SG158858A1 - Preparation of pharmaceutical salts of piperazine compounds - Google Patents

Preparation of pharmaceutical salts of piperazine compounds

Info

Publication number
SG158858A1
SG158858A1 SG201000065-1A SG2010000651A SG158858A1 SG 158858 A1 SG158858 A1 SG 158858A1 SG 2010000651 A SG2010000651 A SG 2010000651A SG 158858 A1 SG158858 A1 SG 158858A1
Authority
SG
Singapore
Prior art keywords
preparation
pharmaceutical salts
salts
piperazine compounds
rotameric
Prior art date
Application number
SG201000065-1A
Other languages
English (en)
Inventor
Wenxue Wu
Loc Thanh Tran
Bosco Daeaesa
Feng Liang
William Leong
Hong-Chang Lee
Kevin Klopfer
Vijay Sabesen
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of SG158858A1 publication Critical patent/SG158858A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SG201000065-1A 2005-01-06 2006-01-05 Preparation of pharmaceutical salts of piperazine compounds SG158858A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US64191005P 2005-01-06 2005-01-06

Publications (1)

Publication Number Publication Date
SG158858A1 true SG158858A1 (en) 2010-02-26

Family

ID=36592935

Family Applications (1)

Application Number Title Priority Date Filing Date
SG201000065-1A SG158858A1 (en) 2005-01-06 2006-01-05 Preparation of pharmaceutical salts of piperazine compounds

Country Status (10)

Country Link
US (2) US7521452B2 (es)
EP (1) EP1836190A2 (es)
JP (1) JP2008526862A (es)
CN (1) CN101133048A (es)
AR (1) AR052865A1 (es)
CA (1) CA2594109A1 (es)
MX (1) MX2007008281A (es)
SG (1) SG158858A1 (es)
WO (1) WO2006074269A2 (es)
ZA (1) ZA200705514B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006074269A2 (en) * 2005-01-06 2006-07-13 Schering Corporation Preparation of pharmaceutical salts of piperazine compounds
WO2009111218A2 (en) * 2008-02-29 2009-09-11 Schering Corporation Ccr5 antagonists as prophylactics for preventing hiv infection and methods of inhibiting transmission of same

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1632479B1 (en) * 1999-05-04 2011-01-12 Schering Corporation Pharmaceutical compositions comprising CCR5 antagonizing piperazine derivatives
US6270325B1 (en) * 1999-09-14 2001-08-07 Hsieh Hsin-Mao Magnetically assembled cooling fan
AUPQ887100A0 (en) 2000-07-19 2000-08-10 Dynamic Digital Depth Research Pty Ltd Image processing and encoding techniques
AU2002255947B8 (en) * 2001-03-29 2005-11-17 Schering Corporation CCR5 antagonists useful for treating AIDS
CA2468525A1 (en) * 2001-11-29 2003-06-12 Schering Corporation Process for the preparation of compositions having an increased amount of pharmaceutically active salts of rotamers of 4-[4-[(1r)-[4-(trifluoromethyl)phenyl]-2-methoxyethyl]-(3s)-methyl-1-piperazinyl]-4-methyl-1-[(4,6-dimethyl-5-pyrimidinyl)carbonyl]
JP2005518424A (ja) * 2001-11-29 2005-06-23 シェーリング コーポレイション Aidsおよび関連するhiv感染の処置のためのccr5−アンタゴニストとしての4((z)−(4−ブロモフェニル)エトキシイミノ)メチル)−1’−((2,4−ジメチル−1−オキシド−3−ピリジニルカルボニル)−4’−メチル−1,4’ビピペリジンの薬学的塩の調製
WO2006074269A2 (en) * 2005-01-06 2006-07-13 Schering Corporation Preparation of pharmaceutical salts of piperazine compounds

Also Published As

Publication number Publication date
US20090093496A1 (en) 2009-04-09
ZA200705514B (en) 2008-09-25
MX2007008281A (es) 2007-09-07
CN101133048A (zh) 2008-02-27
CA2594109A1 (en) 2006-07-13
US20060241295A1 (en) 2006-10-26
AR052865A1 (es) 2007-04-11
US7521452B2 (en) 2009-04-21
JP2008526862A (ja) 2008-07-24
EP1836190A2 (en) 2007-09-26
WO2006074269A2 (en) 2006-07-13
WO2006074269A3 (en) 2006-09-14

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