SG11201809802PA - Compositions for treating or preventing vasomotor symptoms - Google Patents

Compositions for treating or preventing vasomotor symptoms

Info

Publication number
SG11201809802PA
SG11201809802PA SG11201809802PA SG11201809802PA SG11201809802PA SG 11201809802P A SG11201809802P A SG 11201809802PA SG 11201809802P A SG11201809802P A SG 11201809802PA SG 11201809802P A SG11201809802P A SG 11201809802PA SG 11201809802P A SG11201809802P A SG 11201809802PA
Authority
SG
Singapore
Prior art keywords
international
compositions
osaka
treating
pct
Prior art date
Application number
SG11201809802PA
Other languages
English (en)
Inventor
Joseph M Palumbo
Original Assignee
Mitsubishi Tanabe Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Tanabe Pharma Corp filed Critical Mitsubishi Tanabe Pharma Corp
Publication of SG11201809802PA publication Critical patent/SG11201809802PA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Vascular Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SG11201809802PA 2016-06-13 2017-06-12 Compositions for treating or preventing vasomotor symptoms SG11201809802PA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662349179P 2016-06-13 2016-06-13
PCT/JP2017/021569 WO2017217351A1 (en) 2016-06-13 2017-06-12 Compositions for treating or preventing vasomotor symptoms

Publications (1)

Publication Number Publication Date
SG11201809802PA true SG11201809802PA (en) 2018-12-28

Family

ID=59101629

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201809802PA SG11201809802PA (en) 2016-06-13 2017-06-12 Compositions for treating or preventing vasomotor symptoms

Country Status (17)

Country Link
US (2) US10993939B2 (zh)
EP (2) EP4140484A1 (zh)
JP (1) JP6943887B2 (zh)
KR (2) KR20230005413A (zh)
CN (4) CN114748624A (zh)
AU (2) AU2017285609B2 (zh)
BR (1) BR112018075403A2 (zh)
CA (1) CA3022808A1 (zh)
CO (1) CO2018013692A2 (zh)
ES (1) ES2957232T3 (zh)
IL (1) IL262664B (zh)
MX (1) MX2018015399A (zh)
PH (1) PH12018502618A1 (zh)
RU (1) RU2768875C2 (zh)
SG (1) SG11201809802PA (zh)
TW (1) TWI739850B (zh)
WO (1) WO2017217351A1 (zh)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3727383A1 (en) 2017-12-19 2020-10-28 Mitsubishi Tanabe Pharma Corporation Compositions and methods for treating or preventing vasomotor symptoms
CN113677334B (zh) * 2019-02-01 2024-04-09 马歇尔大学科研协会 瞬时受体电位melastatin 8(trpm8)拮抗剂和相关方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006122156A2 (en) * 2005-05-09 2006-11-16 Hydra Biosciences, Inc. Compounds for modulating trpv3 function
WO2009073788A1 (en) 2007-12-07 2009-06-11 Firestone Leigh H Compositions and methods for treating menopausal females
CA2747637A1 (en) 2008-12-18 2010-07-15 Janssen Pharmaceutica Nv Sulfamides as trpm8 modulators
WO2010103381A1 (en) 2009-03-13 2010-09-16 Glenmark Pharmaceuticals S.A. Spirocyclic piperidine derivatives as trpm 8 modulators
EP2424517A4 (en) 2009-05-01 2013-01-23 Raqualia Pharma Inc SULFAMOYLBENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS
TW201103941A (en) 2009-06-10 2011-02-01 Janssen Pharmaceutica Nv Benzimidazole derivatives useful as TRPM8 channel modulators
EP2481727A1 (en) 2011-01-28 2012-08-01 Dompe S.p.A. TRPM8 receptor antagonists
PL2686302T3 (pl) * 2011-03-16 2017-01-31 Mitsubishi Tanabe Pharma Corporation Związki sulfonamidowe mające działanie antagonistyczne dla TRPMS
JP2014527511A (ja) 2011-06-24 2014-10-16 アムジエン・インコーポレーテツド Trpm8拮抗剤及び治療におけるそれらの使用
DK2793883T3 (en) 2011-12-19 2018-07-30 Dompe Farm Spa TRPM8 antagonists
WO2014042238A1 (ja) * 2012-09-14 2014-03-20 田辺三菱製薬株式会社 スルホンアミド化合物
JP5985453B2 (ja) * 2012-09-14 2016-09-06 田辺三菱製薬株式会社 医薬組成物
JP6352413B2 (ja) * 2013-10-22 2018-07-04 エドワード タク ウェイWEI, Edward Tak 感覚的不快感の治療向け局所薬としてのジ−イソプロピル−アルカン(dapa)化合物

Also Published As

Publication number Publication date
EP3468557A1 (en) 2019-04-17
WO2017217351A1 (en) 2017-12-21
AU2017285609B2 (en) 2022-08-18
IL262664B (en) 2021-10-31
CA3022808A1 (en) 2017-12-21
ES2957232T3 (es) 2024-01-15
PH12018502618A1 (en) 2019-10-07
CN113384577A (zh) 2021-09-14
CN113398124A (zh) 2021-09-17
MX2018015399A (es) 2019-04-29
CO2018013692A2 (es) 2019-01-18
JP6943887B2 (ja) 2021-10-06
IL262664A (en) 2018-12-31
TWI739850B (zh) 2021-09-21
EP3468557B1 (en) 2023-07-26
US20210177830A1 (en) 2021-06-17
BR112018075403A2 (pt) 2019-03-19
KR20190017800A (ko) 2019-02-20
US10993939B2 (en) 2021-05-04
AU2022211877A1 (en) 2022-09-01
RU2019100424A (ru) 2020-07-15
US20190142821A1 (en) 2019-05-16
JP2019517573A (ja) 2019-06-24
RU2768875C2 (ru) 2022-03-25
EP4140484A1 (en) 2023-03-01
RU2019100424A3 (zh) 2020-09-24
KR20230005413A (ko) 2023-01-09
AU2017285609A1 (en) 2019-01-03
TW201803595A (zh) 2018-02-01
CN114748624A (zh) 2022-07-15
CN109310689A (zh) 2019-02-05

Similar Documents

Publication Publication Date Title
SG11201909949XA (en) Targeted immunotolerance
SG11201811470PA (en) Pyrazolopyrimidine derivatives as kinase inhibitor
SG11201808566WA (en) Polymorphic form of n-{6-(2-hydroxypropan-2-yl)-2-[2-(methylsulphonyl)ethyl]-2h-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide
SG11201909325RA (en) 2-amino-quinoline derivatives
SG11201804758QA (en) Aqueous pharmaceutical formulation comprising anti-pd-1 antibody avelumab
SG11201906891RA (en) Methods for the administration of certain vmat2 inhibitors
SG11201906386XA (en) Combination therapy involving diaryl macrocyclic compounds
SG11201810280YA (en) Spiro-lactam nmda receptor modulators and uses thereof
SG11201806583XA (en) Compositions containing tucaresol or its analogs
SG11201907023UA (en) Method of reducing neutropenia
SG11201906436VA (en) Novel heterocyclic compound, its preparation method, and pharmaceutical composition comprising the same
SG11201901558VA (en) Pth compounds with low peak-to-trough ratios
SG11201809751XA (en) Egfr inhibitor compounds
SG11201408237YA (en) Compound as wnt signaling inhibitor, composition, and use thereof
SG11201900558RA (en) Spiro-lactam nmda receptor modulators and uses thereof
SG11201408750VA (en) NOVEL FUSED PYRIDINE DERIVATIVES USEFUL AS c-MET TYROSINE KINASE INHIBITORS
SG11201900551WA (en) Spiro-lactam nmda receptor modulators and uses thereof
SG11201900546UA (en) Spiro-lactam and bis-spiro-lactam nmda receptor modulators and uses thereof
SG11201900633XA (en) Piperidine cxcr7 receptor modulators
SG11201805001UA (en) Method of treating influenza a
SG11201808686VA (en) Synthesis of indazoles
SG11201902949PA (en) Pharmaceutical compositions and methods of treating cardiovascular diseases
SG11201907356SA (en) Piperidine-substituted mnk inhibitors and methods related thereto
SG11201805149XA (en) Compositions comprising 15-hepe and methods of using the same
SG11201900214UA (en) Iso-citrate dehydrogenase (idh) inhibitor