl-butyric acid 2,4 , 5-trimetylškoricová

-155--155-

• ·· • · • ··· • ·· • · • ··· ·· • · • · · · • · • · ···· • • ···· • • ·· · • · ·· • · · ·· · • · ·· • · · • · · · • · · · ·· · · ·· · · ·· ·· ·· ··

kyselina 4-metyl-1,2,3-tiadiazol-5-karboxylová kyselina 2-butoxy-5-ferc-oktylbenzénsulfónová kyselina tnp-gama-aminomaslová kyselina 1 -(4-metoxyfenyl)-2-oxopyrolidín-4-karboxylová kyselina 5-chlór-2-(metyltio)pyrimidín-4-karboxylová kyselina /?-(trifluóracetyl)-d/-asparágová kyselina 2'-karbamoylglutáranilová kyselina 2,6-dimetyl-4-oxo-pyran-3-karboxylová kyselina n-etyl-5-sulfoantranilová kyselina c/s-4'-etylhexahydroftalanilová kyselina (2r,4r)-(+)-azetidín-2,4-dikarboxylová kyselina 2-etyl-2-metylbutánová kyselina 4-aminosulfonyl-1-hydroxy-2-naftoová kyselina 3-(3,4-dichlórfenyl)propiónová kyselina 2-(3-chlór-1,4-dioxo-1,4-dihydro-naftalén-2-ylamino)-4-metyl-pentánová kyselina 2,4-dihydroxy-3-metylbenzoová kyselina 2-bróm-4,6-dimetyl-3-hydroxybenzoová kyselina 3,5,7-trimetyl-1 -adamantánoctová kyselina alfa-hydroxybenzylfosfínová kyselina ((2-hydroxy-5-nitro-benzylidén)-amino)-fenyl-octová kyselina 1-valyl-1-glutámová kyselina [2,3-dichlór-4-(2-metylénbutyryl)fenoxy]octová kyselina 9-fluorenón-2-karboxylová kyselina s-4-metoxymandlová kyselina 5-metylsalicylová kyselina 4-acetoxyfenoxyoctová kyselina 2-(o-chlórfenoxy)-2-metyl-propiónová kyselina 4-hydroxytiobenzoová kyselina etánsulfónová kyselina 2-[4-chlór[(4-chlórfenyl)sulfonyl]anilíno]octová kyselina d/-benzyljantárová kyselina (r)-(+)-gama-butyrolaktón-gama-3-propiónová4-methyl-1,2,3-thiadiazole-5-carboxylic acid 2-butoxy-5-tert-octylbenzenesulfonic acid 1- (4-methoxyphenyl) -2-oxopyrrolidine-4-carboxylic acid 5 - Chloro-2- (methylthio) pyrimidine-4-carboxylic acid N- (trifluoroacetyl) - d] -aspartic acid 2'-Carbamoylglutaranilic acid 2,6-dimethyl-4-oxo-pyran-3-carboxylic acid n-ethyl -5-sulfoantranilic acid cis-4'-ethylhexahydrophthalanilic acid (2r, 4r) - (+) - azetidine-2,4-dicarboxylic acid 2-ethyl-2-methylbutanoic acid 4-aminosulfonyl-1-hydroxy-2- 3- (3,4-Dichloro-phenyl) -propionic acid 2- (3-chloro-1,4-dioxo-1,4-dihydro-naphthalen-2-ylamino) -4-methyl-pentanoic acid 2,4-dihydroxy 3-methylbenzoic acid 2-bromo-4,6-dimethyl-3-hydroxybenzoic acid 3,5,7-trimethyl-1-adamantanacetic acid alpha-hydroxybenzylphosphinic acid ((2-hydroxy-5-nitro-benzylidene) -amino) -phenyl-acetic acid 1-valyl-1-glutamic acid [2,3-dichloro- 4- (2-methylenebutyryl) phenoxy] acetic acid 9-fluorenone-2-carboxylic acid s-4-methoxymandelic acid 5-methylsalicylic acid 4-acetoxyphenoxyacetic acid 2- (o-chlorophenoxy) -2-methylpropionic acid 4-hydroxythiobenzoic acid ethanesulfonic acid 2- [4-chloro [(4-chlorophenyl) sulfonyl] anilino] acetic acid d-benzylsuccinic acid (r) - (+) - gamma-butyrolactone-gamma-3-propionic acid

-156 --156 -

• ·· • ·· ·· · · ···· ···· ·· · ·· · • · • · • · • · • · · · • · · · • ··· • ··· e · e · • · · • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 5-(4-metoxy-benzénsulfonyl)-tiofén-2-karboxylová kyselina 2-kyano-5-fenyl-2,4-pentadiénová kyselina (-)-4'-fluórtartranilová kyselina 3,4-dichlór-2-furoová kyselina 4-(2,4-dipentyl-fenoxy)-maslová kyselina 4,5.5-trifluór-2,4-pentadiénová kyselina 2’-metoxy-3,4,4’,5,6-pentachlórftalanilová kyselina eruková kyselina 3-jódftalová kyselina 4'-(2-benzoylacetamido)sukcínanilová kyselina (4-metoxy-benzoylamino)-octová kyselina 4-fenylazobenzoová kyselina 3-(2-metyl-benzotiazot-6-ylkarbamoyl)-akrylová kyselina 4-oxo-4h,9h-1-tia-4a,10-diaza-indeno(1,2-a)indén-2-karboxylová kyselina n-(2-fenyletyl)-3,4,5,6-tetrachlórŤtalámová kyselina 4-metyl-3-sulfobenzoová kyselina 5-hydroxypentadekánová kyselina 4-hydroxy-3-metoxyfenylpyrohroznová kyselina 2'-fluórmaleanilová kyselina 2-karbamoyl-2-propylvalérová kyselina metylén-bis(tiooctová) kyselina 4-(4-hydroxymetyl-3-metoxyfenoxy)-maslová kyselina 2-fluór-5-(trifluórmetyl)škoricová kyselina 5-sulfónamid kyseliny 2-chlórbenzoová kyselina 1,6-diaminohexán-/?,/?,n’,n’-teraoctová kyselina 4-(trifenylsilyl)benzoová kyselina 5-chlór-2-metylimidazo[1,2-a]pyridín-3-karboxylová kyselina d/-4-hydroxy-3-metoxymandlová kyselina 2-naftylsulfínová kyselina 1 .ľ-binaftyl-e.e'-dikarboxylová kyselina ŕrans-3-chlórakrylová kyselina 3-(4-chlórbenzoyl)-2-(2,4-dichlórfenyl)propiónová ·· ·· ···· ·· • · · · · · · ··· 9 9 9 9 95- (4-Methoxy-benzenesulfonyl) -thiophene-2-carboxylic acid 2-cyano-5-phenyl-2,4-pentadienoic acid (-) - 4'-Fluoro-tartranilic acid 3,4-dichloro-2-furoic acid 4- (2,4-dipentyl-phenoxy) -butyric acid 4,5,5-trifluoro-2,4-pentadienoic acid 2'-methoxy-3,4,4 ', 5,6-pentachlorophthalanilic acid erucic acid 3-iodophthalic acid 4 '- (2-benzoylacetamido) succinilic acid (4-methoxy-benzoylamino) -acetic acid 4-phenylazobenzoic acid 3- (2-methyl-benzothiazol-6-ylcarbamoyl) -acrylic acid 4-oxo-4h, 9h-1- thia-4a, 10-diaza-indeno (1,2-a) indene-2-carboxylic acid n- (2-phenylethyl) -3,4,5,6-tetrachloro-phthalic acid 4-methyl-3-sulfobenzoic acid 5- hydroxypentadecanoic acid 4-hydroxy-3-methoxyphenylpyruvic acid 2'-fluoromaleanilic acid 2-carbamoyl-2-propylvaleric acid methylene-bis (thioacetic) 4- (4-hydroxymethyl-3-methoxyphenoxy) butyric acid 2-fluoro-5- (trifluoromethyl) cinnamic acid 5-sulf 2-chlorobenzoic acid amide 1,6-diaminohexane-p, p, n ', n'-teraacetic acid 4- (triphenylsilyl) benzoic acid 5-chloro-2-methylimidazo [1,2-a] pyridin-3 - 4-hydroxy-3-methoxy-butyric acid 2-naphthylsulphonic acid 1,1'-binaphthyl-e-e'-dicarboxylic acid trans-3-chloroacrylic acid 3- (4-chlorobenzoyl) -2- (2, 4-chlorobenzoyl) 4-Dichlorophenyl) propionic acid 9 9 9 9 9

-157• ·· ·· ·· ·· · kyselina 3-benzo(1,3)dioxol-5-yl-2-etyl-akrylová kyselina indol-7-karboxylová kyselina 11-(4-(metoxykarbonyl)fenoxy)undekánová kyselina 4-(2,5-dimetyl-fenyl)-2-metyl-maslová kyselina 3-(4,5I6,6a-tetrahydro-fluorantén-3-yl)-propiónová kyselina n-(4,6-dimetylpyrimidín-2-yl)-n-metyl-3-aminobenzoová kyselina n-(3,4-dikyano-fenyl)-5-nitro-ftalámová kyselina indazolon-4-karboxylová kyselina (r)-2-chlór-3-metylmaslová kyselina 2-metyl-3-naftalén-1 -yl-akrylová kyselina tionikotínová kyselina 2-hydroxyoktánová kyselina 6-(4-chlórfenyl)-2-hydroxy-315-pyridíndikarboxylová kyselina 2-(4-metyl-1 -cyklohexylidén)octová kyselina 2-hydroxy-2-(2-aminotiazol)-4-octová kyselina (2-chlór-5-metyl-fenyl)-fosfónová kyselina 4-nitro-alfa-(orto-tolyl)škoricová kyselina alfa-propyl-1 -cyklopentén-1 -octová kyselina d/-2-amino-6-fosfonohexánová kyselina 4-(3-hydroxyfenoxy)benzoová kyselina (+/-)-2-acetoxypropiónová kyselina 4-(3-metylureido)benzoová kyselina 5-chlór-2-hydroxypyridín-3-karboxylová kyselina 2,3,4,5-furántetrakarboxylová kyselina 2-bróm-3-ftalimidopropiónová kyselina 3-chlór-4-metoxybenzoová kyselina 2,4,6-trifluórbenzoová kyselina 5-(acetamido)-2-nitrobenzoová kyselina 5-(4-nitrofenyl)-2-furoová kyselina 2-chlór-2-(3,4-dihydroftalazin-4-ón-1 -yljoctová kyselina 3-(4-jódfenyl)propiónová kyselina 4-fenyltetrahydropyrán-4-karboxylová • ·· ·· ···· ·· ··· · · ···· • ··· · · · · ·-157 3-Benzo (1,3) dioxol-5-yl-2-ethyl-acrylic acid Indole-7-carboxylic acid 11- (4- (methoxycarbonyl) phenoxy) undecanoic acid 4- (2,5-Dimethyl-phenyl) -2-methyl-butyric acid 3- (4,5 L 6,6a-tetrahydro-fluoroanten-3-yl) -propionic acid n- (4,6-dimethyl-pyrimidine- 2-yl) n-methyl-3-aminobenzoic acid n- (3,4-dicyano-phenyl) -5-nitro-phthalic acid indazolone-4-carboxylic acid (r) -2-chloro-3-methylbutyric acid 2 methyl-3-naphthalen-1-yl-acrylic acid tionikotínová acid, 2-hydroxyoctanoic acid 6- (4-chlorophenyl) -2-hydroxy-3-pyridine-5 1 2- (4-methyl-1-cyclohexylidene) -acetic acid 2-hydroxy-2- (2-aminothiazole) -4-acetic acid (2-chloro-5-methylphenyl) -phosphonic acid 4-nitro-alpha- (ortho-tolyl) cinnamic acid alpha-propyl-1-cyclopentene -1-acetic acid d -2-amino-6-phosphonohexanoic acid 4- (3-hydroxyphenoxy) benzoic acid (+/-) - 2-acetoxypropionic acid 4- (3-methylurei) do) benzoic acid 5-chloro-2-hydroxypyridine-3-carboxylic acid 2,3,4,5-furanetetracarboxylic acid 2-bromo-3-phthalimidopropionic acid 3-chloro-4-methoxybenzoic acid 2,4,6-trifluorobenzoic acid 5- (Acetamido) -2-nitrobenzoic acid 5- (4-nitrophenyl) -2-furoic acid 2-chloro-2- (3,4-dihydrophthalazin-4-one-1-yl) acetic acid 3- (4-iodophenyl) propionic acid 4-phenyl-tetrahydropyran-4-carboxylic acid

-158kyselina 3-fenyl-3-(toluén-4-sulfonylamino)-propiónová kyselina 5,7-dioxooktánová kyselina (4-aminobenzyl)fosfónová kyselina 4-(4-chlór-o-tolyloxy)maslová kyselina n-boc-d/-1 -aminoindán-1 -karboxylová kyselina n-ftaloyl-d/-alfa-aminomaslová kyselina 4-jód-3-metylbenzoová kyselina 2-(n-(1 -naftyl)karbamoyl)cyklohexánkarboxylová kyselina bis(boc-3,5-diaminobenzoová) kyselina (d)-n-benzylglutámová kyselina 4-(4-chlór-m-tolyloxy)-maslová kyselina 6-benzamidohexánová kyselina 11-bróm-undekánová kyselina 2-(2-karboxy-cyklohexa-2,5-diénylamino)-4-nitro-benzoová kyselina 1,4-dioxo-2,5-metano-pentalén-2,3a,5,6a-tetrakarboxylová kyselina 3-(tetradecyloxy)benzoová kyselina trifluóroctová kyselina cyklohexánmaslová kyselina 5,5-dimetyl-2,4-tiazolidíndikarboxylová kyselina 2,2,3,3-tetrametylcyklopropánkarboxylová n-karbamyl-1-leucín kyselina 2-chlór-4-metytsulfonylbenzoová kyselina 2-( 1,8-naftyridín-2-yl)benzoová kyselina 5-[[(4-metylfenyl)sulfonyl]amino]-5-oxopentánová kyselina ŕrans-cyklobután-1,2-dikarboxylová kyselina exo-2-bróm-5-oxo-bicyklo[2.2.1)heptán-syn-7-karboxylová kyselina diamyloctová kyselina (3-fosfono-adamantán-1 -yl)-fosfónová kyselina 4-(3-[2,2,2-trichlór-1-(2,2-d/-me-propionylamino)-et]-tioureido)-benzoová kyselina 1 h, 1 h,2h,2h-perfluóroktánsulfónová kyselina c/s-2,4-piperidín-dikarboxylová kyselina 4-(3-(2,4-xylyl)ureido)benzoová-158 3-phenyl-3- (toluene-4-sulfonylamino) -propionic acid 5,7-dioxooctanoic acid (4-aminobenzyl) phosphonic acid 4- (4-chloro-o-tolyloxy) butyric acid n-boc-d] 1-aminoindan-1-carboxylic acid n-phthaloyl-N-alpha-aminobutyric acid 4-iodo-3-methylbenzoic acid 2- (n- (1-naphthyl) carbamoyl) cyclohexanecarboxylic acid bis (boc-3,5- (d) -n-benzylglutamic acid 4- (4-chloro-m-tolyloxy) butyric acid 6-benzamidohexanoic acid 11-bromo-undecanoic acid 2- (2-carboxy-cyclohexa-2,5-dienylamino) -4-nitro-benzoic acid 1,4-dioxo-2,5-methano-pentalen-2,3a, 5,6a-tetracarboxylic acid 3- (tetradecyloxy) benzoic acid trifluoroacetic acid cyclohexanebutyric acid 5,5-dimethyl-2, 4-thiazolidinedicarboxylic acid 2,2,3,3-tetramethylcyclopropanecarboxylic acid n-carbamyl-1-leucine 2-chloro-4-methylsulfonylbenzoic acid 2- (1,8-naphthyridin-2-yl) benzoic acid 5 - [[(4 methylphenyl) sulfonyl] amino] -5-oxopentanoic acid trans-cyclobutane-1,2-dicarboxylic acid exo-2-bromo-5-oxo-bicyclo [2.2.1] heptane-syn-7-carboxylic acid diamylacetic acid (3-phosphono-adamantane- 1-yl) -phosphonic acid 4- (3- [2,2,2-trichloro-1- (2,2-d-metropionylamino) -ethyl] -thioureido) -benzoic acid 1 h, 1 h, 2h, 2h-Perfluorooctane sulfonic acid cis-2,4-piperidine-dicarboxylic acid 4- (3- (2,4-xylyl) ureido) benzoic acid

-159--159-

• ·· • · • ··· • · · • ·· • · • ··· • · · ·· ···· • · · • · · • · · · · ·· ···· • · · • · · • · · · · ·· • c • · • · · · • c • · • · ·· · · ·· Φ· ·· Φ · ·· ·· ·· ·· ·· · · ·· · ·

kyselina 3',5'-dichlórftalanilová kyselina 2,4-dihydroxypyrimidín-5-karboxylová kyselina cyklobután-1,1,3,3-tetrakarboxylová kyselina 4-metyl-2-(orto-tolyl)-valérová kyselina (s)-(-)-alfa-metoxyfenyloctová kyselina (-)-4'-metyltartranilová kyselina 5-(2-hydroxy-3-metoxy-fenyl)-pentánová kyselina c/s,c/s-mukonová kyselina 2-(2,7-dichlór-6-hydroxy-3-oxo-2,3-dihydro-1h-xantén-9-yl)-benzoová kyselina (e)-2-oktadecénová kyselina d/-2-amino-4-metyl-5-fosfono-3-penténová kyselina 5-(2,5-dioxo-pyrolidín-1 -yl)-4-oxo-pentánová kyselina 2,4-di(decyloxy)benzoová kyselina 3,5-dijód-4-hydroxybenzoová kyselina 3-(4-chlórbenzoyl)-2-(3-chlórfenyl)propiónová kyselina 2-(2-benzotiazol-2-yl-vinyl)-benzoová kyselina 11-(9-antroyloxy)undekánová kyselina 1,3-adamantándikarboxylová kyselina myristolejová kyselina 3-(2,2-difluór-1,3-benzodioxol-5-yl)-(2e)-propénová kyselina neooktánová kyselina 4-(2-benzoylamino-3-fenyl-akryloylamino)-maslová kyselina 2-[(4I6-dimetoxypyrimidín-2-yl)tio]benzoová beta-benzyl-ester kyseliny n-boc-d-asparágovej kyselina n-(4-metoxyfenyl)-1,2,5,6-tetrahydroftalámová kyselina 1 -(2-chlór-4-fluórfenyl)cyklopentánkarboxylová kyselina 2-metoxy-4-metylbenzoová kyselina 1 -adamantánkarboxylová kyselina 3-(2-nitrofenoxy)-2-tiofénkarboxylová kyselina 3-chlór-2,6-dimetoxybenzoová kyselina 2,3-dimetoxy-5-jódbenzoová kyselina 2,4-dichlór-5-fluórbenzoová • ·· ·· ···· 88 • 8 · 88 8 888 • 888 8 · 8 883 ', 5'-dichlorophthalanic acid 2,4-dihydroxypyrimidine-5-carboxylic acid cyclobutane-1,1,3,3-tetracarboxylic acid 4-methyl-2- (ortho-tolyl) -valeric acid (s) - ( -) - alpha-Methoxyphenylacetic acid (-) - 4'-methyltartranilic acid 5- (2-hydroxy-3-methoxyphenyl) -pentanoic acid cis / cis-muconic acid 2- (2,7-dichloro) -6-hydroxy-3-oxo-2,3-dihydro-1H-xanthen-9-yl) -benzoic acid (e) -2-octadecenoic acid d -2-amino-4-methyl-5-phosphono-3 -pentenoic acid 5- (2,5-dioxo-pyrrolidin-1-yl) -4-oxo-pentanoic acid 2,4-di (decyloxy) benzoic acid 3,5-diiodo-4-hydroxybenzoic acid 3- (4- chlorobenzoyl) -2- (3-chlorophenyl) propionic acid 2- (2-benzothiazol-2-yl-vinyl) -benzoic acid 11- (9-antroyloxy) undecanoic acid 1,3-adamantanedicarboxylic acid myristoleic acid 3- (2, 2-Difluoro-1,3-benzodioxol-5-yl) - (2e) -propenoic acid neooctanoic acid 4- (2-benzoylamino-3-phenyl-acryloylamino) -butyric acid 2 - [(4 I 6-dimetho) xypyrimidin-2-yl) thio] benzoic n-boc-d-aspartic acid beta-benzyl ester n- (4-methoxyphenyl) -1,2,5,6-tetrahydrophthalic acid 1- (2-chloro-4- fluorophenyl) cyclopentanecarboxylic acid 2-methoxy-4-methylbenzoic acid 1-adamantanecarboxylic acid 3- (2-nitrophenoxy) -2-thiophenecarboxylic acid 3-chloro-2,6-dimethoxybenzoic acid 2,3-dimethoxy-5-iodobenzoic acid 2, 4-Dichloro-5-fluorobenzoic acid 88,88,888,888 888 8,888

-160kyselina n-(5-chlórfenyl)-1,2,5,6-tetrahydroftalámová kyselina 2,3-difenyl-maslová kyselina 3,5-dimetylbenzoová kyselina d/-alfa-hydroxyizokaprónová kyselina 5-(4-chlórfenyl)-2-furoová kyselina (2-guanidínoetytmerkapto)jantárová kyselina 7-nitro-4-fluorénkarboxylová kyselina karbobenzyloxy-d/-glutámová kyselina 8-bróm-1-naftoová kyselina 12-(n-(7-nitrobenz-2-oxa-1,3-diazol-4-yl)amino)dodekánová kyselina n-hexadecylmalónová kyselina 2,5-dichlórtereftalová kyselina hexakozánová kyselina heptaglukónová kyselina 2,3,5,6-tetrachlórbenzoová kyselina beta-4-metoxybenzylmerkapto-beta,beta-cyklopentametylénpropiónová-160 n- (5-chlorophenyl) -1,2,5,6-tetrahydrophthalic acid 2,3-diphenylbutyric acid 3,5-dimethylbenzoic acid N-alpha-hydroxyisocaproic acid 5- (4-chlorophenyl) -2 (2-guanidinoethylmercapto) succinic acid 7-nitro-4-fluorenecarboxylic acid carbobenzyloxy-d-glutamic acid 8-bromo-1-naphthoic acid 12- (n- (7-nitrobenz-2-oxa-1,3) -diazol-4-yl) amino) dodecanoic acid n-hexadecylmalonic acid 2,5-dichloro-terephthalic acid hexacosanoic acid heptagluconic acid 2,3,5,6-tetrachlorobenzoic acid beta-4-methoxybenzylmercapto-beta, beta-cyclopentamethylenepropionic acid

N-(fosfonometyl)glycín kyselina c/s-azetidín-2,4-dikarboxylová kyselina 6-merkaptonikotinová kyselina 2-[2-[3-chlór-5-(trifluórmetyl)-2-pyridyl]hydrazóno]octová kyselina 2-(2-metoxyetoxy)octová n-cbz-d-norleucín kyselina 2-chlórbenzoová kyselina n-(2,6-dinitro-4-trifluórmetyl)izonipekotínová kyselina 2-hydroxyamino-maslová kyselina brómchlóroctová kyselina 1 -alfa-glutamyl-terc-gtulámová kyselina 8-brómoktánová kyselina 3-fluórfenyloctová kyselina fmoc-1 -indolín-2-karboxylová kyselina 2,3-dibróm-4,-etoxysukcínanilová kyselina 3-(4-(2,2-dimetylpropionyl)benzoyl)propiónová • ·· ·· · ·· · · · ·« · 9 · ···· • ··· 9 · · · ·N- (phosphonomethyl) glycine cis-azetidine-2,4-dicarboxylic acid 6-mercaptonicotinic acid 2- [2- [3-chloro-5- (trifluoromethyl) -2-pyridyl] hydrazono] acetic acid 2- ( 2-methoxyethoxy) acetic acid n-cbz-d-norleucine 2-chlorobenzoic acid n- (2,6-dinitro-4-trifluoromethyl) isonipecotinic acid 2-hydroxyamino-butyric acid bromochloroacetic acid 8-bromooctanoic acid 3-fluorophenylacetic acid fmoc-1-indoline-2-carboxylic acid 2,3-dibromo-4 , -ethoxy-succinic acid 3- (4- (2,2-dimethylpropionyl) benzoyl) propionic acid · ·· ·· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ·

-161 kyselina 2-nitrotiofén-4-karboxylová kyselina 2-fenyl-2-adamantán-octová kyselina 7-fenyl-618-dioxa-spiro(3,5)nonán-2,2-dikarboxylová kyselina 5,5'-tiodisalicylová kyselina (s)-(-)-2-chlórpropiónová kyselina 7-nitro-9-oxo-4-fluorénkarboxylová kyselina z-(+)-alfa-amino-4-fenylmaslová kyselina alfa-kyano-3,4-dimetoxyškoricová kyselina salicylsalicylová kyselina 4-brómmandlová kyselina 2-(3-fenylureido)benzoová kyselina 4-(izopropylsulfonyl)tiofén-2-karboxylová kyselina 3-metyl-2-fenylacetylamino-maslová kyselina 5-antracén-2-yl-pentánová kyselina 3-[1,2-dihydro-2-oxo-5-(trifluórmetyl)-pyrid-1 -yljpropiônová kyselina 3'-nitrosukcínanilová kyselina fmoc-d/-beta-aminomaslová kyselina d/-3,4-dihydroxymandlová kyselina (2-benzylsulfanyl-6-metyl-pyrimidín-4-yloxy)-octová kyselina 5-metyl-2-(trifluórmetyl)furán-3-karboxylová kyselina 3-metyl-4-nitrobenzoová kyselina 1-propánsulfónová kyselina 5-indán-akrylová kyselina 3-acetamido-4-hexadecyloxybenzoová kyselina sebaková kyselina (10-karboxymetyl-antracén-9-yl)-octová kyselina 3-(4,5-dimetoxy-2-nitro-fenyl)-akrylová kyselina pentadekánová kyselina 4-chlór-3-metylbenzoová kyselina n-(3-chlórfenyl)malonámová kyselina 2-fosfonomaslová kyselina 3-(3-trifliiórmetylbenzyloxy)tiofén-2-karboxylová-161 acid 2-nitro-thiophene-4-carboxylic acid 2-phenyl-2-adamantane acetic acid, 7-phenyl-6-one 8-dioxa-spiro (3,5) nonane-2,2-dicarboxylic acid, 5,5 ' thiodisalicylic acid (s) - (-) - 2-chloropropionic acid 7-nitro-9-oxo-4-fluorenecarboxylic acid from - (+) - alpha-amino-4-phenylbutyric acid alpha-cyano-3,4-dimethoxycinnamic acid salicylsalicylic acid 4-bromo-butyric acid 2- (3-phenylureido) benzoic acid 4- (isopropylsulfonyl) thiophene-2-carboxylic acid 3-methyl-2-phenylacetylamino-butyric acid 5-anthracen-2-yl-pentanoic acid 3- [1 2-dihydro-2-oxo-5- (trifluoromethyl) -pyrid-1-yl] propionic acid 3'-nitrosuccinilic acid fmoc-d-beta-aminobutyric acid d] -3,4-dihydroxymandelic acid (2-benzylsulfanyl-6) -methyl-pyrimidin-4-yloxy) -acetic acid 5-methyl-2- (trifluoromethyl) furan-3-carboxylic acid 3-methyl-4-nitrobenzoic acid 1-propanesulfonic acid 5-indan-acrylic acid 3-acetamido-4 -hexadecyloxyb enzoic acid sebacic acid (10-carboxymethyl-anthracen-9-yl) -acetic acid 3- (4,5-dimethoxy-2-nitro-phenyl) -acrylic acid pentadecanoic acid 4-chloro-3-methylbenzoic acid n- (3 3-Trifluoromethylbenzyloxy) thiophene-2-carboxylic acid

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B · · B · B ···B · B · B ···

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-162kyselina 2-ketomaslová kyselina 4-chlórpikolínová kyselina 414I4-trifluór-3-fenylacetylamino-maslová kyselina 4-acetamido-3,5-dichlórbenzoová kyselina gama(2-pyridyl)-maslová kyselina 2-aminofenol-6-sulfónová kyselina )-oxo-1,8-oktándikarboxylová kyselina 1-naftoxymliečna kyselina (l)-n-benzylglutámová kyselina 4-metyl-2-fenyl-pentánová kyselina (5-hydroxy-5h-dibenzo(a,d)cykloheptén-5-yl)-octová kyselina 2-pyrid í n-3-yl-chinol í η-4-karboxy lová kyselina cŕ/-p-toluoyl-1-vínna kyselina 2-hydroxy-cyklohexánkarboxylová kyselina 4-nitroizoftalová kysel ina 3,3,3-tris(4-chlórfenyl )propiónová kyselina 6-[(4-amino-3-sulfofenyl)amino]-4-hydroxy-2-naftalénsulfónová kyselina (chlór-fosfono-metyl)-fosfónová kyselina (s)-(+)-2-fenylmaslová kyselina 1 -oxy-pyridín-4-sulfónová kyselina 4-chlór-2,5-dimetyltiofénoxyoctová kyselina beta-metyl-3-nitroškoricová kyselina d/-2-(4-hydroxyfenyl)-2-fenyloctová kyselina 4-metyltio-3-nitrobenzoová kyselina 1-izoleucyl-1-gtutámová kyselina 3-chlórbenzoová kyselina 6-bróm-3,4-metyléndioxyškoricová kyselina n-(4-bróm-2-chlórfenyl)maleámová kyselina 1 -karboxy-4-(trimetylsilyl)cyklohexánoctová kyselina 10,12-trikozadiínová kyselina (+/-)-2-hydroxytridekánová kyselina ľ-oxo^.S.e.ľ-tetrahydro-benzofurán-S-karboxylová-162 2-ketobutyric acid 4-chloropicolinic acid 4 1 4 1 4-Trifluoro-3-phenylacetylamino-butyric acid 4-acetamido-3,5-dichlorobenzoic acid Gamma (2-pyridyl) butyric acid 2-aminophenol-6-sulfonic acid (1) -n-benzylglutamic acid 4-methyl-2-phenyl-pentanoic acid (5-hydroxy-5h-dibenzo (a, d) cycloheptene-5-) - oxo-1,8-octanedicarboxylic acid yl) -acetic acid 2-pyridin-3-yl-quinoline-4-carboxylic acid cis-p-toluoyl-1-tartaric acid 2-hydroxy-cyclohexanecarboxylic acid 4-nitroisophthalic acid 3,3, 3-Tris (4-chlorophenyl) propionic acid 6 - [(4-amino-3-sulfophenyl) amino] -4-hydroxy-2-naphthalenesulfonic acid (chloro-phosphono-methyl) -phosphonic acid (s) - (+) -2-phenylbutyric acid 1-oxy-pyridine-4-sulfonic acid 4-chloro-2,5-dimethylthiophenoxyacetic acid beta-methyl-3-nitrocinnamic acid d -2- (4-hydroxyphenyl) -2-phenylacetic acid 4- methylthio-3-nitrobenzoic acid 1-isoleucyl-1-gtutamic acid 3-chlorobenzoic acid 6-bromo-3,4-methylenedioxycinnamic acid n- (4-bromo-2-chlorophenyl) maleic acid 1-carboxy-4- (trimethylsilyl) cyclohexaneacetic acid 10,12 (+/-) - 2-hydroxytridecanoic acid 1'-oxo-4'-S-tetrahydro-benzofuran-5-carboxylic acid

-163 --163 -

a ·· A · • ··· and ·· A · • ··· • · • · • · • · • · • · • ·· · ♦ • • ·· · ♦ • • · 9 9 9 99 9 9· • · 9 9 9 9 · ·· c· ·· c · ·· · · • · • · 99 9 9 99 9 9

kyselina 5-chlór-2-fenylimidazo[1,2-a]-pyrimidín-3-karboxylovä kyselina 2-(orto-tolyl)-maslová kyselina 4-(4-azidofenyl)maslová kyselina 2-(4-(3-oxo-3-fenyl-1 -propén-1 -yl)fenoxy)octová kyselina 9-oxo-6,7,8,9-tetrahydro-5h-benzocykloheptén-6-karboxylová kyselina (3-brómpropyl)fosfónová kyselina (+/-)-9-hydroxy-(5z,7e,11z,14z)-eikozatetraénová kyselina o-krotylfenoxyoctová kyselina 5-fenylacetylamino-benzoová kyselina 2-metoxy-4-nitroškoricová kyselina 1-indánylmalónová kyselina 2,3,5-trifluórbenzoová kyselina 5-bróm-orotová kyselina 3-metoxy-2-nitrobenzoová kyselina 2,3-dimetoxy-9-oxo-6,7,8I9-tetrahydro-5h-benzocykloheptén-5-karboxylová kyselina 5-(4-chlórfenyl)-2-metylfurán-3-karboxylová kyselina dibenzoyl-d-vínna kyselina 3-(difluórmetoxy)benzoová kyselina 3-ureidopropiónová kyselina omega-3-arachidónová kyselina 1,3-propándisulfónová kyselina 3-(toluén-4-sulfonylamino)-propiónová kyselina 3-(4-metoxy-benzo(1,3)dioxol-5-yl)-akrylová kyselina 4-hydroxymetyl-3-metoxy-fenoxyoctová kyselina cyklopropán-1,2-dikarboxylová kyselina 4-(4-(4-(2-karboxy-etyl)-cyklohexylmetyl)-cyklohexyl)-maslová kyselina 17-bróm-heptadekánová kyselina 4-(3-(2,3-xylyl)ureido)benzoová fmoc-alfa-metylalanín kyselina d/-erytro-4-fluórglutámová kyselina fra/7s-2-penténová kyselina 3-(2-benzoxazolín-2-ón-3-yl)propiónová • ·· ·· ···· «· • · ·» · · · ··· • ··· · · · · ·5-chloro-2-phenylimidazo [1,2-a] pyrimidine-3-carboxylic acid 2- (ortho-tolyl) butyric acid 4- (4-azidophenyl) butyric acid 2- (4- (3-oxo) 3-Phenyl-1-propen-1-yl) phenoxy) acetic acid 9-oxo-6,7,8,9-tetrahydro-5h-benzocycloheptene-6-carboxylic acid (3-bromopropyl) phosphonic acid (+/- ) -9-hydroxy- (5z, 7e, 11z, 14z) -eicosatetraenoic acid o-crotylphenoxyacetic acid 5-phenylacetylamino-benzoic acid 2-methoxy-4-nitrocinnamic acid 1-indanylmalonic acid 2,3,5-trifluorobenzoic acid 5- bromo-orotic acid 3-methoxy-2-nitrobenzoic acid, 2,3-dimethoxy-9-oxo-6,7,8-I, 9-tetrahydro-5H-benzocyclohepten-5-carboxylic acid 5- (4-chlorophenyl) -2- methylfuran-3-carboxylic acid dibenzoyl-d-tartaric acid 3- (difluoromethoxy) benzoic acid 3-ureidopropionic acid omega-3-arachidonic acid 1,3-propanedisulfonic acid 3- (toluene-4-sulfonylamino) -propionic acid 3- ( 4-Methoxy-benzo (1,3) dioxol-5-yl) -acrylic acid 4-hydroxymethyl-3-methoxy-phenoxyacetic acid cyclopropane-1,2-dicarboxylic acid 4- (4- (4- (2-carboxy-ethyl) -cyclohexylmethyl) -cyclohexyl) -butyric acid 17-bromo-heptadecanoic acid 4 - (3- (2,3-xylyl) ureido) benzoic fmoc-alpha-methylalanine d -erythro-4-fluoroglutamic acid fra / 7s-2-pentenoic acid 3- (2-benzoxazolin-2-one-3- yl) propionic prop prop ión ión prop ión prop ión prop prop prop) ión prop prop prop) prop)

-164kyselina 3,4,5-trifluórškoricová kyselina benzén-1,3,5-trikarboxylová kyselina 2-(azokán-1 -karbotioylsulfanyl)-2-metyl-propiónová kyselina c/s-n-(dodecyl)hexahydroftalámová kyselina 3-kyanoetylbenzoová kyselina 4I5,5I5-tetrafluór-4-(trifluórmetyl)pentánová kyselina 5-(3-(trifluórmetyl)fenyl)-2-furoová kyselina 4-(2-(3-benzyloxy-4-metoxy-fenyl)-etylkarbamoyl)-maslová kyselina alfa-metyl-2-tiofén-octová kyselina 3-(n-(m-tolyl)karbamoyl)-5-norbornén-2-karboxylová kyselina n-alfa-(ŕerc-butyloxykarbonyl)-alfa-(metylester)-1-glutámová kyselina 2-metyl-3-furoová kyselina 2,4,5-trichlórfenoxyoctová kyselina cyklohexylfosfónová kyselina c/s-chrysantémum-rnonokarboxylová kyselina 12-metyltridekánová kyselina 4,10-dioxo-9-oxa-tricyklo(6.2.1.0(1,5))undekán-2-karboxylová kyselina 4-acetoxyškoricová kyselina 4-(tetradekánamido)benzoová kyselina (s)-(-)-fenyljantárová kyselina o-toluylová kyselina (-)-cŕ/-p-toluoyl-d-vínna kyselina (s)-(-)-2-brómmaslová kyselina 2,2-azoxydibenzoová kyselina n-formyl-1 -2-aminomaslová kyselina n-fmoc-2-amino-4-(dimetoxyfosfono)-butánová kyselina 3-amino-5-(trifluórmetyl)benzoová kyselina 4,4,-[(metándiyl)bis(iminokarbonyl)]bis-benzoová kyselina 3-(trifluórmetyl)hydroškoricová kyselina 12-tridecénová kyselina 12,12,12-trifluórdodekánová kyselina fosfonooctová • · ·· ···· ·· • · · · e · · · · • ··· « · · · ·-164 3,4,5-trifluorocinnamic acid benzene-1,3,5-tricarboxylic acid 2- (azocane-1-carbothioylsulfanyl) -2-methyl-propionic acid cis- (dodecyl) hexahydrophthalic acid 3-cyanoethylbenzoic acid 4 I 5.5 L 5-tetrafluoro-4- (trifluoromethyl) pentanoic acid 5- (3- (trifluoromethyl) phenyl) -2-furoic acid 4- (2- (3-benzyloxy-4-methoxy-phenyl) ethylcarbamoyl) butyric acid alpha-methyl-2-thiophene-acetic acid 3- (n- (m-tolyl) carbamoyl) -5-norbornene-2-carboxylic acid n-alpha- (tert-butyloxycarbonyl) -alpha- (methyl ester) - 1-glutamic acid 2-methyl-3-furoic acid 2,4,5-trichlorophenoxyacetic acid cyclohexylphosphonic acid cis-chrysanthemum-monocarboxylic acid 12-methyltridecanoic acid 4,10-dioxo-9-oxa-tricyclo (6.2.1.0 ( 1,5)) undecane-2-carboxylic acid 4-acetoxycinnamic acid 4- (tetradecanamido) benzoic acid (s) - (-) - phenylsuccinic acid o-toluic acid (-) - N-p-toluoyl-d-tartaric acid (s) - (-) - 2-bromoic acid 2,2-azoxydibenzoic acid n-formyl-1-2-aminobutyric acid n-fmoc-2-amino-4- (dimethoxyphosphono) butanoic acid 3-amino-5- (trifluoromethyl) benzoic acid 4,4 , - [(methanediyl) bis (iminocarbonyl)] bis-benzoic acid 3- (trifluoromethyl) hydrocinnamic acid 12-tridecenic acid 12,12,12-trifluorododecanoic acid phosphonoacetic acid · · ············· · · · ···

-165kyselina 2,5-bis(2,2,2-trifluóretoxy)benzoová kyselina metanilsulfonyl-salicylová kyselina 3-fluórškoricová kyselina 5-ketoglukónová kyselina 12(r)-hydroxyeikoza-5z,8z, 10e, 14z-tetraénová kyselina (+/-)-gáforkarboxylová kyselina 3-benzoylpropiónová kyselina 10,10,10-trifluórdekánová kyselina 1 -metyl-2-oxocyklohexánpropiónová kyselina gama-metylén-ď/-glutámová kyselina pth-cysteínová kyselina 7-nitro-9-oxo-2-fluorénkarboxylová kyselina 3-(n-(4-metoxyfenyl)karbamoyl)-5-norbornén-2-karboxylová kyselina alph-beta-dibróm-2-nitrohydroškoricová kyselina 4'-bróm-2'-metyl-1,2,3,6-tetrahydroftalanilová kyselina izoftalová kyselina n-propylfosfónová kyselina 14-metylhexadekánová kyselina 2-bróm-3-metylvalérová kyselina ŕrans-škoricová kyselina 2,4,6-trimetoxyškoricová kyselina 2-(3,5-dinitro-tiofén-2-ylamino)-propiónová kyselina 4-pyridínbutylová kyselina 5-(4-(4-karboxy-butyl)-fenyl)-pentánová kyselina n-(4-brómfenyl)malonámová kyselina 2,2’-dichlórdifenylglykolová kyselina 2,5-dimetyl-benzén-1,3-disulfínová kyselina 4,5-dibróm-2-hexénová kyselina 4-karboxyfenoxyoctová kyselina 3-(oktyloxy)-propiónová kyselina 3'-chlór-4'-fluórftalanilová kyselina 5-chlórvanilová-165 2,5-bis (2,2,2-trifluoroethoxy) benzoic acid methanilsulfonyl-salicylic acid 3-fluorocinnamic acid 5-ketogluconic acid 12 (r) -hydroxyeicose-5z, 8z, 10e, 14z-tetraenoic acid (+/-) -) - Camphoric acid 3-benzoylpropionic acid 10,10,10-trifluorodecanoic acid 1-Methyl-2-oxocyclohexanepropionic acid Gamma-methylene- N -glutamic acid p-Cysteic acid 7-nitro-9-oxo-2-fluorenecarboxylic acid 3- (n- (4-Methoxyphenyl) carbamoyl) -5-norbornene-2-carboxylic acid alph-beta-dibromo-2-nitrohydrocinnamic acid 4'-bromo-2'-methyl-1,2,3,6-tetrahydrophthalanilic acid isophthalic acid n-propylphosphonic acid 14-methylhexadecanoic acid 2-bromo-3-methylvaleric acid trans-cinnamic acid 2,4,6-trimethoxycinnamic acid 2- (3,5-dinitro-thiophen-2-ylamino) -propionic acid 4 5- (4- (4-Carboxy-butyl) -phenyl) -pentanoic acid- (4-bromophenyl) malonamic acid 2,2'-Dichloro-diphenylglycolic acid 2,5-dimethyl-benzene-1,3-disulphonic acid 4,5-dibromo-2-hexenoic acid 4-carboxyphenoxyacetic acid 3- (octyloxy) -propionic acid 3'-chloro-4 5-Chloroanilic acid

-166--166-

• · · • · · 99 99 9999 9999 ·· B ·· B 9 · 9 · 9 9 9 9 9 9 • · · · • · · · • ··· • ··· 9 · 9 · 9 9 • · · • · · 99 99 99 99 ·· · · • · • · ·· 99 ·· 99

kyselina 5,6-dehydroarachidónová kyselina 3-(3-metoxyfenyl)propiónová kyselina nonylfenoxyoctová kyselina (1 s,3s)-1 -amino-1 -karboxycyklopentán-3-octová kyselina 3-(2-fluór-4-nitrofenoxy)-2-tiofénkarboxylová kyselina alfa-brómdietyloctová kyselina 1-izoleucínová (kyselina 2-hydroxy-3-metylvalérová) kyselina 4-karboxy-1,1 -cyklohexándioctová kyselina sulfanilid-dikarboxylová kyselina 6-acetamidohexánová kyselina 3-chlórfenyloctová kyselina 2-(2-propinyl)malónová kyselina 3-hydroxy-2-trifluórmetylpropiónová kyselina n-tetradecylfosfónová kyselina ŕrans-styryloctová kyselina 3-(metyltio)benzoová kyselina 2-(3,5-dinitro-tiofén-2-ylamino)-3-fenyl-propiónová kyselina 4*-etyl-4-bifenylkarboxylová kyselina 2,2-bis(trifluórmetyl)propiónová kyselina 3-benzoyl-2-(2,3-dichlórfenyl)propiónová kyselina 2,4-dimetyltiazol-5-karboxylová kyselina 4-fenyl-1,2,3-tiadiazol-5-karboxylová kyselina n-alfa-z-1-alanyl-1-asparágová kyselina 3-(pivaloylamino)tiofén-2-karboxylová kyselina 11-(toluén-4-sulfonyl)-undekánová kyselina 4-hydroxyfenylpyrohroznová kyselina 5-chlór-6-hydroxy-2-metyl-pyrimidín-4-karboxylová kyselina 1,1-cyklobutándikarboxylová kyselina ŕerc-butyl-(1,2,2-trichlór-vinyl)-fosfínová kyselina 2',3'-dichlórftalanilová kyselina 3-metyléncyklopropán-ŕrans-1,2-dikarboxylová kyselina 1 -alfa-hydroxyizovalérová5,6-dehydroarachidonic acid 3- (3-methoxyphenyl) propionic acid nonylphenoxyacetic acid (1s, 3s) -1-amino-1-carboxycyclopentane-3-acetic acid 3- (2-fluoro-4-nitrophenoxy) -2 -thiophenecarboxylic acid alpha-bromo diethylacetic acid 1-isoleucinic acid (2-hydroxy-3-methylvaleric acid) 4-carboxy-1,1-cyclohexanediacetic acid sulfanilide-dicarboxylic acid 6-acetamidohexanoic acid 3-chlorophenylacetic acid 2- (2-propynyl) malonic acid 3-hydroxy-2-trifluoromethylpropionic acid n-tetradecylphosphonic acid trans-styrylacetic acid 3- (methylthio) benzoic acid 2- (3,5-dinitro-thiophen-2-ylamino) -3-phenylpropionic acid 4 * - ethyl 4-biphenylcarboxylic acid 2,2-bis (trifluoromethyl) propionic acid 3-benzoyl-2- (2,3-dichlorophenyl) propionic acid 2,4-dimethylthiazole-5-carboxylic acid 4-phenyl-1,2,3 -thiadiazole-5-carboxylic acid n-alpha-z-1-alanyl-1-aspartic acid 3- (pivaloylamino) thiophene n-2-carboxylic acid 11- (toluene-4-sulfonyl) -undecanoic acid 4-hydroxyphenylpyruvic acid 5-chloro-6-hydroxy-2-methyl-pyrimidine-4-carboxylic acid 1,1-cyclobutanedicarboxylic acid tert-butyl- (1,2,2-Trichloro-vinyl) -phosphinic acid 2 ', 3'-dichlorophthalanilic acid 3-methylene-cyclopropane-trans-1,2-dicarboxylic acid 1-alpha-hydroxyisovaleric acid

-167• 9-167 • 9

999 * ·· kyselina c/s-hexahydro-n-(4-metoxyfenyl)ftalámová kyselina 4-nitrobenzoová kyselina 4-undecyloxybenzoová kyselina bifenylénakrylová kyselina metylfenylfosfínová kyselina 4-(4'-n-hexylfenyl)benzoová kyselina 4'-bróm-2’-metylftalanilová kyselina n-(4-metoxyfenyl)glutáramová kyselina 3,5-diacetamidobenzoová kyselina 2,4,5-trimetoxybenzoová kyselina 2-(2-alylfenoxy)octová kyselina 2-trifluórmetyl-alfa-acetamidoškoricová kyselina 1-amino-ŕrans-cyklobután-1,3-dikarboxylová kyselina 4-(2-antranoyl)maslová kyselina 16-doxyl-stearová kyselina 4,8-dioxo-adamantán-1,2,5,7-tetrakarboxylová kyselina ŕrans-2-benzoyl-1 -cyklohexánkarboxylová kyselina 2-(4-(6-bróm-1 -hydroxy-2-naftylazo)fenoxy)octová kyselina 4-nitrofenyloctová kyselina 3,5-dibróm-4-hydroxyfenoxyoctová kyselina 2,3-difluórmandlová kyselina 3,5-bis(trifluórmetyl)fenyloctová kyselina benzénsulfínová n-gl utaryl-1 -fenylalanín, p-nitroanilid kyselina (s)-(-)-brómjantárová kyselina fenyletinyl-fosfónová kyselina n-alylmaleámová kyselina 3-benzoylamino-3-(2-fluór-fenyl)-propiónová kyselina 1-naftalénsulfónová kyselina xylénsulfónová semialdehyd kyseliny jantárovej kyselina 6-(4-benzyl-fenyl)-hexánová999 * ·· cis-hexahydro-n- (4-methoxyphenyl) phthalic acid 4-nitrobenzoic acid 4-undecyloxybenzoic acid biphenylene-acrylic acid methylphenylphosphinic acid 4- (4'-n-hexylphenyl) benzoic acid 4'-bromo-2 n-(4-methoxyphenyl) glutaramic acid 3,5-diacetamidobenzoic acid 2,4,5-trimethoxybenzoic acid 2- (2-allylphenoxy) acetic acid 2-trifluoromethyl-alpha-acetamido cinnamic acid 1-amino-trans- cyclobutane-1,3-dicarboxylic acid 4- (2-anthranoyl) butyric acid 16-doxyl-stearic acid 4,8-dioxo-adamantane-1,2,5,7-tetracarboxylic acid trans-2-benzoyl-1-cyclohexanecarboxylic acid 2- (4- (6-bromo-1-hydroxy-2-naphthylazo) phenoxy) acetic acid 4-nitrophenylacetic acid 3,5-dibromo-4-hydroxyphenoxyacetic acid 2,3-difluoromandelic acid 3,5-bis (trifluoromethyl) ) Phenylacetic benzenesulfinic acid n-gl utaryl-1-phenylalanine, p-nitroanilide (s) - (-) - bromosuccinic acid phenylethynyl-phosphonic acid n-allylmaleamic acid 3-benzoylamino-3- (2-fluoro-phenyl) -propionic acid 1-naphthalenesulfonic acid xylenesulfonic acid succinic acid semialdehyde 6- (4-benzyl-phenyl) -hexanoic acid

-168 --168 -

• · · • 9 • ··· • · · • 9 • ··· 99 9 · • 9 99 9 · • 9 999 9 9 • 999 9 9 • 99 • 9 9 9 99 • 9 9 9 • 9 • 9 • 9 ·· • 9 ·· • 9 • 9 99 99 99 99 9 9 9 9

kyselina S'-chlóM'-fluórmaleanilová kyselina dnp-d/-glutámová kyselina c/s-hexahydro-n-(4-chlór-3-nitrofenyl)ftalámová kyselina 1,3,4,5,6,5,5-heptametyl-7-oxo-bicyklo(2.2.2)okta-2,5-dién-2-karboxylová kyselina 2,3-difluór-4-(trifluórmetyl)fenyloctová kyselina n-boc-1 -aminocyklopropán-1 -karboxylová kyselina 4-metoxy-3-oxo-indán-1 -karboxylová kyselina (r)-2-hydroxy-4-fenylmaslová kyselina 4-(trifluórmetyl)ftalová kyselina 3,4,4-trifenyl-but-3-énová kyselina 6-chlór-2-nitrofenol-4-sulfónová kyselina n-terc-boc-(2s,3r)-3-amino-2-hydroxy-5-metylhexánová kyselina 4-metoxy-beta-metylškoricová kyselina 3,3-dichlór-2-(4-metyl-benzoylamino-akrylová kyselina 1 -(4-chlórfenyl)-5-oxo-3-pyrolidínkarboxylová kyselina 4-hydroxyfenylmalónová kyselina 4[[4-[(4,6-dimetylpyrimidín-2-yl)oxy]fenyl]amino]-4-oxo-(2z)-buténová kyselina 9-(4-metylfenyl)benzizoxazol-6-propénová kyselina (+/-)-1-aminocyklopentán-c/s-1,2-dikarboxylová kyselina 7-oxo-16-heptadecénová kyselina c/s-/?-(3-chlórfenyl)hexahydroftalárnová kyselina diendo-3-benzoylbicyklo[2.2.1]heptán-2-karboxylová kyselina hexaoxa-bicyklo(18.3.1 )tetrakoza-1 (23),20(24),21-trién-24-karboxylová kyselina 2-metyl-3-(2,4,6-trimetyl-3,5-dinitro-fenyl)-akrylová kyselina (+/-)-1-aminocyklopentán-ŕrans-1,2-dikarboxylová kyselina 2-nitroškoricová kyselina 3-hydroxy-4-metoxybenzoová kyselina 1 -benzocyklobuténkarboxylová kyselina didodecylfosfátS'-chloro-N'-fluoro-maleanoic acid dnp-d-glutamic acid cis-hexahydro-1- (4-chloro-3-nitrophenyl) phthalic acid 1,3,4,5,6,5,5-heptamethyl -7-oxo-bicyclo (2.2.2) octa-2,5-diene-2-carboxylic acid 2,3-difluoro-4- (trifluoromethyl) phenylacetic acid n-boc-1-aminocyclopropane-1-carboxylic acid 4- Methoxy-3-oxo-indan-1-carboxylic acid (R) -2-hydroxy-4-phenylbutyric acid 4- (trifluoromethyl) phthalic acid 3,4,4-triphenyl-but-3-enoic acid 6-chloro-2 -nitrophenol-4-sulfonic acid n-tert-boc- (2s, 3r) -3-amino-2-hydroxy-5-methylhexanoic acid 4-methoxy-beta-methyl cinnamic acid 3,3-dichloro-2- (4- methyl-benzoylamino-acrylic acid 1- (4-chlorophenyl) -5-oxo-3-pyrrolidinecarboxylic acid 4-hydroxyphenylmalonic acid 4 [[4 - [(4,6-dimethylpyrimidin-2-yl) oxy] phenyl] amino] - 4-Oxo- (2z) -butenoic acid 9- (4-methylphenyl) benzisoxazole-6-propenoic acid (+/-) -1-aminocyclopentane-cis-1,2-dicarboxylic acid 7-oxo-16-heptadecenoic acidcis - p - (3-chlorophenyl) hexahydrophthalic acid diendo-3-benzoylbicyclo [2.2.1] heptane-2-carboxylic acid hexaoxabicyclo (18.3.1) tetracoza-1 (23), 20 (24) 21-Triene-24-carboxylic acid 2-methyl-3- (2,4,6-trimethyl-3,5-dinitro-phenyl) -acrylic acid (+/-) -1-aminocyclopentane-trans-1,2 -dicarboxylic acid 2-nitrocinnamic acid 3-hydroxy-4-methoxybenzoic acid 1-benzocyclobutenecarboxylic acid didodecyl phosphate

5-etoxy-1,3-benzéndikarboxylová kyselina 3-(n-(2-fenyletyl)karbamoyl)-5-norbornén-2-karboxylová kyselina 3-fenyl-spiro(5.5)undekán-3-karboxylová5-Ethoxy-1,3-benzenedicarboxylic acid 3- (n- (2-phenylethyl) carbamoyl) -5-norbornene-2-carboxylic acid 3-phenyl-spiro (5.5) undecane-3-carboxylic acid

-169e · · · · · ·· · ·· ··· · · · · · · • ··· g · · · · kyselina 2,5-pyridíndikarboxylová kyselina p-chlórfenyl(benzyl)octová kyselina 4-metyl-3b,4,4a,5-tetrahydro-cyklopropa(a)fenalén-4-karboxylová kyselina alfa-etyl-m-nitroškoricová kyselina 3-amino-5-sulfo-salicylová kyselina 19-brómnonadekánová kyselina 1,2,3,4-tetrahydro-2-naftalénmaslová kyselina 4-benzyloxyškoricová kyselina 3-benzoyl-2-fenylpropiónová kyselina 4'-chlórsukcínanilová kyselina metafenyléndiamín-2-sulfónová kyselina 1 -metyl-5-oxo-3-pyrolidínkarboxylová kyselina 2-(4-(2-hydroxy-1 -naftylazo)fenoxy)octová kyselina 3,4-dimetoxy-2-hydroxybenzoová kyselina n-fenyl-malonámová kyselina 1,6-naftyridín-2-karboxylová kyselina 3-etoxykarbonylmetyl-1 h-indol-2-karboxylová kyselina 2’-etoxyftalanilová kyselina 2,5-dibenzyloxyfenyloctová kyselina 2',4,-dimetylsukcínanilová kyselina n-(2-fluórfenyl)glutarámová kyselina 1 -(2,4-dimetylfenyl)-6-metyl-4-oxo-1,4-dihydro-3-pyridínkarboxylová kyselina farnesyltiooctová kyselina 3-hydroxy-4-metylbenzoová kyselina 1 -metyl-4,9-dihydro-3h-beta-karbolín-3-karboxylová kyselina 4,4-dichlór-5,5,5-trifluórpentánová kyselina 5-brómsalicylová kyselina 2-karbamoyl-6-nitrobenzoová kyselina 4-naftalimidomaslová kyselina 9(10)-brómstearová kyselina glutaranilová kyselina 3-trifluórmetyl-3-hydroxymaslová • ·· ·· · ·· · ·· ··· · · · · · · • ··· · · · · ·-169e 2,5-pyridinedicarboxylic acid p-chlorophenyl (benzyl) acetic acid 4-methyl-3b 4,4a, 5-tetrahydro-cyclopropa (a) phenalene-4-carboxylic acid alpha-ethyl-m-nitro-cinnamic acid 3-amino-5-sulfo-salicylic acid 19-bromonadadecanoic acid 1,2,3,4-tetrahydro 2-naphthalenebutyric acid 4-benzyloxycinnamic acid 3-benzoyl-2-phenylpropionic acid 4'-chlorosuccinilic acid metaphenylenediamine-2-sulfonic acid 1-methyl-5-oxo-3-pyrrolidinecarboxylic acid 2- (4- (2-hydroxy- 1-naphthylazolphenoxy) acetic acid 3,4-dimethoxy-2-hydroxybenzoic acid n-phenyl-malonamic acid 1,6-naphthyridine-2-carboxylic acid 3-ethoxycarbonylmethyl-1H-indole-2-carboxylic acid 2'- etoxyftalanilová dibenzyloxyfenyloctová of 2,5-2 ', 4, -dimetylsukcínanilová n- (2-fluorophenyl) glutaramic acid 1 - (2,4-dimethylphenyl) -6-methyl-4-oxo-1,4- dihydro-3-pyridinecarboxylic acid farnesylthioacetic acid 3-hydroxy-4-methylbenzoic acid 1-methyl-4,9-dihydro-3h-beta-carboline-3-carboxylic acid 4,4-dichloro-5,5,5-trifluoropentanoic acid 5-bromosalicylic acid 2-carbamoyl-6-nitrobenzoic acid 4-naphthalimidobutyric acid 9 (10) -bromostearic acid glutaranilic acid 3-trifluoromethyl-3-hydroxybutyric acid · · · ··· · · · · · ·

-170kyselina fmoc-1-1,2,3,4-tetrahydronorharman-3-karboxylová kyselina 2,4-pyridíndikarboxylová kyselina 3-(3-(2,3-dichlórfenyl)ureido)benzoová kyselina 3-deoxy-d-glycero-d-galakto-2-nonulosonová kyselina 2-(4-chlórfenoxy)propiónová kyselina (+)-n-pinakolylftalámová kyselina d-gama-karboxyglutámová kyselina (s)-14-benzodioxán-2-karboxylová kyselina fmoc-(d,I)-2-aminotetralíη-2-karboxylová kyselina (s)-3-acetoxy-4-brómmaslová kyselina 2-hexadecyloxy-5-sulfobenzoová kyselina podokaprínová kyselina (-)-c/s,ŕrans-abscisová ([S]-5-[1 -hydroxy-2,6,6-trometyl-4-oxocyklohex-2-én--170 fmoc-1-1,2,3,4-tetrahydronorharman-3-carboxylic acid 2,4-pyridinedicarboxylic acid 3- (3- (2,3-dichlorophenyl) ureido) benzoic acid 3-deoxy-d-glycero- d-galacto-2-nonulosonic acid 2- (4-chlorophenoxy) propionic acid (+) - n-pinacolylphthalic acid d-gamma-carboxyglutamic acid (s) -14-benzodioxane-2-carboxylic acid fmoc- (d, I) -2-aminotetraline-2-carboxylic acid (s) -3-acetoxy-4-bromobutyric acid 2-hexadecyloxy-5-sulfobenzoic acid podocaproic acid (-) - cis, trans-abscisic acid ([S] -5- [ 1-Hydroxy-2,6,6-tromethyl-4-oxocyclohex-2-ene

1-yl]-3-metyl-[2z,4e]pentadiénová) kyselina fmoc-alfa-aminomaslová kyselina 2-(3-nitro-benzylidén)-tridec-12-énová kyselina [1 -(4-hydroxyfenoxy)etylidén]bisfosfónová kyselina 3-etoxyfenyloctová kyselina 3-(hexadekánamido)benzoová kyselina (4,5-dimetoxy-3-oxo-1,3-dihydro-izobenzofurán-1 -yl)-octová kyselina 2-(3-acetyl-4-hydroxy-fenylkarbamoyl)-cyklohex-1-énkarboxylová kyselina 4-(bróm-metyl)fenyloctová kyselina 2-butoxy-5-ŕerc-pentylbenzénsulfónová kyselina metafosforečná kyselina ŕrans-4-hydroxy-2-buténová kyselina 1,3,5-pentántrikarboxylová kyselina 4-aminobutylfosfónová kyselina 3,4-dimetoxyškoricová kyselina n-(2-fenetyl)ftalámová kyselina 2,6-heptadiénová kyselina 6-oxo-1,12-dodekándikarboxylová kyselina 2-chlór-3,5-dinitrobenzénsulfónová * ΦΦ ΦΦ ΦΦΦΦ ··1-yl] -3-methyl- [2z, 4e] pentadienoic) fmoc-alpha-aminobutyric acid 2- (3-nitro-benzylidene) -tridec-12-enoic acid [1- (4-hydroxyphenoxy) ethylidene] bisphosphonic acid 3-Ethoxyphenylacetic acid 3- (hexadecanamido) benzoic acid (4,5-dimethoxy-3-oxo-1,3-dihydro-isobenzofuran-1-yl) -acetic acid 2- (3-acetyl-4-hydroxyphenylcarbamoyl) ) -cyclohex-1-enecarboxylic acid 4- (bromomethyl) phenylacetic acid 2-butoxy-5-tert-pentylbenzenesulfonic acid metaphosphoric acid trans-4-hydroxy-2-butenoic acid 1,3,5-pentanetricarboxylic acid 4-aminobutylphosphonic acid 3,4-dimethoxycinnamic acid n- (2-phenethyl) phthalic acid 2,6-heptadienoic acid 6-oxo-1,12-dodecanedicarboxylic acid 2-chloro-3,5-dinitrobenzenesulfonic acid * ΦΦ ΦΦ ΦΦΦΦ ··

ΦΦΦ ** φ«·8 ··· φ · 8 88ΦΦΦ ** φ «· 8 ··· φ · 8 88

-171 n-ftaloylglycín kyselina 2-naftol-3,6,8-trisulfónová kyselina 2,2,4,4,5,5,7,7,8,8,10,10,10-tridekafluór-3,6,9-trioxadekánová kyselina 2,3,4,6-di-o-izopropylidén-2-keto-1 -gulónová kyselina c/s-2-(4-fluórbenzoyl)-1 -cyklohexán-karboxylová kyselina dichlórmetylfosfónová kyselina n-oktylmaleámová kyselina ftalid-3-octová kyselina 2,3-dibróm-3,,4,-dichlórsukcínanilová kyselina 2-acetamido-5-brómbenzoová kyselina (2-bróm-4-metyl-fenyl)-fosfónová kyselina 2-hydroxy-4,6-dimetoxybenzoová kyselina boc-iminodioctová kyselina metylén-bis(3-tiopropiónová) kyselina ditiotereftalová kyselina domoiová (C15H21NO6) kyselina 3-metylfenoxyoctová kyselina 2-metyl-3-(3-nitro-fenyl)-akrylová kyselina 4-metyl-1,1-cyklohexándioctová kyselina 2-acetamido-4-fluórbenzoová kyselina 1 -metyl-2-cyklohexén-1 -karboxylová kyselina 4'-chlórftalanilová kyselina 3-formylfenoxyoctová kyselina alfa-truxilová kyselina 4-(2-nitrofenyl)maslová kyselina n-metyl-sukcínamová kyselina 2'-benzylkarbamoyl-bifenyl-2-karboxylová kyselina 3-(1,3-dioxo-1,3-dihydro-izoindol-2-yl)-benzoová kyselina 2-metyl-5-norbornén-2-karboxylová kyselina 3-etoxy-4-metoxybenzoová kyselina 2-(fluórantén-8-karbonyl)-benzoová kyselina 3-(2,3-dimetoxyfenyl)propiónová • ·· ·· «··· ·· ··· · · · ··· • ··· · · · · I-171 n-phthaloylglycine 2-naphthol-3,6,8-trisulfonic acid 2,2,4,4,5,5,7,7,8,8,10,10,10-tridecafluoro-3,6 9-trioxadecanoic acid 2,3,4,6-di-o-isopropylidene-2-keto-1-gulonic acid cis-2- (4-fluorobenzoyl) -1-cyclohexanecarboxylic acid dichloromethylphosphonic acid n-octylmaleamic acid phthalide-3-acetic acid, 2,3-dibromo-3, 4, -dichlórsukcínanilová acid 2-acetamido-5-bromobenzoic acid (2-bromo-4-methyl-phenyl) -phosphonic acid 2-hydroxy-4,6- dimethoxybenzoic acid boc-iminodiacetic acid methylene-bis (3-thiopropionic) dithioterephthalic acid, domioic acid (C15H21NO6) 3-methylphenoxyacetic acid 2-methyl-3- (3-nitro-phenyl) -acrylic acid 4-methyl-1,1- cyclohexanediacetic acid 2-acetamido-4-fluorobenzoic acid 1-methyl-2-cyclohexene-1-carboxylic acid 4'-chlorophthalanilic acid 3-formylphenoxyacetic acid alpha-truxilic acid 4- (2-nitrophenyl) butyric acid n-methyl-succinamine 2'-Benzylcarbamoyl-biphenyl-2-carboxylic acid 3- (1,3-dioxo-1,3-dihydro-isoindol-2-yl) -benzoic acid 2-methyl-5-norbornene-2-carboxylic acid 3 -ethoxy-4-methoxybenzoic acid 2- (fluoroanthene-8-carbonyl) -benzoic acid 3- (2,3-dimethoxyphenyl) propionic acid • ··· ··· ··· ··· I

-172kyselina r-4-brómmandlová kyselina 4-acetamidoškoricová kyselina (2-metoxy-fenyl)-fenyl-fosfínová kyselina 6-hydroxy-2-naftoová kyselina (s)-(+)-n-(4-((aminoiminometyl)amino)-1-karboxybutyl)-d-glutámová kyselina 2,4,6-trimetoxyfenyloctová kyselina 3-metylpyrazolo-[3,4-b]-chinolin-4-karboxylová kyselina 3-aminometylalizarin-n,n-dioctová kyselina n-(5-chlór-2-metylfenyl)maleámová kyselina dnp-1-glutámová kyselina 2-(4-bifenylyloxy)propiónová kyselina 4-hydroxy-6-(trifluórmetyl)-3-chinolín-karboxylová kyselina anilín-2,4-disulfónová kyselina (s)-(-)-alfa-fenetylsulfámová kyselina 2-(4-nitrofenyl)maslová kyselina 4-(4-metoxy-2-metyl-fenyl)-4-oxo-maslová kyselina 3-(2-oxo-1,3,3-trimetylcyklohexyl)propiónová kyselina 4’-butyl-1,2,3,6-tetrahydroftalanilová kyselina (r)-1,4-benzodioxán-2-karboxylová kyselina 2-(2-etoxyfenylkarbamoyl)cyklohexánkarboxylová kyselina 6-hydroxy-3-oxo-3h-xantén-9-karboxylová kyselina fenylfosfínová kyselina 4-metylškoricová kyselina n-naftalén-1 -yl-sukcínamová kyselina 2-metyl-5,6-dihydro-[1.4]oxatiín-3-karboxylová kyselina 3-bróm-4-hydroxyfenyloctová kyselina tricyklo(2.2.1.0(2,6))heptán-1 -karboxylová kyselina 3-metyl-3-fenyl-pentánová kyselina 1 -(2-chlórbenzoyl)piperazín-2,3-dikarboxylová etyl-mandlan kyselina 2-propyldekánová kyselina (r)-(+)-alfa-fenetylsulfámová • ·· ·· ···· ·· ·· · · · · · · • ··· · 9 · · ·-172 r-4-Bromo-mandelic acid 4-acetamido-cinnamic acid (2-methoxy-phenyl) -phenyl-phosphinic acid 6-hydroxy-2-naphthoic acid (s) - (+) - n- (4 - ((aminoiminomethyl) amino) -1-carboxybutyl) -d-glutamic acid 2,4,6-trimethoxyphenylacetic acid 3-methylpyrazolo- [3,4-b] quinoline-4-carboxylic acid 3-aminomethylalizarin-n, n-diacetic acid n- ( 5-chloro-2-methylphenyl) maleic acid dnp-1-glutamic acid 2- (4-biphenylyloxy) propionic acid 4-hydroxy-6- (trifluoromethyl) -3-quinoline carboxylic acid aniline-2,4-disulfonic acid ( s) - (-) - alpha-Phenethylsulfamic acid 2- (4-nitrophenyl) butyric acid 4- (4-methoxy-2-methylphenyl) -4-oxo-butyric acid 3- (2-oxo-1,3 (3) -1,4-benzodioxane-2-carboxylic acid 2- (2-ethoxyphenylcarbamoyl) cyclohexanecarboxylic acid 6-hydroxy-3, 3-trimethylcyclohexyl) propionic acid 4'-butyl-1,2,3,6-tetrahydrophthalanic acid -oxo-3h-xanthene-9-carboxylic acid phenylphosphinic acid 4-methylscor n-Naphthalen-1-yl-succinic acid 2-methyl-5,6-dihydro- [1,4] oxathiine-3-carboxylic acid 3-bromo-4-hydroxyphenylacetic acid tricyclo (2.2.1.0 (2,6)) heptane-1-carboxylic acid 3-methyl-3-phenylpentanoic acid 1- (2-chlorobenzoyl) piperazine-2,3-dicarboxylic ethyl mandanic acid 2-propyldecanoic acid (r) - (+) - alpha-phenethylsulfamic acid • ····················· · 9

-173kyselina 3,5-dimetyl-1-cyklohexén-1,2-dikarboxylová kyselina 3-(pyrolidín-1 -karbotioylsulfanyl)-propiónová kyselina 2,2,-ditiodipropiónová kyselina 2-[3,5-bis(trifluórmetyl)benzoyl]benzoová kyselina 4-fluórbenzoová kyselina 2-fluórizoftalová kyselina 3-[5-(2-chlór-5-trifluórmetyl-fenyl)furán-2-yl]-2-kyanoakrylová kyselina 5-(4-chlór-fenylsulfanyl)-furán-2-karboxylová kyselina (s)-(-)-2-chlórjantárová kyselina 5-(tiobenzoyl)tioglykolová kyselina 5-hydroxy-2-nitrobenzoová kyselina alfa-metyl-p-[2-tenoyl]fenyloctová kyselina 3h-tetrafluórpropiónová kyselina 4-etyl-tiomaslová kyselina 3-fluór-2,4-dimetyl-benzoová kyselina (2-metyl-4-nitro-fenyl)-fosfónová kyselina 2-etyl-3-(2-metoxy-fenyl)-akrylová kyselina 3,5-dinitro-o-toluylová kyselina 2-(4-chlórfenyl)-3-(3-metylbenzoyl)propiónová kyselina 4-fenylvalérová kyselina (4-jód-fenyl)-fenyl-fosfínová kyselina benzofenón-2,4'-dikarboxylová kyselina 2-ftalimidoglutaranilová kyselina 5-butylhydantoínová kyselina (2-hydroxynorbornán-2-yl)-fenyloctová kyselina 2-[(5-oxotetrahydro-1 h-2-pyrolyl)sulfanyl]octová kyselina 1,4-fenylén-dipropiónová kyselina n-furfurylmaleámová kyselina 4-metoxymandlová kyselina oktahydro-6-oxo-6h-pyrido(3,2,1-jk)karbazol-11 b-propiónová kyselina 1 -chlór-3-metyl-izochinolín-4-karboxylová beta-benzylester kyseliny benzyloxykarbonyl-1-asparágovej-173 3,5-Dimethyl-1-cyclohexene-1,2-dicarboxylic acid 3- (pyrrolidine-1-carbothioylsulfanyl) -propionic acid 2,2 , -dithiodipropionic acid 2- [3,5-bis (trifluoromethyl) benzoyl] benzoic acid 4-fluorobenzoic acid 2-fluoroisophthalic acid 3- [5- (2-chloro-5-trifluoromethyl-phenyl) furan-2-yl] -2-cyanoacrylic acid 5- (4-chloro-phenylsulfanyl) -furan-2 (s) - (-) - 2-chlorosuccinic acid 5- (thiobenzoyl) thioglycolic acid 5-hydroxy-2-nitrobenzoic acid alpha-methyl-p- [2-tenoyl] phenylacetic acid 3h-tetrafluoropropionic acid 4-ethyl 3-fluoro-2,4-dimethyl-benzoic acid (2-methyl-4-nitro-phenyl) -phosphonic acid 2-ethyl-3- (2-methoxy-phenyl) -acrylic acid 3,5-dinitro -o-toluic acid 2- (4-chlorophenyl) -3- (3-methylbenzoyl) propionic acid 4-phenylvaleric acid (4-iodo-phenyl) -phenyl-phosphinic acid benzophenone-2,4'-dicarboxylic acid 2-phthalimidoglutaranilic acid 5-butylh (2-hydroxynorboranen-2-yl) -phenylacetic acid 2 - [(5-oxotetrahydro-1H-2-pyrrolyl) sulfanyl] acetic acid 1,4-phenylene dipropionic acid n-furfurylmaleamic acid 4-methoxy-butyric acid octahydro 6-oxo-6h-pyrido (3,2,1-jk) carbazole-11b-propionic acid 1-Chloro-3-methyl-isoquinoline-4-carboxylic acid benzyloxycarbonyl-1-aspartic acid beta-benzyl ester

-174--174-

• ·· • · • ··· • ·· • · • ··· ·· • · • · · · • · • · ···· • • ···· • • ·· · • · ·· • e e ·· · • · ·· • e e ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 2-chlórakrylová kyselina 2,3-dimetylfurán-5-karboxylová kyselina 2,6-dimetyl-3,5-pyridíndikarboxylová kyselina c/s-2,6-piperidín-dikarboxylová kyselina c/s-hexahydro-n-(3-(trifluórmetyl)fenyl)ftalámová kyselina trans-dl-1,2-cyklopentán-dikarboxylová kyselina 2-hydroxy-3-izopropylbenzoová kyselina fenoxyoctová kyselina n-(2-etyl-6-metyl-fenyl)-3-nitro-ftalámová kyselina 2-jód-5-nitro-benzoová kyselina 5-(4-chlór-3-nitro-fenylsulfamoyl)-izoftalová kyselina 6-metyl-2,3-pyridíndikarboxylová kyselina n-formyl-1-asparágová kyselina 5-hydroxypyrazín-2-karboxylová kyselina 2-(2,4-dimetylbenzoyl)benzoová kyselina 5-bróm-2-chlórbenzoová kyselina 2-(9h-xantén-9-yl)-malónová kyselina c/s-2’,4'-dimetylhexahydroftalanilová kyselina 2,3,4,5-tetrametyl-benzoová kyselina 2-(7-oxo-7h-benz(de)antracén-3-yltio)octová kyselina n-(p-tolyl)ftalámová kyselina 4,4'-izopropylidéndifenoxyoctová kyselina (1 r,2r)-(-)-1,2-cyklohexándikarboxylová kyselina 4-fluór-3-(trifluórmetyl)škoricová kyselina d-pantoténová kyselina 4,5-imidazoldikarboxylová kyselina 4-(2,4-dichlórbenzylidénamino)benzoová kyselina 2-metyltio-5-benzotiazolsulfónová kyselina benzo[b]tiofén-2-karboxylová kyselina 5-benzoyl-7-bróm-2,3-dihydro-1 h-py rolizí n-1 -karboxylová kyselina 1 -(3-fliiórfenyl)cyklopentánkarboxylová kyselina brómdichlóroctová2-chloroacrylic acid 2,3-dimethylfuran-5-carboxylic acid 2,6-dimethyl-3,5-pyridinedicarboxylic acid cis-2,6-piperidine-dicarboxylic acid cis-hexahydro-n- (3- (trifluoromethyl) phenyl) phthalic acid trans-dl-1,2-cyclopentane-dicarboxylic acid 2-hydroxy-3-isopropylbenzoic acid phenoxyacetic acid n- (2-ethyl-6-methylphenyl) -3-nitrophthalic acid 2 5- (4-chloro-3-nitro-phenylsulfamoyl) -isophthalic acid 6-methyl-2,3-pyridinedicarboxylic acid iodo-5-nitro-benzoic acid n-formyl-1-aspartic acid 5-hydroxypyrazine-2-carboxylic acid 2- (2,4-dimethylbenzoyl) benzoic acid 5-bromo-2-chlorobenzoic acid 2- (9h-xanthen-9-yl) malonic acid cis-2 ', 4'-dimethylhexahydrophthalanic acid 2,3, 4,5-tetramethylbenzoic acid 2- (7-oxo-7h-benz (de) anthracen-3-ylthio) acetic acid n- (p-tolyl) phthalic acid 4,4'-isopropylidenediphenoxyacetic acid (1 r, 2r - (-) - 1,2-Cyclohexanedicarboxylic acid 4-flu orth-3- (trifluoromethyl) cinnamic acid d-pantothenic acid 4,5-imidazole dicarboxylic acid 4- (2,4-dichlorobenzylidenamino) benzoic acid 2-methylthio-5-benzothiazolesulfonic acid benzo [b] thiophene-2-carboxylic acid 5- Benzoyl-7-bromo-2,3-dihydro-1H-pyrrolidine-1-carboxylic acid 1- (3-fluorophenyl) cyclopentanecarboxylic acid bromodichloroacetic acid

-175kyselina (+/-)-2-hydroxyundekánová kyselina 2-butoxyoctová kyselina 3-eténsulfonyl-propiónová kyselina pentafluórfenoxyoctová kyselina 3-metyl-4-cyklohexén-c/s-1,2-dikarboxylová kyselina bicyklo[2.2.1 )heptán-2-karboxylová kyselina 3-(4-metylsulfanyl-fenyl)-akrylová kyselina 5-norbornén-2-akrylová kyselina 3,5-dimetyl-4-nitrobenzoová kyselina 2-propylpentánová kyselina 1-cysteínová kyselina cinamylidénmalónová kyselina 5-formyl-2-tiofénkarboxylová kyselina d/-4-hydroxymandlová kyselina 5-(hydroxyimino)azelainová kyselina 2,3-naftaléndikarboxylová n-butyl-pyrofosfát kyselina n-oktadecylglutarámová kyselina n-cyklohexylmaleámová kyselina dansyl-1-cysteinová kyselina m-krezyl-glutárová kyselina 3-hexadecyloxy-4-nitrobenzoová kyselina 5-nitro-2-propiónamidobenzoová kyselina n, n-dibenzylhexahydroftalámová kyselina 4-karboxymetylsulfanyl-3-nitro-benzoová kyselina ricínolejová kyselina c/s-12-oktadecénová kyselina 3-(metylfosfornan)-propiónová kyselina metylénbistioglykolová kyselina 2-metylškoricová kyselina (s)-2-chlór-n-maslová kyselina 2-brómpropiónová-175 (+/-) - 2-hydroxyundecanoic acid 2-butoxyacetic acid 3-Ethenesulfonyl-propionic acid pentafluorophenoxyacetic acid 3-methyl-4-cyclohexene-cis-1,2-dicarboxylic acid bicyclo [2.2.1] heptane- 2-carboxylic acid 3- (4-methylsulfanyl-phenyl) -acrylic acid 5-norborene-2-acrylic acid 3,5-dimethyl-4-nitrobenzoic acid 2-propylpentanoic acid 1-cysteine cinamylidenemalonic acid 5-formyl-2- thiophenecarboxylic acid d-4-hydroxymandelic acid 5- (hydroxyimino) azelaic acid 2,3-naphthalenedicarboxylic acid n-butylpyrophosphate n-octadecylglutaramic acid n-cyclohexylmaleamic acid dansyl-1-cysteic acid m-cresyl-glutaric acid 3-hexadecyloxy 4-nitrobenzoic acid 5-nitro-2-propionamidobenzoic acid n, n-dibenzylhexahydrophthalic acid 4-carboxymethylsulfanyl-3-nitro-benzoic acid ricinoleic acid cis-12-octadecenic acid 3- (methylphosphonate) -propionic acid Methylenebistioglycolic acid 2-methylcinnamic acid (s) -2-chloro-n-butyric acid 2-bromopropionic acid

-176- • 99 99 999999-176- 99 99 999999

9 9 9 9 9 99 • ··· · · ·· t kyselina 5-chlór-2-metoxybenzoová kyselina 2-metylhexánová kyselina 2,6-bis(trifluórmetyl)benzoová kyselina A'-fluór-SAS.e-tetrachlórftalanilová kyselina 3-(3,4-dichlór-fenylamino)-maslová kyselina dimetylfosfínová kyselina 2-hydroxy-3-buténová kyselina 2,3I4-trimetyl-5-nitro-benzoová kyselina 2-hydroxy-3(s)-(n-terc-boc-amino)-4-metoxybutánová kyselina 2-(3,4-dichlórbenzoyl)benzoová kyselina 3,5-dibenzyloxybenzoová kyselina 4-(4-(4-chlór-benzénsulfonyl)-fenoxy)-benzoová kyselina 1-naftol-5-sulfónová kyselina 2-acetyl-3,6-difluórbenzoová (r)-(+)-trolox(r) (kyselina 6-hydroxy-2,5,7,8-tetrametylchroman-2-karboxylová) kyselina krezol-sulfónová kyselina 2-oxo-1,1,3,3-cyklohexántetrapropiónová kyselina (dI)-2-(4-bifenylyl)propiónová kyselina palmitelaidová kyselina (10,11 -dihydro-dibenzo(a,d)cykloheptén-5-ylidén)-octová kyselina 5-bróm-2-metoxyizoftalová kyselina(s)-2-etyldodekánová kyselina 2-benzoylamino-3-(4-izopropoxy-fenyl)-akrylová kyselina 16-heptadecénová kyselina 1,2,3,4-tetrahydro-gama-oxo-2-pyrido[4,3-b][1,8]naftyridinbutánová kyselina (1r,3r)-1-aminocyklopentán-1,3-dikarboxylová kyselina 2-hydroxy-5-metoxybenzoová kyselina tnp-alfa-aminomaslová kyselina 2-[1 -(6-chlór-3-pyridazinyl)-1 h-3-indolyl]octová kyselina 2,3,4-trimetoxybenzoová kyselina (+)-s-2-amino-5-jódacetamidopentánová kyselina 4,-bróm-2'-metylsukcínanilová • ·· ·· ···· ·· ··· ·· ···· • ··· 9 9 9 9 99 9 9 9 9 99 5-chloro-2-methoxybenzoic acid 2-methylhexanoic acid 2,6-bis (trifluoromethyl) benzoic acid A'-fluoro-SAS.e-tetrachlorophthalanic acid 3 - (3,4-dichloro-phenylamino) -butyric acid, dimethylphosphinic acid 2-hydroxy-3-butenoic acid 2.3 L 4-trimethyl-5-nitro-benzoic acid 2-hydroxy-3 (s) - (n-t -boc-amino) -4-methoxybutanoic acid 2- (3,4-dichlorobenzoyl) benzoic acid 3,5-dibenzyloxybenzoic acid 4- (4- (4-chlorobenzenesulfonyl) phenoxy) -benzoic acid 1-naphthol-5 sulfonic acid 2-acetyl-3,6-difluorobenzoic acid (r) - (+) - trolox (r) (6-hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acid) cresol sulfonic acid 2 -oxo-1,1,3,3-cyclohexanetetrapropionic acid (dI) -2- (4-biphenylyl) propionic acid palmitelaidic acid (10,11-dihydro-dibenzo (a, d) cyclohepten-5-ylidene) -acetic acid 5-Bromo-2-methoxyisophthalic acid (s) -2-ethyldodecanoic acid 2-benzoylamino-3- (4-Isopropoxy-phenyl) -acrylic acid 16-Heptadecenoic acid 1,2,3,4-tetrahydro-gamma-oxo-2-pyrido [4,3-b] [1,8] naphthyridinobutanoic acid (1r, 3r) -1-aminocyclopentane-1,3-dicarboxylic acid 2-hydroxy-5-methoxybenzoic acid β-alpha-aminobutyric acid 2- [1- (6-chloro-3-pyridazinyl) -1H-3-indolyl] acetic acid 2 3,4-trimethoxybenzoic acid (+) - s-2-amino-5-iodoacetamidopentanoic acid 4 , -bromo-2'-methylsuccinic acid • ···················· 9 9 9 9 9

-177kyselina n-(2-fenetyl)glutarámová kyselina 2,4,5-trimetoxyškoricová kyselina 3,3-dichlórglutárová kyselina 3-(7-metoxy-2,2-difenyl-benzo(1,3)dioxol-5-yl)-akrylová kyselina 1-tetrazol-octová kyselina 3-hydroxy-7-oxo-7h-benzo(de)antracén-2-karboxylová kyselina 3-(6-metoxy-2-metyl-1 -oxo-1,2,3,4-tetrahydro-naftalén-2-yl)propiónová kyselina (+)-mentoxyoctová kyselina 4-(4-(3,4-dimetylfenyl)-benzénsulfonyl)-ftalová kyselina 2,5-dimetyl-4-nitrobenzoová kyselina 3-(4-metoxy-1 -naftoyl)-propiónová kyselina 2-bróm-2-buténová kyselina (r)-(+)-2-chlórjantárová kyselina 4,5,5,6,6,6-hexafluór-4-(trifluórmetyl)hexánová kyselina 2-oxo-1 -(3-trifluórmetylfenyl)pyrolidín-4-karboxylová kyselina 4-(2-karbamoyl-acetylamino)-benzoová kyselina 4,5-difluór-2-nitrobenzoová kyselina 9-kyanopelargónová kyselina 1-antracénkarboxylová kyselina 3-ftalimidopropiónová kyselina 5-(2-tienyl)pentánová kyselina 3-feny I-1 -indanón-3-karboxylová kyselina (s)-(+)-2-amino-2-metylbutándiová kyselina 2-(2-metoxy-fenyl)-propiónová kyselina 3-amino-5-nitro-2,4,6-trimetylbenzénsulfónová kyselina 2,2-(diacetamido)propiónová kyselina d/-3-metoxymandlová kyselina 4-bróm-3-fluórbenzoová kyselina 1,2-aminokorková kyselina 2-(orto-tolyl)-propiónová kyselina 8(s), 15(s)-dihydroxyeikoza-5z,9e, 11 e, 13e-tetraénová kyselina 2,2-bis(hydroxymetyl)propiónová • ·· ·· ···· ·· ··· ·· ···· • ··· · · · · ·-177 n- (2-phenethyl) glutaramic acid 2,4,5-trimethoxycinnamic acid 3,3-dichloroglutaric acid 3- (7-methoxy-2,2-diphenyl-benzo (1,3) dioxol-5-yl) -acrylic acid 1-tetrazole-acetic acid 3-hydroxy-7-oxo-7h-benzo (de) anthracene-2-carboxylic acid 3- (6-methoxy-2-methyl-1-oxo-1,2,3), 4-Tetrahydro-naphthalen-2-yl) propionic acid (+) - Mentoxyacetic acid 4- (4- (3,4-dimethylphenyl) -benzenesulfonyl) -phthalic acid 2,5-dimethyl-4-nitrobenzoic acid 3- (4 -methoxy-1-naphthoyl) -propionic acid 2-bromo-2-butenoic acid (r) - (+) - 2-chlorosuccinic acid 4,5,5,6,6,6-hexafluoro-4- (trifluoromethyl) hexanoic acid 2-oxo-1- (3-trifluoromethylphenyl) pyrrolidine-4-carboxylic acid 4- (2-carbamoyl-acetylamino) -benzoic acid 4,5-difluoro-2-nitrobenzoic acid 9-cyanopelargonic acid 1-anthracenecarboxylic acid 3- 5- (2-Thienyl) pentanoic acid phthalimidopropionic acid 3-Phenyl-1-indanone-3-carboxylic acid (s) - (+) - 2-amino-2 2- (2-methoxyphenyl) -propionic acid 3-amino-5-nitro-2,4,6-trimethylbenzenesulfonic acid 2,2- (diacetamido) propionic acid d--3-methoxymandelic acid 4-bromo-methylbutanedioic acid -3-fluorobenzoic acid 1,2-aminocorkic acid 2- (ortho-tolyl) -propionic acid 8 (s), 15 (s) -dihydroxyeicoza-5z, 9e, 11e, 13e-tetraenoic acid 2,2-bis ( Hydroxymethyl) propionic acid ·) · • · · · · · · · · · · · ·

-178kyselina 1-alfa-aspartyl-1 -asparágová kyselina 2-undec-10-ényl-malónová kyselina 2-(4-metylbenzoyl)-akrylová kyselina (5-(2-chlór-fenyl)-pyrimidín-4-ylsulfanyl)octová kyselina pinová kyselina 9(10)-jódstearová kyselina 2-(4-chlórfenyl)-2-adamantán-octová kyselina (2-acetylamino-fenyl)-octová kyselina 2-[(fenylsulfonyl)(2-pyridyl)amino]octová kyselina 5-(4-chlórfenyl)-2-(trifluórmetyl)furán-3-karboxylová kyselina dihydrokainová (kyselina kainová = 2-karboxy-3-karboxymetyl-4-izopropenylpyrolidín) kyselina n-alfa-fmoc-n-beta-aloc-1 -diaminopropiónová kyselina 2’-metoxy- 5'-metylglutaranilová kyselina 2-fluór-6-(trifluórmetyl)benzoová kyselina 2-metyl-3-(1 -naftoyl)propiónová kyselina tiodiglykolová kyselina 1,2-diaminopropán-n,n,n’,n’-tetraoctová kyselina 4-(2-(2-chlórbenzoyl)acetamido)benzoová kyselina izomaslová kyselina 3-metyl-4-p-tolyl-maslová kyselina 2-antracénkarboxylová kyselina 4’-chlór-3,415,6-tetrachlórftalanilová kyselina 1 -hydroxycykloheptánkarboxylová kyselina 4-acetylfenoxyoctová kyselina 3-fluór-4-(trifluórmetyl)škoricová kyselina c/s-hexahydro-n-fenylftalámová kyselina c/s-13,16,19-dokozatriénová kyselina hexakozándiová kyselina 2'- metyl-3,4,5,6-tetrachlórftalanilová kyselina 4-(6-hydroxy-3-oxo-3h-xantén-9-yl)benzoová kyselina (4-(4-etyl-fenoxy)-fenoxy)-octová-178 1-alpha-aspartyl-1-aspartic acid 2-undec-10-enyl-malonic acid 2- (4-methylbenzoyl) -acrylic acid (5- (2-chloro-phenyl) -pyrimidin-4-ylsulfanyl) -acetic acid 9 (10) -iodo-stearic acid 2- (4-chloro-phenyl) -2-adamantane-acetic acid (2-acetylamino-phenyl) -acetic acid 2 - [(phenylsulfonyl) (2-pyridyl) amino] -acetic acid 5 - (4-chlorophenyl) -2- (trifluoromethyl) furan-3-carboxylic acid dihydrocaic acid (kainic acid = 2-carboxy-3-carboxymethyl-4-isopropenylpyrrolidine) n-alpha-fmoc-n-beta-aloc-1 - diaminopropionic acid 2'-methoxy-5'-methylglutaranilic acid 2-fluoro-6- (trifluoromethyl) benzoic acid 2-methyl-3- (1-naphthoyl) propionic acid thiodiglycolic acid 1,2-diaminopropane-n, n, n ' , n'-tetraacetic acid 4- (2- (2-chlorobenzoyl) acetamido) benzoic acid isobutyric acid 3-methyl-4-p-tolylbutyric acid 2-anthracenecarboxylic acid 4'-chloro-3,4 1 5,6 -tetrachlorophthalic acid 1 - hydroxycycloheptanecarboxylic acid 4-acetylphenoxyacetic acid 3-fluoro-4- (trifluoromethyl) cinnamic acid cis-hexahydro-n-phenylphthalic acid cis-13,16,19-docosatrienoic acid hexacosanedioic acid 2'-methyl-3,4, 4- (6-Hydroxy-3-oxo-3H-xanthen-9-yl) benzoic acid (4- (4-ethyl-phenoxy) -phenoxy) -acetic acid

-179 --179 -

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · ···· • • ···· • • ·· • · • · ·· • · • · • · • · ·· ·· ·· ·· ·· · · ·· · · ·· · · • · • ·

kyselina (+/-)-c/s-9,10-metylénoktadekánová kyselina 2-benzoylamino-3-(etoxy-fenyl-fosfinoyl)-3-fenyl-akrylová kyselina 5-(4-chlórbenzoyl)tiofén-2-octová kyselina 9-antracénpropiónová kyselina 4-fenetidín-2-sulfónová kyselina 2-(brómmetyl)akrylová kyselina 2-hepténová kyselina 2,4-dibrómfenoxyoctová kyselina benzo(c)fenantrén-5-karboxyiic kyselina 9-( 10)-hydroxyfenylstearová kyselina r-4-chlórmandlová kyselina 5-fluór-2,3-dihydro-gama-oxo-1-(1h)-indolbutánová kyselina (s)-tetrahydrofurán-2-karboxylová kyselina p-butoxybenzoová kyselina 2-(4-nitro-benzoylamino)-3-fenyl-akrylová kyselina 4-hydroxy-7-metoxy-1-(3-metoxy-fenyl)-naftalén-2-karboxylová kyselina 3-(4-izopropyl-fenyl)-2-metyl-akrylová kyselina difluóroctová kyselina c/s,c/s,c/s,c/s-1,2,3,4-cyklopentántetrakarboxylová kyselina 3-metyldekánová kyselina boc-d-pipekolínová kyselina (+/-)-2-endo-aminobicyklo[2.2.1]heptán-2-exo-7-anti-dikarboxylová kyselina 4,-fluór-3,3’,4,5,6-pentachlórftalanilová kyselina 4-fluór-3-nitrobenzoová kyselina 2-metyl-3,4,6-pyridíntrikarboxylová kyselina 3-metylsulfonylbenzoová kyselina 2-(hexadecylsulfonyl)benzoová kyselina izoindolín-1 -ón-2-(2-propiónová) kyselina c/s-5-norbornén-endo-2,3-dikarboxylová kyselina 9-fenylnonánová kyselina 2-fluór-5-(trifluórmetyl)benzoová kyselina 2,,4’,5,-trichlórglutaranilová(+/-) - cis-9,10-methylenoctadecanoic acid 2-benzoylamino-3- (ethoxy-phenyl-phosphinoyl) -3-phenyl-acrylic acid 5- (4-chloro-benzoyl) -thiophene-2-acetic acid 9-anthracenepropionic acid 4-phenetidine-2-sulfonic acid 2- (bromomethyl) acrylic acid 2-heptenoic acid 2,4-dibromophenoxyacetic acid benzo (c) phenanthrene-5-carboxylic acid 9- (10) -hydroxyphenylstearic acid r-4 5-fluoro-2,3-dihydro-gamma-oxo-1- (1h) -indole-butanoic acid (s) -tetrahydrofuran-2-carboxylic acid p-butoxybenzoic acid 2- (4-nitro-benzoylamino) -3 4-hydroxy-7-methoxy-1- (3-methoxy-phenyl) -naphthalene-2-carboxylic acid-phenyl-acrylic acid 3- (4-isopropyl-phenyl) -2-methyl-acrylic acid difluoroacetic acid c / s c / s, c / s, cis / 1,2,3,4-cyclopentanetetracarboxylic acid 3-methyldecanoic acid boc-d-pipecolinic acid (+/-) - 2-endo-aminobicyclo [2.2.1] heptane 2-exo-7-anti-dicarboxylic acid 4-fluoro-3,3 ', 4,5,6-pentachló rftalanilic acid 4-fluoro-3-nitrobenzoic acid 2-methyl-3,4,6-pyridine tricarboxylic acid 3-methylsulfonylbenzoic acid 2- (hexadecylsulfonyl) benzoic acid isoindolin-1-one-2- (2-propionic acid) cis / s 5-norbornene-endo-2,3-dicarboxylic acid 9-fenylnonánová acid 2-fluoro-5- (trifluoromethyl) benzoic acid, 2, 4 ', 5, -trichlórglutaranilová

-180--180-

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · ···· • • ···· • • ·· t • · ·· • · · ·· t • · ·· • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

meta-sulfo-fenyl-gama kyselina kyselina alfa-metyl-2-tiofénakrylová kyselina siričitá kyselina 6-amino-1,3-naftaléndisulfónová kyselina 6,9,12,15-oktadekatetraénová kyselina 3-(2-etoxyfenyl)propiónová kyselina 3-karboxy-1,4-dimetyl-1 h-pyrol-2-octová kyselina rodanín-n-karboxylová fmoc-3-abz-oh kyselina 1 -amino-9,10-dihydro-4-hydroxy-9,10-dioxo-2-antracénsulfónová kyselina 4-bróm-1 -hydroxy-2-naftoová kyselina chelidónová kyselina n-(2-kyanofenyl)tetrachlórftalámová kyselina (4-chlórfenyltio)octová kyselina 4-oxo-1,9-nonándikarboxylová kyselina n-(3,4-dichlórfenyl)maleámová kyselina 4-acetoxy-3-metoxybenzoová kyselina 2-metoxy-5-metylbenzoová kyselina 2-hydroxy-3-(p-tolylimino-metyl)-benzoová kyselina 2-metyldodekánová kyselina formamidínsulfínová kyselina boc-4-fenyl-piperidín-4-karboxylová kyselina 4-hydroxy-alfa-fenylškoricová kyselina 4-etoxymetyl-benzoová kyselina 3,4-dichlórškoricová kyselina 3-(4-chlórfenyltio)tiofén-4-karboxylová kyselina (s)-(-)-2-hydroxy-3,3-dimetylmaslová kyselina /?-(3-brómfenyl)maleámová kyselina n-(3-chlór-4-metylfenyl)glutarámová kyselina 4-(p-tolyl)maslová kyselina 3-bróm-2-fluórbenzoová kyselina 4-nitro-1-naftalénoctovámeta-sulfo-phenyl-gamma alpha-methyl-2-thiophenacrylic acid sulfuric acid 6-amino-1,3-naphthalenedisulfonic acid 6,9,12,15-octadecatetraenoic acid 3- (2-ethoxyphenyl) propionic acid 3- carboxy-1,4-dimethyl-1H-pyrrole-2-acetic acid rhodanine-n-carboxylic acid fmoc-3-abz-oh 1-amino-9,10-dihydro-4-hydroxy-9,10-dioxo- 2-anthracenesulfonic acid 4-bromo-1-hydroxy-2-naphthoic acid chelidonic acid n- (2-cyanophenyl) tetrachlorophthalic acid (4-chlorophenylthio) acetic acid 4-oxo-1,9-nonanedicarboxylic acid n- (3,4) -dichlorophenyl) maleic acid 4-acetoxy-3-methoxybenzoic acid 2-methoxy-5-methylbenzoic acid 2-hydroxy-3- (p-tolylimino-methyl) -benzoic acid 2-methyldodecanoic acid formamidinesulfonic acid boc-4-phenyl-piperidine 4-carboxylic acid 4-hydroxy-alpha-phenyl cinnamic acid 4-ethoxymethyl-benzoic acid 3,4-dichlorocinnamic acid 3- (4-chlorophenylthio) thiophene-4-carboxylic acid (S) - (-) - 2-hydroxy-3,3-dimethylbutyric acid N- (3-bromophenyl) maleic acid n- (3-chloro-4-methylphenyl) glutaramic acid 4- (p-tolyl) Butyric acid 3-bromo-2-fluorobenzoic acid 4-nitro-1-naphthaleneacetic acid

-181 --181 -

• ·· • · • ··· • · · • ·· • · • ··· • · · • · • • • · • · • • • · ···· • · • · t · ···· • · • · t · ·· • · • · • · · · · • · • · • · · ·· ·· ·· ·· ·· · · • · • · ·· · ·

kyselina 6,7-dichlór-3-hydroxy-2-chinoxalínkarboxylová kyselina n-(3-hydroxy-fenyl)-5-nitro-ftalámová kyselina 2,4-furándikarboxylová kyselina n-benzoyl-8-hydroxyl-naftylamín-3,6-disulfónová kyselina 3-((s)-2-karboxypiperazín-4-yl)-propyl-1 -fosfónová kyselina 3,5-dibróm-2-furoová kyselina 5-fluórorotová kyselina (s)-(-)-metyljantárová kyselina 4-(2-chlóracetamido)benzoová kyselina 2'-metyl-3,4,5,6,6,-pentachlórftalanilová kyselina ftaloyl-d/-alanín kyselina 4,5,5,5-tetrafluór-4-heptafluórpropoxy-2-penténová kyselina [n-(4-etoxy-benzoylamino)-3-fenyl-akryloylamino)-octová kyselina d/-2-aminoazelainová kyselina 2,4,6-trimetoxybenzoová kyselina n-(2-kyanoacetyl)antranilová kyselina 3-metoxysalicylová kyselina n-(2,6-dietylfenyl)maleámová kyselina 2-acetamino-4-nitrobenzoová kyselina 3,3,4,4,4-pentachlór-maslová kyselina 4-hydroxyškoricová kyselina 3-o-metylgalová kyselina 3-izo-propylglutárová kyselina (+)-n-benzénsulfonylglutámová kyselina n-karbamyl-1-glutámová kyselina 6-nitro-1 h-benzoimidazol-5-karboxylová kyselina 2-fenylimidazo[1,2-a]pyridín-3-karboxylová kyselina 7-oxotetrakozánová kyselina 3,3-bis-(4-metoxy-fenyl)-akrylová kyselina (-)-2,3:4,6-di-o-izopropylidén-2-keto-1 -gulónová kyselina 4,-bróm-2'-chlórglutaranilová kyselina d-2-aminokorková6,7-Dichloro-3-hydroxy-2-quinoxaline carboxylic acid n- (3-hydroxy-phenyl) -5-nitro-phthalic acid 2,4-furanedicarboxylic acid n-benzoyl-8-hydroxyl-naphthylamine-3,6 Disulfonic acid 3 - ((s) -2-carboxypiperazin-4-yl) -propyl-1-phosphonic acid 3,5-dibromo-2-furoic acid 5-Fluoroorotic acid (s) - (-) - methylsuccinic acid 4 - (2-chloroacetamido) benzoic acid 2'-methyl-3,4,5,6,6 , -pentachlorophthalanic acid phthaloyl-d-alanine 4,5,5,5-tetrafluoro-4-heptafluoropropoxy-2-pentenoic acid [n- (4-ethoxy-benzoylamino) -3-phenyl-acryloylamino) -acetic acid d] -2-aminoazelaic acid 2,4,6-trimethoxybenzoic acid n- (2-cyanoacetyl) anthranilic acid 3-methoxysalicylic acid n - (2,6-diethylphenyl) maleic acid 2-acetamino-4-nitrobenzoic acid 3,3,4,4,4-pentachlorobutyric acid 4-hydroxycinnamic acid 3-o-methylgalic acid 3-isopropylglutaric acid (+ -n-benzenesulfonylglutamic acid n-carbamyl-1-glutamic acid 6-nitro-1H-benzoimidazole-5-carboxylic acid 2-phenylimidazo [1,2-a] pyridine-3-carboxylic acid 7-oxotetracosanoic acid 3,3-bis- (4- methoxy-phenyl) -acrylic acid (-) - 2,3: 4,6-di-o-isopropylidene-2-keto-1 -gulónová acid 4-bromo-2 ' chlórglutaranilová d-2-aminosuberic

-182--182-

• · · • · • ··· • · · • · • ··· • · · · · · • · · Φ · · • · · · · · • · · Φ · · • · · • · ·· Φ · · • · · • · ·· Φ · · • · · · • · · · • · ·· • · ·· ·· ·· ·· ··

kyselina fmoc-1-1,2,3,4-tetrahydroizochulolín-7-karboxylová d/-o-fosfoserín kyselina 4-etoxyfenylfosfónová kyselina 4-(4-(4-karboxy-fenoxy)-benzoyl)-ftalová kyselina 2,7-dimetylimidazo[1,2-a]pyridín-3-karboxylová kyselina 1,4-dihydroxy-2-naftoová kyselina (rs)-jasmonová kyselina karboxyetyl-gama-aminomaslová kyselina 2-chlór-4-fluórfenyloctová kyselina d/-dihydroorotová kyselina c/s-n-(hexadecyl)hexahydroftalámová kyselina 3-(1h-indol-3-yl)-2-(4-metoxy-benzoylamino)-propiónová kyselina 9-tiastearová kyselina 6-metyl-azulén-2-karboxylová kyselina 2,,3'-dichlórglutaranilová kyselina 3-(2-jódfenyl)propiónová kyselina 5-metyl-4-nitroizoftalová kyselina 5-chlórbenzofurán-2-karboxylová kyselina 1 -(4-chlórfenyl)-1 -cyklohexánkarboxylová kyselina 5-chlór-2-fluórbenzoová kyselina 7-hydroxy-1,3,4-triazindolizín-6-karboxylová kyselina 1-pyréndodekánová kyselina 3-(4-chlórbenzoyl)-2-(2-chlór-6-fluórfenyl)propiónová kyselina 2-chlór-6-metylbenzoová kyselina n-(4-bróm-2-metylfenyl)maleámová kyselina vinylfosfónová kyselina 4-(2-o-tolyloxy-acetylamino)-benzoová kyselina 3-ŕerc-butyl-6-metylsalicylová karboxypyrazolón kyselina 3-nitroftalová kyselina 2-bróm-4-hydroxy-5-metoxy-fenyloctová kyselina undekánováfmoc-1-1,2,3,4-tetrahydroisoquinoline-7-carboxylic acid d-o-phosphoserine 4-ethoxyphenylphosphonic acid 4- (4- (4-carboxy-phenoxy) -benzoyl) -phthalic acid 2,7 -dimethylimidazo [1,2-a] pyridine-3-carboxylic acid 1,4-dihydroxy-2-naphthoic acid (Rs) -asonic acid carboxyethyl-gamma-aminobutyric acid 2-chloro-4-fluorophenylacetic acid d -dihydroorotic acid c / sn (hexadecyl) hexahydroftalámová 3- (1H-indol-3-yl) -2- (4-methoxy-benzoylamino) -propionic acid 9-tiastearová 6-methyl-azulene-2-carboxylic acid 2, 3'-Dichloroglutaranilic acid 3- (2-iodophenyl) propionic acid 5-methyl-4-nitroisophthalic acid 5-chlorobenzofuran-2-carboxylic acid 1- (4-chlorophenyl) -1-cyclohexanecarboxylic acid 5-chloro-2-fluorobenzoic acid 7-hydroxy-1,3,4-triazindolizine-6-carboxylic acid 1-pyrene dodecanoic acid 3- (4-chlorobenzoyl) -2- (2-chloro-6-fluorophenyl) propionic acid 2-chloro-6-methylbenzoic acid n- (4-bromo-2-methylphenyl) maleic acid vinylphosphonic acid 4- (2-o-tolyloxyacetylamino) -benzoic acid 3-tert-butyl-6-methylsalicylic carboxypyrazolone 3-nitrophthalic acid 2-bromo-4 -hydroxy-5-methoxy-phenylacetic acid undecanoic acid

-183--183-

• ·· • ·· ·· · · ···· ···· ·· · ·· · • a • a • · • · e a · · e a · · • ··· • ··· • · • · • a · • a · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 1,3-diamino-2-hydroxypropán-n,n,n’,/7-tetraoctová kyselina pent-3-énoylamino-octová kyselina 2,3-dimetylmaslová kyselina S’^'-dimetyl-SAS.e-tetrachlórftalanilová kyselina 2-hydroxyamino-3-metyl-pentánová kyselina n-(4'-(toluén-4-sulfonylamino)-bifenyl-4-yl)-sukcínamová kyselina 4-(/?-(2-oxo-1-(toluén-4-sulfonyl)-propylidén)-hysrazino)-benzoová kyselina 11-(fenyltio)undekánová kyselina 2-hydroxyamino-2-metyl-propiónová kyselina 14,15-epoxy-(5z,8z, 11 z)-eikozatriénová kyselina 2-fenoxymetylbenzoová kyselina (3-ho-3-ph-4h-4h-1-tia-3a,7-diaza-cyklopenta(a)pentalén-2-yl)-octová kyselina 4*-sulfamoylglutaranilová kyselina [[2-(3,4-dimetoxy-fenyl)-etyl]-(toluén-4-sulfonyl)-amirio]-octová kyselina 2-[4-(trifluórmetyl)fenyltio]octová kyselina 15-brómpentadekánová kyselina 2-hexyl-3-(2-metoxy-fenyl)-akrylová kyselina (trimetylsilyl)octová kyselina 2-(4-hydroxyfenyl)propiónová kyselina pyrol-3-karboxylová kyselina n-(3-indolylacetyl)-d/-asparágová kyselina fenyl(3,5-xylyl)fosfínová kyselina 3*,4'-dichlórsukcínanilová kyselina 1,6-dihydro-6-oxo-1,2,5-trimetyl-3-pyridínkarboxylová kyselina 1 -(4-izopropylfenyl)-6-metyl-4-oxo-1,4-dihydro-3-pyridínkarboxylová kyselina 3-chlór-4-hydroxymandlová kyselina 3-(karboxymetyltio)propiónová kyselina 3-(3,4-dimetoxyfenyl)-2-formylamino-propiónová kyselina 3-(p-metoxyfenyl)-2-fenylpropiónová kyselina c/s-11-eikozénová kyselina 4-(ac-(5-nitro-1,3-dioxo-1,3-dihydro-izoindol-2-ylmetyl)-amino)-benzoová kyselina 5,-izopropyl-2'-metyl-3,4,5,6-tetrachlórftalanilová1,3-diamino-2-hydroxypropane-n, n, n ', 7-tetraacetic acid pent-3-enylamino-acetic acid 2,3-dimethylbutyric acid S', 4'-dimethyl-SAS.e-tetrachlorophthalanic acid 2-hydroxyamino-3-methyl-pentanoic acid n- (4 '- (toluene-4-sulfonylamino) -biphenyl-4-yl) -succinamic acid 4 - (R - (2-oxo-1- (toluene-4)) (sulfonyl) -propylidene) -hysrazino) -benzoic acid 11- (phenylthio) undecanoic acid 2-hydroxyamino-2-methyl-propionic acid 14,15-epoxy- (5z, 8z, 11z) -eicosatrienoic acid 2-phenoxymethylbenzoic acid (3-ho-3-ph-4h-4h-1-thia-3α, 7-diaza-cyclopenta (a) pentalen-2-yl) -acetic acid 4'-sulfamoylglutaranilic acid [[2- (3,4- dimethoxy-phenyl) -ethyl] - (toluene-4-sulfonyl) -amirio] -acetic acid 2- [4- (trifluoromethyl) phenylthio] acetic acid 15-bromopentadecanoic acid 2-hexyl-3- (2-methoxy-phenyl) -acrylic acid (trimethylsilyl) acetic acid 2- (4-hydroxyphenyl) propionic acid pyrrole-3-carboxylic acid n- (3-indolylacetyl) -d-aspartic acid phenyl (3,5-xylyl) phosphinic acid 3 *, 4'-dichlorosuccinilic acid 1,6-dihydro-6-oxo-1,2,5-trimethyl-3-pyridinecarboxylic acid 1- (4-isopropylphenyl) -6 methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid 3-chloro-4-hydroxy-butyric acid 3- (carboxymethylthio) propionic acid 3- (3,4-dimethoxyphenyl) -2-formylamino-propionic acid 3- (p-Methoxyphenyl) -2-phenylpropionic acid cis-11-eicosenoic acid 4- (ac- (5-nitro-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl) amino) - benzoic acid, 5-isopropyl-2-methyl-3,4,5,6-tetrachlórftalanilová

-184 --184 -

• ·· • ·· ·· · · ···· ···· ·· · ·· · • · • · • · ·· • · ·· • ··· • ··· • · · • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 5-bróm-2-fluórbenzoová kyselina tetrahydro-2-furoová kyselina (r)-(-)-alfa-(((4-etyl-2,3-dioxo-1-piperazinyl)karbonyl)amino)benzénoctová kyselina (trans,trans)-abscisová ([S]-5-[ 1 -hydroxy-2,6,6-trimetyl-4-oxocyklohex-2-én-5-Bromo-2-fluorobenzoic acid tetrahydro-2-furoic acid (R) - (-) - alpha - (((4-ethyl-2,3-dioxo-1-piperazinyl) carbonyl) amino) benzeneacetic acid (trans , trans) -abscis ([S] -5- [1-hydroxy-2,6,6-trimethyl-4-oxocyclohex-2-ene-

1-yl]-3-metyl-[2z,4e]pentadiénová) kyselina 3-chlórpropiónová kyselina (-)-mentoxyoctová kyselina 4'-butylglutaranilová kyselina 4'-hydroxyglutaranilová kyselina 4-oxo-2,3,4-trifenylmaslová kyselina 1,2,4-butántrikarboxylová kyselina c/s-3-hexénová kyselina allo-gibberová (C18H20O3) kyselina 2-(1,3-dioxo-1,2,3,4-tetrahydro-2-izochinolinyl)octová kyselina 4-decyloxybenzoová kyselina (3-et-9,10-dimetoxy-4-oxo-pyrido(2,1 -a)izochinolín-2-yl)-octová kyselina (z)-2-(2-chlóracetamido)-alfa-(metoxyimino)-4-tiazoloctová kyselina 2-metoxy-9-oxo-6,7,8,9-tetrahydro-5h-benzocykloheptén-6-karboxylová kyselina 4-(3-(2-fenoxyacetyl)-2-tioureido)benzoová kyselina 9,10-epoxyoktadekánová kyselina d/-beta-fenylmliečna kyselina imidazo[2,1 -b]benzotiazol-2-karboxylová kyselina 3-metoxy-4-nitrobenzoová kyselina 2,4-difenyl-furán-3-karboxylová kyselina 1,2-dihydro-2-metyl-1-oxo-3-izochinolínmaslová kyselina 2-(cyklohexánkarbonyl-amino)-benzoová kyselina 2,3-difenyl-jantárová kyselina cis-7,10,13,16,19-dokoza-penténová kyselina 3,3’-tolidín-5-sulfónová kyselina 2-metoxy-1-naftoová kyselina 3-(2-metoxyfenyl)propiónová kyselina n-(4-fluórfenyl)malonámová1-yl] -3-methyl- [2z, 4e] pentadienoic acid 3-chloropropionic acid (-) - Mentoxyacetic acid 4'-butylglutaranilic acid 4'-hydroxyglutaranilic acid 4-oxo-2,3,4-triphenylbutyric acid 1 2,4-butanetricarboxylic acid cis-3-hexenoic allo-gibberic acid (C18H20O3) 2- (1,3-dioxo-1,2,3,4-tetrahydro-2-isoquinolinyl) acetic acid 4-decyloxybenzoic acid (3-Et-9,10-dimethoxy-4-oxo-pyrido (2,1-a) isoquinolin-2-yl) -acetic acid (z) -2- (2-Chloroacetamido) -alpha- (methoxyimino) 4-thiazoleacetic acid 2-methoxy-9-oxo-6,7,8,9-tetrahydro-5h-benzocycloheptene-6-carboxylic acid 4- (3- (2-phenoxyacetyl) -2-thioureido) benzoic acid 9, 10-epoxyoctadecanoic acid d-beta-phenyl-lactic acid imidazo [2,1-b] benzothiazole-2-carboxylic acid 3-methoxy-4-nitrobenzoic acid 2,4-diphenyl-furan-3-carboxylic acid 1,2-dihydro 2-Methyl-1-oxo-3-isoquinolinebutyric acid 2- (cyclohexanecarbonylamino) -benzoic acid 2,3-diphenyl-succinic acid cis-7,10,13,16,19-docosopentenoic acid 3,3'-tolidine-5-sulfonic acid 2-methoxy-1-naphthoic acid 3- (2-methoxyphenyl) propionic acid n- (4) fluorophenyl) -malonamic

-185--185-

• M • · • ··· • M • · • ··· ·· • · • · ·· • · • · ···· • • ···· • • • e · • · ·« • 9 9 • e · • · · « • 9 9 ·· ·· ·· ·· ·· · · • · • · • · · · • · · ·

kyselina -(-)-perilová kyselina gama-1 -glutamyl-1 -glutámová kyselina tartronová kyselina 4-benzyloxyfenyloctová kyselina n-(3,5,5)-trimetylcyklohexyl)maleámová kyselina (S.S-dimetyl-S-oxo-cyklohexylidénaminoJ-octová kyselina d-treo-4-fluórglutámová kyselina (z)-styryltiopropiónová kyselina beta-maleimidopropiónová kyselina chlórfumárová kyselina 4-chlór-3-nitro-5-sulfónamidobenzoová kyselina fenylfosforečná kyselina 1,2-etyléndifosfónová kyselina fmoc-(3-aminometyl)-benzoová kyselina boc-d-beta-aminomaslová kyselina 3-(4-hydroxyfenyl)propiónová kyselina 4,4’-(trichlórmetyl-metylén)-disalicylová kyselina (4-formyl-3-metoxy-fenoxy)octová kyselina (4-nitro-fenyl)-fosfónová kyselina (1 rs)-ŕrans-permetrinová kyselina 4-izobutylškoricová kyselina 3,4-dibrómbenzoová kyselina 4'-metyl-3,-nitrosukcínanilová kyselina ftalámová kyselina 5-chlórsulfonyl-2-hydroxybenzoová kyselina 3,4,5-tribrómbenzoová kyselina 2'-nitromaleanilová kyselina d-(-)-alfa-azido-fenyloctová kyselina 2,2-dihydroxy-3,3,3-trichlórpropiónová kyselina 3’,4'-dimetylglutaranilová kyselina 2,6-dichlórškoricová kyselina 3-nitrohipurová- (-) - Perilic acid gamma-1-glutamyl-1-glutamic acid tartronic acid 4-benzyloxyphenylacetic acid n- (3,5,5) -trimethylcyclohexyl) maleic acid (SS-dimethyl-S-oxo-cyclohexylidenamino) acetic acid d-threo-4-fluoroglutamic acid (z) -styrylthiopropionic acid beta-maleimidopropionic acid chlorofumaric acid 4-chloro-3-nitro-5-sulfonamidobenzoic acid phenylphosphoric acid 1,2-ethylenediphosphonic acid fmoc- (3-aminomethyl) -benzoic acid boc-d-beta-aminobutyric acid 3- (4-hydroxyphenyl) propionic acid 4,4 '- (trichloromethyl-methylene) -disalicylic acid (4-formyl-3-methoxy-phenoxy) acetic acid (4-nitro-phenyl) ) phosphonic acid (1 RS) -trans-4-permethrin acid izobutylškoricová 3,4-dibromobenzoic acid, 4'-methyl-3, -nitrosukcínanilová acid phthalamic acid 5-chlorosulfonyl-2-hydroxybenzoic acid, 3,4,5-tribromobenzoic 2'-nitromaleanilic acid d- ( -) - alpha-azido-phenylacetic acid 2,2-dihydroxy-3,3,3-trichloropropionic acid 3 ', 4'-dimethylglutaranilic acid 2,6-dichlorocinnamic acid 3-nitrohipuric acid

-186--186-

• ·· • · • ··· • ·· • · • ··· • · • · • · • · • · • · ···· • e ···· • e ·· · • · · · • · 9 ·· · • · 9 • c ·· • c ·· ·· · · • · • · ·· ·· ·· ··

kyselina 3,4-dimetoxy-6-nitroškoricová kyselina boc-1-indolín-2-karboxylová kyselina 2-chlór-4-fluórbenzoová kyselina 10-oxoundekánová kyselina (3- metyl-5-nitro-fenyl)-fosfónová kyselina 3-(1,1,2,3,3,3-hexafluór-propyl)-adamantán-1-karboxylová kyselina tricyklo(8.2.2.2(4,7))hexadeka-hexaén-2-karboxylová kyselina 3,4-dimetoxybenzoová kyselina 4-bróm-3,5-dihydroxybenzoová kyselina o-(2,6-dichlóranilíno)benzoová kyselina n-karbamyl-alfa-amino-izomaslová n-1-trifenylmetyl-deamino-histidín kyselina 4-fenoxybenzoová kyselina 4-(3-fluór-4-hydroxyfenyl)maslová kyselina 4-etyloxybifenyl-4'-karboxylová kyselina (s)-(+)-3-(benzyloxykarbonyl)-5-oxo-4-oxazolidínpropiónová kyselina 2-(3-karboxymetánsulfonyl-benzoylamino)-benzoová kyselina 2-acetoxyškoricová kyselina 4-(3,4-dimetylfenyl)maslová kyselina 2-(trifluórmetyl)fenyloctová kyselina 5-[3-(2-metoxykarbonyltienyl)]-2-furoová kyselina 4-hydroxy-1 -metyl-2-oxo-1,2-dihydro-chinolín-3-sulfónová kyselina 4-(4-hexadecytfenyl)maslová kyselina 10-fluór-1-oxo-5,6-dihydro-1h-azepino[3,2,1-ij)chinolín-2-karboxylová kyselina 3-(4-metylbenzyloxy)tiofén-2-karboxylová kyselina 2-(2-íerc-butoxykarbonylamino-3-ph-propionylamino)-4-metylsulfanyl-maslová3,4-dimethoxy-6-nitrocinnamic acid boc-1-indoline-2-carboxylic acid 2-chloro-4-fluorobenzoic acid 10-oxoundecanoic acid (3-methyl-5-nitro-phenyl) -phosphonic acid 3- ( 1,1,2,3,3,3-hexafluoro-propyl) -adamantane-1-carboxylic acid tricyclo (8.2.2.2 (4,7)) hexadeca-hexaene-2-carboxylic acid 3,4-dimethoxybenzoic acid 4- bromo-3,5-dihydroxybenzoic acid o- (2,6-dichloroanilino) benzoic acid n-carbamyl-alpha-amino-isobutyric acid n-1-triphenylmethyl-deamino-histidine 4-phenoxybenzoic acid 4- (3-fluoro-4) 4-ethyloxybiphenyl-4'-carboxylic acid (s) - (+) - 3- (benzyloxycarbonyl) -5-oxo-4-oxazolidinepropionic acid 2- (3-carboxymethanesulfonyl-benzoylamino) -benzoic acid 2- acetoxycinnamic acid 4- (3,4-dimethylphenyl) butyric acid 2- (trifluoromethyl) phenylacetic acid 5- [3- (2-methoxycarbonylthienyl)] - 2-furoic acid 4-hydroxy-1-methyl-2-oxo-1, 2-Dihydro-quinoline-3-sulfonic acid 4- (4-Hexadecylphenyl) butyric acid 10-fluoro-1-oxo-5,6-dihydro-1H-azepino [3,2,1-ij] quinoline-2-carboxylic acid 3- (4-methylbenzyloxy) thiophene-2- 2- (2-tert-butoxycarbonylamino-3-ph-propionylamino) -4-methylsulfanyl-butyric acid

5-sulfosalicylidén-anilin kyselina 5-(2,4-dichlórbenzoyl)tiofén-2-octová kyselina 4-metylpentánová kyselina (4-chlór-2-metylfenoxy)octová kyselina 2-(hexadecyloxy)-p-anízová5-Sulfosalicylidene-aniline 5- (2,4-dichlorobenzoyl) -thiophene-2-acetic acid 4-methylpentanoic acid (4-chloro-2-methylphenoxy) acetic acid 2- (hexadecyloxy) -p-anisic acid

-187--187-

• ·· • ·· b e b e BBBB BBBB BB B BB B • · • · B B B · · · B · · · • BBB • BBB B B B B BBB BBB • B BB • B BB • B • B B · B · BB BB BB BB

kyselina glukónová kyselina (1 s.3s)-1 -etyl-2,3,4,9-tetrahydro-1 h-pyrido[3,4-b]indol-3-karboxylová kyselina 9,10-dihydro-12-fenyl-9,10-etanoantracén-11-karboxylová kyselina 5-nitrosalicylová kyselina 2,3,3-trifenylpropiónová kyselina 3-benzoyl-izonikotínová kyselina 2-nitrofenylpyrohroznová kyselina 13(s)-hydroxyoktadeka-9z,11e-diénová kyselina 2,3-difluórbenzoová kyselina 2-[3-(n-izobutyryl-hydrazíno)-3-oxo-propionylamino]-benzoová kyselina fmoc-d-2-aminomaslová kyselina 2-hydroxyškoricová kyselina 2,6-dichlór-3,5-dinitrobenzoová kyselina s-4-hydroxymandlová kyselina (4,5-difenylimdazol-2-yltio)octová kyselina 6-hydroxy-2-(metyltio)-4-pyrimidínkarboxylová kyselina 3-(1-naftoxy)propiónová kyselina alfa-chlór-5-metyl-1,3-adamantándioctová kyselina 2-fenoxypropiónová kyselina 4,4-dimetyl-itakónová kyselina alfa.beta-dibrómhydroškoricová kyselina n-naftalén-2-yl-5-nitro-ftalámová kyselina 3-bróm-4-metylbenzoová kyselina 2-karboxybenzénpropánová kyselina glycy l-glycy 1-1 -glutámová kyselina ζ-1-asparágová kyselina 4-karbetoxy-3,5-dimetoxybenzoová kyselina 1,6-difenyl-1,3,5-hexatrién-4'-propiónová kyselina 4-(p-jódfenyl)maslová kyselina 9-fluorenón-2,7-dikarboxylová kyselina syringová kyselina hexafluórglutárovágluconic acid (1 s 3s) -1-ethyl-2,3,4,9-tetrahydro-1H-pyrido [3,4-b] indole-3-carboxylic acid 9,10-dihydro-12-phenyl -9,10-ethanoanthracene-11-carboxylic acid 5-nitrosalicylic acid 2,3,3-triphenylpropionic acid 3-benzoyl-isonicotinic acid 2-nitrophenylpyruvic acid 13 (s) -hydroxyoctadeca-9z, 11e-dienoic acid 2,3- Difluorobenzoic acid 2- [3- (n-isobutyryl-hydrazino) -3-oxo-propionylamino] -benzoic acid fmoc-d-2-aminobutyric acid 2-Hydroxycinnamic acid 2,6-dichloro-3,5-dinitrobenzoic acid s- 4-hydroxy-butyric acid (4,5-diphenylimidazol-2-ylthio) acetic acid 6-hydroxy-2- (methylthio) -4-pyrimidinecarboxylic acid 3- (1-naphthoxy) propionic acid alpha-chloro-5-methyl-1, 3-adamantanediacetic acid 2-phenoxypropionic acid 4,4-dimethyl-itaconic acid alpha-beta-dibromocinnamic acid n-naphthalen-2-yl-5-nitro-phthalic acid 3-bromo-4-methylbenzoic acid 2-carboxybenzenepropano Glycic acid 1-Glycic acid 1-1-glutamic acid ζ-1-aspartic acid 4-Carbethoxy-3,5-dimethoxybenzoic acid 1,6-Diphenyl-1,3,5-hexatriene-4'-propionic acid 4- ( p-iodophenyl) butyric acid 9-fluorenone-2,7-dicarboxylic acid syringic acid hexafluoroglutaric acid

-18899 ··· • ·· kyselina 2-nitro-5-tiokyanátobenzoová kyselina (s)-(-)-2-chlórhexánová kyselina (r)-(+)-metyljantárová kyselina 4,5-dihydro-1-metánsulfonylbenzo[c]tiofén-3-karboxylová kyselina 2-metyl-2-hexénová kyselina 4-(o-jódfenyl)maslová kyselina alfa-kyano-beta-5-dimetyl-2-(metyltio)škoricová kyselina 3,3'-dimetyl-bifenyl-2,2'-dikarboxylová kyselina n.n-anilíndioctová kyselina 4-(4-chlór-benzénsulfonyl)-4-kyano-heptándiová kyselina p-acetaminobenzénsulfínová kyselina d/-beta-metylasparágová kyselina alfa-acetylmandlová kyselina 3-(5-nitro-2-furyl)akrylová kyselina S'.S'-dimetoxymaleanilová kyselina 3,5-dinitro-p-toluylová kyselina 4’-metyl-2l-nitromaleanilová kyselina 2-brómfenoxy-octová kyselina 2-chlór-izomaslová kyselina 3,5-dibrómlevulová kyselina c/s-13,16-dokozadiénová kyselina 4'-acetylftalanilová kyselina 2-chlórhipurová kyselina 4-(4'-hydroxyfenyl)benzoová kyselina 1-naftoová kyselina 12(s)-hydroxy-16-heptadecínová kyselina (2-cyklopentén-1 -yl)-malónová kyselina 2'-metoxyftalanilová kyselina 3'-metyl-3,4,5,6-tetrachlórftalanilová kyselina 5-doxyl-stearová kyselina 3,4-xylylfosfónová kyselina (2-sek-butyl-fenoxy)-octová • ·· ·· ···· ·· ··· · · ···· • ··· · · · · ·-18899 ··· • ·· 2-Nitro-5-thiocyanato-benzoic acid (s) - (-) - 2-chlorohexanoic acid (r) - (+) - methylsuccinic acid 4,5-dihydro-1-methanesulfonylbenzo [c ] Thiophene-3-carboxylic acid 2-methyl-2-hexenoic acid 4- (o-iodophenyl) butyric acid alpha-cyano-beta-5-dimethyl-2- (methylthio) cinnamic acid 3,3'-dimethyl-biphenyl- 4- (4-Chloro-benzenesulfonyl) -4-cyano-heptanedioic acid p-acetaminobenzenesulfonic acid 2,2'-dicarboxylic acid n-aniline-di-acetic acid α-acetyl-butyric acid alpha-acetyl-butyric acid 3- (5-nitro-2) furyl) acrylic acid S'.S' dimetoxymaleanilová-3,5-dinitro-p-toluic acid, 4'-methyl-2 l -nitromaleanilová acid 2-bromophenoxy-acetic acid 2-chloro-isobutyric acid, 3,5-dibrómlevulová cis-13,16-docosadienoic acid 4'-acetylphthalanilic acid 2-chlorohippuric acid 4- (4'-hydroxyphenyl) benzoic acid 1-naphthoic acid 12 (s) -hydroxy-16-heptadecinic acid (2-Cyclopenten-1-yl) -malonic acid 2'-methoxyphthalanic acid 3'-methyl-3,4,5,6-tetrachlorophthalanic acid 5-doxyl-stearic acid 3,4-xylylphosphonic acid (2-sec- Butyl-phenoxy) -acetic • ··· ···············

-189kyselina adamantán-1 -yl-fosfónová kyselina 1 -(2,4-dichlórfenyl)-4-karboxytriazol-octová kyselina 2,6-dichlór-5-fluór-3-pyridínkarboxylová kyselina tridekánová kyselina (2-etylfenyl)fosfónová kyselina (s)-2-fluór-2-metylhexánová kyselina 3-hydroxy-1 -adamantánoctová kyselina 3-(4-chlórbenzoyl)-2-(2,3-dichlórfenyl)propiónová kyselina 2-[(3-karboxy-propyl)-(toluén-4-sulfonyl)-amino]-4-chlór-benzoová kyselina (2,6-xylyl)fosfónová kyselina 1 -aminoantrachinón-2-sulfónová kyselina 5-(2,5-dimetoxy-fenyl)-5-oxo-pentánová kyselina 4-(4-metyl-2,6-dinitro-fenylamino)-maslová kyselina 3,5-dichlórbenzoová kyselina 3-sulfobenzoová kyselina bis(fenacyl)octová kyselina (3-benzyl-fenyl)octová kyselina (1 r,3s)-1-aminocyklopentán-1,3-dikarboxylová kyselina cbz-d-1,2,3,4-tetrahydroizochinolín-3-karboxylová kyselina p-fenolsulfónová kyselina perhydrocyklobuta(1,2:3,4)dicyklopentén-2,5-dikarboxylová kyselina 2-(2-oxo-1,2-dihydro-indol-3-ylidénamino)-benzoová kyselina nonadekánová kyselina 4-aminoftalová kyselina 4-acetylmaslová kyselina chaulmoogrová kyselina 3-(n-hexadecylkarbamoyl)-5-norbornén-2-karboxylová kyselina fenylfosfónová kyselina n-propylmaleámová kyselina benzyloxykarbonyl-2-aminobutánová (kyselina 1-z-2-aminomaslová) kyselina 1 -(4-metoxyfenyl)-1 -cyklopropánkarboxylová kyselina 3-chlórdodekándiová-189 adamantan-1-yl-phosphonic acid 1- (2,4-dichlorophenyl) -4-carboxytriazole-acetic acid 2,6-dichloro-5-fluoro-3-pyridinecarboxylic acid tridecanoic acid (2-ethylphenyl) phosphonic acid ( s) -2-fluoro-2-methylhexanoic acid 3-hydroxy-1-adamantaneacetic acid 3- (4-chlorobenzoyl) -2- (2,3-dichlorophenyl) propionic acid 2 - [(3-carboxypropyl) - ( toluene-4-sulfonyl) amino] -4-chloro-benzoic acid (2,6-xylyl) phosphonic acid 1-aminoanthraquinone-2-sulfonic acid 5- (2,5-dimethoxyphenyl) -5-oxo-pentanoic acid 4- (4-methyl-2,6-dinitro-phenylamino) -butyric acid 3,5-dichlorobenzoic acid 3-sulfobenzoic acid bis (phenacyl) acetic acid (3-benzylphenyl) acetic acid (1 r, 3s) 1-aminocyclopentane-1,3-dicarboxylic acid cbz-d-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid p-phenolsulfonic acid perhydrocyclobutane (1,2: 3,4) dicyclopentene-2,5-dicarboxylic acid 2- (2-oxo-1,2-dihydro-indol-3-ylideneamino) -benzic acid oic acid nonadecanoic acid 4-aminophthalic acid 4-acetylbutyric acid chaulmogronic acid 3- (n-hexadecylcarbamoyl) -5-norbornene-2-carboxylic acid phenylphosphonic acid n-propylmaleamic acid benzyloxycarbonyl-2-aminobutanoic acid (1-z-2-aminobutyric acid) ) 1- (4-Methoxyphenyl) -1-cyclopropanecarboxylic acid 3-chlorododecanedioic acid

-190--190-

8 88 8 88 8 8 8 8 8888 8888 88 8 88 8 8 8 8 8 8 8 8 8 8 8 8 8 88 8 8 88 • 888 • 888 8 8 8 8 8 8 8 8 8 8 88 88 88 88 88 88 8 8 8 8 M 88 M 88

kyselina (2-imino-4-oxo-tiazolidín-5-yl)-octová kyselina etyléndiamin-n,n’-di-octová-n,n’-di-alfa-propiónová kyselina 2-hydroxy-2-trifluórmetyl-dec-4-énová kyselina 3-nitro-5-sulfosalicylová kyselina 9-hydroxy-9h-fluorén-1 -karboxylová kyselina n-m-tolylftalámová kyselina fenyljantárová kyselina (s)-(-)-2-metylglutárová kyselina 4-fluór-3-metoxybenzoová kyselina 3,5-pyrazoldikarboxylová kyselina 2,3-dibróm-3-(p-chlórfenyl)propiónová kyselina 1,6-difenyl-1,3,5-hexatrién-4'-octová kyselina 2h-(1,2,4)-triazol-3-karboxylová kyselina 9,10-dihydro-9,10-dioxo-2,3-antracéndikarboxylová kyselina 4-izopropylfenyloctová kyselina 2-brómtetradekánová kyselina 2-(3,5-di-ŕerc-butyl-benzoylamino)-benzoová kyselina valérová kyselina 2-fenyl-1 h-imidazol-4,5-dikarboxylová kyselina 2-hydroxyoktadekánová kyselina bisakrylamidooctová kyselina 4,-metyl-3'-nitroftalanilová kyselina 2-fosfonopropiónová kyselina chlóracetyl-1 -gama-glu-p-aminobenzoová kyselina 3-etoxyškoricová kyselina 3-metyl-3h-imidazo(415-b)pyridín-2-sulfónová kyselina 7-chlór-2,2,3,34,4,5,5,6,6,7,7-dodekafluórheptánová kyselina 3,5-dichlór-4-hydroxybenzoová kyselina 3-(3,5-dimetyl-fenyl)-3-metyl-maslová kyselina 3,5-dibróm-4-hydroxybenzoová kyselina tricyklo(8.2.2.2(4,7))hexadeka-hexaén-5-yl-octová kyselina alfa-kyanoškoricová(2-Imino-4-oxo-thiazolidin-5-yl) -acetic acid ethylenediamine-n, n'-di-acetic acid, n'-di-alpha-propionic acid 2-hydroxy-2-trifluoromethyl-dec 4-enoic acid 3-nitro-5-sulfosalicylic acid 9-hydroxy-9h-fluorene-1-carboxylic acid nm-tolylphthalic acid phenylsuccinic acid (s) - (-) - 2-methylglutaric acid 4-fluoro-3-methoxybenzoic acid 3,5-pyrazoleicarboxylic acid 2,3-dibromo-3- (p-chlorophenyl) propionic acid 1,6-diphenyl-1,3,5-hexatriene-4'-acetic acid 2h- (1,2,4) -triazole-3-carboxylic acid 9,10-dihydro-9,10-dioxo-2,3-anthracenedicarboxylic acid 4-isopropylphenylacetic acid 2-bromotetradecanoic acid 2- (3,5-di-tert-butyl-benzoylamino) -benzoic acid acid, valeric acid, 2-phenyl-1H-imidazole-4,5-dicarboxylic acid 2-hydroxyoctadecanoic acid, bisacrylamidoacetic acid, 4-methyl-3 &apos; nitroftalanilová acid, 2-phosphonopropionic acid chloroacetyl-1-gamma-glu-p-aminobenzoic acid 3 3-methyl-3h-imidazo (4 1 5-b) pyridine-2-sulfonic acid ethoxycinnamic acid 7-chloro-2,2,3,34,4,5,5,6,6,7,7-dodecafluoroheptanoic acid 3,5-Dichloro-4-hydroxybenzoic acid 3- (3,5-dimethylphenyl) -3-methylbutyric acid 3,5-dibromo-4-hydroxybenzoic acid tricyclo (8.2.2.2 (4,7)) hexadeca -hexaen-5-yl-acetic acid alpha-cyano cinnamic acid

-191 --191 -

• · · • · • ··» • · · • · • ·· » • · • · • · • · • · • · ···· • • ···· • • ·· · • · · · • · · ·· · • · · ·· ·· ·· ·· ·· · · • · • · ·· ·· ·· ··

kyselina 2-brómizovalérová kyselina 3-chlór-benzo(b)tiofén-2-karboxylová kyselina 7-hydroxy-4-metylkumarín-3-octová kyselina n-(4,6-dimetylpyrimidin-2-yl)-n-metyl-4-aminobenzoová kyselina metándisulfónová kyselina izatín-n-octová kyselina (2-benzyloxy-3-metoxy-fenyl)-octová kyselina 3-kyanobenzoová kyselina 2,5-difluórfenyloctová kyselina citronelová kyselina ximeninová kyselina 5-chlór-2,6-dimetoxy-5-nitrobenzoová kyselina 3-metylsalicylová kyselina pyrofosforečná kyselina xantén-9-karboxylová kyselina 7-metoxybenzofurán-2-karboxylová kyselina 7,4,5-trichlórbenzénsulfónová kyselina m-jódfenyloctová kyselina 2-benzoyl-3,4,5,6-tetrachlórbenzoová kyselina fenyltiohydantoínová kyselina myrist-elaidová kyselina 4*-(etoxykarbonyl)sukcínanilová kyselina (r)-(-)-2,2-dimetyl-5-oxo-1,3-dioxolán-4-octová kyselina 4-acetylbenzoová kyselina 4-amino-2-nitrobenzoová kyselina 2-(2,5-dimetylbenzoyl)-akrylová kyselina gama-oxo-2-naftalénmaslová kyselina 2-bróm-3-chlórbenzoová kyselina p-toluénsulfinová kyselina 1-benzyl-1,2,3-triazol-4,5-dikarboxylová kyselina 12(s),20-dihydroxyeikoza-5z,8z, 10c, 14z-tetraénová kyselina 7-benzoylheptánová • ·· ·· ···· ·· ··· · · · · · · • ··· · · · · ·2-Bromoisovaleric acid 3-chloro-benzo (b) thiophene-2-carboxylic acid 7-hydroxy-4-methylcoumarin-3-acetic acid n- (4,6-dimethylpyrimidin-2-yl) -n-methyl-4 -aminobenzoic acid methanesulfonic acid isatin-n-acetic acid (2-benzyloxy-3-methoxyphenyl) -acetic acid 3-cyanobenzoic acid 2,5-difluorophenylacetic acid citric acid ximenic acid 5-chloro-2,6-dimethoxy-5 -nitrobenzoic acid 3-methylsalicylic acid pyrophosphoric acid xanthene-9-carboxylic acid 7-methoxybenzofuran-2-carboxylic acid 7,4,5-trichlorobenzenesulfonic acid m-iodophenylacetic acid 2-benzoyl-3,4,5,6-tetrachlorobenzoic acid phenylthiohydantoic acid 4 * - (ethoxycarbonyl) succinilic acid (R) - (-) - 2,2-dimethyl-5-oxo-1,3-dioxolane-4-acetic acid 4-acetylbenzoic acid 4-amino-2 -nitrobenzoic acid 2- (2,5-dimethylbenzoyl) -acrylic acid gamma-oxo-2-naphthalenebutyric acid 2-bromo-3-chlorobenzoic acid p-toluenesulfinic acid 1-benzyl-1,2,3-triazole-4,5-dicarboxylic acid 12 (s), 20-dihydroxyeicoza-5z, 8z, 10c, 14z-tetraenoic acid 7 -benzoylheptane • ·····················

-192kyselina 2,6-dihydroxybenzoová kyselina 4-chlór-2-metylbenzoová kyselina 3'-nitroglutaranilová kyselina 2,5-dimetyl-3-furoová kyselina (s)-2-metyldodekánová kyselina 1 -boc-piperidín-4-karboxylová kyselina dichlóroctová kyselina alfa-fenylškoricová gama-ŕerc-butylester kyseliny benzyloxykarbonyl-1-glutámovej kyselina dokozándiová kyselina 1 -(2,4-dichlórfenyl)cyklopropánkarboxylová kyselina m-nitrobenzén-sulfónová kyselina (r,s)-alfa-metoxy-alfa-trifluórmetylfenyloctová kyselina n-ftaloyl-1-glutámová kyselina (5-(1-ho-2,2,6,6-tetrametyl-1,2,3,6-4h-pyridín-4-yl)tiofén-2-yl)octová kyselina 3-(3-metoxybenzoyl)adipová kyselina 3,6-epoxycyklohexán-1,2-dikarboxylová kyselina 2-bróm-1 -naftalénsulfónová kyselina 4-(trifluórmetoxy)benzoová n-alfa-(benzyloxykarbonyl)-alfa-(benzylester)-1-asparágovej kyseliny kyselina d/-treo-beta-hyd roxyasparágová kyselina 3-(2-metylsulfanyl-benztiazol-6-ylamino)-propiónová kyselina 5-bróm-2,3-dihydrobenzofurán-7-karboxylová kyselina 3-(2,3,5,6-tetrametylbenzoyl)-akrylová kyselina 2-(1,3-benzodioxol-5-yl)-1 -metyl-5-oxo-3-pyrolidínkarboxylová kyselina 3-(2-(2-karboxy-benzoylamino)-etyl)-5-chlór-1h-indol-2-karboxylová kyselina 2,4-dihydroxybenzoová kyselina 3-(4-fluórfenoxy)propiónová kyselina 6-oxo-1,11-undekándikarboxylová kyselina 2,4-difluórškoricová kyselina 5-chlór-n-(2-chlóracetyl)antranilová kyselina 3-(4-nitro-1,3-dioxo-1,3-dihydro-izoindol-2-yl)-benzoová « ·· ·· ···· ·· ··· · ♦ · · · · • ··· · · · · ·-192 2,6-dihydroxybenzoic acid 4-chloro-2-methylbenzoic acid 3'-nitroglutaranilic acid 2,5-dimethyl-3-furoic acid (s) -2-methyldodecanoic acid 1 -boc-piperidine-4-carboxylic acid dichloroacetic acid alpha-phenyl cinnamic acid gamma-tert-butyl benzyloxycarbonyl-1-glutamic acid docosanedioic acid 1- (2,4-dichlorophenyl) cyclopropanecarboxylic acid m-nitrobenzenesulfonic acid (r, s) -alpha-methoxy-alpha-trifluoromethylphenylacetic acid n -phthaloyl-1-glutamic acid (5- (1-ho-2,2,6,6-tetramethyl-1,2,3,6-4h-pyridin-4-yl) thiophen-2-yl) acetic acid 3 - (3-Methoxybenzoyl) adipic acid 3,6-epoxycyclohexane-1,2-dicarboxylic acid 2-bromo-1-naphthalenesulfonic acid 4- (trifluoromethoxy) benzoic acid n-alpha- (benzyloxycarbonyl) -alpha- (benzyl ester) -1- Aspartic acid d-threo-beta-hydroxyaspartic acid 3- (2-methylsulfanyl-benzothiazol-6-ylamino) -propionic acid 5-bromo-2,3-dihydrobenzofuran -7-Carboxylic acid 3- (2,3,5,6-tetramethylbenzoyl) -acrylic acid 2- (1,3-benzodioxol-5-yl) -1-methyl-5-oxo-3-pyrrolidinecarboxylic acid 3- ( 2- (2-carboxy-benzoylamino) -ethyl) -5-chloro-1H-indole-2-carboxylic acid 2,4-dihydroxybenzoic acid 3- (4-fluorophenoxy) propionic acid 6-oxo-1,11-undecanedicarboxylic acid 2,4-Difluoro cinnamic acid 5-chloro-1- (2-chloroacetyl) anthranilic acid 3- (4-nitro-1,3-dioxo-1,3-dihydro-isoindol-2-yl) -benzoic acid · ·· · · ·····················

-193kyselina kvarcetínsulfónová kyselina 6-metyl-1 -(3-metylfenyl)-4-oxo-1,4-dihydro-5-pyridínkarboxylová n-(4-karboxy-3-hydroxyfenyl)maleimid kyselina 2,3-dihydroxy-4-metoxyškoricová kyselina fmoc-gama-aminomaslová kyselina 2-(2,4-dichlórfenyltio)octová kyselina 2,2’-oxydibenzoová kyselina 1-pyrénkarboxylová kyselina 9-fluorenón-1 -karboxylová kyselina (2-acetyl-6,7-dimetoxy-1,2,3,4-tetrahydro-izochinolín-1 -yl)-octová kyselina 3-n-propoxypikolínová kyselina s-benzyltioglykolová kyselina 4-(4-(3-(4-brómfenyl)-3-oxo-propyl)-fenyl)-4-oxo-maslová kyselina n-benzylmaleámová kyselina n-(4-chlórbenzoyl)aminooctová kyselina undecylénová kyselina 2-(2,4-dimetylbenzoyl)-3-metylbenzoová kyselina 2-acetylamino-4,5-dimetyl-tiofén-3-karboxylová kyselina cyklohexán-1,1-bis(meraptooctová) kyselina 2-(3,4-dimetoxybenzoyl)benzoová kyselina 2-(3-oxo-1 -indányl)octová kyselina 2-chlór-4-toluidín-6-sulfónová kyselina 2-(1 -karboxy-etylamino)-benzoová kyselina n-(2,4-difluórfenyl)maleámová kyselina 1-aminocyklobután-c/s-1,3-dikarboxylová kyselina 6,8-nonadekadiínová kyselina 3-fenyl-7-fluór-1 -oxoindán-3-karboxylová kyselina boc-1 -amino-1 -cyklohexán-karboxylová kyselina 3,3'-ditiobisbenzoová kyselina 3-dodekanoylamino-benzoová kyselina 4-(3-(2,2,2-trichlór-1-izobutyrylamino-etyl)-tioureido)-benzoová kyselina 2-fenyl-levulová • 9 99 9999 996-methyl-1- (3-methylphenyl) -4-oxo-1,4-dihydro-5-pyridinecarboxylic acid 4- (4-carboxy-3-hydroxyphenyl) maleimide 2,3-dihydroxy-4- fmoc-gamma-aminobutyric acid 2- (2,4-dichlorophenylthio) acetic acid 2,2'-oxydibenzoic acid 1-pyrene carboxylic acid 9-fluorenone-1-carboxylic acid (2-acetyl-6,7-dimethoxy-1) 2,3,4-tetrahydro-isoquinolin-1-yl) -acetic acid 3-n-propoxypicolinic acid s-benzylthioglycolic acid 4- (4- (3- (4-bromophenyl) -3-oxo-propyl) -phenyl ) -4-Oxo-butyric acid n-benzylmaleamic acid n- (4-chlorobenzoyl) aminoacetic acid undecylenic acid 2- (2,4-dimethylbenzoyl) -3-methylbenzoic acid 2-acetylamino-4,5-dimethylthiophene-3 carboxylic acid cyclohexane-1,1-bis (mercaptoacetic) 2- (3,4-dimethoxybenzoyl) benzoic acid 2- (3-oxo-1-indanyl) acetic acid 2-chloro-4-toluidine-6-sulfonic acid 2- (1-carboxy-ethylamino) -benzoic acid n- (2,4-Difluorophenyl) maleic acid 1-Aminocyclobutane-cis-1,3-dicarboxylic acid 6,8-Nonadecadioic acid 3-phenyl-7-fluoro-1-oxoindane-3-carboxylic acid boc-1-amino -1-cyclohexanecarboxylic acid 3,3'-dithiobisbenzoic acid 3-dodecanoylamino-benzoic acid 4- (3- (2,2,2-trichloro-1-isobutyrylamino-ethyl) -thioureido) -benzoic acid 2-phenyl- left • 9 99 9999 99

9 9 9 9 9 99 9 9 9 9

999 9 9 9 9 9999 9 9 9 9 9

-19499 99 99 9 kyselina 3-bróm-5-metoxy-benzoová kyselina 3-acetimidoylsulfanyl-propán-1 -sulfónová kyselina 4-benzyloxybenzoová kyselina 9,10,15-trihydroxy-oktadekánová kyselina 3-[3,4-(trimetyléndioxy)benzoyl]propiónová kyselina (s)-2-benzyljantárová kyselina (2-oxo-bicyklopentyl-1 '-én-1 -yl)-octová kyselina 4-(2-(4-chlórbenzoyl)acetamido)benzoová kyselina n-boc-d-1,2,3,4-tetrahydroizochinolín-3-karboxylová kyselina 4-(4-chlórfenylsulfonyl)-benzoová kyselina boc-1,2-aminokorková kyselina farnesylová (farnesol) kyselina 2-bróm-4,5-dimetoxyškoricová kyselina n-alfa-boc-glycyl-1 -asparágová kyselina 4,6-fenoxatindikarboxylová kyselina 3-nitro-4-(3-chlórfenoxy)škoricová kyselina 3-brómpyrohroznová kyselina pentafluórfenylpropiónová laktón kyseliny d/-izocitrónovej kyselina 3-(4-(5-(4-(2-karboxy-etyl)-fenyl)-pentyl)-fenyl)-propiónová kyselina 2-metoxyfenoxyoctová kyselina 1,2-etándisulfónová kyselina 3,5-dinitro-2-fluórbenzoová kyselina 2-etoxyfenyloctová kyselina 3-fluór-4-(trifluórmetyl)benzoová kyselina 2-p-tolyl-maslová kyselina 2-(5-nitro-1,3-dioxo-1,3-dihydro-izoindol-2-yl)-benzoová kyselina 4-acetamido-salicylová kyselina 7-doxyl-stearová kyselina 2',4,-dimetylftalanilová kyselina n-alfa-fmoc-n-alfa'-boc-diaminooctová kyselina undekándiová-19499 99 99 9 3-bromo-5-methoxy-benzoic acid 3-acetimidoylsulfanyl-propane-1-sulfonic acid 4-benzyloxybenzoic acid 9,10,15-trihydroxy-octadecanoic acid 3- [3,4- (trimethylenedioxy) benzoyl] propionic acid (s) -2-benzylsuccinic acid (2-oxo-bicyclopentyl-1'-en-1-yl) -acetic acid 4- (2- (4-chlorobenzoyl) acetamido) benzoic acid n-boc-d -1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid 4- (4-chlorophenylsulfonyl) -benzoic acid boc-1,2-aminocorkic acid farnesylic acid (farnesol) 2-bromo-4,5-dimethoxycinnamic acid n- alpha-boc-glycyl-1-aspartic acid 4,6-phenoxatindicarboxylic acid 3-nitro-4- (3-chlorophenoxy) cinnamic acid 3-bromopyruvic acid pentafluorophenylpropionic lactone d -isocitric acid 3- (4- (5- ( 4- (2-carboxy-ethyl) -phenyl) -pentyl) -phenyl) -propionic acid 2-methoxyphenoxyacetic acid 1,2-ethanedisulfonic acid 3,5-dinitro-2-fluorobenzoic acid 2-et 3-Fluoro-4- (trifluoromethyl) benzoic acid 2-p-tolyl-butyric acid 2- (5-nitro-1,3-dioxo-1,3-dihydro-isoindol-2-yl) -benzoic acid 4 acetamido-7-salicylic acid, stearic acid, DOXYL-2 ', 4, -dimetylftalanilová n-a-fmoc-n-boc-alpha' diaminoacetic acid undecanedioic

-195 --195 -

• ·· • · • ··· • ·· • · • ··· ·· • · • · ·· • · • · ···· • 9 ···· • 9 ·· · • · ·· 9 9 · ·· · • · ·· 9 9 · ·· ·· ·· ·· • · • · ·· · · ·· ·· ·· ··

kyselina 4-chlór-3-metoxybenzoová kyselina (r)-(+)-2-chlórpropiónová kyselina 2,3-dibróm-2'-etoxysukcínanilová kyselina 3-(3-(2,5-dioxo-2,5-dihydro-pyrol-1-yl)-fenyl)-akrylová kyselina 3,3-tetrametylénglutárová kyselina (1s)-(+)-(1-aminopropyl)fosfónová kyselina 4-(4-metoxy-fenyl)-but-2-énová kyselina 3-etyladipová kyselina mezo-2,3-dimetyljantárová kyselina 3,4,5,6-tetrachlór-2',4',6’-trimetylftalanilová kyselina 2,4,5-trimetylbenzoová metyl-beta-d-glukuronid, monohydrát voľnej kyseliny4-chloro-3-methoxybenzoic acid (R) - (+) - 2-chloropropionic acid 2,3-dibromo-2'-ethoxy-succinic acid 3- (3- (2,5-dioxo-2,5-dihydro- pyrrol-1-yl) -phenyl) -acrylic acid 3,3-tetramethyleneglutaric acid (1s) - (+) - (1-aminopropyl) phosphonic acid 4- (4-methoxy-phenyl) -but-2-enoic acid 3 -ethyladipic acid meso-2,3-dimethylsuccinic acid 3,4,5,6-tetrachloro-2 ', 4', 6'-trimethylphthalanilic acid 2,4,5-trimethylbenzoic acid methyl beta-d-glucuronide, free acid monohydrate

4-hydroxy-3-metyl(alfa-aminooctová kyselina)benzoová kyselina kyselina benzénsulfónová kyselina fenylpropargylová kyselina 2,5-dimetylbenzoová kyselina 4,4,8,8-tetrafluór-adamantán-1,3-dikarboxylová kyselina n-fmoc-d-1,2,3,4-tetrahydroizochinolín-3-karboxylová kyselina (+/-)-ŕrans-1 -amino-1 -karboxycyklopentán-2-octová kyselina 11-benzénsulfonyl-undekánová kyselina n-((s)-1-(1-naftyl)etyl)ftalámová kyselina (ij-3-hydroxymaslová kyselina 19-fenyl-nonadekánová kyselina 2-[3-(n’-butyrylhydrazíno)-3-oxo-propionylamino]-benzoová kyselina 4-oxo-1-fenyl-1,4-dihydro-pyridín-2,6-dikarboxylová kyselina chorismová kyselina n-(4-jódfenyl)ftalámová kyselina 4-oxo-4h-1 -tia-4a,9-diaza-fluorén-2-karboxylová kyselina 3-hydroxyftalid-7-karboxylová kyselina 5-(3-hydroxy-4-metoxy-fenyl)-pentánová kyselina 4-[[4-[(4,6-dimetylpyrimidín-2-yl)tio]fenyl]amino]-2-metyl-4-oxo-(2z)buténová4-hydroxy-3-methyl (alpha-aminoacetic acid) benzoic acid benzenesulfonic acid phenylpropargylic acid 2,5-dimethylbenzoic acid 4,4,8,8-tetrafluoro-adamantane-1,3-dicarboxylic acid n-fmoc-d- 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (+/-) - trans-1-amino-1-carboxycyclopentane-2-acetic acid 11-benzenesulfonyl-undecanoic acid n - ((s) -1- ( 1-naphthyl) ethyl) phthalic acid (1'-3-hydroxybutyric acid) 19-phenyl-nonadecanoic acid 2- [3- (n'-butyrylhydrazino) -3-oxo-propionylamino] -benzoic acid 4-oxo-1-phenyl- 1,4-dihydro-pyridine-2,6-dicarboxylic acid chorismic acid n- (4-iodophenyl) phthalic acid 4-oxo-4h-1-thia-4a, 9-diaza-fluorene-2-carboxylic acid 3-hydroxyphthalid -7-carboxylic acid 5- (3-hydroxy-4-methoxyphenyl) -pentanoic acid 4 - [[4 - [(4,6-dimethylpyrimidin-2-yl) thio] phenyl] amino] -2-methyl- 4-oxo- (2z) butenoic acid

-196 --196 -

• ·· • ·· ·· · · ···· ···· • · • · • · • · • · • · • · • · • · • · • ··· • ··· • · • · • · • · ·· ·· ·· ·· ·· · · • · • · ·· · · ·· · ·

kyselina 5,6-dichlór-3-indoloctová kyselina 3-(2,5-dimetylbenzoyl)-akrylová kyselina 7-oxo-11-dodecénová kyselina n,n'-dodekametylénbis(maleámová kyselina) kyselina treo-9,10-dihydroxystearová kyselina n-acetyl-d/-asparágová kyselina 1-pyroglutámová kyselina 2-metyl-3-m-tolyl-akrylová kyselina (2-acetyl-fenyl)-octová kyselina n-fenylacetyl-p-aminobenzoová kyselina 12-brómdodekánová kyselina chryzantémum-monokarboxylová kyselina (1 -benzoylamino-2,2-dichlór-vinyl)-fosfónová kyselina 3-metyl-3-(5,6,7,8-tetrahydro-naftalén-2-yl)-maslová kyselina 4-(2-hydroxy-1 -naftylmetylénamino)salicylová kyselina (2-fenyl-eténsulfonylamino)-octová kyselina 3-hydroxyadamantánkarboxylová kyselina 5-bróm-2-benzofuránkarboxylová kyselina 4-acetoxy-3-metoxyškoricová kyselina chicago kyselina 5-formylsalicylová kyselina 3-etyl-3-metylglutárová kyselina 2-(3,5-d/-ŕerc-butyl-4-hydroxy-benzylidén)-malónová kyselina 4-(2-hydroxyhexafluór-izopropyl)benzoová kyselina (r)-(+)-n-(1 -fenyletyl)ftalámová kyselina 2-acetylamino-4,5,6,7-tetrahydro-benzo(b)tiofén-3-karboxylová kyselina 2,5-diizotiokyanátobenzénsulfónová kyselina 3-(dodecyltio)-propiónová kyselina 10-fenyldekánová kyselina 4-formylfenoxyoctová kyselina 6-metyl-1 -(3-nitroanilíno)-4-oxo-1,4-dihydro-3-pyridínkarboxylová kyselina 4-metyl-2-(2-nitro-4-trifluórmetyl-fenylamino)-pentánová • ·· ·· ···· ·· ··· · · · · · · • ··· · · · · ·5,6-dichloro-3-indole acetic acid 3- (2,5-dimethylbenzoyl) -acrylic acid 7-oxo-11-dodecenoic acid n, n'-dodecamethylenebis (maleic acid) threo-9,10-dihydroxystearic acid n-acetyl-d-aspartic acid 1-pyroglutamic acid 2-methyl-3-m-tolyl-acrylic acid (2-acetyl-phenyl) -acetic acid n-phenylacetyl-p-aminobenzoic acid 12-bromododecanoic acid chrysanthemum-monocarboxylic acid (1-Benzoylamino-2,2-dichloro-vinyl) -phosphonic acid 3-methyl-3- (5,6,7,8-tetrahydro-naphthalen-2-yl) -butyric acid 4- (2-hydroxy- 1-naphthylmethyleneamino) salicylic acid (2-phenyl-etenesulfonylamino) -acetic acid 3-hydroxyadamantanecarboxylic acid 5-bromo-2-benzofuranecarboxylic acid 4-acetoxy-3-methoxycinnamic acid chicago 5-formylsalicylic acid 3-ethyl-3-methylglut 3 2- (3,5-tert-Butyl-4-hydroxy-benzylidene) -malonic acid 4- (2-hydroxy-hexafluoro-isopropyl) -benzoic acid ( r) - (+) - N- (1-phenylethyl) phthalic acid 2-acetylamino-4,5,6,7-tetrahydro-benzo (b) thiophene-3-carboxylic acid 2,5-diisothiocyanatobenzenesulfonic acid 3- (dodecylthio) 4-formylphenoxyacetic acid 6-methyl-1- (3-nitroanilino) -4-oxo-1,4-dihydro-3-pyridinecarboxylic acid 4-methyl-2- (2-nitro-4) -propionic acid -trifluoromethyl-phenylamino) -pentanoic acid

-197kyselina 2-chlór-6-metoxybenzoová kyselina 4-hydroxy-3-jód-5-nitrobenzoová kyselina 5-(4-(3-karboxy-propyl)-fenyl)-5-oxo-pentánová kyselina 3-(3,4-dimetoxy-6-nitrobenzoyl)propiónová kyselina 6-amino-2,3-dibróm-benzoová kyselina 2-(2,4,6-trichlórfenoxy)propiónová kyselina 3-(5-mtetyl-furán-2-yl)-akrylová kyselina (2-fluórfenyl)fosfónová kyselina 2-(2-(4-hydroxyfenyl)propyl)benzoová kyselina c/s-hexahydro-n-(4-metylfenyl)ftalámová kyselina 4-bifenylsulfónová kyselina 5-fenyl-2h-tetrazol-2-octová kyselina c/s-2-metoxyškoricová kyselina 4-metyldodekánová kyselina 3-(4-n-butylbenzoyl)propiónová kyselina (s)-(+)-2-fenylpropiónová kyselina 12-doxyl-stearová kyselina (1,2,3-trifenyl-cykloprop-2-enyl)-octová kyselina 1 -(4-chlórbenzoyl)piperazín-2,3-dikarboxylová kyselina 17-metyloktadekánová kyselina 2,4-dichlórškoricová kyselina 2-bróm-6-chlórbenzoová kyselina 3-metoxy-5-metyl-4-oxo-2,5-hexadiénová kyselina 2,3-dibrómpropiónová kyselina 3-(3-(2,4-dimetoxyfenyl)ureido)benzoová kyselina 2- [(2-karboxy-etyl)-(toluén-4-siilfonyl)-amino]-benzoová kyselina 2,5-diamino-1,4-benzéndisulfónová kyselina 2-brómmetyl-benzoová kyselina alfa-(brómmetyl)škoricová kyselina 3-benzoyl-2 pyridínkarboxylová kyselina 2-fenyl-2-etylmaslová kyselina 4-[[(4,6-dimetyl-2-pyrimidinyl)amino]karbonyl]-5-metyl-3-izoxazolkarboxylo-198-2-chloro-6-methoxybenzoic acid 4-hydroxy-3-iodo-5-nitrobenzoic acid 5- (4- (3-carboxypropyl) phenyl) -5-oxo-pentanoic acid 3- (3,4) 6-amino-2,3-dibromo-benzoic acid 2- (2,4,6-trichlorophenoxy) propionic acid 3- (5-methyl-furan-2-yl) -acrylic acid-dimethoxy-6-nitrobenzoyl) propionic acid (2-Fluorophenyl) phosphonic acid 2- (2- (4-hydroxyphenyl) propyl) benzoic acid cis-hexahydro-1- (4-methylphenyl) phthalic acid 4-biphenylsulfonic acid 5-phenyl-2h-tetrazole-2- acetic acid cis-2-methoxycinnamic acid 4-methyldodecanoic acid 3- (4-n-butylbenzoyl) propionic acid (s) - (+) - 2-phenylpropionic acid 12-doxyl-stearic acid (1,2,3- Triphenyl-cycloprop-2-enyl) -acetic acid 1- (4-chlorobenzoyl) piperazine-2,3-dicarboxylic acid 17-methyloctadecanoic acid 2,4-dichlorocinnamic acid 2-bromo-6-chlorobenzoic acid 3-methoxy-5- methyl 4-oxo-2,5-hexadienoic acid 2,3-dibromopropionic acid 3- (3- (2,4-Dimethoxyphenyl) ureido) benzoic acid 2 - [(2-carboxyethyl) - (toluene-4-sulfonyl) amino] benzoic acid 2,5-diamino-1,4-benzenedisulfonic acid 2-Bromomethyl-benzoic acid alpha- (bromomethyl) cinnamic acid 3-Benzoyl-2 pyridinecarboxylic acid 2-phenyl-2-ethylbutyric acid 4 - [[(4,6-dimethyl-2-pyrimidinyl) amino] carbonyl] -5- methyl-3-izoxazolkarboxylo-198-

• ·· • · • ··· • ·· • · • ··· • · • · • · • · • · • · ···· • • ···· • • ·· • · • · ·· • · • · ·· · · ·· ·· ·· ·· ·· · · ·· · · ·· · · • · • ·

vá kyselina 5-(3-hydroxyfenyl)valérová kyselina 8,9-epoxy-(5z,11z,14z)-eikozatriénová kyselina 3’-chlór-2'-metylmaleanilová kyselina ŕrans-4-metyl-1 -cyklohexánkarboxylová kyselina n-decylfosfónová kyselina hexadekándiová kyselina n-alfa-boc-(n-beta-fmoc)-diaminopropiónová kyselina 2-hydroxymyristová kyselina 4,4’-dihydroxybifenyl-2-karboxylová kyselina 8-chlórnaftalén-1 -sulfónová kyselina 2,3-bis-(4-metoxy-benzylidén)-jantárová kyselina 3,5-dihydroxy-4-metylbenzoová alfa-benzyl-ester kyseliny n-boc-1-asparágovej5- (3-hydroxyphenyl) valeric acid 8,9-epoxy- (5z, 11z, 14z) -eicosatrienoic acid 3'-chloro-2'-methylmaleanilic acid trans-4-methyl-1-cyclohexanecarboxylic acid n-decylphosphonic acid hexadecanedioic acid n-alpha-boc- (n-beta-fmoc) -diaminopropionic acid 2-hydroxymyristic acid 4,4'-dihydroxybiphenyl-2-carboxylic acid 8-chloronaphthalene-1-sulfonic acid 2,3-bis- (4 -methoxy-benzylidene) -succinic acid 3,5-dihydroxy-4-methylbenzoic acid n-boc-1-aspartic acid alpha-benzyl ester

4-karboxybenzénsulfonamid kyselina n-furfuryl-1,2,3,6-tetrahydroftalámová kyselina 2,5-dihydroxytereftalová kyselina 6-[(4,5-d/-meo-3-oxo-3h-izobenzofurán-1-ylidén)-ho-me]-2,3-d/-nneo-benzoová kyselina n-(1 -etoxykarbonyl-2-hydroxy-2-fenyl-etyl)jantárová kyselina 2-metyl-4-penténová kyselina ((5-bróm-furán-2-karbonyl)-amino)-octová kyselina alfa,alfa'-dibróm-1 ,3-adamantándioctová kyselina d/-4-(benzoylamino)-5-(dipropylamino)-5-oxo-pentánová kyselina 1 -(2-chlór-4-fluórfenyl)cyklohexánkarboxylová kyselina 3-metoxy-3-fenyl-propiónová kyselina ŕerc-butyl-perftalová kyselina 1-pyréndekánová kyselina ŕrans-2-(2-metoxyfenyl)-5-oxo-tetrahydrofurán-3-karboxylová kyselina 2-hydroxy-6-[4-(trifluórmetyl)fenyl]-3,5-pyridíndikarboxylová kyselina 5-brómferulová kyselina 3-(acetylmerkapto)-maslová4-carboxybenzenesulfonamide n-furfuryl-1,2,3,6-tetrahydrophthalic acid 2,5-dihydroxyterephthalic acid 6 - [(4,5-d-Meo-3-oxo-3h-isobenzofuran-1-ylidene) - 2-methyl-4-pentenoic acid ((5-bromo-furan) -2,3-di-non-benzoic acid n- (1-ethoxycarbonyl-2-hydroxy-2-phenyl-ethyl) -succinic acid -2-carbonyl) amino) -acetic acid alpha, alpha'-dibromo-1,3-adamantanediacetic acid d] -4- (benzoylamino) -5- (dipropylamino) -5-oxo-pentanoic acid 1- (2- chloro-4-fluorophenyl) cyclohexanecarboxylic acid 3-methoxy-3-phenyl-propionic acid tert-butyl-perfthalic acid trans-2- (2-methoxyphenyl) -5-oxo-tetrahydrofuran-3-carboxylic acid 2- hydroxy-6- [4- (trifluoromethyl) phenyl] -3,5-pyridinedicarboxylic acid 5-bromo-ferulic acid 3- (acetylmercapto) -butyric acid

-199--199-

• ·· • · • ··· • ·· • · • ··· • · • · • · • · • · • · ···· • • ···· • • ·· · • · ·· • · · ·· · • · ·· • · · ·· ·· ·· ·· ·· · · ·· · · ·· ·· ·· ··

kyselina 4-(acetyl-1,3-dioxo-1,3-dihydro-izoindol-2-ylmetyl)-amino)benzoová kyselina d/-cysteínová kyselina 5,7-dimetoxy-1 -oxo-2-indánkarboxylová kyselina 4-hydroxy-3-metylbenzoová kyselina 3-(3-chlór-fenyl)-2-metyl-akrylová kyselina 3-(o-tolyltio)propiónová kyselina 2-amino-6-sulfo-1 -naftalénmetánsulfónová kyselina n-(p-toluénsulfonyl)-d-glutámová kyselina 5-norbornén-2,3-dikarboxylová kyselina 3-bróm-1 -adamantánoctová kyselina 5-(5-indanylmetylénamino)-salicylová kyselina 4-(4-benzyloxykarbonylamino-butyrylamino)-maslová kyselina 3-(dichlór-metánsulfonyl)-propiónová kyselina hydantoínová kyselina 4-hydroxy-3-nitrofenyloctová kyselina 3’-chlór-6'-metoxymaleanilová kyselina 2-chlór-5-(fluórsulfónyl)benzoová kyselina 3-metyl-2-oxovalérová kyselina 2-anilíno-5-brómtereftalová kyselina benzoová kyselina cyklohexylidénkyanooctová kyselina 1,4-butánbis-(tioglykolová) kyselina 2,-metoxy-4'-nitromaleanilová kyselina 4-(3-metyl-4-hydroxyfenylazo)benzénsulfónová kyselina 2-(3-karboxy-propylamino)-benzoová kyselina 2-(brómmetyl)-2,3-dimetyl-4-oxocyklohexánkarboxylová kyselina 11-(3-(3-(trifluórmetyl)fenyl)ureido)undekánová kyselina 3-(3-benzyloxy-4-metoxy-fenyl)-propiónová kyselina 2,3,4-tribrómmaslová kyselina hexánová kyselina 4-fluór-2-metoxybenzoová kyselina benzylmalónová4- (acetyl-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl) amino) benzoic acid d -cysteic acid 5,7-dimethoxy-1-oxo-2-indanecarboxylic acid 4- hydroxy-3-methylbenzoic acid 3- (3-chloro-phenyl) -2-methyl-acrylic acid 3- (o-tolylthio) propionic acid 2-amino-6-sulfo-1-naphthalenemethanesulfonic acid n- (p-toluenesulfonyl) -d-glutamic acid 5-norbornene-2,3-dicarboxylic acid 3-bromo-1-adamantanacetic acid 5- (5-indanylmethyleneamino) -salicylic acid 4- (4-benzyloxycarbonylamino-butyrylamino) -butyric acid 3- (dichloro- methanesulfonyl) propionic acid hydantoic acid 4-hydroxy-3-nitrophenylacetic acid 3'-chloro-6'-methoxymaleanilic acid 2-chloro-5- (fluorosulfonyl) benzoic acid 3-methyl-2-oxovaleric acid 2-anilino-5- bromo-terephthalic acid benzoic acid cyclohexylidene cyanoacetic acid 1,4-butanebis- (thioglycolic) 2 , -methoxy-4'-nitromaleanilic acid 4- (3-methyl-4-hydroxyphenol) Ylazo) benzenesulfonic acid 2- (3-carboxy-propylamino) -benzoic acid 2- (bromomethyl) -2,3-dimethyl-4-oxocyclohexanecarboxylic acid 11- (3- (3- (trifluoromethyl) phenyl) ureido) undecanoic acid 3 - (3-Benzyloxy-4-methoxy-phenyl) -propionic acid 2,3,4-Tribromobutyric acid Hexanoic acid 4-Fluoro-2-methoxybenzoic acid Benzyl malonic acid

-200--200-

• ·· • · • ··· • ·· • · • ··· 99 • · • · 99 • · • · ···· • • ···· • • ·· • · • · · · • · • · 99 99 ·· ·· ·· ·· ·· · · ·· · · ·· · · 99 99

kyselina 2-naftyloctová kyselina c//-2-amino-8-fosfonooktánová kyselina 2-bróm-5-chlórfenyloctová kyselina 6-oxo-15-hexadecénová kyselina 1,2-fenyléndioctová boc-1-norleucín kyselina mezo-2,3-dibrómjantárová kyselina 3-(bután-1 -sulfonyl)-propiónová kyselina chlórsulfónová kyselina 4-chlór-3,5-dihydroxybenzoová kyselina izovalérová kyselina 3-(3-fluór-4-metoxybenzoyl)propiónová kyselina gama-d-glutamylaminometyl-fosfónová kyselina 2-metyl-4-oxo-4-fenylmaslová kyselina n-(2,4-dichlórfenyl)-2,3-dihydroxyjantárová kyselina 2-anizidín-4-sulfónová kyselina 2-(2’-pyridyl)-etylmalónová kyselina 4-etoxyfenyloctová kyselina 3-furoová kyselina 4’-acetyl-bifenyl-4-karboxylová kyselina diizooktyltiofosfínová kyselina (2,4-dinitro-fenylimino)-octová kyselina metylén-bis(tiomliečna) kyselina n-dodecylmaleámová kyselina n-acetyl-muramová kyselina benzénsulfonylamino-octová kyselina 1-metyl-2-aminotereftalát-4-pentyloxybifenyl-4'-karboxylová kyselina 3-[2-(benzoyloxy)fenyl]propiónová kyselina 5-nitrotiofén-2-karboxylová kyselina 4'-etylglutaranilová kyselina 4-(3-metyl-benzoylamino)-benzoová kyselina 1 -alfa-aspartyl-1 -glutámová ·· ······ ·· • · · 8 · · · • 88 8 8 8 8 82-naphthylacetic acid cis-2-amino-8-phosphonoctanoic acid 2-bromo-5-chlorophenylacetic acid 6-oxo-15-hexadecenoic acid 1,2-phenylenediacetic acid boc-1-norleucine meso-2,3- dibromosuccinic acid 3- (butane-1-sulfonyl) -propionic acid chlorosulfonic acid 4-chloro-3,5-dihydroxybenzoic acid isovaleric acid 3- (3-fluoro-4-methoxybenzoyl) propionic acid gamma-d-glutamylaminomethylphosphonic acid 2 methyl-4-oxo-4-phenylbutyric acid 2- (2'-pyridyl) ethylmalonic acid 4-ethoxyphenylacetic acid 2- (2'-pyridyl) -2,3-dihydroxysuccinic acid 3-furoic acid 4'-acetyl-biphenyl-4-carboxylic acid diisoctylthiophosphinic acid (2,4-dinitro-phenylimino) -acetic acid methylene-bis (thiomylic) n-dodecylmaleamic acid n-acetyl-muramic acid benzenesulfonylamino-acetic acid 1-methyl-2-aminoterephthalate-4-pentyloxybiphenyl-4'-carboxylic acid 3- [2- (benzoyloxy) phenyl] propionic acid 5-nitrothiophene-2-carboxylic acid 4'-ethylglutaranilic acid 4- (3-methyl-benzoylamino) -benzoic acid 1-alpha-aspartyl-1-glutamic acid ·· · 8 8 8 8 8 8

-201 kyselina 3,5-dimetylizoxazol-4-karboxylová kyselina (4-(4-karboxymetylsulfanyl-fenoxy)-fenylsulfanyl)-octová kyselina n-(4-adamantán-1 -yl-fenyl)-ftalámová kyselina 2-bróm-4-fluórbenzoová kyselina 3-fluór-4-n-oktyloxybenzoová kyselina 4-chlór-2,3,5,6-tetrametyl-benzoová kyselina p-chlórmandlová kyselina 2-metyl-benzén-1,3,5-trikarboxylová kyselina (+/-)-10-metyloktadekánová kyselina 2-jód-5-oxo-4-oxa-tricyklo(4.2.1.0(3,7))nonán-9-karboxylová kyselina 2-(2,4-d/-ŕerc-pentylfenoxy)maslová kyselina s-4-brómmandlová kyselina c/s-5-dodecénová kyselina 3-acenaftén-5-yl-propiónová kyselina 2'-benzoyl-2-bifenylkarboxylová kyselina 4-nitrotoluén-2-sulfónová kyselina 4-(2-metoxyanilíno)-4-oxo-2-buténová kyselina n-alfa-(9-fluorenylmetyloxykarbonyl)-alfa-(ŕerc-butylester)-1-glutámová kyselina 11 (r), 12(r)-epoxy-13(s)-hydroxy-9z-oktadecénová kyselina 2-hydroxy-1-naftoová kyselina 3-(2-nitro-fenyl)-2-o-tolylakrylová kyselina 3,5-dinitrosalicylová kyselina 4-(3-(2,6-xylyl)ureido)salicylová kyselina 3-okténová kyselina dehydrotio-4-toluidinsulfónová kyselina 5-(4-nitrofenyl)-2h-tetrazol-2-octová kyselina cyklohexánsulfámová kyselina 2,3-norbornándikarboxylová kyselina 12-tridecínová kyselina r-4-hydroxymandlová kyselina 3-(4-butyl-benzoylamino)-benzoová kyselina 2-bifenylénkarboxylová • ·· ·· ···· ·· ·· · · · · · · • ··· · · · · ·-201 3,5-dimethylisoxazole-4-carboxylic acid (4- (4-carboxymethylsulfanyl-phenoxy) -phenylsulfanyl) -acetic acid n- (4-adamantan-1-yl-phenyl) -phthalic acid 2-bromo-4 -fluorobenzoic acid 3-fluoro-4-n-octyloxybenzoic acid 4-chloro-2,3,5,6-tetramethylbenzoic acid p-chloromandelic acid 2-methylbenzene-1,3,5-tricarboxylic acid (+ / -) - 10-methyloctadecanoic acid 2-iodo-5-oxo-4-oxa-tricyclo (4.2.1.0 (3,7)) nonane-9-carboxylic acid 2- (2,4-di-tert-pentylphenoxy) s-4-bromo-butyric acid cis-5-dodecenoic acid 3-acenaphthen-5-yl-propionic acid 2'-benzoyl-2-biphenylcarboxylic acid 4-nitrotoluene-2-sulfonic acid 4- (2-methoxyanilino) -4-oxo-2-butenoic acid n-alpha- (9-fluorenylmethyloxycarbonyl) -alpha- (tert-butyl ester) -1-glutamic acid 11 (r), 12 (r) -epoxy-13 (s) -hydroxy- 9z-Octadecenic acid 2-hydroxy-1-naphthoic acid 3- (2-nitro-phenyl) -2-o-tolylacrylic acid 3,5-dinitrosalicylic acid 4- (3- (2,6-xylyl) ureido) salicylic acid 3-octenoic acid dehydrothio-4-toluidinesulfonic acid 5- (4-nitrophenyl) -2h-tetrazole-2-acetic acid cyclohexanesulfamic acid 2,3-norboranedicarboxylic acid 12-tridecinic acid r-4-Hydroxy-butyric acid 3- (4-butyl-benzoylamino) -benzoic acid 2-biphenylenecarboxylic acid • ······················ · · · ·

-202kyselina 2-(2-kyano-etylamino)-3-metyl-maslová kyselina 3-aminoftalová kyselina 3-hydroxy-o-toluylová kyselina 7-oxo-7h-benzo(e)pirimidín-4-karboxylová kyselina 3-bróm-4-hydroxybenzoová kyselina [3-(4-bróm-2-fluórbenzyl)-4-oxo-3h-ftalazín-1-yl]octová kyselina 3-(1-kyanoetyl)benzoová kyselina r?-(6-metyl-2-pyridyl)glutarámová kyselina n-(4-acetamidobenzylidén)antranilová kyselina chinolín-5-karboxylová kyselina 4,5-dichlóranilín-2-sulfónová kyselina 4-amino-3,5-dichlórbenzoová kyselina 3-(n-(3-pyridyl)karbamoyl)-5-norbornén-2-karboxylová kyselina o-naftiónová kyselina 4-imidazol-karboxylová kyselina 1 -amino-8-naftol-2,4-disulfónová kyselina n-(5-nitro-3-pyridyl)ftalámová kyselina 4-aminobenzoová kyselina 3-(3-pyridyl)akrylová kyselina nbd-aminohexánová kyselina n-(5,7-dimetyl-18-naftyridín-2-vl)-sukcínamová kyselina 5-amino-3-chlór-o-toluénsulfónová kyselina 5-nitro-4-chinolínkarboxylová kyselina n-(2-naftyl)-3,4,5,6-tetrachlórftalámová kyselina 2-amino-3-metoxybenzoová kyselina 4-bróm-2,5-dimetylpyrol-3-karboxylová kyselina 4-(2-benzimidazolyl)-benzénsulfónová kyselina 2,6-diaminomezitylén-4-sulfónová kyselina 4-pyridyloctová kyselina n-amino-3,4,5-trimetoxybenzoová kyselina dnp-alfa-aminoizomaslová kyselina 3-amino-2-naftoová ·· φφ ΦΦΦ· Φ· • · · · · · φφφ φφφ 9 φ-202 2- (2-cyano-ethylamino) -3-methyl-butyric acid 3-aminophthalic acid 3-hydroxy-o-toluic acid 7-oxo-7h-benzo (e) pirimidine-4-carboxylic acid 3-bromo- 4-Hydroxybenzoic acid [3- (4-bromo-2-fluorobenzyl) -4-oxo-3h-phthalazin-1-yl] acetic acid 3- (1-cyanoethyl) benzoic acid R 6 - (6-methyl-2- pyridyl) glutaramic acid n- (4-acetamidobenzylidene) anthranilic acid quinoline-5-carboxylic acid 4,5-dichloroaniline-2-sulfonic acid 4-amino-3,5-dichlorobenzoic acid 3- (n- (3-pyridyl) carbamoyl ) -5-Norbornene-2-carboxylic acid o-Naphthionic acid 4-Imidazole-carboxylic acid 1-amino-8-naphthol-2,4-disulfonic acid n- (5-nitro-3-pyridyl) phthalic acid 4-aminobenzoic acid 3- (3-pyridyl) acrylic acid nbd-aminohexanoic acid n- (5,7-Dimethyl-18-naphthyridin-2-yl) -succinamic acid 5-amino-3-chloro-o-toluenesulfonic acid 5-nitro- 4-quinolinecarboxylic acid n- (2-naphthyl) -3,4,5,6-tetrachlorophthalamo 2-Amino-3-methoxybenzoic acid 4-bromo-2,5-dimethylpyrrole-3-carboxylic acid 4- (2-benzimidazolyl) -benzenesulfonic acid 2,6-diaminomezitylene-4-sulfonic acid 4-pyridylacetic acid n- amino-3,4,5-trimethoxybenzoic acid dnp-alpha-aminoisobutyric acid 3-amino-2-naphthoic acid ··· 9 · · · φ · φφ 9 9φ 9

-203kyselina 6-metylnikotínová kyselina 6-(1,2,4-triazol-l -yl)nikotínová kyselina 5-metylindol-2-karboxylová kyselina 3-(n-metylanilíno)-1-propánsulfónová kyselina 2-amino-3,6-dimetylbenzoová kyselina 2,3-dichlór-4-[2-[3-chlór-5-(trifluórmetyl)-2-pyridyl]hydrazóno]-2-buténová kyselina 8-amino-2-naftalénsulfónová kyselina 2-amino-5-metoxybenzoová kyselina 5,6-dimetylmetanilová kyselina 5-amino-2,4-xylénsulfónová kyselina metanilová kyselina 4-(butylamino)benzoová kyselina 3-aminopyridín-4-karboxylová kyselina 1,2-fenyléndiamín-4-sulfónová kyselina 2-(2,5-dimetoxyfenyltio)pyridín-3-karboxylová kyselina n-[4-[(aminoiminometyl)-amino]-1 -karboxybutyl]-1 -glutámová kyselina 4h-1,2,4-triazol-3-karboxylová kyselina 2-dimetylaminobenzoová kyselina n-(3-pyridyl)-maleámová kyselina 2-propionyl-3-indoloctová kyselina 6-[n-metylamino]-1 -naftol-3-sulfónová kyselina 2-(2-pyridyl)etánsulfónová kyselina n-metylsulfanilová kyselina dnp-c//-alfa-amino-n-maslová kyselina 4-(hexadecyloxy)- 3-nitroškoricová kyselina 2-(4-chlórfenyltio)pyridín-3-karboxylová-203 6-methylnicotinic acid 6- (1,2,4-triazol-1-yl) nicotinic acid 5-methylindole-2-carboxylic acid 3- (n-methylanilino) -1-propanesulfonic acid 2-amino-3,6 -dimethylbenzoic acid 2,3-dichloro-4- [2- [3-chloro-5- (trifluoromethyl) -2-pyridyl] hydrazono] -2-butenoic acid 8-amino-2-naphthalenesulfonic acid 2-amino-5- methoxybenzoic acid 5,6-dimethylmethanilic acid 5-amino-2,4-xylenesulfonic acid metanilic acid 4- (butylamino) benzoic acid 3-aminopyridine-4-carboxylic acid 1,2-phenylenediamine-4-sulfonic acid 2- (2, 5-Dimethoxyphenylthio) pyridine-3-carboxylic acid N- [4 - [(aminoiminomethyl) amino] -1-carboxybutyl] -1-glutamic acid 4h-1,2,4-triazole-3-carboxylic acid 2-dimethylaminobenzoic acid n- (3-pyridyl) -maleamic acid 2-propionyl-3-indole acetic acid 6- [n-methylamino] -1-naphthol-3-sulfonic acid 2- (2-pyridyl) ethanesulfonic acid n-methylsulfanilic acid dnp-c // - a-amino-nm 4- (hexadecyloxy) -3-nitrocinnamic acid 2- (4-chlorophenylthio) pyridine-3-carboxylic acid

2-metyl-3-hydroxy-4-karboxy-5-hydroxy-metylpyridín kyselina dianilínotereftalová kyselina 2-hydroxychinolín-4-karboxylová kyselina 5-[aminometyl]-4-[karboxymetyl)-1 h-pyrol-3-propánová kyselina n-(3-nitrofenyl)antranilová kyselina 5-amino-4-metoxybenzoová2-methyl-3-hydroxy-4-carboxy-5-hydroxymethylpyridine dianiline-terephthalic acid 2-hydroxyquinoline-4-carboxylic acid 5- [aminomethyl] -4- [carboxymethyl] -1H-pyrrole-3-propanoic acid n - (3-Nitrophenyl) anthranilic acid 5-amino-4-methoxybenzoic acid

-204--204-

Φ · · • · • ··· • · · Φ · · • · • ··· • · · • · • • • · • · • • • · ···· • · • · • · ···· • · • · • · t· • · • · • · · t · • · • · • · · • · • · ·· ·· ·· ·· ·· · · • · • · ·· · · • e • e

kyselina anilin-2,5-disulfónová kyselina 7-amino-2-naftalénsulfónová, monosódna soľ kyselina 6-fluór-7-morfolín-4-yl-4-oxo-1,4-dihydro-chinolín-3-karboxylová kyselina 3,5-diaminobenzoová kyselina 8-hydroxychinolín-2-karboxylová kyselina 4-(5-(2,5-xylyl)ureido)salicylová kyselina 5-(3-amino-5-oxo-2-pyrazolín-1-yl)-2-fenoxybenzénsulfónová kyselina 3-hydroxypikolínová kyselina 4-hydroxychinolín-2-karboxylová kyselina p-toluidín-o-sulfónová kyselina oxolinová kyselina 3-(3-nitro-4-pyrolidínofenyl)akrylová kyselina 2-pyridyloctová kyselina 2-chlórnikotínová kyselina meta-fenyléndiamín-4,6-disulfónová kyselina 3-pyridyloctová kyselina 2-merkapto-4-metyl-5-tiazoloctová kyselina pyrol-2-karboxylová kyselina 4-(4-chlórfenyl)-6,8-dimetyl-1,9-diaza-indén-3-karboxylová kyselina 4-metylnikotínová kyselina 1 -(4-metylfenyl)-4-hydroxy-6-pyridazinón-karboxylová kyselina 1-indoloctová kyselina 4,8-dihydroxychinolín-2-karboxylová kyselina benzoová kyselina 2-nafto-o-toluidín-3-fosforečná kyselina 4-metoxy-2-chinolínkarboxylová kyselina 2-(4-dimetylamino-fenyl)-tiazolidín-4-karboxylová kyselina 1 -metylpyrol-2-karboxylová kyselina 3-indol-mliečna kyselina ftalová kyselina 5-benzyloxyindol-3-octová kyselina (z)-2-amino-alfa-(1 -(íerc-butoxykarbonyl)-l-metyletoxyimino)-4-tiazoloctová • ·· ·· ···· ·· • · · ·· · ··· • ··· · · · * ·aniline-2,5-disulfonic acid 7-amino-2-naphthalenesulfonic acid, 6-fluoro-7-morpholin-4-yl-4-oxo-1,4-dihydroquinoline-3-carboxylic acid, monosodium salt 3, 5-Diaminobenzoic acid 8-hydroxyquinoline-2-carboxylic acid 4- (5- (2,5-xylyl) ureido) salicylic acid 5- (3-amino-5-oxo-2-pyrazolin-1-yl) -2- phenoxybenzenesulfonic acid 3-hydroxypicolinic acid 4-hydroxyquinoline-2-carboxylic acid p-toluidine-o-sulfonic acid oxolinic acid 3- (3-nitro-4-pyrrolidinophenyl) acrylic acid 2-pyridylacetic acid 2-chloronicotinic acid meta-4-phenylenediamine 6-disulfonic acid 3-pyridylacetic acid 2-mercapto-4-methyl-5-thiazoleacetic acid pyrrole-2-carboxylic acid 4- (4-chlorophenyl) -6,8-dimethyl-1,9-diaza-indene-3 4-methylnicotinic acid 1- (4-methylphenyl) -4-hydroxy-6-pyridazinone-carboxylic acid 1-indole acetic acid 4,8-dihydroxyquinoline-2-carboxylic acid benzoic acid 2-naphtho-o-toluidine-3-phosphoric acid 4-methoxy-2-quinolinecarboxylic acid 2- (4-dimethylamino-phenyl) -thiazolidine-4-carboxylic acid 1-methylpyrrole-2-carboxylic acid 3-indole-lactic acid phthalic acid 5-Benzyloxyindole-3-acetic acid (z) -2-amino-alpha- (1- (tert-butoxycarbonyl) -1-methylethoxyimino) -4-thiazoleacetic acid • ·· ·· ······· · · ··· · ··· · ··· · · ·

-205kyselina 2-(4-chlórfenoxy)pyridín-3-karboxylová kyselina 2-amino-1 -naftalénsulfónová kyselina 5-amino-2(p-aminoanilíno)-benzénsulfónová kyselina alfa-(n-etylanilíno)-m-toluénsulfónová kyselina 2-chlór-4-karboxychinolin kyselina 6-(p-toluidíno)-2-naftalénsulfónová kyselina n-(n-metyl-n-(2-(3-chlór-5-trifluórmetyl)pyridyl)maleámová kyselina 3-amino-4-íerc-butylbenzoová kyselina 4-etyl-5-formyl-5-metyl-2-pyrolkarboxylová kyselina 5-metyl-benzo(1,2,5)tiadiazol-4-sulfónová kyselina dnp-gama-aminomaslová kyselina 6-(2,4,5-trichlórfenoxy)-metanilová kyselina 7-anilíno-4-hydroxy-2-naftalénsulfónová kyselina 4-amino-3,5,6-trichlórpicolínová kyselina 3-hydroxyantranilová kyselina 2-metoxynikotínová kyselina n-(4-metyl-2-pyridyl)sukcínamová kyselina 8-aminonaftalén-1,3,6-trisulfónová kyselina 4-(2,3-dihydro-2-tioxo-1-benzimidazolylmetylamino)-benzoová kyselina 2-formyl-4-metyl-3-pyrolpropiónová kyselina 4-amidínobenzoová kyselina 4-amino-5-chlór-m-toluén-sulfónová kyselina 2-amino-3,4,5,6-tetrafluórbenzoová kyselina 5-formyl-4-metyl-3-pyrolpropiónová kyselina 5-(2,5-dihydroxybenzylamino)-2-hydroxybenzoová kyselina 2-(4-aminofenoxy)-2-metylpropiónová kyselina 1-metyl-3-indoloctová kyselina n-amino-3,5-dibróm-6-fluórbenzoová kyselina pikrová kyselina 2-(4-metylfenyltio)pyridin-3-karboxylová kyselina n-(3-pyridylmetyl)glutarámová kyselina 1 -metylindol-2-karboxylová • · · ·· · ··· • ··· φ φ · φ φ-205 2- (4-chlorophenoxy) pyridine-3-carboxylic acid 2-amino-1-naphthalenesulfonic acid 5-amino-2 (p-aminoanilino) -benzenesulfonic acid alpha- (n-ethylanilino) -m-toluenesulfonic acid 2- chloro-4-carboxyquinoline 6- (p-toluidino) -2-naphthalenesulfonic acid n- (n-methyl-n- (2- (3-chloro-5-trifluoromethyl) pyridyl) maleic acid 3-amino-4-tert -butylbenzoic acid 4-ethyl-5-formyl-5-methyl-2-pyrrolecarboxylic acid 5-methyl-benzo (1,2,5) thiadiazole-4-sulfonic acid dnp-gamma-aminobutyric acid 6- (2,4, 5-Trichlorophenoxy) -methanilic acid 7-Anilino-4-hydroxy-2-naphthalenesulfonic acid 4-amino-3,5,6-trichloropicolic acid 3-hydroxyantranilic acid 2-methoxynicotinic acid n- (4-methyl-2-pyridyl) 8-aminonaphthalene-1,3,6-trisulfonic acid 4- (2,3-dihydro-2-thioxo-1-benzimidazolylmethylamino) -benzoic acid 2-formyl-4-methyl-3-pyrrolepropionic acid 4-amidinobenzoic acid 4-amino-5-C 2-Amino-3,4,5,6-tetrafluorobenzoic acid 5-formyl-4-methyl-3-pyrropropionic acid 5-2,5-dihydroxybenzylamino) -2-hydroxybenzoic acid (4-aminophenoxy) -2-methylpropionic acid 1-methyl-3-indoleacetic acid n-amino-3,5-dibromo-6-fluorobenzoic acid picric acid 2- (4-methylphenylthio) pyridine-3-carboxylic acid n- ( 3-pyridylmethyl) glutaramic acid 1-methylindole-2-carboxylic acid • • · · φ φ

-206kyselina 6-dimetylamino-4-hydroxy-2-naftalénsulfónová kyselina 4-amino-difenylamín-2-sulfónová kyselina 1 -izochinolínkarboxylová kyselina 3-(3-aminofenyl)propiónová kyselina 3-acetamido-5-aminobenzoová kyselina 4-hydroxychinolín-2-karboxylová kyselina 1,4-dihydro-1-etyl-7-metyl-4-oxo-1,8-naftyridín-3-karboxylová kyselina (2-benzimidazolytio)octová kyselina 5-izochinolínsulfónová kyselina 4-(4-anilínofenylazo)benzénsulfónová kyselina 4-dimetylaminonaftalén-1 -karboxylová kyselina dinitrofenyl-pipekolínová kyselina n-(2-pyridyl)-1,2,5,6-tetrahydroftalámová kyselina n-sulfanilylsulfanilová kyselina 4-aminobenzénsulfónová kyselina 5-aminosalicylic kyselina 2-aminobenzoová, 5-sulfamid kyselina pyrazol-3-karboxylová kyselina n-amino-4-chlórfenol-6-sulfónová kyselina 4,4’-diaminobifenyl-2l2,-dikarboxylová kyselina 8-amino-1,6-naftaléndisulfónová kyselina n-(2,5-dichlórfenyl)antranilová kyselina ftalylsulfatiazol-4-nitroantranilová kyselina indol-3-glyoxylová kyselina n-(2-nitrofenyl)antranilová kyselina 2,3-dimetyl-7-indolkarboxylová kyselina 2-(p-chlórfenyl)-chinolíne-4-karbxylová kyselina 1-nafíylamín-5-sulfónová kyselina 2,4-diaminobenzoová kyselina c/s-hexahydro-n-(3-pyridylmetyl)ftalámová kyselina 2-amino-3,4-dimetylbenzoová kyselina 3-izotioureidopropiónová ·· ·· ···· ·· • · · · · · ··· · · · · ·-206 6-dimethylamino-4-hydroxy-2-naphthalenesulfonic acid 4-amino-diphenylamine-2-sulfonic acid 1-isoquinolinecarboxylic acid 3- (3-aminophenyl) propionic acid 3-acetamido-5-aminobenzoic acid 4-hydroxyquinoline-2 1,4-dihydro-1-ethyl-7-methyl-4-oxo-1,8-naphthyridine-3-carboxylic acid (2-benzimidazolytio) acetic acid 5-isoquinolinesulfonic acid 4- (4-anilino-phenylazo) benzenesulfonic acid 4-dimethylaminonaphthalene-1-carboxylic acid dinitrophenyl-pipecolinic acid n- (2-pyridyl) -1,2,5,6-tetrahydrophthalic acid n-sulfanilylsulfanilic acid 4-aminobenzenesulfonic acid 5-aminosalicylic 2-aminobenzoic acid, 5-sulfamide of the pyrazole-3-carboxylic acid n-amino-4-chlorophenol-6-sulfonic acid 4,4-diamino-2 l 2, -dicarboxylic acid, 8-amino-1,6-disulfonic acid, N- (2,5- dichlorophenyl) anthranilic acid phthalylsulfathiazole-4-nitroantranilic acid indole-3-glyoxylic acid n- (2-nitrophenyl) anthranilic acid 2,3-dimethyl-7-indolecarboxylic acid 2- (p-chlorophenyl) quinoline-4-carboxylic acid 1-naphthylamine-5-sulfonic acid 2,4 -diaminobenzoic acid cis-hexahydro-1- (3-pyridylmethyl) phthalic acid 2-amino-3,4-dimethylbenzoic acid 3-isothioureidopropionic acid ··· ··············· · · · · · ·

-207kyselina n-(2-(n-metylanilíno)etyl)-1,2,3,6-tetrahydroftalámová kyselina 2-aminofenol-4-sulfónová kyselina citrazínová kyselina 3-indolpropiónová kyselina alfa(2-amino-4-(trifluórmetyl)fenyl)-4-(trifluórmetyl)škoricová kyselina 5-(pyrid-2-yl)tiofén-2-karboxylová kyselina 2-metyl-4-trifluórmetyltiazol-5-karboxylová kyselina 2-amino-6-hydroxybenzénsulfónová kyselina 5-chlór-6-hydroxynikotínová kyselina 5-metyl-3-pyridínsulfónová kyselina 5-amino-2-chlórbenzoová kyselina 2-fenyl-4-chinolínkarboxylová n-fenylglycín-207 n- (2- (n-methylanilino) ethyl) -1,2,3,6-tetrahydrophthalamic acid 2-aminophenol-4-sulfonic acid citrazic acid 3-indolpropionic acid alpha (2-amino-4- (trifluoromethyl) phenyl) -4- (trifluoromethyl) cinnamic acid 5- (pyrid-2-yl) thiophene-2-carboxylic acid 2-methyl-4-trifluoromethylthiazole-5-carboxylic acid 2-amino-6-hydroxybenzenesulfonic acid 5-chloro-6 -hydroxynicotinic acid 5-methyl-3-pyridinesulfonic acid 5-amino-2-chlorobenzoic acid 2-phenyl-4-quinolinecarboxylic acid n-phenylglycine

4-amino-2’-nitro-4,-sulfodifenylamín kyselina 8-hydroxychinolín-5-sulfónová kyselina 4,4,-diamino-5,5,-dimetyl-2,2'-bifenyldisulfónová kyselina n-etylnaftyl-2-amino-6-sulfónová kyselina 2'- metyl-3,3’,4,5,6-pentachlórftalanilová kyselina (z)-(2-aminotiazol-4-yl)hydroxyinninooctová kyselina nikotínurová kyselina 4-(veratrylidénamino)benzoová kyselina chinaldínová kyselina 5-metoxyindol-5-octová kyselina 4-anizidín-2-sulfónová kyselina 2(/?-metylamino)-8-hydroxynaftalén-6-sulfónová kyselina indol-5-karboxylová kyselina 1-(3-trifluórmetylfenyl)-4-hydroxy-6-pyridazinón-karboxylová kyselina 4-(2,3-dihydro-2-tioxo-3-benzoxazolylmetylamino)-salicylová kyselina 8-amino-1 -naftol-3,6-disulfónová kyselina 4-nitro-4,-aminodifenylamin-2-sulfónová 4-amino-2-nitro-4 -sulfodifenylamín 8-hydroxyquinoline-5-sulfonic acid 4,4'-diamino-5,5, dimethyl-2,2'-N-bifenyldisulfónová ethylnaphthyl-2-amino 6-sulfonic acid 2'-methyl-3,3 ', 4,5,6-pentachlorophthalanilic acid (z) - (2-aminothiazol-4-yl) hydroxyinninoacetic acid nicotinuric acid 4- (veratrylidenamino) benzoic acid quinaldic acid 5 -methoxyindole-5-acetic acid 4-anisidine-2-sulfonic acid 2 (R-methylamino) -8-hydroxynaphthalene-6-sulfonic acid indole-5-carboxylic acid 1- (3-trifluoromethylphenyl) -4-hydroxy-6 pyridazinone carboxylic acid 4- (2,3-dihydro-2-thioxo-3-benzoxazolylmethylamino) -salicylic acid, 8-amino-1-naphthyl-3,6-disulfonic acid 4-nitro-4-2 -aminodifenylamin sulfonic

2-(4-sulfobutylamino)-4-chlórfenol kyselina 4-pyridylhydroxymetánsulfónová2- (4-sulfobutylamino) -4-chlorophenol 4-pyridylhydroxymethanesulfonic acid

-208·· ·· ···· ·· • · · · · · · ··· · · · · · kyselina 4-(2,3-dihydro-2-tioxo-1-benzimidazolylmetylamino)-salicylová kyselina akridón-10-octová kyselina 6-metoxy-2-(5-nitrofenyl)-4-chinolínkarboxylová kyselina 1 -amino-2-naftol-4-sulfónová kyselina 4-imidazol-akrylová kyselina 4-chlór-n-fenylantranilová kyselina anilíno-4-hydroxy-2-naftalénsulfónová kyselina 2-((2-hydroxy-benzilidén)-amino)-3-(3h-imidazol-4-yl)propiónová kyselina n-(6-metyl-2-pyridyl)-3,4,5,6-tetrachlórftalámová kyselina 1 -benzylindol-5-karboxylová kyselina 5-bróm-4-chlór-3-indolyl-beta-d-glukurónová kyselina 4l-anilínohexahydroftalanilová kyselina 4-(etoxykarbonylamino)antranilová kyselina indol-4-karboxylová kyselina 4-(metylamino)benzoová kyselina 2,5-diaminobenzoová kyselina 2-amino-3-nitrobenzoová kyselina 5-brómindol-3-octová kyselina n-(4-etoxyfenyl)-4-nitroantranilová kyselina 5-nitro-3-fenylindol-2-karboxylová kyselina (2-benzimidazolylmetyltio)-octová kyselina 5-nitrochinaldínová-208 4- (2,3-dihydro-2-thioxo-1-benzimidazolylmethylamino) -salicylic acid acridone- 10-acetic acid 6-methoxy-2- (5-nitrophenyl) -4-quinolinecarboxylic acid 1-amino-2-naphthol-4-sulfonic acid 4-imidazole-acrylic acid 4-chloro-n-phenylanthranilic acid anilino-4- hydroxy-2-naphthalenesulfonic acid 2 - ((2-hydroxy-benzilidene) -amino) -3- (3h-imidazol-4-yl) propionic acid n- (6-methyl-2-pyridyl) -3,4,5 6-tetrachlorophthalic acid 1-benzylindole-5-carboxylic acid 5-bromo-4-chloro-3-indolyl-beta-d-glucuronic acid 4- l- anilino-hexahydrophthalanilic acid 4- (ethoxycarbonylamino) anthranilic acid indole-4-carboxylic acid 4 - (methylamino) benzoic acid 2,5-diaminobenzoic acid 2-amino-3-nitrobenzoic acid 5-bromoindole-3-acetic acid n- (4-ethoxyphenyl) -4-nitroantranilic acid 5-nitro-3-phenylindole-2- carboxylic acid (2-benzimidazolylmethylthio) - acetic acid 5-nitrochinaldic acid

6-benzyloxy-5-metoxy-2-karboxyindol kyselina indol-5-maslová kyselina 6-metoxy-4-chinolínkarboxylová kyselina (s)-2-[6-hydroxy-2-benzotiazolyl]-2-tiazolén-4-karboxylová kyselina n-(1 -naftyl)-5-nitroantranilová kyselina 4-amino-3,5-dijódsalicylová kyselina chinolín-8-sulfónová kyselina 1 -metylbenzimidazol-2-sulfónová kyselina 5-metyl-3-fenylizoxazol-4-karboxylová kyselina indol-2-karboxylová • ·· ·· ···· ·· ··· ·· · ··· • ··· · · · · ·6-benzyloxy-5-methoxy-2-carboxyindole indole-5-butyric acid 6-methoxy-4-quinolinecarboxylic acid (s) -2- [6-hydroxy-2-benzothiazolyl] -2-thiazolene-4-carboxylic acid n- (1-naphthyl) -5-nitroantranilic acid 4-amino-3,5-diiodosalicylic acid quinoline-8-sulfonic acid 1-methylbenzimidazole-2-sulfonic acid 5-methyl-3-phenylisoxazole-4-carboxylic acid indole- 2-carboxylic • ···················

-209chloramben kyselina 4-dimetylaminobenzoová kyselina 1,5-dihydroxy-9-akridínkarboxylová kyselina c/s-hexahydro-/7-(4-metyl-2-pyridyl)ftalámová kyselina 4-(etylamino)benzoová kyselina benztiazol-6-karboxylová kyselina 6-aminonikotínová kyselina 5-(4-aminobenzamido)valérová kyselina n-(4-metyl-2-pyridyl)ftalámová kyselina 2-(n-propyltio)nikotínová kyselina n-(3-pyridyl)glutarámová kyselina 2,3,5,6-tetrachlór-4-pyridínkarboxylová kyselina 2-(4-pyridyl)etánsulfónová kyselina 4-amino-2,3,5,6-tetrafluórbenzoová kyselina 3-chlór-5-trifluórmetyl-pyridín-2-propénová kyselina 5-(3-(4-chlór-fenyl)-4,5-dihydro-pyrazol-1-yl)-izoftalová kyselina n-(3-metyl-2-pyridyl)ftalámová kyselina 4-metylmetanilová kyselina 2-amino-6-chlórbenzoová kyselina n-etylantranilová kyselina 4-tioureido-benzoová kyselina 1-naftylamín-6-sulfónová kyselina 5-amino-2-p-toluidínobenzénsulfónová kyselina 4-(di-n-hexylamino)benzoová kyselina 4-(4-chinolylazo)benzénsulfónová kyselina 2-fluórnikotínová kyselina 2-(benzo(1l2,5)tiadiazol-4-sylfonylamino)-5-bróm-benzoová kyselina 5-fluórindol-2-karboxylová kyselina o-anizidín-5-sulfónová kyselina dehydrotio-p-toluidínsulfónová kyselina 3,5-diamino-2-metylbenzoová kyselina 4,-(dimetylamino)glutaranilová ·· ·· ···· ·· • · · · · · · ··· · φ · · ·4-dimethylaminobenzoic acid 1,5-dihydroxy-9-acridinecarboxylic acid cis-hexahydro- [7- (4-methyl-2-pyridyl) phthalic acid] 4- (ethylamino) benzoic acid benzothiazole-6-carboxylic acid 6-aminonicotinic acid 5- (4-aminobenzamido) valeric acid n- (4-methyl-2-pyridyl) phthalic acid 2- (n-propylthio) nicotinic acid n- (3-pyridyl) glutaramic acid 2,3,5, 6-Tetrachloro-4-pyridinecarboxylic acid 2- (4-pyridyl) ethanesulfonic acid 4-amino-2,3,5,6-tetrafluorobenzoic acid 3-Chloro-5-trifluoromethyl-pyridine-2-propenoic acid 5- (3- (4-Chloro-phenyl) -4,5-dihydro-pyrazol-1-yl) -isophthalic acid N- (3-methyl-2-pyridyl) -phthalic acid 4-Methyl-methanilic acid 2-amino-6-chloro-benzoic acid n- 4-Thioureido-benzoic acid, ethylanthranilic acid 1-naphthylamine-6-sulfonic acid 5-amino-2-p-toluidine-benzenesulfonic acid 4- (di-n-hexylamino) benzoic acid 4- (4-quinolylazo) benzenesulfonic acid acid 2-fluoro-nicotinic acid 2- (benzo (1 L 2,5) thiadiazole-4-sylfonylamino) -5-bromo-benzoic acid, 5-fluoroindole-2-carboxylic acid o-anisidine-5-sulfonic acid, p-dehydrotio toluidínsulfónová 3,5-diamino-2-methylbenzoic acid 4 , - (dimethylamino) glutaranilic acid ·· ··········

-210kyselina 6-(1-imidazolyl)nikotínová kyselina 2-(4-hydroxyfenylazo)benzoová kyselina 7-dietylaminokumarín-5-karboxylová kyselina 2-[(2,3-dimetylfenyl)amino]benzoová kyselina 2-(n-(2-(n-metylanilino)etyl)karbamoyl)cyklohexánkarboxylová kyselina 2-(4-izopropyl-4-metyl-5-oxo-2-imidazolín-2-yl)nikotínová kyselina 1-(2I4-dichlórfenyl)-4-hydroxy-6-pyridazinón-karboxylová kyselina n,n-dimetyl-5-nitrosulfanilová kyselina 8-anilíno-1 -naftalénsulfónová kyselina 5-amino-3-chlór-2,4-dihydroxybenzoová kyselina n,4-dimetylmetanilová kyselina n-(2-tioxobenzotiazolín-3-ylmetyl)-antranilová kyselina 2-chlór-6-metylnikotinová kyselina 4-dimetylaminoazobenzén-4'-karboxylová kyselina 2-(fenyltio)pyridín-5-karboxylová kyselina 5-(1 -pyrolidino)-2h-tetrazol-2-octová kyselina 2,4-dichlór-3,5-dinitrobenzoová kyselina 4’-metyl-2,-nitro-3,4,5,6-tetrachlórftalanilová kyselina 2-(4-(dibutylamino)-2-hydroxybenzoyl)benzoová kyselina 3-pyridyloctová kyselina 4-aminoacetanilid-3-sulfónová n-acetyl-d/-tryptofán kyselina 2-[[2-(6-chlór-2-pyridyl)hydrazíno]karbonyl]benzoová kyselina 7-jód-8-hydroxychinolín-5-sulfónová kyselina 4-amino-3-nitrobenzoová kyselina 2-amino-5-metylbenzoová kyselina 4-(dietylamino)benzoová kyselina 4-chlóranilín-5-sulfónová kyselina antranilová chlóracetyl-d/-tryptofán kyselina 1 -(3-chlórfenyl)-4-hydroxy-6-pyridazinón-3-karboxylová kyselina 5-butyl-2-pyridinkarboxylová • ·· ·· ···· ·· • · · ·· · ··· • ··· · · · · ·-210 acid 6- (1-imidazolyl) nicotinic acid 2- (4-hydroxyphenylazo) benzoic acid 7-diethylaminocoumarin-5-carboxylic acid 2 - [(2,3-dimethylphenyl) amino] benzoic acid 2- (n- (2- (n-methylanilino) ethyl) carbamoyl) cyclohexanecarboxylic acid 2- (4-isopropyl-4-methyl-5-oxo-2-imidazolin-2-yl) -nicotinic acid 1- (2 L 4-dichlorophenyl) -4-hydroxy 6-pyridazinone-carboxylic acid n, n-dimethyl-5-nitrosulfanilic acid 8-anilino-1-naphthalenesulfonic acid 5-amino-3-chloro-2,4-dihydroxybenzoic acid n, 4-dimethylmethanilic acid n- (2-thioxobenzothiazoline) 3-ylmethyl) -antranilic acid 2-chloro-6-methylnicotinic acid 4-dimethylaminoazobenzene-4'-carboxylic acid 2- (phenylthio) pyridine-5-carboxylic acid 5- (1-pyrrolidino) -2h-tetrazole-2- Acetic acid 2,4-dichloro-3,5-dinitrobenzoic acid 4'-methyl-2 , -nitro-3,4,5,6-tetrachlorophthalanilic acid 2- (4- (dibutylamino) -2-hydroxybenzoyl) benzoic acid 3 -pyridylacetic acid 4-aminoacetane 3-sulfonic acid n-acetyl-d-tryptophan 2 - [[2- (6-chloro-2-pyridyl) hydrazino] carbonyl] benzoic acid 7-iodo-8-hydroxyquinoline-5-sulfonic acid 4-amino 3-nitrobenzoic acid 2-amino-5-methylbenzoic acid 4- (diethylamino) benzoic acid 4-chloroaniline-5-sulfonic acid anthranilic chloroacetyl-d -tryptophanic acid 1- (3-chlorophenyl) -4-hydroxy-6- 5-Butyl-2-pyridinecarboxylic acid pyridazinone-3-carboxylic acid.

-211 kyselina n-(5-metyl-3-izoxazolyl)-3,4,5,6-tetrachlórftalámová kyselina 5-(fenyletinyl)pyridín-5-karboxylová kyselina 2-metyl-2-(1,2,4-triazol-1-yl)propiónová kyselina 8-acetoxy-2-fenyl-4-chinolínkarboxylová kyselina 4-(4-(dimetylamino)benzylidénamino)salicylová kyselina 2-(4-ŕerc-butylfenoxy)pyridin-5-karboxylová kyselina 6-(trifluóretoxy)pyridín-3-karboxylová kyselina d/-alfa-bróm-beta-(5-imidazolyl)-propiónová kyselina 2-amino-5-bróm-5-metylbenzoová kyselina 1 -amino-8-naftalénsulfónová kyselina 5-chlórindol-2-karboxylová kyselina 4-(4-metoxybenzylamino)benzoová kyselina 4-(4-(dietylamino)benzylidénamino)salicylová kyselina 2-(4-dietylamino-2-hydroxybenzoyl)benzoová kyselina 2-karbamylnikotínová kyselina indolín-2-karboxylová o-dianizidín kyselina n-(3-amino-4-hydroxyfenylsulfonyl)-antranilová kyselina 3-metyl-5-pyrazolkarboxylová kyselina trans-1 -benzidín-3,3'-dikarboxylová kyselina 2-aminonikotínová kyselina 4-(2,5-dimetyl-3-formyl-1 -pyrolyl)-benzoová kyselina 3-amino-4-hydroxybenzoová kyselina 5-fluórindol-3-octová kyselina n-(2-(2-pyridyl)etyl)-3I4,5,6-tetrachlórftalámová kyselina 1 -(d iety Imetyl)-1,2,3,4-tetrahydronorharmán-5-karboxylová kyselina 4-hydroxy-8-(trifluórmetyl)-3-chinolín-karboxylová kyselina n-(3-pyridyl)ftalámová kyselina 2-fn-amyltio)nikotínová kyselina 2-(4-hydroxyfenyl)-6-metoxy-4-chinolínkarboxylová kyselina 4-(4-metoxybenzylidénamino)benzoová kyselina merkaptotetrazolyloctová-211 N- (5-methyl-3-isoxazolyl) -3,4,5,6-tetrachlorophthalic acid 5- (phenylethynyl) pyridine-5-carboxylic acid 2-methyl-2- (1,2,4-triazole) -1-yl) propionic acid 8-acetoxy-2-phenyl-4-quinolinecarboxylic acid 4- (4- (dimethylamino) benzylideneamino) salicylic acid 2- (4-tert-butylphenoxy) pyridine-5-carboxylic acid 6- (trifluoroethoxy) 1-Amino-8-naphthalenesulfonic acid 5-chloroindole-2- 2-amino-5-bromo-5-methyl-benzoic acid 1-amino-8-naphthalenesulfonic acid 1 H -alpha-bromo-beta- (5-imidazolyl) -propionic acid 4- (4-Methoxybenzylamino) benzoic acid 4- (4- (diethylamino) benzylideneamino) salicylic acid 2- (4-diethylamino-2-hydroxybenzoyl) benzoic acid 2-carbamylnicotinic acid indoline-2-carboxylic acid o-dianisidine n - (3-amino-4-hydroxyphenylsulfonyl) -antranilic acid 3-methyl-5-pyrazolecarboxylic acid trans-1-benzidine-3,3'-dicarboxylic acid 2-aminonicotinic acid 4- (2,5-dimethyl-3-formyl) -1 - pyrrolyl) benzoic acid, 3-amino-4-hydroxybenzoic acid, 5-fluoroindole-3-acetic acid N- (2- (2-pyridyl) ethyl) -3-4,5,6 tetrachlórftalámová I, 1 - (dimethyl iety d ) -1,2,3,4-tetrahydronorharman-5-carboxylic acid 4-hydroxy-8- (trifluoromethyl) -3-quinoline-carboxylic acid n- (3-pyridyl) phthalic acid 2-n-amylthio) nicotinic acid 2 - (4-hydroxyphenyl) -6-methoxy-4-quinolinecarboxylic acid 4- (4-methoxybenzylideneamino) benzoic acid mercaptotetrazolylacetic acid

-212--212-

• ·· • ·· ·· · · ···· ···· ·· · · • · • · • · • · • ··· • ··· ·· ·· ·· ·· ·· · · ·· · · ·· · · ·· · ·

kyselina 6,6'-ditiodinikotínová kyselina 6-amino-1 -naftol-5-sulfónová kyselina 4-amino-2-chlórbenzoová kyselina c/s-hexahydro-n-(2-pyridyl)ftalámová kyselina 2-(3-(1 '-fenylaminotiazol)benzoová kysel ina 5-(metoxykarbonyl )py rid í η-2-karboxylová kyselina 2-amino-5-nitrobenzoová kyselina 4-(trifluórmetyl)nikotínová kyselina 8-hydroxychinolín-4-karboxylová kyselina 3-amino-2,4,6-tribrómbenzoová kyselina 3-(n-etyl-5-hydroxy-4-nitrózoanilíno)propánsulfónová kyselina 2-amino-3,5-dijódbenzoová kyselina 3-amino-2-metylbenzoová kyselina 2-((2-hydroxy-3-nitro-benzylidén)-amino)-3-(1h-imidazol-2-yl)-propiónová kyselina 2-(2-furyl)-4-chinolínkarboxylová kyselina 2,6-dichlórnikotínová kyselina p-[[(n-tioxobenzotiazolín-5-yl)-metyl]amino]benzoová kyselina 2’-metoxy-4-nitrodifenylamín-2-sulfónová kyselina n-metylantranilová kyselina 4’-metyl-3,3,,4,5,6-pentachlórftalanilová kyselina 6-amino-2-naftalénsulfónová kyselina 2-hydroxynikotínová kyselina 1 -dimetylaminonaftalén-5-sulfónová kyselina 3-anilino-1 -propánsulfónová kyselina 5-bróm-2-(etoxykarbonyl)-3-indolmaslová kyselina 2-amino-3-metylbenzoová kyselina 4-aminohipurová kyselina indol-5-octová kyselina 3-metoxy-4-amino-azobenzén-sulfónová kyselina 2-amino-3,6-dichlórbenzoová kyselina n-veratrylidénantranilová kyselina n-(2-pyridyl)ftalámová6,6'-Dithiodinicotinic acid 6-amino-1-naphthol-5-sulfonic acid 4-amino-2-chlorobenzoic acid cis-hexahydro-1- (2-pyridyl) phthalic acid 2- (3- (1) 5-Methoxycarbonyl) pyridine-2-carboxylic acid 2-amino-5-nitrobenzoic acid 4- (trifluoromethyl) nicotinic acid 8-hydroxyquinoline-4-carboxylic acid 3-amino-2, 1-phenylaminothiazole) benzoic acid 4,6-Tribromobenzoic acid 3- (n-ethyl-5-hydroxy-4-nitrosoanilino) propanesulfonic acid 2-amino-3,5-diiodobenzoic acid 3-amino-2-methylbenzoic acid 2 - ((2-hydroxy-3) -nitro-benzylidene) -amino) -3- (1H-imidazol-2-yl) -propionic acid 2- (2-furyl) -4-quinolinecarboxylic acid 2,6-dichloronicotinic acid p - [[(n-thioxobenzothiazoline- 5-yl) methyl] amino] benzoic acid 2'-methoxy-4-nitrodiphenylamine-2-sulfonic acid n-methylanthranilic acid 4'-methyl-3,3,, 4,5,6-pentachlórftalanilová 6-amino- 2-Naphthalenesulfonic acid 2-hydroxynicotinic acid and 1-dimethylaminonaphthalene-5-sulfonic acid 3-anilino-1-propanesulfonic acid 5-bromo-2- (ethoxycarbonyl) -3-indolebutyric acid 2-amino-3-methylbenzoic acid 4-aminohippuric acid indole-5-acetic acid 3 -methoxy-4-amino-azobenzene-sulfonic acid 2-amino-3,6-dichlorobenzoic acid n-veratrylidenantranilic acid n- (2-pyridyl) phthalic acid

-213--213

• ·· • · • ··· • · · • ·· • · • ··· • · · ·· ···· • · · • · · • · · · · ·· ···· · · · • · · · · · · · · · · · ·· • · • · • · ·· • · • · • · ·· ·· ·· ·· ·· ·· ·· ·· ·· · ·

kyselina toluén-sulfónová kyselina 1,2,3,4-tetrahydro-akridín-9-karboxylová kyselina 2-amino-5-brómbenzoová kyselina 1-beta-imidazolmliečna kyselina 9-fluór-2-metyl-1 -azaxantán-3-karboxylová kyselina 2-metoxy-5-metylanilín-4-sulfónová kyselina 4-amino-3-metoxybenzoová kyselina n-(2,4-dinitrofenyl)-6-aminohexánová kyselina 5-etyl-2-indolkarboxylová kyselina 2,6-dimetylimidazo[1,2-a]pyridín-5-karboxylová kyselina 5-hydroxy-2-metyl-4-chinolinkarboxylová kyselina n,n-etyléndiantranilová kyselina 2-chlór-6-metoxypyridín-4-karboxylová kyselina n-anilínosukcínamová kyselina 6-metoxy-4-chinolínakrylová kyselina n-(2-amino-4-chlórfenyl)antranilová kyselina 5-nitro-n-fenylantranilová kyselina 1-tryptofyl-1-glutámová kyselina 4-amino-5-metoxytoluén-2-sulfónová kyselina 2-amino-4-fluórbenzoová kyselina 5-(2,3-dihydro-2-tioxo-3-benzoxazolylmetylamino)-salicylová kyselina 2-(a,a,a-trifluór-m-toluidíno)-nikotínová kyselina 3-aminofenyloctová kyselina 2-chlóranilín-4-sulfónová kyselina 4-nitroanilín-2-sulfónová kyselina beta-karbolín-3-karboxylová kyselina chinolin-8-karboxylová kyselina chinolín-4-karboxylová kyselina 3-(4-pyridyl)akrylová kyselina meta-xylidín-6-sulfónová kyselina 5-benzimidazolkarboxylová kyselina 4-amino-azobenzén-4-sulfónováToluene-sulfonic acid 1,2,3,4-tetrahydro-acridine-9-carboxylic acid 2-amino-5-bromobenzoic acid 1-beta-imidazole-lactic acid 9-fluoro-2-methyl-1-azaxantane-3-carboxylic acid 2-methoxy-5-methylaniline-4-sulfonic acid 4-amino-3-methoxybenzoic acid n- (2,4-dinitrophenyl) -6-aminohexanoic acid 5-ethyl-2-indolecarboxylic acid 2,6-dimethylimidazo [1 2-a] pyridine-5-carboxylic acid 5-hydroxy-2-methyl-4-quinolinecarboxylic acid n, n-ethylenediantranilic acid 2-chloro-6-methoxypyridine-4-carboxylic acid n-anilino succinamic acid 6-methoxy-4 quinolinacrylic acid n- (2-amino-4-chlorophenyl) anthranilic acid 5-nitro-n-phenylanthranilic acid 1-tryptophyll-1-glutamic acid 4-amino-5-methoxy-toluene-2-sulfonic acid 2-amino-4- 5- (2,3-Dihydro-2-thioxo-3-benzoxazolylmethylamino) -salicylic acid 2- (α, α, α-trifluoro-m-toluidino) -nicotinic acid 3-aminophenylacetic acid 2- chloroaniline-4-sulfonic acid 4-nitroaniline-2-sulfonic acid beta-carboline-3-carboxylic acid quinoline-8-carboxylic acid quinoline-4-carboxylic acid 3- (4-pyridyl) acrylic methoxylidine-6-sulfonic acid 5-Benzimidazolecarboxylic acid 4-amino-azobenzene-4-sulfonic acid

-214·· ·· ·· · kyselina 2,6-toluyléndiamín-4-sulfónová kyselina n-(2-(3-chlór-5-trifluórmetyl-pyridyl)-4-amino-maslová kyselina imidazol-4-octová kyselina 1 -[4-(4-metoxyfenyl)-1,3-tiazol-2-yl]-5-(trifl uórmety 11)-1 h-4-pyrazolkarboxylová kyselina p-aminooxanilová kyselina 2,5-dibróm-2'-metoxy-4,-nitrosukcínanilová kyselina 9-chlór-2-metyl-1 -azaxantán-3-karboxylová kyselina 4-amino-3-hydroxybenzoová kyselina 2-chlóranilín-5-sulfónová kyselina 5-benzyloxyindol-2-karboxylová kyselina 4-chlór-n-(4-tolyl)antranilová kyselina 2-amino-5-chlór-p-toluén-sulfónová kyselina 2-etoxynikotínová kyselina 4-amino-5-metylbenzoová kyselina 4-dimetylamino-3,5-dinitrobenzoová kyselina 1 -(4-etoxyanilíno)-2-antrachinónkarboxylová kyselina 3-amino-4-metylbenzoová kyselina 4-(1 h-benzotriazol-1-ylmetylamino)benzoová kyselina 7-chlór-6-fluór-1 -cyklopropyl-1,4-dihydro-4-oxochinolín-3-karboxylová kyselina 7-amino-1 -naftalénsulfónová kyselina n-(5-nitro-2-pyridyl)-3,4,5,6-tetrachlórftalámová kyselina difenylaminsulfónová kyselina 2-naftylamín-5-sulfónová kyselina 6-acetyl-n-fenylantranilová kyselina 3,5-dibrómsulfanilová kyselina 2-amino-3,5-dibrómbenzoová kyselina 3-(amidínotio)-1 -propánsulfónová kyselina 3-(2-metyl-4-nitroimidazol-1 -yl)propiónová kyselina 4-nitro-2-aminofenol-6-sulfónová kyselina 5,6-dichlórnikotínová kyselina 3,4-diaminobenzoová • ·· ·· ···· ·· · · · · · · · • ··· · · · · ·-214 ·· ·· ·· · 2,6-Toluylenediamine-4-sulfonic acid n- (2- (3-chloro-5-trifluoromethyl-pyridyl) -4-amino-butyric acid imidazole-4-acetic acid 1 - [4- (4-methoxyphenyl) -1,3-thiazol-2-yl] -5- (trifluoromethyl) -1H-4-pyrazolecarboxylic acid p-aminooxanilic acid 2,5-dibromo-2'-methoxy -4, -nitrosukcínanilová 9-chloro-2-methyl-1 -azaxantán-3-carboxylic acid 4-amino-3-hydroxybenzoic acid 2-chloroaniline-5-sulfonic acid 5-benzyloxy-indole-2-carboxylic acid 4-chloro- n- (4-tolyl) anthranilic acid 2-amino-5-chloro-p-toluenesulfonic acid 2-ethoxynicotinic acid 4-amino-5-methylbenzoic acid 4-dimethylamino-3,5-dinitrobenzoic acid 1- (4- ethoxyanilino) -2-anthraquinone carboxylic acid 3-amino-4-methylbenzoic acid 4- (1H-benzotriazol-1-ylmethylamino) benzoic acid 7-chloro-6-fluoro-1-cyclopropyl-1,4-dihydro-4-oxoquinoline 3-Carboxylic acid 7-amino-1-naphthalenesulfonic acid n- (5-nitro- 2-Pyridyl) -3,4,5,6-tetrachlorophthalic acid Diphenylamine sulfonic acid 2-Naphthylamine-5-sulfonic acid 6-Acetyl-n-phenylanthranilic acid 3,5-Dibromosulfanilic acid 2-Amino-3,5-dibromobenzoic acid 3 - (amidinothio) -1-propanesulfonic acid 3- (2-methyl-4-nitroimidazol-1-yl) propionic acid 4-nitro-2-aminophenol-6-sulfonic acid 5,6-dichloronicotinic acid 3,4-diaminobenzoic acid • ···························

-215kyselina 3-(n-(2-pyridyl)karbamoyl)-5-norbornén-2-karboxylová kyselina 6-acetamido-3-pyridínsulfónová kyselina 3-(4-chlór-2-nitroanilíno)-propiónová kyselina n-cyklohexylidénantranilová kyselina 2-benzimidazolpropiónová kyselina cytozín-5-karboxylová kyselina 6-acetylamino-2-aminofenol-4-sulfónová kyselina 2,6-dimetylpyridín-3-sulfónová kyselina dinitropyridyI-1 -asparágová kyselina 2-amino-3-chlórbenzoová-215 3- (n- (2-pyridyl) carbamoyl) -5-norbornene-2-carboxylic acid 6-acetamido-3-pyridinesulfonic acid 3- (4-chloro-2-nitroanilino) -propionic acid n-Cyclohexylidenenantranilic acid 2 -benzimidazole propionic acid cytosine-5-carboxylic acid 6-acetylamino-2-aminophenol-4-sulfonic acid 2,6-dimethylpyridine-3-sulfonic acid dinitropyridyl-1-aspartic acid 2-amino-3-chlorobenzoic acid

8-(3-karboxy propy I)-1,3-d i mety Ixa ntí n kyselina indol-5-pyrohroznová kyselina 2,2,-bipyridin-4,4,-dikarboxylová kyselina 2-(alyltio)nikotínová kyselina 2,3,4,-tnbrómsukcínanilová kyselina n-(6-metyl-2-pyridyl)ftalámová kyselina 7-nitroindol-2-karboxylová kyselina 4-(3-metyl-5-oxo-2-pyrazolín-1 -yl)benzoová kyselina 4-(n-hexylamino)benzoová kyselina n-anilínoglutarámová kyselina 3-anilínopropiónová kyselina 2-metoxyamino-2-(2-aminotiazol-4-yl)-octová kyselina n-(4-metyl-2-pyridyl)glutarámová kyselina 2-acetamidobenzoová kyselina 2-pyrolopyridín-5-karboxylová kyselina 4,4'-dikarboxy-2,2'-bichinolín kyselina 3,4,5-trichlór-2-pyridínkarboxylová kyselina 2,5-diaminobenzénsulfónová kyselina aristolochová kyselina n-(4,6-disulfo-8-hydroxy-1 -naftyl)-benzamid kyselina 4-hydroxy-7-(trifluórmetyl)-3-chinolín-karboxylová kyselina 2-amino-7-naftalénsulfónová ·· ·· ···· ·· ··· ·· · ··· • ··· 9 9 9 9 98- (3-carboxypropyl) -1,3-dimethoxyindole-5-pyruvic acid 2,2 , -bipyridine-4,4 , -dicarboxylic acid 2- (allythio) nicotinic acid 2,3 4, -tnbrómsukcínanilová n- (6-methyl-2-pyridyl) phthalamic acid 7-nitroindole-2-carboxylic acid 4- (3-methyl-5-oxo-2-pyrazolin-1-yl) benzoic acid, 4- (n-hexylamino) benzoic acid n-anilino-glutaramic acid 3-anilino-propionic acid 2-methoxyamino-2- (2-aminothiazol-4-yl) -acetic acid n- (4-methyl-2-pyridyl) glutaramic acid 2-acetamidobenzoic acid 2-pyrrolopyridine-5-carboxylic acid 4,4'-dicarboxy-2,2'-quinoline 3,4,5-trichloro-2-pyridinecarboxylic acid 2,5-diaminobenzenesulfonic acid aristolochic acid n- (4,6-disulfo) -8-hydroxy-1-naphthyl) -benzamide 4-hydroxy-7- (trifluoromethyl) -3-quinoline-carboxylic acid 2-amino-7-naphthalenesulfonic acid ·· ·· ···· ·· ··· ·· · ··· 9 9 9 9 9

-216• 0 » 0000 00 0 • 00 00 ·* 99 99 999 kyselina 4-amino-2-metylškoricová kyselina 2-[2-(4-chlórbenzénsulfonyl)etyltio]pyridín-3-karboxylová kyselina 2-amino-3,4-dimetoxy-benzoová kyselina 4,6-biantranilová kyselina nikotínová kyselina 6-amino-4-hydroxy-2-naftalénsulfónová kyselina 2-amino-4,5-dimetoxybenzoová kyselina 4-acetyl-3,5-dimetfiyl-2-pyrolkarboxylová kyselina 3-aminosalicylová kyselina 3,3,,4,4’-tetrametyl-(2,2,-bipyrol)-5I5,-dikarboxylová kyselina 3-benzyloxy[tieno 1,2,5-b]pyridín-karboxylová kyselina 4-amino-1 -naftalénsulfónová kyselina 6-hydroxynikotínová kyselina 3-amino-4-chlórbenzoová kyselina m-toluidín-4-sulfónová kyselina 213-dichlór-4-(2,4-dinitrofenylhydrazóno)-2-buténová kyselina 4-nitropyrol-2-karboxylová kyselina 4-(dimetylamino)fenyloctová kyselina 2-(2,6-dimetylmorfolíno)-5-nitrobenzoová n-(4-chlórfenyl)-maleimid kyselina 4-azidobenzoová kyselina teofylín-7-octová kyselina 6-amino-3-pyridínsulfónová kyselina o-nitroanilín-p-sulfónová kyselina 2-(3-amino-4-chlórbenzoyl)benzoová kyselina n-(2,4-dinitrofenyl)-antranilová kyselina 4-(4-amino-m-tolylazo)-m-toluénsulfónová kyselina 3-(3-hydropxy-4-nitrózo-n-propylanilíno)propánsulfónová kyselina 3-amino-2,4,5-trifluórbenzoová kyselina 4-amino-2-metoxyškoricová kyselina 5-fenyl-2-pyrolpropiónová kyselina 7-anilíno-1 -naftol-3-sulfónová • ·· ·· ···· ·· ··· * · · · · · • ··· · · · · t-216 • 0 »0000 00 0 • 00 00 · * 99 99 999 4-amino-2-methylcinnamic acid 2- [2- (4-chlorobenzenesulfonyl) ethylthio] pyridine-3-carboxylic acid 2-amino-3,4 -dimethoxybenzoic acid 4,6-biantranilic acid nicotinic acid 6-amino-4-hydroxy-2-naphthalenesulfonic acid 2-amino-4,5-dimethoxybenzoic acid 4-acetyl-3,5-dimethylphenyl-2-pyrrolecarboxylic acid 3 aminosalicylic acid, 3,3,, 4,4-tetramethyl (2,2, -bipyrol) -5 I, 5-dicarboxylic acid 3-benzyloxy [thieno 1,2,5-b] pyridine-4-carboxylic acid amino-1-naphthalenesulfonic acid 6-hydroxynicotinic acid 3-amino-4-chlorobenzoic acid m-toluidine-4-sulfonic acid 2 1 3-dichloro-4- (2,4-dinitrophenylhydrazono) -2-butenoic acid 4-nitropyrole- 2-carboxylic acid 4- (dimethylamino) phenylacetic acid 2- (2,6-dimethylmorpholino) -5-nitrobenzoic acid 4- (4-chlorophenyl) -maleimide 4-azidobenzoic acid theophylline-7-acetic acid 6-amino-3- pyridinesulfonic o-nitroaniline-p-sulfonic acid 2- (3-amino-4-chlorobenzoyl) benzoic acid n- (2,4-dinitrophenyl) -antranilic acid 4- (4-amino-m-tolylazo) -m-toluenesulfonic acid 3- (3-hydropxy-4-nitroso-n-propylanilino) propanesulfonic acid 3-amino-2,4,5-trifluorobenzoic acid 4-amino-2-methoxycinnamic acid 5-phenyl-2-pyrrolepropionic acid 7-anilino-1 -naphthol-3-sulfonic acid · naphthol-3-sulfonic acid

-217kyselina pyridín-3-sulfónová kyselina 2-[2-(benzénsulfonyl)etyltio]pyridín-3-karboxylová kyselina 2-(etyltio)nikotínová kyselina n-(3-metyl-n-pyridyl)glutarámová kyselina 2-amino-2-tiazolín-4-karboxylová kyselina 9-metyl-2-metyl-1 -azaxantón-5-karboxylová kyselina 5-amino-2-nitrobenzoová kyselina 3-nitropyrid-2-yltiooctová kyselina 2,3-dibróm-4,,5’-dichlór-2‘-metylsukcínanilová kyselina 3,5-dichlórantranilová kyselina 8-amino-1 -naftol-5-sulfónová kyselina n-etyl-4-metylmetanilová kyselina 2-aminobenzofenón-2’-karboxylová-217 pyridine-3-sulfonic acid 2- [2- (benzenesulfonyl) ethylthio] pyridine-3-carboxylic acid 2- (ethylthio) nicotinic acid n- (3-methyl-n-pyridyl) glutaramic acid 2-amino-2- thiazoline-4-carboxylic acid 9-methyl-2-methyl-1 -azaxantón-5-carboxylic acid 5-amino-2-nitrobenzoic acid 3-nitro-pyridin-2-yltiooctová 2,3-dibromo-4, 5 &apos;dichloro-2'-methylsuccinilic acid 3,5-dichloroantranilic acid 8-amino-1-naphthol-5-sulfonic acid n-ethyl-4-methylmethanilic acid 2-aminobenzophenone-2'-carboxylic acid

3-nitroanilín-4-sulfónová kyselina n-(1-naftyl)antranilová kyselina 2-(2,-amino-4,-trifluórmetylfenyltio)benzoová kyselina 6-metylpikolínová kyselina 2-(pyrid-3-yl)tiazol-4-karboxylová kyselina 2-hydroxy-3-(2'-aminofenyltio)-3-(4-metoxyfenyl)propiónová kyselina 1,2,5-trimetylpyrol-3-karboxylová3-nitroaniline-4-sulfonic acid N- (1-naphthyl) anthranilic acid, 2- (2-amino-4, -trifluórmetylfenyltio) benzoic acid 6-methylpicolinic acid 2- (pyrid-3-yl) -thiazole-4-carboxylic acid 2-hydroxy-3- (2'-aminophenylthio) -3- (4-methoxyphenyl) propionic acid 1,2,5-trimethylpyrrole-3-carboxylic acid

6-metoxycinchofén kyselina 4-aminoškoricová kyselina 4-[n-(2-amino-3-kyano-5-pyrazinylmetyl)-amino)benzoová kyselina S'-chlór^.S-dibróm-Z-metoxysukcínanilová kyselina 2-metyl-3-indoteoctová kyselina (2-aminobenzénsulfónová) kyselina 3,5-dioxo-2,3,4,5-tetrahydro-(1,2,4)triazin-6-sulfónová kyselina 2-amino-4-fenyl-5-tiazolyloctová kyselina indol-3-karboxylová kyselina 8-metylpyrido[1,2-a]pyrimidín-4-ón-3-karboxylová kyselina 2-(4-metylfenoxy)pyridín-3-karboxylová kyselina 8-hydroxychinolín-7-sulfónová ·· BB BBBB ·· • B B · · · ·6-Methoxycinchophene 4-Amino-cinnamic acid 4- [n- (2-amino-3-cyano-5-pyrazinylmethyl) -amino) benzoic acid S'-chloro-4'-dibromo-2-methoxy-succinilic acid 2-methyl-3 (2-Aminobenzenesulfonic acid) -indoteacetic acid 3,5-dioxo-2,3,4,5-tetrahydro- (1,2,4) triazine-6-sulfonic acid 2-amino-4-phenyl-5-thiazolylacetic acid 8-methylpyrido [1,2-a] pyrimidin-4-one-3-carboxylic acid indole-3-carboxylic acid 2- (4-methylphenoxy) pyridine-3-carboxylic acid 8-hydroxyquinoline-7-sulfonic acid ·· BB BBBB ·· • BB · · · ·

BBB · B · B BBBB · B · B · B

-218B BB BB BB BBB kyselina 2-amino-4-chlórbenzoová kyselina n-(4-metoxybenzylidén)antranilová kyselina 5-brómnikotínová kyselina 2-piperidínocinchonínová kyselina 7-chlórkynurénová kyselina [+/-]-6-chlór-alfa-metylkarbazol-2-octová kyselina n-(2,4.6-tri n itrofenyl )-12-aminolaurová kyselina 2-(2-aminotiazol-4-yl)-2-metoxyiminooctová kyselina 11-(amidínotio)-undekánová kyselina 4-amino-3,5-dibrómbenzoová kyselina 4-(1 h-pyrol-1-yl)benzoová kyselina n-(2-pyridyl)sukcínamová kyselina 3-indolakrylová kyselina 5-((3-etyl-2(3h)-benzoxazolylidén)etylidén]-4-oxo-2-tioxo-3-tiazolidínoctová kyselina 8-etoxychinolin-5-sulfónová kyselina bromaminová kyselina n-(6-metyl-2-pyridyl)sukcínamová kyselina 6-chlórnikotínová kyselina 4-(/?,n-dietylamino)škoricová kyselina 3-dimetylaminometyl-1 h-indol-2-karboxylová kyselina 2,2’-metylén-bis(3,4-dimetyl-5-pyrolkarboxylová) kyselina 2,2,-benzidíndisulfónová kyselina 2-[(2,3-dihydroindol-1 -yl)imino]propánová kyselina 214-dinitro-4,-hydroxydifenylamín-3’-sulfónová kyselina 4-aminotoluén-3-sulfónová kyselina 4-(4-aminofenyl)maslová kyselina n,/?-tereftalylidéndiantranilová kyselina 2,2'-tiobis(5-aminobenzénsulfónová) kyselina 6-nitro-2-aminofenol-4-sulfónová kyselina 2-metylnikotínová kyselina 2-(5,6-dihydro-4h-1,3-oxazín-2-yl)benzoová kyselina 1 -metyl-4-(2,4-dichlórbenzoyl)pyrol-2-karboxylová • ·· ·· ···· ·· ·· · · · · ♦ · • ··· · · · · ·-218B BB BB BB BBB 2-Amino-4-chlorobenzoic acid n- (4-methoxybenzylidene) anthranilic acid 5-bromonicotinic acid 2-piperidinocinchoninic acid 7-Chloro-cyanoic acid [+/-] - 6-chloro-alpha-methylcarbazole- 2- (2-Aminothiazol-4-yl) -2-methoxyiminoacetic acid 2- (2-aminothiazol-4-yl) -2- (2,4,6-trifluorophenyl) -12-aminolauric acid 11- (amidinothio) -undecanoic acid 4-amino-3, 5-Dibromobenzoic acid 4- (1H-pyrrol-1-yl) benzoic acid n- (2-pyridyl) succinamic acid 3-indolacrylic acid 5 - ((3-ethyl-2 (3h) -benzoxazolylidene) ethylidene] -4 -oxo-2-thioxo-3-thiazolidineacetic acid 8-ethoxyquinoline-5-sulfonic acid bromamic acid n- (6-methyl-2-pyridyl) succinamic acid 6-chloronicotinic acid 4- (R, n-diethylamino) cinnamic acid 3-dimethylaminomethyl-1H-indole-2-carboxylic acid 2,2'-methylene-bis (3,4-dimethyl-5-pyrrolecarboxylic acid) 2,2 , -benzidinedisulfonic acid 2 - [(2,3-dihydroindole- 1-yl) imino] propanes and the 2 1 4-dinitro-4, -hydroxydifenylamín-3'-sulfonic acid, 4-aminotoluene-3-sulfonic acid 4- (4-aminophenyl) butyric acid n, /? - tereftalylidéndiantranilová 2,2'-thiobis (5 6-nitro-2-aminophenol-4-sulfonic acid 2-methylnicotinic acid 2- (5,6-dihydro-4h-1,3-oxazin-2-yl) benzoic acid 1-methyl-4- ( 2,4-Dichlorobenzoyl) pyrrole-2-carboxylic acid · 2,4-dichlorobenzoyl) pyrrole-2-carboxylic acid

-219kyselina 2-amino-5-chlórbenzoová kyselina 1 -etyl-3-metyl-1 h-pyrazol-5-karboxylová kyselina 4’-(dimetylamino)-3,4,5,6-tetrachlórftalanilová-219-2-amino-5-chlorobenzoic acid 1-ethyl-3-methyl-1H-pyrazole-5-carboxylic acid 4 '- (dimethylamino) -3,4,5,6-tetrachlorophthalanilic acid

3-karboxy-4-hydroxy-6-metoxychinolín kyselina 2-amino-6-chlór-3,5-dibrómbenzoová kyselina (4-pyridyltio)octová kyselina 2-pyridylhydroxymetánsulfónová kyselina 2,6-dimetoxynikotínová kyselina 2-chlór-6-metylpyridín-4-karboxylová kyselina 4-(2,6-dichlórbenzylidénamino)-benzoová kyselina p-anizidín-2-sulfónová kyselina 4-(4-amino-3-metylfenoxy)-1-butánsulfínová kyselina (5,6-dimetyl-2-benzimidazolyltio)-octová kyselina 4-(3-indolylmetylamino)benzoová kyselina 4-amino-2-butoxybenzoová kyselina 4-amino-3,5-dijódbenzoová n-jódacetyl-n-(5-sulfo-1-naftyl)etyléndiamín kyselina 4,4'-diaminostilbén-2,2,-disulfónová kyselina (2-amino-4-tiazolyl)octová kyselina 2-amino-5-hydroxybenzoová kyselina 4'-anilínoglutaranilová kyselina 2-(2-pyridylkarbonyl)benzoová kyselina n-(2-kyanoetyl)antranilová kyselina 6-chlór-3-aminoetylbenzén-4-sulfónová kyselina 1,3-fenyléndiamin-4-sulfónová kyselina 4’-amino-2’-hydroxysukcínanilovákyselina 7-benzyl-1-etyl-1,4-dihydro-4-oxo-1,8-naftyridín-3-karboxylová kyselina 4-nitrodifenylamín-2-sulfónová kyselina 2,3-dihydro-5-oxotiazolo[3.2-a]pyrimidín-6-karboxylová kyselina 2-amino-5-bróm-4-nitrobenzoová kyselina 5-nitro-2-(3-fenylpropylamino)benzoová kyselina izonikotínová3-carboxy-4-hydroxy-6-methoxyquinoline 2-amino-6-chloro-3,5-dibromobenzoic acid (4-pyridylthio) acetic acid 2-pyridylhydroxymethanesulfonic acid 2,6-dimethoxynicotinic acid 2-chloro-6-methylpyridine 4-carboxylic acid 4- (2,6-dichlorobenzylideneamino) -benzoic acid p-anisidine-2-sulfonic acid 4- (4-amino-3-methylphenoxy) -1-butanesulfonic acid (5,6-dimethyl-2- benzimidazolylthio) acetic acid 4- (3-indolylmethylamino) benzoic acid 4-amino-2-butoxybenzoic acid 4-amino-3,5-diiodobenzoic acid n-iodoacetyl-N- (5-sulfo-1-naphthyl) ethylenediamine acid 4, 4'-diaminostilbene-2,2-disulfonic acid acid (2-amino-4-thiazolyl) acetic acid 2-amino-5-hydroxybenzoic acid 4 ' anilínoglutaranilová 2- (2-pyridylcarbonyl) benzoic acid, n- (2- 6-chloro-3-aminoethylbenzene-4-sulfonic acid 1,3-phenylenediamine-4-sulfonic acid 4'-amino-2'-hydroxysuccinic acid 7-benzyl-1-ethyl-1,4-dianoic acid hydro-4-oxo-1,8-naphthyridine-3-carboxylic acid 4-nitrodiphenylamine-2-sulfonic acid 2,3-dihydro-5-oxothiazolo [3,2-a] pyrimidine-6-carboxylic acid 2-amino-5- Bromo-4-nitrobenzoic acid 5-nitro-2- (3-phenylpropylamino) benzoic acid isonicotinic acid

-220--220-

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kyselina 2-hydroxy-6-metylpyridín-3-karboxylová kyselina 6-chlór-2-(4-chlórfenyl)-4-chinolínkarbxylová kyselina 4-amino-3,5-dinitrobenzoová kyselina 2-metoxy-4-nitroanilín-5-sulfónová kyselina 2-amino-3,5-dimetylbenzoová kyselina 2-(1 -imidazolylkarbonyl)benzoová kyselina 5-hydroxyindol-2-karboxylová kyselina 4,5-dibrómantranilová kyselina (s)-(-)-indolín-2-karboxylová kyselina 2-amino-4-metylbenzoová kyselina 5-metoxy-2-metyl-5-indoloctová kyselina 2,5-dichlórsulfanilová kyselina 2-fenylbenzimidazol-5-sulfónová kyselina 3-amino-2,5,6-trifluórbenzoová kyselina 3-amino-5-nitrobenzoová kyselina 6-chlór-2-aminofenol-4-sulfónová kyselina 4-(dimetylamino)škoricová kyselina benzoová kyselina 2-[(3-chlór-2-metylfenyl)amino]-5-dimetylamino-1-naftalénsulfónová kyselina 5-amino-1 -naftol-3-sulfónová kyselina 3-(4-aminofenyl)propiónová kyselina 2-hydroxy-1 -(2-hydroxy-4-sulfo-1 -naftylazo)-3-naftoová kyselina 4-amino-5-chlór-2-metoxybenzoová kyselina pikolínová kyselina 4'-anilínomaleanilová kyselina p-[n,/?-bis(2-chlóretyl)amino]benzoová kyselina izoxazol-5-karboxylová kyselina 7-chlór-4-hydroxychinolín-3-karboxylová kyselina [(3,5,6-trichlór-2-pyridinyl)oxy]-octová kyselina 7,8-dimetyl-4-hydroxy-3-chinolínkarboxylová kyselina 2-naftylamín-1,5-disulfónová kyselina 5-metoxy-indol-2-karboxylová ·· · ···· • · · ·2-hydroxy-6-methylpyridine-3-carboxylic acid 6-chloro-2- (4-chlorophenyl) -4-quinolinecarboxylic acid 4-amino-3,5-dinitrobenzoic acid 2-methoxy-4-nitroaniline-5-sulfonic acid 2-amino-3,5-dimethylbenzoic acid 2- (1-imidazolylcarbonyl) benzoic acid 5-hydroxyindole-2-carboxylic acid 4,5-dibromantranilic acid (s) - (-) - indoline-2-carboxylic acid 2- amino-4-methylbenzoic acid 5-methoxy-2-methyl-5-indole acetic acid 2,5-dichlorosulfanilic acid 2-phenylbenzimidazole-5-sulfonic acid 3-amino-2,5,6-trifluorobenzoic acid 3-amino-5- nitrobenzoic acid 6-chloro-2-aminophenol-4-sulfonic acid 4- (dimethylamino) cinnamic acid benzoic acid 2 - [(3-chloro-2-methylphenyl) amino] -5-dimethylamino-1-naphthalenesulfonic acid 5-amino- 1-Naphthol-3-sulfonic acid 3- (4-aminophenyl) propionic acid 2-hydroxy-1- (2-hydroxy-4-sulfo-1-naphthylazo) -3-naphthoic acid 4-amino-5-chloro-2 -methoxybenzoic acid pic isoxazole-5-carboxylic acid 4'-anilinoomaleanilic acid p- [N, R-bis (2-chloroethyl) amino] benzoic acid 7-chloro-4-hydroxyquinoline-3-carboxylic acid [(3,5,6) -trichloro-2-pyridinyl) oxy] -acetic acid 7,8-dimethyl-4-hydroxy-3-quinolinecarboxylic acid 2-naphthylamine-1,5-disulfonic acid 5-methoxy-indole-2-carboxylic acid ·· · ·· ·· · · · ·

-221 kyselina 3-aminobenzoová kyselina 5,7-dichlórkynurénová kyselina 4-(8-hydroxy-5-chinolylazo)-1 -naftalénsulfónová kyselina 5-hydroxy-indol-3-octová kyselina 2-metyl-1 -azanton-5-karboxylová kyselina 5-acetamidoantranilová kyselina 4-amino-2-chlórtoluén-5-sulfónová-221 3-Aminobenzoic acid 5,7-Dichlorkynurenic acid 4- (8-hydroxy-5-quinolylazo) -1-naphthalenesulfonic acid 5-hydroxy-indole-3-acetic acid 2-methyl-1-azantone-5-carboxylic acid 5-Acetamidoantranilic acid 4-Amino-2-chlorotoluene-5-sulfonic acid

1-(2’,5,-dichlór-4'-sulfofenyl)-3-metyl-5-pyrazolón kyselina 4'-anilínosukcínanilová kyselina n-(2-tiazolyl)-1,2,3,6-tetrahydroftalámová kyselina 7-amino-4-metyl-3-kumarinyloctová kyselina 2,5-dimetylpyrol-3-karboxylová kyselina 3-chinolínkarboxylová kyselina imidazol-4-akrylová kyselina 2-amino-6-metylbenzoová kyselina 2-naft-o-anizidín-3-fosforečná kyselina beta-n-indolpropiónová kyselina 1 -diazo-2-naftol-4-sulfónová kyselina 3-hydroxy-2-fenylcinchonínová kyselina 4'-(dimetylamino)hexahydroftalanilová kyselina 2-amino-alfa,beta-dibrómhydroškoricová kyselina (1,3-dimetyl-2,6-dioxo-2,3,6,7-tetrahydro-1 h-purín-8-yl)-octová kyselina 4,5-difluórantranilová kyselina 3-(4-dimetylamino-1 -naftylazo)-4-metoxybenzénsulfónová kyselina 2-amino-5-fluórbenzoová kyselina 6-chinolínkarboxylová kyselina 3-aminobenzylmetylamín-4-sulfónová kyselina 2-nitrózo-1 -naftol-4-sulfónová kyselina 2-metylmerkaptonikotínová kyselina n-(3-pyridyl)hexahydroftalámová kyselina 5-(2,3-dihydro-2-tioxo-1-benzimidazolylmetylamino)-salicylová kyselina 2-chlór-6-metyl-nikotínová1- (2 ', 5'-dichloro-4'-sulfophenyl) -3-methyl-5-pyrazolone-4'anilínosukcínanilová N- (2-thiazolyl) -1,2,3,6-tetrahydroftalámová 7- amino-4-methyl-3-coumarinylacetic acid 2,5-dimethylpyrrole-3-carboxylic acid 3-quinolinecarboxylic acid imidazole-4-acrylic acid 2-amino-6-methylbenzoic acid 2-naphth-o-anisidine-3-phosphoric acid beta-n-indolpropionic acid 1-diazo-2-naphthol-4-sulfonic acid 3-hydroxy-2-phenylcinchoninic acid 4 '- (dimethylamino) hexahydrophthalanilic acid 2-amino-alpha, beta-dibromo-cinnamic acid (1,3-dimethyl -2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl) -acetic acid 4,5-difluoroantranilic acid 3- (4-dimethylamino-1-naphthylazo) -4-methoxybenzenesulfonic acid 2-amino-5-fluorobenzoic acid 6-quinolinecarboxylic acid 3-aminobenzylmethylamine-4-sulfonic acid 2-nitroso-1-naphthol-4-sulfonic acid 2-methylmercaptonicotinic acid n- (3-pyridyl) hexahydrophthalaams α 5- (2,3-Dihydro-2-thioxo-1-benzimidazolylmethylamino) -salicylic acid 2-chloro-6-methyl-nicotinic acid

-222--222-

9 99 9 9 • ··· 9 99 9 9 • ··· 99 9 9 • · 99 9 9 • · 9999 9 • 9999 9 • 99 9 • · · · • 9 · 99 9 • · · · • 9 · • » · · • »· · • · • · ·· · · ·· 99 ·· 99

kyselina 2-amino-5-jódbenzoová kyselina 5-metyl-4-[[3-(trifluórmetyl)anilíno]karbonyl]-3-izoxazol-karboxylová kyselina 4-aminosalicylová kyselina 5-brómindol-2-karboxylová kyselina 2-chlór-6-nitrofenol-4-sulfónová kyselina 4-(bis(2-chlóretyl)amino)benzénmaslová kyselina (4-aminofenyltio)octová kyselina n-benzylantranilová kyselina 3-pyridylhydroxymetánsulfónová kyselina 4-chlór-n-(6-metoxy-3-pyridyl)antranilová kyselina 4-aminofenyloctová kyselina 4-benzotiazol-2-yl-maslová kyselina 2-(4-pyridyl)tiazol-4-karboxylová kyselina 3-(4-dietylamino-2-hydroxyfenylazo)-4-hydroxybenzénsulfónová kyselina 1 -fenyl-4-hydroxy-6-pyridazinón-karboxylová kyselina 2-aminotoluén-5-sulfónová kyselina pyrazol-1-yl-octová kyselina n-(3-pyridyl)sukcínamová kyselina 5-(benzyloxykarbonyl)-2,4-dimetyl-3-pyrolpropiónová kyselina 4-dimetylaminosalicylová kyselina 3-chlór-2-toluidín-5-sulfónová kyselina 2,4-dimetyl-5-(ŕerc-butoxykarbonyl)-3-pyrolpropiónová kyselina 5-amino-2-hydroxybenzénsulfónová, a kyselina 3-aminopyridín-2-karboxylová.2-amino-5-iodobenzoic acid 5-methyl-4 - [[3- (trifluoromethyl) anilino] carbonyl] -3-isoxazole-carboxylic acid 4-aminosalicylic acid 5-bromoindole-2-carboxylic acid 2-chloro-6 -nitrophenol-4-sulfonic acid 4- (bis (2-chloroethyl) amino) benzenebutyric acid (4-aminophenylthio) acetic acid n-benzylanthranilic acid 3-pyridylhydroxymethanesulfonic acid 4-chloro-n- (6-methoxy-3-pyridyl) 4-Aminophenylacetic acid 4-benzothiazol-2-yl-butyric acid 2- (4-pyridyl) thiazole-4-carboxylic acid 3- (4-diethylamino-2-hydroxyphenylazo) -4-hydroxybenzenesulfonic acid 1-phenyl-4 -hydroxy-6-pyridazinone-carboxylic acid 2-aminotoluene-5-sulfonic acid pyrazol-1-yl-acetic acid n- (3-pyridyl) succinamic acid 5- (benzyloxycarbonyl) -2,4-dimethyl-3-pyrrolepropionic acid 4-dimethylaminosalicylic acid 3-chloro-2-toluidine-5-sulfonic acid 2,4-dimethyl-5- (tert-butoxycarbonyl) -3-pyrrolepropionic acid 5-am ino-2-hydroxybenzenesulfonic acid, and 3-aminopyridine-2-carboxylic acid.

Táto skupina sa ďalej označuje ako „Skupina kyselín.This group is hereinafter referred to as the "Acid group.

Ak kyselina vybraná zo „Skupiny kyselín“ je multifunkčná kyselina, soli tvorené s paroxetínom môžu obsahovať premenlivé podiely paroxetínu, v závislosti od počtu kyselinových skupín, ktoré sú naviazané na molekulu paroxetínu. Všetky takéto soli sú zahrnuté v rozsahu tohto vynálezu.If the acid selected from the "Acid group" is a multifunctional acid, the salts formed with paroxetine may contain varying proportions of paroxetine, depending on the number of acid groups that are bound to the paroxetine molecule. All such salts are included within the scope of this invention.

Stérické hľadiská všeobecne diktujú, že v prípade multifunkčnej kyseliny, ktorá má väzbovosť väčšiu než dva, anión kyseliny nebude spojený s viac než s dvoma molekulami paroxetínu.The steric aspects generally dictate that in the case of a multifunctional acid having a binding greater than two, the acid anion will not be associated with more than two molecules of paroxetine.

• ·· ·· ···· ·· ··· · · · · · · • ··· 9 9 9 99• 9 9 9 99

-223Preto vzhľadom na všetky kyseliny v „Skupine kyselín“, vo výhodnom uskutočnení vynález poskytuje paroxetínovú soľ, v ktorej pomer paroxetínu ku kyseline (molový) je 1:1.Therefore, with respect to all acids in the "Acid Group", in a preferred embodiment, the invention provides a paroxetine salt wherein the ratio of paroxetine to acid (molar) is 1: 1.

Vzhľadom na multifunkčné kyseliny v „Skupine kyselín, v ďalšom výhodnom uskutočnení vynález poskytuje paroxetínovú soľ, v ktorej je pomer paroxetínu ku kyseline (molový) 2:1.With respect to the multifunctional acids in the "Acid Group", in another preferred embodiment, the invention provides a paroxetine salt wherein the ratio of paroxetine to acid (molar) is 2: 1.

V soliach s multifunkčnými kyselinami môže byť kyselinový anión spojený s protónom (vodíkovým atómom) okrem paroxetínu alebo sa môže naviazať na iný katión, napríklad katión alkalického kovu alebo amónia, čím sa tvorí zmiešaná soľ.In salts with multifunctional acids, the acidic anion may be coupled to a proton (hydrogen atom) other than paroxetine, or it may bind to another cation, for example an alkali metal or ammonium cation, to form a mixed salt.

Keď kyselina v „Skupine kyselín existuje v enantiomérnych formách, tento vynález zahrnuje soli aj D-kyselín aj L-kyselín individuálne aj racemické zmesi oboch solí, a tiež diastereoizoméry.When the acid in the "Acid group" exists in enantiomeric forms, the present invention includes both D-acid and L-acid salts, both individual and racemic mixtures of both salts, as well as diastereoisomers.

V jednom aspekte nové soli tohto vynálezu sú poskytované v nekryštalickej forme, ktorou môže byť tuhá látka alebo olej. Tento olej sa výhodne absorbuje na tuhom nosiči, zvlášť na nosiči, ktorý je použiteľný ako zložka farmaceutickej zmesi.In one aspect, the novel salts of the invention are provided in a non-crystalline form, which may be a solid or an oil. The oil is preferably absorbed on a solid carrier, especially on a carrier which is useful as a component of a pharmaceutical composition.

V inom uskutočnení sa nové soli podľa tohto vynálezu poskytujú v kryštalickej forme. Keď kryštalická forma existuje ako viac než jedna polymorfná forma, každá polymorfná forma tvorí ďalší uskutočnenie tohto vynálezu.In another embodiment, the novel salts of the invention are provided in crystalline form. When a crystalline form exists as more than one polymorphic form, each polymorphic form forms a further embodiment of the invention.

Paroxetínové soli sa môžu pripraviť pomocou kontaktovania stechiometrických množstiev kyseliny a paroxetinovej voľnej zásady. Výhodne je zásada v roztoku, výhodnejšie sú obe v roztoku. Kyselina môže tiež byť v tuhej forme, za predpokladu, že výsledná soľ nie je tak nerozpustná, že tvorí povlak na pridanej tuhej látke, že bráni ďalšej reakcii. Zmiešané soli sa môžu pripraviť pomocou tvorby prekurzorovej 1:1 soli in situ (alebo 2:1 soľ pre trojfunkčné a vyššie kyseliny), alebo sa použijú vopred pripravené, a kontaktujú sa v roztoku s roztokom obsahujúcim kovový alebo amóniový ión.Paroxetine salts can be prepared by contacting stoichiometric amounts of acid and paroxetine free base. Preferably, the base is in solution, more preferably both are in solution. The acid may also be in solid form, provided that the resulting salt is not so insoluble that it forms a coating on the added solid that prevents further reaction. The mixed salts may be prepared by forming a precursor 1: 1 salt in situ (or a 2: 1 salt for the trifunctional and higher acids), or may be used previously prepared and contacted in solution with a solution containing a metal or ammonium ion.

Najbežnejšie používané rozpúšťadlá sú vhodné na tvorbu pohyblivej formy paroxetinovej voľnej zásady, napríklad toluén, alkoholy, ako napríklad metanol, etanol, propán-2-ol, estery, ako napríklad etylacetát, ketóny, ako napríklad acetón a butanón, halogenované uhľovodíky, ako napríklad dichlórmetán, a étery, ako napríklad tetrahydrofurán a dietyléter. Kyselina zo „Skupiny kyselín“ sa výhodne pridáva ako roztok, výhodne vodný, ak je rozpustná vo vode, voliteľne sa ďalejThe most commonly used solvents are suitable for forming the mobile form of the paroxetine free base, for example toluene, alcohols such as methanol, ethanol, propan-2-ol, esters such as ethyl acetate, ketones such as acetone and butanone, halogenated hydrocarbons such as dichloromethane , and ethers such as tetrahydrofuran and diethyl ether. The acid of the "Acid group" is preferably added as a solution, preferably aqueous, if it is water soluble, optionally further

-224--224-

• ·· • 9 • ··· • ·· • 9 • ··· ·· • · • · ·· • · • · ···· • • ···· • • • · · • · · · • e · • · · • · · · • e · ·· ·· ·· ·· ·· · · • · • · ·· ·· ·· ··

zrieďuje s miešateľným organickým rozpúšťadlom. Kyselina sa môže tiež pridať vo forme rozpustnej soli, napríklad amónna soľ, alebo soľ amíriu, napríklad etylamínu alebo dietylamínu.Dilute with miscible organic solvent. The acid may also be added in the form of a soluble salt, for example, an ammonium salt, or an ammonium salt, for example, ethylamine or diethylamine.

Koncentrácia paroxetínovej zásady je výhodne v rozsahu 5 až 50 % hmotnosť/objem, výhodnejšie v rozsahu 10 až 30%. Koncentrácia kyseliny je výhodne v rozsahu 0,1 až 2 mol/l. Na zvýšenie rozpustnosti sa môžu použiť zvýšené teploty.The concentration of the paroxetine base is preferably in the range of 5 to 50% w / v, more preferably in the range of 10 to 30%. The acid concentration is preferably in the range of 0.1 to 2 mol / l. Elevated temperatures may be used to increase solubility.

Soli sa môžu izolovať v tuhej forme pomocou konvenčných prostriedkov z ich roztoku získaného ako je uvedené vyššie. Napríklad nekryštalická soľ sa môže pripraviť pomocou zrážania z roztoku, sušením rozstrekovaním a sušením vymrazovaním roztokov, odparovaním roztoku na sklo alebo vákuovým sušením olejov, alebo tuhnutím tavenín získaných z reakcie voľnej zásady a kyseliny.The salts can be isolated in solid form by conventional means from their solution obtained as above. For example, a non-crystalline salt may be prepared by precipitation from solution, spray drying and freeze-drying solutions, evaporation of the solution to glass or vacuum drying of oils, or solidification of melts obtained from the reaction of the free base and acid.

Kryštalická soľ sa môže pripraviť pomocou priamej kryštalizácie z rozpúšťadla, v ktorom má produkt obmedzenú rozpustnosť, alebo rozotieraním alebo inou kryštalizáciou nekryštalickej soli. Vo všeobecnosti rozpúšťadlové systémy, ktoré sú vhodné na prípravu paroxetínovej soli, môžu tiež byť použité na rekryštalizáciu. Zlepšený výťažok soli sa získa odparením časti alebo všetkého rozpúšťadla alebo kryštalizáciou pri zvýšenej teplote nasledovanej riadeným chladením, výhodne po etapách. Starostlivé riadenie teploty zrážania a naočkovanie sa môžu použiť na zlepšenie reprodukovateľnosti výrobného procesu a distribúcie veľkosti častíc a formy produktu. Individuálne polymorfné formy sa výhodne kryštalizujú priamo z roztoku soli, hoci sa tiež môže uskutočniť rekryštalizácia roztoku jednej polymorfnej formy použitím očkovania druhej polymorfnej formy.The crystalline salt may be prepared by direct crystallization from a solvent in which the product has limited solubility, or by trituration or other crystallization of the non-crystalline salt. In general, solvent systems that are suitable for preparing the paroxetine salt can also be used for recrystallization. The improved salt yield is obtained by evaporating some or all of the solvent or crystallizing at an elevated temperature followed by controlled cooling, preferably in stages. Careful precipitation temperature control and seeding can be used to improve the reproducibility of the production process and the particle size distribution and product form. The individual polymorphic forms are preferably crystallized directly from the salt solution, although recrystallization of a solution of one polymorphic form can also be performed using seeding of the other polymorphic form.

Alternatívny spôsob prípravy soli paroxetínu s kyselinou zo „Skupiny kyselín“ je začatie so soľou paroxetínu s organickou kyselinou, ako napríklad octová kyselina alebo maleínová kyselina. Použitie inej soli paroxetínu ako východiskového materiálu je vhodné na prípravu kryštalickej soli alebo, ak sa používa prchavá kyselina, ako napríklad kyselina octová, nekryštalickej soli spôsobmi, ktoré zahrnujú odparenie (ako napríklad sušenie vymrazovaním a sušenie striekaním).An alternative method of preparing a salt of paroxetine with an acid from the "Acid group" is to start with a salt of paroxetine with an organic acid such as acetic acid or maleic acid. The use of a paroxetine salt other than the starting material is suitable for preparing the crystalline salt or, if a volatile acid such as acetic acid is used, the non-crystalline salt by methods which include evaporation (such as freeze-drying and spray-drying).

Soľ sa môže získať ako solvát, ak sa počas izolácie z roztoku stáva naviazanou na rozpúšťadlo, v ktorom je rozpustená. Akékoľvek takéto solváty tvoria ďalší aspekt podľa tohto vynálezu. Solváty sa môžu premeniť späť na ·« ·· ···· ·· • · · · · · · ··· · · · t ·A salt can be obtained as a solvate if, during isolation from the solution, it becomes bound to the solvent in which it is dissolved. Any such solvates form another aspect of the invention. Solvates can be converted back to · «·· ······ · · · · · · ···

-225··· ·· ·· ··· nesolvatovanú soľ pomocou zahrievania, napríklad pomocou sušenia v piecke, alebo pomocou opracovania s náhradným rozpúšťadlom, ktoré netvorí solvát.Unsolvated salt by heating, for example by oven drying, or by treatment with a non-solvate substitute solvent.

Pred izoláciou paroxetínovej soli sa z roztoku obsahujúceho soľ môže odstrániť voda pomocou azeotropickej destilácie na zabránenie tvorby hydrátov alebo na získanie produktu v bezvodej forme. V tom prípade sú vhodné rozpúšťadlá pre roztok soli tie, ktoré tvoria s vodou azeotropickú zmes, ako napríklad toluén a propán-2-ol. Treba si tiež všimnúť, že sa môžu na pomoc pri azeotropickom odstraňovaní vody tiež použiť zmesi rozpúšťadiel.Before the isolation of the paroxetine salt, water can be removed from the salt-containing solution by azeotropic distillation to prevent the formation of hydrates or to obtain the product in anhydrous form. In this case, suitable solvents for the salt solution are those that form an azeotropic mixture with water, such as toluene and propan-2-ol. It should also be noted that solvent mixtures can also be used to aid in the azeotropic removal of water.

Paroxetínová voľná zásada sa môže pripraviť podľa postupov všeobecne uvedených v US patente č. 4007196 a EP-B-0223403. Kyseliny v „Skupine kyselín“ sú komerčne dostupné alebo uvedené v literatúre.The paroxetine free base may be prepared according to the procedures generally set forth in U.S. Pat. 4007196 and EP-B-0223403. The acids in the "Acid Group" are commercially available or listed in the literature.

Látky podľa tohto vynálezu nasledujúcich porúch:The substances according to the invention of the following disorders:

Alkoholizmusalcoholism

Depresiadepression

Panické poruchyPanic disorders

Obezita sa môžu použiť na liečenie a prevenciuObesity can be used for treatment and prevention

Úzkosťanxiety

Obsedantno-kompulzívna poruchaObsessive-compulsive disorder

Chronická bolesťChronic pain

Starecká demenciaStarecká dementia

Bulímiabulimia

Sociálna fóbiaSocial phobia

Depresia adolescentov TrudnomyseľnosťDepression of adolescents

Migrénamigraine

Anorexiaanorexia

Pred menštruačný syndróm (PMS)Pre menstrual syndrome (PMS)

Trichotilomániatrichotillomania

Zneužívanie návykových látokSubstance Abuse

Tieto poruchy sú v tomto dokumente ďalej označované ako Poruchy.These disorders are hereinafter referred to as Disorders.

Tento vynález ďalej poskytuje spôsob liečenia a/alebo prevencie jednej alebo viacerých „Porúch“ podávaním účinného a/alebo profylakčného množstva soli podľa tohto vynálezu pacientom, ktorí to potrebujú.The invention further provides a method of treating and / or preventing one or more "Disorders" by administering an effective and / or prophylactic amount of a salt of the invention to a patient in need thereof.

Tento vynález ďalej poskytuje farmaceutické prostriedky na použitie na liečenie a/alebo prevenciu „Porúch“, ktoré obsahujú zmes soli podľa tohto vynálezu s farmaceutický prijateľným nosičom.The invention further provides pharmaceutical compositions for use in the treatment and / or prevention of "Disorders" comprising a mixture of a salt of the invention with a pharmaceutically acceptable carrier.

Tento vynález tiež poskytuje použitie soli podľa tohto vynálezu na liečenie a/alebo prevenciu „Porúch“.The invention also provides the use of a salt of the invention for the treatment and / or prevention of "Disorders".

Tento vynález tiež poskytuje použitie soli podľa tohto vynálezu pri výrobeThe invention also provides the use of a salt of the invention in the manufacture

-226--226-respectively

• ·· • 8 • ··· 8 • ··· ·· · · 8888 9 8 8888 9 8 88 8 8 9 99 8 8 8 88 8 8 9 99 8 8 8 • • • • • 8 • 8 88 88 88 88 88 88 8 e 8 e 88 88 88 88

liekov na liečenie a/alebo prevenciu „Porúch“.medicines to treat and / or prevent “Disorders”.

Najvhodnejšie sa tento vynález aplikuje na liečenie depresie, OCD a paniky.Most preferably, the present invention is applied to the treatment of depression, OCD and panic.

Zmesi podľa tohto vynálezu sú obvykle upravené pre orálne podávanie, ale prípravky na rozpustenie pre parenterálne podávanie sú tiež v rozsahu tohto vynálezu.The compositions of the invention are generally adapted for oral administration, but dissolution formulations for parenteral administration are also within the scope of the invention.

Farmaceutické prostriedky obvykle predstavujú prostriedky v jednotkovej dávke obsahujúcej od 1 do 200 mg aktívnej zložky, počítané vzhľadom na voľnú zásadu, obvyklejšie od 5 do 100 mg, napríklad 10 až 50 mg, napríklad 10, 12,5, 15, 20, 25, 30 alebo 40 mg pre ľudských pacientov. Najvýhodnejšie jednotkové dávky obsahujú 20 mg aktívnej zložky počítané vzhľadom na voľnú zásadu. Takéto zmesi sa normálne berú 1 až 6 krát denne, napríklad 2, 3 alebo 4 krát denne, takže celkové množstvo podaného aktívneho činidla je v rozsahu 5 až 400 mg aktívnej zložky počítané vzhľadom na voľnú zásadu. Najvýhodnejšie sa jednotková dávka berie raz za deň.The pharmaceutical compositions usually represent unit dose formulations containing from 1 to 200 mg of active ingredient, calculated on the free base, more usually from 5 to 100 mg, for example 10 to 50 mg, for example 10, 12.5, 15, 20, 25, 30 or 40 mg for human patients. Most preferred unit doses contain 20 mg of active ingredient calculated on the free base. Such mixtures are normally taken 1 to 6 times a day, for example 2, 3 or 4 times a day, so that the total amount of active agent administered is in the range of 5 to 400 mg of active ingredient calculated with respect to the free base. Most preferably, the unit dose is taken once a day.

Výhodné jednotkové dávkové formy zahrnujú tablety alebo kapsuly.Preferred unit dosage forms include tablets or capsules.

Farmaceutické prostriedky podľa tohto vynálezu sa môžu upravovať pomocou konvenčných spôsobov primiešavania ako napríklad zmiešanie, plnenie a lisovanie.The pharmaceutical compositions of the invention may be formulated by conventional mixing methods such as mixing, filling and compression.

Vhodné nosiče na použitie v tomto vynáleze zahrnujú zried’ovadlo, spojivo, dezintegračné činidlo, farbivo, ochucovadlo a/alebo konzervačnú látku. Tieto činidlá sa môžu používať konvenčným spôsobom, napríklad v spôsobom podobným na spôsoby doteraz používané pre predávané anti-depresívne činidlá.Suitable carriers for use in the present invention include a diluent, a binder, a disintegrant, a colorant, a flavoring, and / or a preservative. These agents may be used in a conventional manner, for example, in a manner similar to those previously used for marketed anti-depressant agents.

Vhodné farmaceutické prostriedky zahrnujú prostriedky opísané v EP-B0223405 a US patente 4,007,196, v ktorých sa produkty podľa tohto vynálezu môžu použiť ako aktívne zložky.Suitable pharmaceutical compositions include those described in EP-B0223405 and US Patent 4,007,196, in which the products of the invention can be used as active ingredients.

Nasledujúce Príklady ilustrujú tento vynález.The following Examples illustrate the invention.

Príklady uskutočnenia vynálezuDETAILED DESCRIPTION OF THE INVENTION

Príklad 1Example 1

Príprava tablietPreparation of tablets

99 9999 9999 9900 99

9 9 9 9 9 99 9 9 9 9

999 9 9 9 9 9999 9 9 9 9 9

-22799-22,799

99 99 999 99 9

Zložky ingredients 20 mg tableta 20 mg tablet 30 mg tableta 30 mg tablet Paroxetínová soľ Paroxetine salt 20,00 mg (počítané ako voľná zásada) 20,00 mg (calculated as free base) 30,00 mg (počítané ako voľná zásada) 30,00 mg (calculated as free base) Hydrogenfosforečnan vápenatý (DCP) Calcium hydrogen phosphate (DCP) 83,34 mg 83.34 mg 125,0 mg 125.0 mg Mikrokryštalická celulóza Microcrystalline cellulose 50,67 mg 50.67 mg 76,0 mg 76.0 mg Škrobglykolát sodný Sodium starch glycolate 8,34 mg 8.34 mg 12,5 mg 12.5 mg Stearan horečnatý Magnesium stearate 1,67 mg 1,67 mg 2,5 mg 2.5 mg

Komerčný zdroj zložiekCommercial source components

Hydrogenfosforečnan vápenatý, dihydrát - Emcompress alebo Ditab*Calcium hydrogen phosphate dihydrate - Emcompress or Ditab *

Mikrokryštalická celulóza - Avicel PH 102*Microcrystalline cellulose - Avicel PH 102 *

Škrobglykolát sodný - Explotab.* * Obchodné značkySodium starch glycolate - Explotab. * * Trademarks

Metódamethod

1. Prechod DCP cez sito a váhu do planétového mixéra.1. Pass the DCP through a sieve and weight into a planetary mixer.

2. Pridanie 30 mesh Paroxetínovej soli do nádoby.2. Add 30 mesh Paroxetine salt to the vessel.

3. Pridanie 20 mesh Avicel a Explotab a miešanie práškov počas 10 minút.3. Add 20 mesh Avicel and Explotab and mix the powders for 10 minutes.

4. Pridanie stearanu horečnatého a miešanie počas 5 minút4. Add magnesium stearate and mix for 5 minutes

Tabletovanie na pentagonálne tablety použitím nasledujúcich otvorov:Tableting into pentagonal tablets using the following holes:

mg tablety 9,5 mm kruhový prierez mg tablety 8,25 mm kruhový prierezmg tablets 9.5 mm circular cross section mg tablets 8.25 mm circular cross section

Tablety sa vyrábajú uspokojivo na jednootvorovom alebo a rotačnom lise.The tablets are produced satisfactorily on a single-hole or rotary press.

Príklad 2Example 2

Príprava tabliet • ·· ·· ···· ·· ··· · · ···· • ··· · · · · ·Preparing Tablets

-228··· ·· ·· ·· ·· ···-228 ··· ·· ·· ·· ·· ···

Zložky ingredients 10 mg tableta 10 mg tablet 20 mg tableta 20 mg tablet 30 mg tableta 30 mg tablet Paroxetínová soľ Paroxetine salt 10,00 mg (počítané, ako voľná zásada) 10.00 mg (calculated as free base) 20,00 mg (počítané, ako voľná zásada) 20,00 mg (calculated as free base) 30,00 mg (počítané, ako voľná zásada) 30,00 mg (calculated as free base) Škrobglykolát sodný Sodium starch glycolate 2,98 mg 2,98 mg 5,95 mg 5,95 mg 8,93 mg 8.93 mg Granulovaný hydrogenfosforečnan vápenatý (DCP) Granular calcium hydrogen phosphate (DCP) 158,88 mg 158.88 mg 317,75 mg 317.75 mg 476,63 mg 476.63 mg (DITAB) alebo Dicafos Stearan horečnatý (DITAB) or Dicafos Magnesium Stearate 1,75 mg 1.75 mg 3,50 mg 3,50 mg 5,25 mg 5,25 mg

Metódamethod

1. Paroxetínová soľ, škrobglykolát sodný a hydrogenfosforečnan vápenatý, dihydrát sa preosiali a zmiešali vo vhodnom zmiešavači.1. Paroxetine salt, sodium starch glycolate and dibasic calcium phosphate, dihydrate are sieved and mixed in a suitable mixer.

(Planetový, Cuble alebo mixér s vysokou energiou strihu) Pridanie stearanu horečnatého a lisovanie na tablety použitím jednootvorového alebo a rotačného tabletovacieho stroja.(Planetary, Cuble or High Energy Shear Mixer) Add magnesium stearate and compress into tablets using a single-hole or rotary tabletting machine.

Claims (11)

1. Paroxetínová soľ kyseliny vybranej zo Skupiny kyselín.A paroxetine salt of an acid selected from the group of acids. 2. Paroxetínová soľ podľa nároku 1,vyznačujúca sa tým, že je to soľ s D-kyselinou.Paroxetine salt according to claim 1, characterized in that it is a salt with D-acid. 3. Paroxetínová soľ podľa nároku 1, v y z n a č u j ú c a sa tým, že je to soľ s L-kyselinou.A paroxetine salt according to claim 1, characterized in that it is an L-acid salt. 4. Paroxetínová soľ podľa nároku 1, 2 alebo 3, vyznačujúca sa t ý m, že molový pomer paroxetínovej voľnej zásady ku kyseline je 1:1.A paroxetine salt according to claim 1, 2 or 3, characterized in that the molar ratio of paroxetine free base to acid is 1: 1. 5. Paroxetínová soľ podľa nároku 1, 2 alebo 3, vyznačujúca sa t ý m, že molový pomer paroxetínovej voľnej zásady ku kyseline je 2:1.A paroxetine salt according to claim 1, 2 or 3, characterized in that the molar ratio of paroxetine free base to acid is 2: 1. 6. Paroxetínová soľ podľa nároku 1, 2, 3,4 alebo 5 v nekryštalickej forme.The paroxetine salt of claim 1, 2, 3, 4 or 5 in non-crystalline form. 7. Paroxetínová soľ podľa nároku 1, 2, 3, 4 alebo 5 v kryštalickej forme.The paroxetine salt of claim 1, 2, 3, 4 or 5 in crystalline form. 8. Spôsob prípravy paroxetínovej soli podľa nároku 1, 2, 3, 4, 5 alebo 6, v yznačujúci sa tým, že zahŕňa zrážanie z roztoku paroxetínovej soli, sušenie striekaním alebo sušenie vymrazovaním roztoku paroxetínovej soli, odparovanie roztoku paroxetínovej soli na sklo, alebo vákuové sušenie olejov paroxetínovej soli, alebo tuhnutie tavenín paroxetínovej soli.A process for preparing a paroxetine salt according to claim 1, 2, 3, 4, 5 or 6, comprising precipitating from a paroxetine salt solution, spray drying or freeze-drying the paroxetine salt solution, evaporating the paroxetine salt solution onto the glass, or vacuum drying the paroxetine salt oils, or solidifying the melts of the paroxetine salt. 9. Spôsob prípravy paroxetínovej soli podľa nároku 1, 2, 3, 4, 5 alebo 7, v yznačujúci sa tým, že zahŕňa kryštalizáciu alebo rekryštalizáciu z roztoku paroxetínovej soli.A process for preparing a paroxetine salt according to claim 1, 2, 3, 4, 5 or 7, characterized in that it comprises crystallization or recrystallization from a solution of the paroxetine salt. 10. Spôsob podľa nároku 8 alebo 9, vyznačujúci sa tým, že roztok, olej alebo tavenina paroxetínovej soli sa pripraví pôsobením kyseliny • ·· ·· ···· ·· ··· · · · · · · • ··· · · · · · ······ · · · · • · · ···· ·· ··· ·· ·· ·· ·· ·Process according to claim 8 or 9, characterized in that the solution, oil or melt of the paroxetine salt is prepared by treatment with an acid. · · · ·········································· -230vybranej zo Skupiny kyselín alebo jej amónnou alebo aminovou soľou na paroxetínovú voľnú zásadu alebo jej soľ s organickou kyselinou.-230 selected from the group of acids or an ammonium or amine salt thereof for paroxetine free base or an organic acid salt thereof. 11. Použitie paroxetínovej soli s kyselinou vybranou zo Skupiny kyselín na výrobu lieku na liečenie a/alebo prevenciu jednej alebo viacerých porúch vybraných zo skupiny zahrnujúcej alkoholizmus, depresiu, panické poruchy, obezitu, migrénu, anorexiu, pred-menštruačný syndróm, trichotilomániu, zneužívanie návykových látok, úzkosť, obsedantno-kompulzívne poruchy, chronickú bolesť, stareckú demenciu, bulímiu, sociálnu fóbiu, depresiu adolescentov a trudnomyseľnosť.Use of a paroxetine salt with an acid selected from the group of acids for the manufacture of a medicament for the treatment and / or prevention of one or more disorders selected from the group consisting of alcoholism, depression, panic disorder, obesity, migraine, anorexia, pre-menstrual syndrome, trichothilomania anxiety, obsessive-compulsive disorder, chronic pain, aging dementia, bulimia, social phobia, adolescent depression, and stomach-related disorder.
SK2024-2000A 1998-07-02 1999-06-30 Salts of paroxetine SK20242000A3 (en)

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