SE7708626L - METHODS OF PREPARING OXIMIN DERIVATIVES OF 3-CARBAMOYLOXIMETHYL-7-AMINOTIAZOLYL-ACETAMIDOCEFALOSPORANIC ACID - Google Patents
METHODS OF PREPARING OXIMIN DERIVATIVES OF 3-CARBAMOYLOXIMETHYL-7-AMINOTIAZOLYL-ACETAMIDOCEFALOSPORANIC ACIDInfo
- Publication number
- SE7708626L SE7708626L SE7708626A SE7708626A SE7708626L SE 7708626 L SE7708626 L SE 7708626L SE 7708626 A SE7708626 A SE 7708626A SE 7708626 A SE7708626 A SE 7708626A SE 7708626 L SE7708626 L SE 7708626L
- Authority
- SE
- Sweden
- Prior art keywords
- acid
- oximin
- carbamoyloximethyl
- aminotiazolyl
- acetamidocefalosporanic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
The syn isomers of the compounds of formula: <IMAGE> , in which R1 represents a saturated or unsaturated C1-C4 alkyl and A represents hydrogen or one equivalent of an alkali metal or alkaline-earth metal or of an amine organic base, are prepared from the syn isomers of the corresponding compounds in which the amino group of the thiazolyl radical is substituted by a group which can be removed by acid hydrolysis or by hydrogenolysis, or by a chloroacetyl group; in the first case, an acid hydrolysis or a hydrogenolysis is carried out, in the second case treatment is carried out with thiourea. The compounds obtained have antibacterial properties; they can be used in the treatment of infectious diseases, especially of staphylococcias and of colibacilloses.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7625326A FR2361895A1 (en) | 1976-08-20 | 1976-08-20 | NEW OXIMES DERIVED FROM 3-CARBAMOYLOXYMETHYL 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SE7708626L true SE7708626L (en) | 1978-02-21 |
Family
ID=9177033
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7708626A SE7708626L (en) | 1976-08-20 | 1977-07-27 | METHODS OF PREPARING OXIMIN DERIVATIVES OF 3-CARBAMOYLOXIMETHYL-7-AMINOTIAZOLYL-ACETAMIDOCEFALOSPORANIC ACID |
Country Status (18)
| Country | Link |
|---|---|
| JP (1) | JPS5325595A (en) |
| AT (1) | AT357671B (en) |
| AU (1) | AU510300B2 (en) |
| BE (1) | BE857933A (en) |
| CH (1) | CH626088A5 (en) |
| DE (1) | DE2737504A1 (en) |
| DK (1) | DK369677A (en) |
| ES (1) | ES461764A1 (en) |
| FR (1) | FR2361895A1 (en) |
| GB (1) | GB1584398A (en) |
| IE (1) | IE45865B1 (en) |
| IL (1) | IL52709A (en) |
| LU (1) | LU77993A1 (en) |
| NL (1) | NL7709258A (en) |
| PT (1) | PT66944B (en) |
| SE (1) | SE7708626L (en) |
| SU (1) | SU700065A3 (en) |
| ZA (1) | ZA775039B (en) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2367756B1 (en) * | 1976-04-12 | 1985-07-05 | Fujisawa Pharmaceutical Co | 2-ALCOXYAMINO-2- (AMINO-1,3-THIAZOLYL) ACETICS DERIVATIVES AND THEIR USE |
| PH17188A (en) * | 1977-03-14 | 1984-06-14 | Fujisawa Pharmaceutical Co | New cephem and cepham compounds and their pharmaceutical compositions and method of use |
| DE2714880A1 (en) * | 1977-04-02 | 1978-10-26 | Hoechst Ag | CEPHEMDER DERIVATIVES AND PROCESS FOR THEIR PRODUCTION |
| SE445350B (en) * | 1978-04-14 | 1986-06-16 | Roussel Uclaf | OXIMO DERIVATIVES OF 3-AZIDOMETHYL-7-AMINO-THIAZOLYL-ACETAMIDO-CEPHALOSPORANIC ACID AND ITS USE AS ANTIBIOTICS |
| IL61458A0 (en) * | 1979-12-07 | 1980-12-31 | Erba Farmitalia | N-substituted thiazolyl derivatives of oximino-substituted cephalosporins, their preparation and pharmalceutical compositions containing them |
| FR2475043A2 (en) * | 1980-02-06 | 1981-08-07 | Roussel Uclaf | Amino:thiazolyl hydroxy:imino acetic ester(s) - protected on the amino gp. are intermediates for cephalosporanic acid antibiotics |
| AU1638183A (en) * | 1982-06-30 | 1984-01-05 | Glaxo Group Limited | Cephalosporin antibiotics |
| JPS60190783A (en) * | 1983-12-21 | 1985-09-28 | Sumitomo Seiyaku Kk | Cephem compound |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1399086A (en) * | 1971-05-14 | 1975-06-25 | Glaxo Lab Ltd | Cephalosporin compounds |
-
1976
- 1976-08-20 FR FR7625326A patent/FR2361895A1/en active Granted
-
1977
- 1977-07-27 SE SE7708626A patent/SE7708626L/en not_active Application Discontinuation
- 1977-08-12 IL IL52709A patent/IL52709A/en unknown
- 1977-08-16 SU SU772511698A patent/SU700065A3/en active
- 1977-08-19 DK DK369677A patent/DK369677A/en not_active Application Discontinuation
- 1977-08-19 BE BE180282A patent/BE857933A/en not_active IP Right Cessation
- 1977-08-19 CH CH1022777A patent/CH626088A5/en not_active IP Right Cessation
- 1977-08-19 AU AU28062/77A patent/AU510300B2/en not_active Expired
- 1977-08-19 LU LU77993A patent/LU77993A1/xx unknown
- 1977-08-19 ES ES461764A patent/ES461764A1/en not_active Expired
- 1977-08-19 GB GB34847/77A patent/GB1584398A/en not_active Expired
- 1977-08-19 IE IE1748/77A patent/IE45865B1/en unknown
- 1977-08-19 PT PT66944A patent/PT66944B/en unknown
- 1977-08-19 DE DE19772737504 patent/DE2737504A1/en not_active Withdrawn
- 1977-08-19 AT AT601677A patent/AT357671B/en not_active IP Right Cessation
- 1977-08-19 ZA ZA00775039A patent/ZA775039B/en unknown
- 1977-08-20 JP JP10007077A patent/JPS5325595A/en active Pending
- 1977-08-22 NL NL7709258A patent/NL7709258A/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| BE857933A (en) | 1978-02-20 |
| IL52709A0 (en) | 1977-10-31 |
| SU700065A3 (en) | 1979-11-25 |
| FR2361895B1 (en) | 1978-12-15 |
| LU77993A1 (en) | 1978-04-27 |
| DK369677A (en) | 1978-02-21 |
| NL7709258A (en) | 1978-02-22 |
| DE2737504A1 (en) | 1978-02-23 |
| ATA601677A (en) | 1979-12-15 |
| CH626088A5 (en) | 1981-10-30 |
| GB1584398A (en) | 1981-02-11 |
| JPS5325595A (en) | 1978-03-09 |
| AT357671B (en) | 1980-07-25 |
| AU2806277A (en) | 1979-02-22 |
| ZA775039B (en) | 1978-09-27 |
| IE45865L (en) | 1978-02-20 |
| IL52709A (en) | 1981-01-30 |
| ES461764A1 (en) | 1978-09-01 |
| IE45865B1 (en) | 1982-12-15 |
| PT66944A (en) | 1977-09-01 |
| PT66944B (en) | 1979-11-12 |
| FR2361895A1 (en) | 1978-03-17 |
| AU510300B2 (en) | 1980-06-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| NAV | Patent application has lapsed |
Ref document number: 7708626-2 |