SG19795G - Piperidyl-substituted indoles - Google Patents

Piperidyl-substituted indoles

Info

Publication number
SG19795G
SG19795G SG19795A SG19795A SG19795G SG 19795 G SG19795 G SG 19795G SG 19795 A SG19795 A SG 19795A SG 19795 A SG19795 A SG 19795A SG 19795 G SG19795 G SG 19795G
Authority
SG
Singapore
Prior art keywords
piperidyl
substituted indoles
methyl
mammals
mammal
Prior art date
Application number
SG19795A
Other languages
English (en)
Inventor
Jens Kristian Perregaard
Brenda Costall
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to DK152090A priority Critical patent/DK152090D0/da
Priority to IE213791A priority patent/IE65421B1/en
Priority to ZA914747A priority patent/ZA914747B/xx
Priority to IL9857491A priority patent/IL98574A/en
Priority to NZ238655A priority patent/NZ238655A/en
Priority to AT91912147T priority patent/ATE113838T1/de
Priority to DK91912147.5T priority patent/DK0533824T3/da
Priority to JP51105091A priority patent/JP3332232B2/ja
Priority to AU80684/91A priority patent/AU650464B2/en
Priority to DE69105135T priority patent/DE69105135T2/de
Priority to EP91912147A priority patent/EP0533824B1/en
Priority to CA002085987A priority patent/CA2085987C/en
Priority to PCT/DK1991/000168 priority patent/WO1992000070A1/en
Priority to US07/999,482 priority patent/US5439922A/en
Priority to FI925801A priority patent/FI925801A/fi
Priority to NO92924949A priority patent/NO924949L/no
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Priority to SG19795A priority patent/SG19795G/en
Priority to HK51395A priority patent/HK51395A/xx
Publication of SG19795G publication Critical patent/SG19795G/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
SG19795A 1990-06-22 1995-02-07 Piperidyl-substituted indoles SG19795G (en)

Priority Applications (18)

Application Number Priority Date Filing Date Title
DK152090A DK152090D0 (da) 1990-06-22 1990-06-22 Piperidylsubstituerede indolderivater
ZA914747A ZA914747B (en) 1990-06-22 1991-06-20 Piperidyl-substituted indoles
IL9857491A IL98574A (en) 1990-06-22 1991-06-20 Pharmaceutical compositions for the treatment of anxiety comprising a piperidyl indole derivative and some such novel compounds
IE213791A IE65421B1 (en) 1990-06-22 1991-06-20 Piperidyl-substituted indoles
CA002085987A CA2085987C (en) 1990-06-22 1991-06-21 Piperidyl-substituted indoles
DK91912147.5T DK0533824T3 (da) 1990-06-22 1991-06-21 Piperidylsubstituerede indoler
JP51105091A JP3332232B2 (ja) 1990-06-22 1991-06-21 ピペリジル―置換されたインドール
AU80684/91A AU650464B2 (en) 1990-06-22 1991-06-21 Piperidyl-substituted indoles
DE69105135T DE69105135T2 (de) 1990-06-22 1991-06-21 Piperidyl-substituierte indole.
NZ238655A NZ238655A (en) 1990-06-22 1991-06-21 Piperidyl-substituted indole derivatives and pharmaceutical compositions
AT91912147T ATE113838T1 (de) 1990-06-22 1991-06-21 Piperidyl-substituierte indole.
PCT/DK1991/000168 WO1992000070A1 (en) 1990-06-22 1991-06-21 Piperidyl-substituted indoles
EP91912147A EP0533824B1 (en) 1990-06-22 1991-06-21 Piperidyl-substituted indoles
US07/999,482 US5439922A (en) 1990-06-22 1992-12-17 Piperidyl-substituted indoles for treating anxiety
FI925801A FI925801A (fi) 1990-06-22 1992-12-21 Piperidyl-substituerade indoler
NO92924949A NO924949L (no) 1990-06-22 1992-12-21 Piperidylsubstituerte indoler
SG19795A SG19795G (en) 1990-06-22 1995-02-07 Piperidyl-substituted indoles
HK51395A HK51395A (en) 1990-06-22 1995-04-06 Piperidyl-substituted indoles.

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK152090A DK152090D0 (da) 1990-06-22 1990-06-22 Piperidylsubstituerede indolderivater
SG19795A SG19795G (en) 1990-06-22 1995-02-07 Piperidyl-substituted indoles

Publications (1)

Publication Number Publication Date
SG19795G true SG19795G (en) 1995-08-18

Family

ID=26065861

Family Applications (1)

Application Number Title Priority Date Filing Date
SG19795A SG19795G (en) 1990-06-22 1995-02-07 Piperidyl-substituted indoles

Country Status (17)

Country Link
US (1) US5439922A (ja)
EP (1) EP0533824B1 (ja)
JP (1) JP3332232B2 (ja)
AT (1) ATE113838T1 (ja)
AU (1) AU650464B2 (ja)
CA (1) CA2085987C (ja)
DE (1) DE69105135T2 (ja)
DK (2) DK152090D0 (ja)
FI (1) FI925801A (ja)
HK (1) HK51395A (ja)
IE (1) IE65421B1 (ja)
IL (1) IL98574A (ja)
NO (1) NO924949L (ja)
NZ (1) NZ238655A (ja)
SG (1) SG19795G (ja)
WO (1) WO1992000070A1 (ja)
ZA (1) ZA914747B (ja)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5643784A (en) * 1990-12-04 1997-07-01 H, Lundbeck A/S Indan derivatives
NZ243065A (en) * 1991-06-13 1995-07-26 Lundbeck & Co As H Piperidine derivatives and pharmaceutical compositions
DK55192D0 (da) * 1992-04-28 1992-04-28 Lundbeck & Co As H 1-piperazino-1,2-dihydroindenderivater
DK78692D0 (da) * 1992-06-12 1992-06-12 Lundbeck & Co As H Dimere piperidin- og piperazinderivater
DK148392D0 (da) * 1992-12-09 1992-12-09 Lundbeck & Co As H Heterocykliske forbindelser
DK148292D0 (da) * 1992-12-09 1992-12-09 Lundbeck & Co As H Forbindelser
US5484788A (en) * 1993-03-26 1996-01-16 Beth Israel Hospital Association Buspirone as a systemic immunosuppressant
US5631017A (en) * 1993-03-26 1997-05-20 Beth Israel Deaconess Medical Center, Inc. Topical application of buspirone for treatment of pathological conditions associated with immune responses
DK123493D0 (da) * 1993-11-01 1993-11-01 Lundbeck & Co As H Compounds
DK139593D0 (da) * 1993-12-16 1993-12-16 Lundbeck & Co As H Compounds
DE19500689A1 (de) * 1995-01-12 1996-07-18 Merck Patent Gmbh Indolpiperidin-Derivate
US5637314A (en) * 1995-06-07 1997-06-10 Beth Israel Deaconess Medical Center, Inc. Topical and systemic application of buspirone or derivatives thereof for treating atopic dermatitis
GB9523583D0 (en) * 1995-11-17 1996-01-17 Merck Sharp & Dohme Therapeutic agents
DE19707628A1 (de) * 1997-02-26 1998-08-27 Merck Patent Gmbh Oxazolidinone
US6489341B1 (en) * 1999-06-02 2002-12-03 Sepracor Inc. Methods for the treatment of neuroleptic and related disorders using sertindole derivatives
US20070212412A1 (en) * 2005-09-08 2007-09-13 H. Lundbeck A/S Stable solid formulation of sertindole
TW200821296A (en) * 2006-06-01 2008-05-16 Lundbeck & Co As H Use of sertindole for the preventive treatment of suicidal behaviour

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2258843B1 (ja) * 1974-01-30 1977-09-09 Roussel Uclaf
US4208417A (en) * 1978-06-29 1980-06-17 Pharmindustrie Indole derivatives and their use as anxiolytics
IE58370B1 (en) * 1985-04-10 1993-09-08 Lundbeck & Co As H Indole derivatives
US4997841A (en) * 1987-08-13 1991-03-05 Glaxo Group Limited Indole derivatives
GB8819024D0 (en) * 1988-08-10 1988-09-14 Glaxo Group Ltd Chemical compounds
DK158590D0 (da) * 1990-07-02 1990-07-02 Lundbeck & Co As H Indolderivater

Also Published As

Publication number Publication date
DE69105135D1 (de) 1994-12-15
ZA914747B (en) 1992-03-25
EP0533824B1 (en) 1994-11-09
FI925801A0 (fi) 1992-12-21
IL98574A0 (en) 1992-07-15
NZ238655A (en) 1993-11-25
NO924949L (no) 1993-02-19
DK152090D0 (da) 1990-06-22
NO924949D0 (no) 1992-12-21
CA2085987A1 (en) 1991-12-23
AU8068491A (en) 1992-01-23
CA2085987C (en) 2000-08-22
ATE113838T1 (de) 1994-11-15
JPH05509080A (ja) 1993-12-16
HK51395A (en) 1995-04-13
DK0533824T3 (da) 1995-05-01
DE69105135T2 (de) 1995-03-23
AU650464B2 (en) 1994-06-23
WO1992000070A1 (en) 1992-01-09
US5439922A (en) 1995-08-08
IE65421B1 (en) 1995-10-18
EP0533824A1 (en) 1993-03-31
JP3332232B2 (ja) 2002-10-07
FI925801A (fi) 1992-12-21
IE912137A1 (en) 1992-01-01
IL98574A (en) 1995-11-27

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